Target-based Classification of Drugs

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 G Protein-coupled receptors
 
 Ion channels
   Ligand-gated ion channels
   Voltage-gated ion channels
     Sodium channels
     Calcium channels
       CACNA1-T [HSA:8911 8912 8913] [KO:K04856 K04855 K04854]
       CACNA1B [HSA:774] [KO:K04849]
       CACNA1-L [HSA:775 776 778 779] [KO:K04850 K04851 K04853 K04857]
         D02537  Dronedarone (INN)
         D03914  Dronedarone hydrochloride (USP) <US>
         D07845  Diltiazem (INN)
         D00616  Diltiazem hydrochloride (JP18/USP) <JP/US>
         D03830  Diltiazem malate (USAN)
         D01369  Bevantolol hydrochloride (JAN/USAN) <JP>
         D07450  Amlodipine (USP/INN)
         D00615  Amlodipine besylate (USP) <JP/US>
         D02914  Amlodipine maleate (USAN)
         D11881  Amlodipine benzoate <US>
         D00319  Felodipine (JP18/USP/INN) <JP/US>
         D00349  Isradipine (USP/INN) <US>
         D08270  Nicardipine (INN)
         D00617  Nicardipine hydrochloride (JP18/USAN) <JP/US>
         D00437  Nifedipine (JP18/USP/INN) <JP/US>
         D00438  Nimodipine (USP/INN) <US>
         D00618  Nisoldipine (JAN/USAN/INN) <US>
         D00629  Nitrendipine (JP18/USAN/INN) <JP>
         D04657  Lacidipine (USAN/INN)
         D01908  Nilvadipine (JP18/USAN/INN) <JP>
         D08155  Manidipine (INN)
         D01553  Manidipine hydrochloride (JP18) <JP>
         D07494  Barnidipine (INN)
         D01104  Barnidipine hydrochloride (JAN) <JP>
         D08111  Lercanidipine (INN)
         D01849  Lercanidipine hydrochloride (JAN/USAN)
         D01173  Cilnidipine (JP18/INN) <JP>
         D07509  Benidipine (INN)
         D02045  Benidipine hydrochloride (JP18) <JP>
         D08892  Clevidipine (USAN/INN) <US>
         D08941  Levamlodipine malate (USAN)
         D11723  Levamlodipine maleate (USAN) <US>
         D08217  Mibefradil (INN)
         D05024  Mibefradil dihydrochloride (USAN)
         D02356  Verapamil (USAN/INN)
         D00619  Verapamil hydrochloride (JP18/USP) <JP/US>
         D08009  Gallopamil (INN)
         D01969  Gallopamil hydrochloride (JAN)
         D07185  Fendiline (INN)
         D07943  Fendiline hydrochloride
         D07520  Bepridil (INN)
         D00631  Bepridil hydrochloride (USAN) <JP>
         D08340  Perhexiline (INN)
         D05442  Perhexiline maleate (USAN)
         D08441  Propiverine (INN)
         D01007  Propiverine hydrochloride (JP18) <JP>
         D00495  Paramethadione (INN)
         D00537  Topiramate (JAN/USP/INN) <JP/US>
         D01145  Azelnidipine (JP18/INN) <JP>
         D01151  Lemildipine (JAN/INN)
         D01171  Monatepil maleate (JAN/USAN)
         D01562  Aranidipine (JAN/INN)
         D01604  Efonidipine hydrochloride ethanolate (JAN) <JP>
         D01933  Vatanidipine hydrochloride (JAN)
         D03067  Belfosdil (USAN/INN)
         D03536  Clentiazem maleate (JAN/USAN)
         D03655  Darodipine (USAN/INN)
         D04193  Flordipine (USAN/INN)
         D04260  Fostedil (USAN/INN)
         D06129  Tiapamil hydrochloride (USAN)
         D07886  Efonidipine (INN)
         D09789  Kirenidipine hydrochloride (JAN)
         D09833  Levosemotiadil fumarate (JAN)
         D10932  Etripamil (USAN/INN)
         D11102  Tamolarizine hydrochloride (JAN)
       CACNA1S [HSA:779] [KO:K04857]
       CACNA2D [HSA:781 9254 55799 93589] [KO:K04858 K04859 K04860 K04861]
       CACNA2D1 [HSA:781] [KO:K04858]
       CACNA2D2 [HSA:9254] [KO:K04859]
     Potassium channels
     Inward rectifier channels (Kir)
     Ryanodine receptors (RYR)
     Transient receptor potential channels
   Other ion channels
 
 Nuclear receptors
 
 Protein kinases
 
 Cytokines and receptors
 
 Cell surface molecules and ligands
 
 Transporters
 
 Enzymes
 
 Nucleic acids
 
 Not elsewhere classified

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Last updated: April 25, 2024

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