| C01996 |
Acetylcholine; O-Acetylcholine |
(P) unclassified |
| C06850 |
Bethanechol |
(P) unclassified |
| C06975 |
Echothiophate |
(P) unclassified |
| C07051 |
Indinavir |
(P) unclassified |
| C07055 |
Isopropamide |
(P) unclassified |
| C07410 |
Pyridostigmine |
(P) unclassified |
| C07471 |
Methacholine; Acetyl-beta-methylcholine |
(P) unclassified |
| C07506 |
Propantheline |
(P) unclassified |
| C07773 |
Ambenonium |
(P) unclassified |
| C07811 |
Hexocyclium |
(P) unclassified |
| C07814 |
Homatropine |
(P) unclassified |
| C07818 |
Mepenzolate |
(P) unclassified |
| C07849 |
Methantheline |
(P) unclassified |
| C07861 |
Tridihexethyl |
(P) unclassified |
| C12768 |
Timepidium bromide; Timepidium bromide anhydrous |
(P) unclassified |
| C16823 |
Distigmine |
(P) unclassified |
| C20131 |
Aclatonium |
(P) unclassified |
| D00043 |
Isoflurophate; Fluostigmine; Floropryl (TN) |
(P) Target: ACHE |
| D00109 |
Aspirin (JP19/USP); Aspalon (JAN); Acetylsalicylic acid; Easprin (TN); Durlaza (TN) |
(P) unclassified |
| D00113 |
Atropine (USP); Atropen (TN) |
(P) unclassified |
| D00118 |
Naproxen (JP19/USP/INN); Naprosyn (TN) |
(P) unclassified |
| D00120 |
Sulindac (JP19/USP/INN); Clinoril (TN) |
(P) unclassified |
| D00126 |
Ibuprofen (JP19/USP/INN); Advil (TN); Motrin (TN) |
(P) unclassified |
| D00127 |
Piroxicam (JP19/USP/INN); Feldene (TN) |
(P) unclassified |
| D00130 |
Diflunisal (JAN/USP/INN); Dolobid (TN) |
(P) unclassified |
| D00132 |
Ketoprofen (JP19/USP/INN); Orudis (TN) |
(P) unclassified |
| D00138 |
Scopolamine (INN); Transderm scop (TN) |
(P) unclassified |
| D00140 |
Erythromycin (JP19/USP/INN); Akne-mycin (TN); Eryc (TN); Erygel (TN); Pce (TN); Staticin (TN); T-stat (TN) |
(P) unclassified |
| D00141 |
Indomethacin (USP); Indometacin (JP19/INN); Aconip (TN); Indocin (TN) |
(P) unclassified |
| D00147 |
Hyoscyamine (USP) |
(P) unclassified |
| D00151 |
Mefenamic acid (JP19/USP/INN); Ponstel (TN) |
(P) unclassified |
| D00158 |
Tolmetin sodium (JAN/USP); Tolmetin sodium dihydrate; Tolectin (TN) |
(P) unclassified |
| D00169 |
Meclofenamate sodium (USP); Meclofenamate sodium monohydrate; Meclomen (TN) |
(P) unclassified |
| D00184 |
Cyclosporine (USP); Ciclosporin (JP19); Gengraf (TN); Neoral (TN); Restasis (TN); Sandimmune (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D00196 |
Physostigmine (USP); Eserine (TN) |
(P) Target: ACHE |
| D00210 |
Norfloxacin (JP19/USP/INN); Noroxin (TN) |
(P) unclassified |
| D00211 |
Rifampin (USP); Rifampicin (JP19/INN); Rifadin (TN); Rimactane (TN) |
(P) CYP induction: CYP3A4 |
| D00232 |
Anisotropine methylbromide (USAN); Octatropine methylbromide (INN); Methyloctatropine bromide (JAN); Valpin (TN); Valpin 50 (TN) |
(P) unclassified |
| D00252 |
Carbamazepine (JP19/USP/INN); Equetro (TN); Tegretol (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
| D00270 |
Chlorpromazine (USP/INN); Thorazine (TN) |
(P) unclassified |
| D00276 |
Clarithromycin (JP19/USP/INN); Biaxin (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D00282 |
Clotrimazole (JP19/USP/INN); Lotrimin (TN); Mycelex (TN) |
(P) CYP inhibition: CYP3A4 |
| D00292 |
Dexamethasone (JP19/USP/INN); Decadron (TN); Maxidex (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
| D00293 |
Diazepam (JP19/USP/INN); Diastat (TN); Valium (TN) |
(P) Enzyme: CYP3A4 |
| D00295 |
Cimetidine (JP19/USP/INN); Tagamet (TN) |
(P) CYP inhibition: CYP3A4 |
| D00315 |
Etodolac (JP19/USP/INN); Lodine (TN) |
(P) unclassified |
| D00322 |
Fluconazole (JP19/USP/INN); Diflucan (TN) |
(P) CYP inhibition: CYP3A4 |
| D00326 |
Fluoxetine (USAN/INN); Fluoxetine (TN) |
(P) unclassified |
| D00330 |
Flurbiprofen (JP19/USP/INN); Ansaid (TN) |
