KEGG   DGROUP: CYP1A2 substrate
Entry
DG01892                     DGroup                                 
Name
CYP1A2 substrate
Type
Metabolism
Member
Alosetron
 D07129  
Alosetron (INN)
 D02829  
Alosetron hydrochloride (USAN)  <US>
Ondansetron
 D00456  
Ondansetron (JAN/USP/INN)  <US>
 D00678  
Ondansetron hydrochloride hydrate (JAN/USP)  <JP/US>
Palonosetron
 D07175  
Palonosetron (INN)
 D05343  
Palonosetron hydrochloride (JAN/USP)  <JP/US>
Fenfluramine
 D07945  
Fenfluramine (INN)
 D04148  
Fenfluramine hydrochloride (JAN/USAN)  <JP/US>
Clopidogrel
 D07729  
Clopidogrel (USP/INN)
 D00769  
Clopidogrel bisulfate (USP); Clopidogrel sulfate (JP18); Clopidogrel sulfate tablets (JP18)  <JP/US>
 D10823  
Clopidogrel hydrochloride
 D10824  
Clopidogrel besilate
D10513  
Clopidogrel sulfate and aspirin  <JP>
Lidocaine
 D00358  
Lidocaine (JP18/USP/INN)  <JP/US>
 D02086  
Lidocaine hydrochloride (JAN/USP)  <JP/US>
 D08127  
Lidocaine hydrochloride monohydrate  <JP/US>
Mexiletine
 D08215  
Mexiletine (INN)
 D00639  
Mexiletine hydrochloride (JP18/USP)  <JP/US>
Propafenone
 D08435  
Propafenone (INN)
 D00640  
Propafenone hydrochloride (JP18/USP)  <JP/US>
Propranolol
 D08443  
Propranolol (INN)
 D00483  
Propranolol hydrochloride (JP18/USP)  <JP/US>
Carvedilol
 D00255  
Carvedilol (JP18/USP/INN)  <JP/US>
 D03415  
Carvedilol phosphate (USAN); Carvedilol phosphate hydrate (JAN)  <US>
Terbinafine
 D02375  
Terbinafine (USAN/INN)
 D02219  
Terbinafine hydrochloride (JP18/USP)  <JP/US>
Doxepin
 D07875  
Doxepin (INN)
 D00814  
Doxepin hydrochloride (USP)  <US>
D05744  
Roflumilast (JAN/USAN/INN)  <US>
Caffeine
 D00528  
Caffeine (USP); Anhydrous caffeine (JP18)  <JP>
 D01453  
Caffeine hydrate (JP18)  <JP>
 D07603  
Caffeine citrate (USP)  <US>
D11976  
Fezolinetant (USAN)  <US>
Norfloxacin
 D00210  
Norfloxacin (JP18/USP/INN)  <JP>
 D08287  
Norfloxacin nicotinate
D04859  
Maribavir (JAN/USAN/INN)  <US>
Erlotinib
 D07907  
Erlotinib (INN)
 D04023  
Erlotinib hydrochloride (JAN/USAN)  <JP/US>
Selumetinib
 D09666  
Selumetinib (USAN/INN)
 D10024  
Selumetinib sulfate (JAN/USAN)  <JP/US>
Momelotinib
 D10315  
Momelotinib (USAN/INN)
 D10358  
Momelotinib dihydrochloride (USAN)
 D10889  
Momelotinib hydrochloride hydrate (JAN)  <US>
Anagrelide
 D07455  
Anagrelide (INN/BAN)
 D02933  
Anagrelide hydrochloride (USP)
 D10255  
Anagrelide hydrochloride hydrate (JAN)  <JP/US>
D11817  
Deucravacitinib (JAN/USAN)  <JP/US>
D01583  
Pirfenidone (JAN/USAN/INN)  <JP/US>
D08976  
Pomalidomide (JAN/USAN/INN)  <JP/US>
D11576  
Naproxen and esomeprazole magnesium  <US>
Tizanidine
 D08611  
Tizanidine (INN)
 D00776  
Tizanidine hydrochloride (JP18/USP)  <JP/US>
Dantrolene
 D02347  
Dantrolene (USAN/INN)
 D02274  
Dantrolene sodium (USP); Dantrolene sodium hydrate (JP18)  <JP/US>
Ropivacaine
 D08490  
Ropivacaine (INN)
 D04048  
Ropivacaine hydrochloride (USP); Ropivacaine hydrochloride hydrate (JAN)  <JP/US>
