| Class I antiarrhythmic agent |
| Class Ia antiarrhythmic agent |
| Quinidine |
| Quinidine (BAN) |
| Quinidine gluconate (USP) <US> |
| Quinidine polygalacturonate |
| Quinidine sulfate (USP); Quinidine sulfate hydrate (JP18) <JP/US> |
| Quinidine phenylethylbarbiturate |
| Procainamide |
| Procainamide (INN) |
| Procainamide hydrochloride (JP18/USP) <JP/US> |
| Disopyramide |
| Disopyramide (JP18/USAN/INN) <JP> |
| Disopyramide phosphate (JAN/USP) <JP/US> |
| Sparteine |
| Sparteine (INN) |
| Sparteine sulfate (JAN/USAN) |
| Ajmaline (JP18) |
| Lorajmine hydrochloride (USAN) |
| Hydroquinidine |
| Hydroquinidine (DCF) |
| Hydroquinidine hydrochloride |
| Cibenzoline |
| Cifenline (USAN); Cibenzoline (INN) |
| Cifenline succinate (USAN); Cibenzoline succinate (JP18) <JP> |
| Pirmenol |
| Pirmenol (INN) |
| Pirmenol hydrochloride hydrate (JAN) <JP> |
| Pirmenol hydrochloride (USAN) |
| Class Ib antiarrhythmic agent |
| Lidocaine |
| Lidocaine (JP18/USP/INN) <JP/US> |
| Lidocaine hydrochloride (JAN/USP) <JP/US> |
| Lidocaine hydrochloride monohydrate <JP/US> |
| Mexiletine |
| Mexiletine (INN) |
| Mexiletine hydrochloride (JP18/USP) <JP/US> |
| Tocainide |
| Tocainide (USAN/INN) |
| Tocainide hydrochloride (USP) |
| Aprindine |
| Aprindine (USAN/INN) |
| Aprindine hydrochloride (JP18/USAN) <JP> |
| Class Ic antiarrhythmic agent |
| Propafenone |
| Propafenone (INN) |
| Propafenone hydrochloride (JP18/USP) <JP/US> |
| Flecainide |
| Flecainide (INN) |
| Flecainide acetate (JP18/USP) <JP/US> |
| Lorcainide |
| Lorcainide (INN) |
| Lorcainide hydrochloride (USAN) |
| Encainide |
| Encainide (INN) |
| Encainide hydrochloride (USAN) |
| Ethacizine |
| Pilsicainide |
| Pilsicainide (INN) |
| Pilsicainide hydrochloride hydrate (JP18) <JP> |
| Class III antiarrhythmic agent |
| Amiodarone |
| Amiodarone (USAN/INN) |
| Amiodarone hydrochloride (JP18/USP) <JP/US> |
| Bretylium tosylate (USP); Bretylium tosilate (INN) |
| Bunaftine (INN) |
| Dofetilide (JAN/USP/INN) <US> |
| Ibutilide |
| Ibutilide (INN) |
| Ibutilide fumarate (USP) <US> |
| Tedisamil |
| Tedisamil (USAN) |
| Tedisamil sesquifumarate (USAN) |
| Dronedarone |
| Dronedarone (INN) |
| Dronedarone hydrochloride (USP) <US> |
| Vernakalant hydrochloride (USAN) |
| Sotalol |
| Sotalol (INN) |
| Sotalol hydrochloride (JAN/USP) <JP/US> |
| Nifekalant hydrochloride (JAN) <JP> |
| Acecainide hydrochloride (USAN) |
| Azimilide dihydrochloride (USAN) |
| Sematilide hydrochloride (USAN) |
| Class II antiarrhythmic agent |
| Alprenolol |
| Alprenolol (INN) |
| Alprenolol hydrochloride (JP18/USAN) |
| Oxprenolol |
| Oxprenolol (INN) |
| Oxprenolol hydrochloride (JP18/USP) |
| Pindolol (JP18/USP/INN) <US> |
| Propranolol |
| Propranolol (INN) |
| Propranolol hydrochloride (JP18/USP) <JP/US> |
| Nadolol (JP18/USP/INN) <JP/US> |
| Carteolol |
| Carteolol (INN) |
| Carteolol hydrochloride (JP18/USP) <JP/US> |
| Tertatolol |
| Tertatolol (INN) |
| Tertatolol hydrochloride |
| Penbutolol |
| Penbutolol (INN) |
| Penbutolol sulfate (JP18/USP) |
| Cloranolol (INN) |
| Practolol (USAN) |
| Metoprolol |
| Metoprolol (USAN/INN) |
| Metoprolol tartrate (JP18/USP) <JP/US> |
| Metoprolol succinate (USP) <US> |
| Metoprolol fumarate (USP) |
| Atenolol (JP18/USP/INN) <JP/US> |
| Acebutolol |
| Acebutolol (USAN/INN) |
| Acebutolol hydrochloride (JP18/USP) <US> |
| Bisoprolol |
| Bisoprolol (JAN/USAN/INN) <JP> |
| Bisoprolol fumarate (JP18/USP) <JP/US> |
| Esmolol |
| Esmolol (INN) |
| Esmolol hydrochloride (JAN/USP) <JP/US> |
| Epanolol (USAN/INN) |
| Talinolol (INN) |
| Landiolol |
| Landiolol (USAN/INN) |
| Landiolol hydrochloride (JAN/USAN) <JP> |
| Bufetolol hydrochloride (JP18) |
| Arotinolol |
| Arotinolol (INN) |
| Arotinolol hydrochloride (JP18) <JP> |
| Indenolol |
| Indenolol (INN) |
| Indenolol hydrochloride (JP18) |
| Bucumolol hydrochloride (JP18) |
| Primidolol (USAN/INN) |
| Dexpropranolol hydrochloride (USAN) |
| Diacetolol hydrochloride (USAN) |
| Flestolol sulfate (USAN) |
| Tiprenolol hydrochloride (USAN) |
| Tolamolol (USAN/INN) |
| Phenylalkylamine derivative |
| Verapamil |
| Verapamil (USAN/INN) |
| Verapamil hydrochloride (JP18/USP) <JP/US> |
| Gallopamil |
| Gallopamil (INN) |
| Gallopamil hydrochloride (JAN) |
| Fendiline |
| Fendiline (INN) |
| Fendiline hydrochloride |
| Bepridil |
| Bepridil (INN) |
| Bepridil hydrochloride (USAN); Bepridil hydrochloride hydrate (JAN) <JP> |
| Tiapamil hydrochloride (USAN) |
| Digoxin (JP18/USP) <JP/US> |
| Deslanoside (JP18/USP/INN) <JP> |
| Metildigoxin |
| Metildigoxin (INN); Medigoxin (BAN) |
| Metildigoxin (JP18) <JP> |
| Moracizine |
| Moricizine (USAN); Moracizine (INN) |
| Moricizine hydrochloride (USP) |
| Diltiazem |
| Diltiazem (INN) |
| Diltiazem hydrochloride (JP18/USP) <JP/US> |
| Diltiazem malate (USAN) |
| Dexsotalol hydrochloride (USAN) |