(P) unclassified |
| D00350 |
Itraconazole (JP19/USP); Itrizole (TN); Sporanox (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D00351 |
Ketoconazole (JP19/USP); Nizoral (TN); Xolegel (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D00377 |
Mesalamine (USP); Mesalazine (JP19/INN); Apriso (TN); Asacol (TN); Canasa (TN); Delzicol (TN); Lialda (TN); Mesalamine (TN); Pentasa (TN); Rowasa (TN); Sfrowasa (TN) |
(P) unclassified |
| D00397 |
Tropicamide (JP19/USP/INN); Mydriacyl (TN) |
(P) unclassified |
| D00416 |
Miconazole (JP19/USP/INN); Monistat (TN); Oravig (TN) |
(P) unclassified |
| D00420 |
Mitotane (JAN/USP/INN); Lysodren (TN) |
(P) unclassified |
| D00422 |
Ranitidine (USAN/INN) |
(P) unclassified |
| D00425 |
Nabumetone (JP19/USP/INN); Relafen (TN) |
(P) unclassified |
| D00427 |
Ritonavir (JAN/USP/INN); Norvir (TN) |
(P) unclassified |
| D00428 |
Salsalate (USP/INN); Sasapyrine (JAN); Disalcid (TN) |
(P) unclassified |
| D00435 |
Nevirapine (JAN/USP/INN); Viramune (TN) |
(P) Enzyme: CYP3A4 |
| D00448 |
Sulfasalazine (USP/INN); Salazosulfapyridine (JP19); Azulfidine (TN) |
(P) unclassified |
| D00452 |
Suprofen (JAN/USP/INN); Profenal (TN) |
(P) unclassified |
| D00463 |
Oxaprozin (JP19/USP/INN); Daypro (TN) |
(P) unclassified |
| D00465 |
Oxybutynin (USAN/INN); Anturol (TN); Oxytrol (TN) |
(P) Enzyme: CYP3A4 |
| D00481 |
Propantheline bromide (JP19/USP/INN); Pro-banthine (TN) |
(P) unclassified |
| D00487 |
Pyridostigmine bromide (JP19/USP/INN); Mestinon (TN) |
(P) Target: ACHE |
| D00506 |
Phenobarbital (JP19/USP/INN); Luminal (TN) |
(P) unclassified |
| D00510 |
Phenylbutazone (JP19/USP/INN); Azolid (TN) |
(P) unclassified |
| D00512 |
Phenytoin (JP19/USP/INN); Dilantin (TN) |
(P) unclassified |
| D00524 |
Carbachol (JAN/USP/INN); Miostat (TN) |
(P) unclassified |
| D00525 |
Pilocarpine (JAN/USP); Ocusert pilo-20 (TN) |
(P) unclassified |
| D00540 |
Glycopyrrolate (USP); Glycopyrronium bromide (JAN/INN); Cuvposa (TN); Robinul (TN); Seebri breezhaler (TN) |
(P) unclassified |
| D00550 |
Midazolam (JAN/USP/INN); Dormicum (TN); Buccolam (TN); Nayzilam (TN) |
(P) Enzyme: CYP3A4 |
| D00554 |
Ethinyl estradiol (USP); Ethinylestradiol (JP19/INN); Estinyl (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D00556 |
Aminopyrine (JAN); Aminophenazone (INN) |
(P) unclassified |
| D00566 |
Sodium salicylate (JP19/USP); Salsonin (TN) |
(P) unclassified |
| D00567 |
Celecoxib (JP19/USP/INN); Celebrex (TN); Onsenal (TN) |
(P) unclassified |
| D00568 |
Rofecoxib (JAN/USAN/INN); Vioxx (TN) |
(P) unclassified |
| D00578 |
Voriconazole (JP19/USP/INN); Vfend (TN) |
(P) unclassified |
| D00585 |
Mifepristone (JAN/USAN/INN); Korlym (TN); Mifeprex (TN) |
(P) Enzyme: CYP3A4 |
| D00619 |
Verapamil hydrochloride (JP19/USP); Calan (TN); Covera-hs (TN); Vasolan (TN); Verelan (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D00636 |
Amiodarone hydrochloride (JP19/USP); Ancaron (TN); Cordarone (TN); Nexterone (TN) |
(P) Enzyme: CYP3A4 |
| D00644 |
Esmolol hydrochloride (JAN/USP); Brevibloc (TN) |
(P) unclassified |
| D00646 |
Tolterodine (USAN/INN) |
(P) Enzyme: CYP3A4 |
| D00661 |
Cevimeline hydrochloride (USAN); Cevimeline hydrochloride hydrate (JAN); Evoxac (TN); Saligren (TN) |
(P) Enzyme: CYP3A4 |
| D00667 |
Demecarium bromide (USP/INN); Humorsol (TN) |
(P) Target: ACHE |
| D00670 |
Donepezil hydrochloride (JP19/USP); Aricept (TN) |
(P) Enzyme: CYP3A4 / Target: ACHE |
| D00672 |
Hydroxyzine hydrochloride (JP19/USP); Hydroxyzine dihydrochloride; Atarax (TN); Vistaril (TN) |
(P) unclassified |
| D00673 |
Ranitidine hydrochloride (JP19/USP); Zantac (TN) |
(P) unclassified |
| D00701 |