Levobupivacaine
 D08116  
Levobupivacaine (INN)
 D01287  
Levobupivacaine hydrochloride (JAN/USAN)  <JP>
D02740  
Lidocaine and prilocaine  <JP/US>
Naratriptan
 D08255  
Naratriptan (INN)
 D00674  
Naratriptan hydrochloride (JAN/USP)  <JP/US>
D00415  
Zolmitriptan (JAN/USP/INN)  <JP/US>
D05928  
Stiripentol (JAN/USAN/INN)  <JP>
Ropinirole
 D08489  
Ropinirole (USAN/INN)
 D00784  
Ropinirole hydrochloride (JAN/USP)  <JP/US>
Rasagiline
 D08469  
Rasagiline (USAN/INN)
 D02562  
Rasagiline mesylate (USAN); Rasagiline mesilate (JAN)  <JP/US>
 D10829  
Rasagiline tartrate
Loxapine
 D02340  
Loxapine (USAN/INN)  <US>
 D00794  
Loxapine succinate (USP)  <US>
 D08148  
Loxapine hydrochloride
D00283  
Clozapine (JAN/USP/INN)  <JP/US>
Olanzapine
 D00454  
Olanzapine (JAN/USP/INN)  <JP/US>
 D06623  
Olanzapine pamoate (USAN)  <US>
Asenapine
 D11769  
Asenapine (INN)  <US>
 D02995  
Asenapine maleate (JAN/USAN)  <JP/US>
Zolpidem
 D08690  
Zolpidem (INN)
 D00706  
Zolpidem tartrate (JP18/USP)  <JP/US>
D08170  
Melatonin (JAN)  <JP>
D02689  
Ramelteon (JAN/USAN/INN)  <JP/US>
D09388  
Tasimelteon (USAN/INN)  <US>
Dexmedetomidine
 D00514  
Dexmedetomidine (USAN/INN)
 D01205  
Dexmedetomidine hydrochloride (JAN/USP)  <JP/US>
Imipramine
 D08070  
Imipramine (INN)
 D00815  
Imipramine hydrochloride (JP18/USP)  <JP/US>
 D08071  
Imipramine pamoate (USP)  <US>
Clomipramine
 D07727  
Clomipramine (INN)
 D00811  
Clomipramine hydrochloride (JP18/USP)  <JP/US>
Amitriptyline
 D07448  
Amitriptyline (INN)
 D00809  
Amitriptyline hydrochloride (JP18/USP)  <JP/US>
Mianserin
 D08216  
Mianserin (INN)
 D01358  
Mianserin hydrochloride (JAN/USAN)  <JP>
Mirtazapine
 D00563  
Mirtazapine (JAN/USP/INN)  <JP/US>
 D11056  
Mirtazapine hydrate (JAN)
Duloxetine
 D07880  
Duloxetine (INN)
 D01179  
Duloxetine hydrochloride (JAN/USP)  <JP/US>
Tacrine
 D08555  
Tacrine (INN)
 D02068  
Tacrine hydrochloride (USP)
D00775  
Riluzole (JAN/USP/INN)  <JP/US>
D08575  
Tetrabenazine (JAN/INN)  <JP/US>
D10687  
Abametapir (USAN/INN)  <US>
D02017  
Oxtriphylline (USP); Choline theophyllinate (INN); Choline theophylline (JAN)
Theophylline
 D00371  
Theophylline (JP18)  <JP/US>
 D01712  
Theophylline sodium acetate (JAN)
 D06103  
Theophylline (USP)
 D06104  
Theophylline sodium glycinate (USP)
Aminophylline
 D00227  
Aminophylline (USP/INN)
 D05429  
Aminophylline hydrate (JP18)  <JP>
 D11630  
Aminophylline dihydrate  <US>
Ramosetron
 D08466  
Ramosetron (INN)
 D02016  
Ramosetron hydrochloride (JAN)  <JP>
Sarpogrelate
 D08508  
Sarpogrelate (INN)
 D01624  
Sarpogrelate hydrochloride (JP18)  <JP>
D04052  
Epinephrine and lidocaine hydrochloride  <JP/US>
D04813  
Lidocaine hydrochloride and epinephrine bitartrate  <JP/US>
D11553  
Lidocaine and tetracaine  <US>
D11851  
Butalbital, acetaminophen, caffeine and codeine phosphate  <US>
 » expand
Class
Metabolizing enzyme substrate
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