Phenobarbital sodium (JAN/USP/INN); Luminal sodium (TN) |
(P) unclassified |
| D00707 |
Fomepizole (JAN/USAN/INN); Antizol (TN) |
(P) CYP inhibition: CYP3A4 |
| D00715 |
Methscopolamine bromide (USP); Hyoscine methobromide (INN); Pamine (TN) |
(P) unclassified |
| D00716 |
Clidinium bromide (USP/INN); Quarzan (TN) |
(P) unclassified |
| D00717 |
Dicyclomine hydrochloride (JAN/USP); Dicycloverine hydrochloride; Bentyl (TN); Urispas (TN) |
(P) unclassified |
| D00719 |
Hyoscyamine sulfate (USP); Hyoscyamine sulfate dihydrate; Egacene (TN) |
(P) unclassified |
| D00720 |
Mepenzolate bromide (JP19/INN); Cantil (TN) |
(P) unclassified |
| D00721 |
Methanthelinium bromide (INN); Methantheline bromide; Banthine (TN) |
(P) unclassified |
| D00722 |
Oxybutynin chloride (USP); Oxybutynin hydrochloride (JP19); Ditropan (TN); Gelnique (TN) |
(P) Enzyme: CYP3A4 |
| D00723 |
Tridihexethyl chloride (BAN); Pathilon (TN) |
(P) unclassified |
| D00727 |
Olsalazine sodium (USAN); Dipentum (TN) |
(P) unclassified |
| D00753 |
Sirolimus (JAN/USAN/INN); Rapamune (TN); Rapamycin (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D00774 |
Orphenadrine citrate (USP); Norflex (TN) |
(P) unclassified |
| D00778 |
Benztropine mesylate (USP); Benztropine mesilate (JAN); Cogentin (TN) |
(P) unclassified |
| D00779 |
Biperiden (JAN/USP/INN); Akineton (TN) |
(P) unclassified |
| D00780 |
Bromocriptine mesylate (USP); Bromocriptine mesilate (JP19); Parlodel (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D00782 |
Procyclidine hydrochloride (USP); Kemadrin (TN) |
(P) unclassified |
| D00787 |
Trihexyphenidyl hydrochloride (JP19/USP); Artane (TN) |
(P) unclassified |
| D00789 |
Chlorpromazine hydrochloride (JP19/USP); Sonazine (TN) |
(P) unclassified |
| D00810 |
Choline salicylate (JAN/USAN/INN); Arthropan (TN) |
(P) unclassified |
| D00813 |
Ketorolac tromethamine (USP); Acular (TN); Toradol (TN) |
(P) unclassified |
| D00823 |
Fluoxetine hydrochloride (JAN/USP); Prozac (TN); Sarafem (TN) |
(P) unclassified |
| D00824 |
Fluvoxamine maleate (JP19/USP); Luvox (TN) |
(P) CYP inhibition: CYP3A4 |
| D00827 |
Magnesium salicylate (USP); Magnesium salicylate tetrahydrate; Magan (TN) |
(P) unclassified |
| D00831 |
Mefloquine hydrochloride (JP19/USP); Lariam (TN) |
(P) unclassified |
| D00851 |
Erythromycin estolate (USP); Erythromycin estorate (JAN); Ilosone (TN) |
(P) unclassified |
| D00854 |
Quinupristin and dalfopristin; Synercid (TN) |
(P) CYP inhibition: CYP3A4 |
| D00882 |
Miconazole nitrate (JP19/USP); Micatin (TN); Monistat (TN) |
(P) unclassified |
| D00894 |
Amprenavir (JAN/USAN/INN); Agenerase (TN) |
(P) Enzyme: CYP3A4 |
| D00895 |
Delavirdine mesylate (USAN); Delavirdine mesilate (JAN); Rescriptor (TN) |
(P) unclassified |
| D00897 |
Indinavir sulfate (USP); Crixivan (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D00899 |
Nelfinavir mesylate (USAN/INN); Nelfinavir mesilate (JAN); Viracept (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D00903 |
Diclofenac potassium (USP); Cambia (TN); Cataflam (TN); Zipsor (TN) |
(P) unclassified |
| D00904 |
Diclofenac sodium (JP19/USP); Solaraze (TN); Voltaren (TN) |
(P) unclassified |
| D00960 |
Anastrozole (JP19/USP/INN); Arimidex (TN) |
(P) CYP inhibition: CYP3A4 |
| D00961 |
Bicalutamide (JP19/USP/INN); Casodex (TN) |
(P) CYP inhibition: CYP3A4 |
| D00968 |
Fenoprofen calcium (JAN/USP); Nalfon (TN) |
(P) unclassified |
| D00969 |
Meloxicam (JAN/USP/INN); Mobic (TN) |
(P) unclassified |
| D00970 |
Naproxen sodium (USP); Anaprox (TN) |
(P) unclassified |
| D00971 |
Sodium thiosalicylate; Thiosalicylic acid sodium salt; Rexolate (TN) |
(P) unclassified |
| D00975 |
Dexamethasone sodium phosphate (JAN/USP); Dalalone (TN); Maxidex (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
| D00994 |
Edrophonium chloride (JP19/USP/INN); Enlon (TN); Tensilon (TN) |
(P) Target: ACHE |
| D00995 |
Neostigmine bromide (JAN/USP/INN); Vagostigmin (TN) |
(P) Target: ACHE |
| D00998 |
Neostigmine methylsulfate (JP19/USP); Bloxiverz (TN); Prostigmin (TN) |
(P) Target: ACHE |
| D00999 |
Acetylcholine chloride (JP19/USP/INN); Miochol (TN) |
(P) Enzyme-Target: ACHE |
| D01000 |
Bethanechol chloride (JP19/USP); Urecholine (TN) |
(P) unclassified |
| D01001 |
Ambenonium chloride (JP19/INN); Mytelase (TN) |
(P) Target: ACHE |
| D01002 |
Cyclopentolate hydrochloride (JP19/USP); Cyclogyl (TN) |
(P) unclassified |
| D01003 |
Hexocyclium metilsulfate (INN); Hexocyclium methyl sulfate; Tral (TN) |
(P) unclassified |
| D01004 |
Homatropine hydrobromide (JP19/USP); Isopto homatropine (TN) |
(P) unclassified |
| D01005 |
Isopropamide iodide (JAN/USP/INN); Darbid (TN) |
(P) unclassified |
| D01006 |
Oxyphencyclimine hydrochloride (JAN); Daricon (TN) |
(P) unclassified |
| D01007 |
Propiverine hydrochloride (JP19); Bup-4 (TN); Mictonorm (TN) |
(P) Enzyme: CYP3A4 |
| D01037 |
1,4-Dimethyl-7-isopropylazulene (JAN); Guaiazulene; Azunol (TN) |
(P) unclassified |
| D01049 |
Nimesulide (JAN/INN) |
(P) unclassified |
| D01077 |
Methylatropine nitrate (USAN); Atropine methonitrate (JAN/INN); Ekomine (TN) |
(P) unclassified |
| D01078 |
Telithromycin (JAN/USAN/INN); Ketek (TN) |
(P) unclassified |
| D01087 |
Methyl salicylate (JP19/NF) |
(P) unclassified |
| D01096 |
Hydroxyzine pamoate (JP19/USP); Atarax-P (TN); Vistaril pamoate (TN) |
(P) unclassified |
| D01103 |
Trospium chloride (JAN/USP/INN); Spasmex (TN); Spasmoplex (TN) |
(P) unclassified |
| D01118 |
Profenamine hydrochloride (JAN); Ethopropazine hydrochloride; Parkin (TN); Parsidol (TN) |
(P) unclassified |
| D01122 |
Ibuprofen piconol (JP19/USAN); Staderm (TN) |
(P) unclassified |
| D01148 |
Tolterodine tartrate (JAN/USP); Detrol (TN); Detrusitol (TN) |
(P) Enzyme: CYP3A4 |
| D01165 |
Piperidolate hydrochloride (JAN); Dactil (TN) |
(P) unclassified |
| D01175 |
Carpronium chloride (JAN/INN); Actinamin (TN) |
(P) unclassified |
| D01183 |
Tolfenamic acid (JAN/INN); Clotam (TN) |
(P) unclassified |
| D01185 |
Protizinic acid (JAN/INN) |
(P) unclassified |
| D01189 |
Metiazinic acid (JAN/INN) |
(P) unclassified |
| D01201 |
Tiemonium iodide (JAN/INN); Visceralgine (TN) |
(P) unclassified |
| D01228 |
Distigmine bromide (JP19/INN); Ubretid (TN) |
(P) Target: ACHE |
| D01231 |
Piroheptine hydrochloride (JAN); Trimol (TN) |
(P) unclassified |
| D01235 |
Josamycin (JP19/USAN/INN); Leucomycin A3; JM |
(P) CYP inhibition: CYP3A4 |
| D01236 |
Conivaptan hydrochloride (JAN/USAN); Vaprisol (TN) |
(P) unclassified |
| D01252 |
Alclofenac (JAN/USP/INN); Mervan (TN) |
(P) unclassified |
| D01253 |
Clobazam (JAN/USAN/INN); Mystan (TN); Onfi (TN) |
(P) Enzyme: CYP3A4 |
| D01267 |
Floctafenine (JAN/USAN/INN); Idarac (TN) |
(P) unclassified |
| D01269 |
Solifenacin succinate (JAN/USAN/INN); Vesicare (TN) |
(P) Enzyme: CYP3A4 |
| D01271 |
Bufexamac (JAN/INN); Anderm (TN) |
(P) unclassified |
| D01276 |
Atazanavir sulfate (JAN/USAN); Reyataz (TN) |
(P) CYP inhibition: CYP3A4 |
| D01289 |
Suxibuzone (JAN/INN) |
(P) unclassified |
| D01297 |
Pirenzepine hydrochloride (USAN) |
(P) unclassified |
| D01305 |
Feprazone (JAN/INN) |
(P) unclassified |
| D01315 |
Methylbenactyzium bromide (JP19/INN) |
(P) unclassified |
| D01322 |
Troleandomycin (USAN/INN); Triacetyloleandomycin (JAN); TAO; Tao (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D01325 |
Tiaprofenic acid (JAN/INN); Surgam (TN) |
(P) unclassified |
| D01330 |
Clidanac (JAN/INN) |
(P) unclassified |
| D01339 |
Midecamycin (JP19/INN); Medemycin (TN) |
(P) CYP inhibition: CYP3A4 |
| D01341 |
Tiaramide hydrochloride (JP19/USAN); Solantal (TN) |
(P) unclassified |
| D01344 |
Fenbufen (JP19/USAN/INN) |
(P) unclassified |
| D01353 |
Emorfazone (JP19/INN); Pentoil (TN) |
(P) unclassified |
| D01359 |
Etomidoline (JAN/INN); Smedolin (TN) |
(P) unclassified |
| D01361 |
Erythromycin ethylsuccinate (JP19/USP); E.E.S. (TN); Eryped (TN); Erythrocin W (TN) |
(P) unclassified |
| D01377 |
Prifinium bromide (JAN/INN); Padrin (TN) |
(P) unclassified |
| D01380 |
Isopropylantipyrine (JP19); Propyphenazone (INN); Yoshipyrin (TN) |
(P) unclassified |
| D01394 |
Epirizole (JP19/USAN); Mebron (TN) |
(P) unclassified |
| D01397 |
Ampiroxicam (JP19/INN); Flucam (TN) |
(P) unclassified |
| D01410 |
Benzydamine hydrochloride (JAN/USAN); Tantum (TN) |
(P) unclassified |
| D01425 |
Lopinavir (JAN/USP/INN) |
(P) unclassified |
| D01429 |
Fosfluconazole (JAN/INN); Prodif (TN) |
(P) CYP inhibition: CYP3A4 |
| D01437 |
Nifenazone (JAN/INN) |
(P) unclassified |
| D01451 |
Scopolamine butylbromide (JP19); Butylscopolamine bromide; Buscopan (TN) |
(P) unclassified |
| D01463 |
Diponium bromide (JAN/INN); Dipenine bromide |
(P) unclassified |
| D01466 |
Ethenzamide (JP19/INN) |
(P) unclassified |
| D01475 |
Flurbiprofen axetil (JAN); FP 83; Ropion (TN) |
(P) unclassified |
| D01491 |
Butropium bromide (JP19/INN); Coliopan (TN) |
(P) unclassified |
| D01510 |
Dexamethasone metasulfobenzoate sodium (JAN); Dexamethazone metasulfobenzoate sodium; Dexapos; Santeson (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
| D01513 |
Alminoprofen (JP19/INN); Minalfen (TN) |
(P) unclassified |
| D01521 |
Pipethanate hydrochloride (JAN); Glymor (TN) |
(P) unclassified |
| D01538 |
Valethamate bromide (JAN); Shinmetane (TN) |
(P) unclassified |
| D01545 |
Aceclofenac (JAN/INN) |
(P) unclassified |
| D01547 |
Zaltoprofen (JP19/INN); CN 100; Peon (TN) |
(P) unclassified |
| D01557 |
Glycol salicylate (JAN); Ethylene glycol salicylate; Norgesic (TN); Phlogont (TN) |
(P) unclassified |
| D01565 |
Indometacin farnesil (JAN); Infree (TN) |
(P) unclassified |
| D01567 |
Ketophenylbutazone (JAN); Kebuzone (INN) |
(P) unclassified |
| D01578 |
Pranoprofen (JP19/INN); Elicapric (TN) |
(P) unclassified |
| D01581 |
Flufenamic acid (JAN/USAN/INN); Arlef (TN) |
(P) unclassified |
| D01582 |
Acemetacin (JP19/INN); Rantudil (TN) |
(P) unclassified |
| D01594 |
Bendazac (JAN/USAN/INN); Iwazac (TN) |
(P) unclassified |
| D01600 |
Diphenylpiperidinomethyldioxolan iodide (JAN); Anacolin; Gastrophyllin-A (TN) |
(P) unclassified |
| D01615 |
Dexamethasone palmitate (JAN); Dexamethasone 21-palmitate; Limethason (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
| D01632 |
Dexamethasone dipropionate (USAN); Dexamethasone propionate (JAN); Hifmeta (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
| D01636 |
Midecamycin acetate (JP19); Miocamycin; Miocamycin (TN) |
(P) CYP inhibition: CYP3A4 |
| D01648 |
Hyoscyamine methylbromide (JAN) |
(P) unclassified |
| D01661 |
Bucolome (JAN/INN); Paramidin (TN) |
(P) unclassified |
| D01675 |
Felbinac (JP19/USAN/INN); Dolinac (TN) |
(P) unclassified |
| D01699 |
Darifenacin hydrobromide (JAN/USAN); Enablex (TN) |
(P) Enzyme: CYP3A4 |
| D01706 |
Migrenin (JP19) |
(P) unclassified |
| D01709 |
Loxoprofen sodium hydrate (JP19); Lorfenamin (TN); Loxonin (TN) |
(P) unclassified |
| D01718 |
Mofezolac (JAN/INN) |
(P) unclassified |
| D01762 |
Dipyrone (USAN); Sulpyrine hydrate (JP19); Metamizole sodium salt monohydrate |
(P) unclassified |
| D01765 |
Proglumetacin maleate (JAN); Miridacin (TN) |
(P) unclassified |
| D01767 |
Tenoxicam (JAN/USAN/INN); Tilcotil (TN) |
(P) unclassified |
| D01776 |
Antipyrine (JP19/USP); Phenazone (INN) |
(P) unclassified |
| D01788 |
Amfenac sodium (USAN); Amfenac sodium hydrate (JAN); Fenazox (TN) |
(P) unclassified |
| D01811 |
Salicylamide (JAN/USP/INN) |
(P) unclassified |
| D01815 |
Oxapium iodide (JP19/INN); Espalexan (TN) |
(P) unclassified |
| D01823 |
Ufenamate (JAN/INN); Flufenamic acid butyl ester; Combec (TN) |
(P) unclassified |
| D01841 |
Felbinac ethyl (JAN); LM 001 |
(P) unclassified |
| D01847 |
Landiolol hydrochloride (JAN/USAN); ONO 1101 hydrochloride; Onoact (TN); Rapiblyk (TN) |
(P) unclassified |
| D01851 |
Mepranoprofen arbamel (JAN); Y-23023 |
(P) unclassified |
| D01865 |
Pelubiprofen (JAN/INN) |
(P) unclassified |
| D01866 |
Lornoxicam (JP19/USAN/INN); Lorcam (TN) |
(P) unclassified |
| D01871 |
Methixene hydrochloride (USAN); Metixene hydrochloride (JAN); Methixene hydrochloride hydrete; Trest (TN) |
(P) unclassified |
| D01874 |
Vedaprofen (JAN/USAN/INN) |
(P) unclassified |
| D01875 |
Tiquizium bromide (JAN/INN); Thiaton (TN) |
(P) unclassified |
| D01929 |
Tiotropium bromide hydrate (JAN); Tiotropium bromide monohydrate; Spiriva (TN) |
(P) unclassified |
| D01946 |
Oxitropium bromide (JAN/INN); Tersigan (TN) |
(P) unclassified |
| D01948 |
Dexamethasone valerate (JAN); Dexamethasone 17-valerate; DV-17; Voalla ointment (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
| D01955 |
Aclatonium napadisilate (JAN); Abovis (TN) |
(P) unclassified |
| D01963 |
Ibufenac (JAN/USAN/INN); Dytransin (TN) |
(P) unclassified |
| D01974 |
Tilmacoxib (JAN/USAN/INN) |
(P) unclassified |
| D01975 |
Fentiazac (JAN/USAN/INN) |
(P) unclassified |
| D01976 |
N-Methylscopolamine methylsulfate (JAN); Daipin (TN) |
(P) unclassified |
| D01980 |
Luliconazole (JAN/USAN/INN); Lulicon (TN); Luzu (TN) |
(P) CYP inhibition: CYP3A4 |
| D02009 |
Erythromycin lactobionate (JP19/USP); Erythrocin (TN) |
(P) unclassified |
| D02068 |
Tacrine hydrochloride (USP); Cognex (TN) |
(P) Target: ACHE |
| D02069 |
Atropine sulfate (JP19/USP); Ryjusea (TN) |
(P) unclassified |
| D02070 |
Homatropine methylbromide (USP); Equipin (TN) |
(P) unclassified |
| D02071 |
Scopolamine hydrobromide (USP); Scopolamine hydrobromide hydrate (JP19); Scopolamine hydrobromide trihydrate; Hysco (TN); Isopto hyoscine (TN) |
(P) unclassified |
| D02075 |
Sodium gualenate (INN); Sodium guaiazulenesulfonate; Azunol ST (TN) |
(P) unclassified |
| D02103 |
Phenytoin sodium (USP); Phenytoin sodium for injection (JP19); Aleviatin (TN); Dilantin (TN) |
(P) unclassified |
| D02110 |
Indomethacin sodium (USP); Indometacin sodium hydrate (JAN); Indomethacin sodium trihydrate; Indometacin sodium; Indocin I.V. (TN) |
(P) unclassified |
| D02173 |
Galantamine hydrobromide (JAN/USP); Razadyne (TN); Reminyl (TN) |
(P) Enzyme: CYP3A4 / Target: ACHE |
| D02174 |
Dexamethasone acetate (JAN/USP); Decadronal (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
| D02184 |
Erythromycin stearate (JP19/USP); Bristamycin (TN) |
(P) unclassified |
| D02193 |
Echothiophate iodide (USP); Ecothiopate iodide (JP19/INN); Phospholine iodide (TN) |
(P) Target: ACHE |
| D02200 |
Pilocarpine hydrochloride (JP19/USP); Isopto carpine (TN); Pilopine HS (TN); Salagen (TN); Sanpilo (TN) |
(P) unclassified |
| D02212 |
Ipratropium bromide (USP); Ipratropium bromide hydrate (JP19); Atrovent (TN) |
(P) unclassified |
| D02246 |
Biperiden hydrochloride (JP19/USP); Tasmolin (TN) |
(P) unclassified |
| D02247 |
Biperiden lactate (JAN/USP); Tasmolin (TN) |
(P) unclassified |
| D02264 |
Dipotassium glycyrrhizinate (JAN); Glycyrrhizinate dipotassium; Neubormitin (TN) |
(P) unclassified |
| D02272 |
Quinidine sulfate (USP); Quinidine sulfate hydrate (JP19); Quinidex (TN) |
(P) Enzyme: CYP3A4 |
| D02275 |
Suxamethonium chloride hydrate (JP19); Suxamethonium chloride dihydrate; Succin (TN) |
(P) unclassified |
| D02290 |
Flurbiprofen sodium (USP); Ocufen (TN) |
(P) unclassified |
| D02341 |
Meclofenamic acid (USAN/INN) |
(P) unclassified |
| D02350 |
Fenoprofen (USAN/INN) |
(P) unclassified |
| D02355 |
Tolmetin (USAN/INN) |
(P) unclassified |
| D02356 |
Verapamil (USAN/INN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D02372 |
Perospirone hydrochloride hydrate (JP19); Lullan (TN) |
(P) unclassified |
| D02417 |
Flutropium bromide (JAN); Flutropium bromide monohydrate; Flubron (TN) |
(P) unclassified |
| D02418 |
Physostigmine salicylate (JAN/USP); Antilirium (TN) |
(P) Target: ACHE |
| D02484 |
Artemether and lumefantrine; Coartem (TN) |
(P) unclassified |
| D02497 |
Fosamprenavir (INN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D02498 |
Lopinavir and ritonavir; Kaletra (TN) |
(P) unclassified |
| D02523 |
Erythromycin acistrate (USAN); Erasis (TN) |
(P) unclassified |
| D02524 |
Erythromycin gluceptate (USP); Erythromycin glucoheptonate; Ilotycin gluceptate (TN) |
(P) unclassified |
| D02525 |
Erythromycin propionate (USAN) |
(P) unclassified |
| D02535 |
Timepidium bromide hydrate (JP19); Sesden (TN) |
(P) unclassified |
| D02537 |
Dronedarone (INN) |
(P) unclassified |
| D02555 |
Posaconazole (JAN/USAN/INN); Noxafil (TN) |
(P) CYP inhibition: CYP3A4 |
| D02556 |
Ravuconazole (prop.INN) |
(P) unclassified |
| D02558 |
Rivastigmine tartrate; Rivastigmine hydrogen tartrate; Exelon (TN); Nimvastid (TN) |
(P) Target: ACHE |
| D02565 |
Dimetacrine (INN) |
(P) Target: ACHE |
| D02591 |
Dexamethasone acefurate (USAN/INN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
| D02592 |
Dexamethasone beloxil (USAN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
| D02599 |
Orphenadrine hydrochloride; Disipal (TN) |
(P) unclassified |
| D02691 |
Somatropin (USP/INN); Somatropin (genetical recombination) (JAN); Human growth hormone (JAN); Asellacrin (TN); Humatrope (TN); Nutropin (TN); Omnitrope (TN) |
(P) unclassified |
| D02706 |
Sodium gualenate hydrate (JAN); Azulene sulfonate sodium hydrate; Sodium guaiazulene sulfonate; Azunol (TN) |
(P) unclassified |
| D02709 |
Valdecoxib (USAN/INN); Bextra (TN) |
(P) unclassified |
| D02715 |
Balsalazide disodium (USP); Colazide (TN) |
(P) unclassified |
| D02729 |
Itopride hydrochloride (JAN); Ganaton (TN) |
(P) Target: ACHE |
| D02732 |
Pranlukast hydrate (JP19); Onon (TN) |
(P) Enzyme: CYP3A4 |
| D02750 |
Aceclidine (USAN/INN); Glaucostat (TN) |
(P) unclassified |
| D02861 |
Indinavir sulfate ethanolate (JAN); Crixivan (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D02867 |
Fosamprenavir calcium hydrate (JAN); Lexiva (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D02876 |
Alvameline maleate (USAN) |
(P) unclassified |
| D02944 |
Anirolac (USAN/INN) |
(P) unclassified |
| D02968 |
Aprepitant (JAN/USP/INN); Aponvie (TN); Emend (TN); Cinvanti (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4 |
| D03080 |
Benoxaprofen (USAN/INN); Oraflex (TN) |
(P) unclassified |
| D03087 |
Benzetimide hydrochloride (USAN); Dioxatrine (TN) |
(P) unclassified |
| D03098 |
Berythromycin (USAN/INN); Erythromycin B |
(P) unclassified |
| D03106 |
Bexarotene (JAN/USAN/INN); Targretin (TN) |
(P) unclassified |
| D03163 |
Bromfenac sodium (USAN); Bromfenac sodium hydrate (JP19); Bromfenac sodium sesquihydrate; Bromday (TN); Prolensa (TN); Xibrom (TN); Yellox (TN) |
(P) unclassified |
| D03165 |
Bromocriptine (USAN/INN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D03239 |
Ladostigil tartrate (USAN) |
(P) Target: ACHE |
| D03254 |
Flufenamate aluminum (JAN); Flufenamic acid aluminum; Opyrin (TN) |
(P) unclassified |
| D03264 |
Mazaticol hydrochloride hydrate (JAN); Mazaticol hydrochloride; Pentona (TN) |
(P) unclassified |
| D03274 |
Chlorpromazine hibenzate (JAN); Contomin (TN) |
(P) unclassified |
| D03276 |
Profenamine hibenzate (JAN); Parkin (TN) |
(P) unclassified |
| D03378 |
Caracemide (USAN) |
(P) unclassified |
| D03385 |
Carbaspirin calcium (USAN); Carbasalate calcium (INN) |
(P) unclassified |
| D03410 |
Carprofen (USP/INN); Rimadyl (TN) |
(P) unclassified |
| D03489 |
Cicloprofen (USAN/INN) |
(P) unclassified |
| D03503 |
Cimetidine hydrochloride (USP) |
(P) CYP inhibition: CYP3A4 |
| D03540 |
Cliprofen (USAN/INN) |
(P) unclassified |
| D03560 |
Clopirac (USAN/INN) |
(P) unclassified |
| D03652 |
Darbufelone mesylate (USAN) |
(P) unclassified |
| D03654 |
Darifenacin (USAN/INN) |
(P) Enzyme: CYP3A4 |
| D03656 |
Darunavir (USAN/INN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D03658 |
Dasatinib (JAN/INN) |
(P) Enzyme: CYP3A4 |
| D03669 |
Deferasirox (JAN/USAN/INN); Exjade (TN); Jadenu (TN) |
(P) CYP induction: CYP3A4 |
| D03689 |
Deracoxib (USAN) |
(P) unclassified |
| D03710 |
Etoricoxib (USAN/INN) |
(P) unclassified |
| D03711 |
Dexetimide (USAN/INN); (+)-Benzetimide |
(P) unclassified |
| D03712 |
Firocoxib (USAN/INN); Equioxx (TN) [veterinary] |
(P) unclassified |
| D03714 |
Lumiracoxib (USAN/INN) |
(P) unclassified |
| D03715 |
Dexibuprofen (USAN/INN) |
(P) unclassified |
| D03716 |
Parecoxib (USAN/INN) |
(P) unclassified |
| D03717 |
Parecoxib sodium (USAN); Dynastat (TN) |
(P) unclassified |
| D03718 |
Dexibuprofen lysine (USAN); Dexibuprofen lysine monohydrate; Doctrin (TN) |
(P) unclassified |
| D03727 |
Dexpemedolac (USAN/INN) |
(P) unclassified |
| D03751 |
Icopezil maleate (USAN) |
(P) Target: ACHE |
| D03791 |
Dichlorvos (USAN/INN); Atgard (TN) |
(P) unclassified |
| D03814 |
Atropine methylbromide (JAN) |
(P) unclassified |
| D03822 |
Rivastigmine (JAN/USP/INN); Exelon (TN); Prometax (TN) |
(P) Target: ACHE |
| D03824 |
Dihexyverine hydrochloride (USAN) |
(P) unclassified |
| D03826 |
Physostigmine sulfate (USP); Eserine sulfate (TN) |
(P) Target: ACHE |
| D03833 |
Indinavir (USAN); Indinavir hydrate |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D03835 |
Fosamprenavir calcium (USAN); Lexiva (TN); Telzir (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D03837 |
Fosamprenavir sodium (USAN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D03914 |
Dronedarone hydrochloride (USP); Multaq (TN) |
(P) unclassified |
| D03960 |
Aspirin and dialuminate; Aspirin, aluminum glycinate and magnesium carbonate; Bufferin (TN) |
(P) unclassified |
| D04003 |
Enolicam sodium (USAN); Enolicam sodium monohydrate |
(P) unclassified |
| D04024 |
Lapatinib ditosylate (USAN); Lapatinib tosilate hydrate (JAN); Lapatinib ditosylate monohydrate; Tykerb (TN); Tyverb (TN) |
(P) Enzyme: CYP3A4 |
| D04034 |
Chlorpromazine phenolphthalinate (JAN); Wintermin (TN) |
(P) unclassified |
| D04054 |
Erythromycin salnacedin (USAN); Erythromycin salnacedin dihydrate |
(P) unclassified |
| D04057 |
Esoxybutynin chloride (USAN) |
(P) unclassified |
| D04087 |
Ethybenztropine (USAN); Etybenzatropine (INN); Panolid (TN) |
(P) unclassified |
| D04102 |
Etofenamate (USAN/INN) |
(P) unclassified |
| D04116 |
Eucatropine hydrochloride (USP XXXII) |
(P) unclassified |
| D04142 |
Fenclofenac (USAN/INN) |
(P) unclassified |
| D04144 |
Fenclorac (USAN/INN) |
(P) unclassified |
| D04145 |
Fendosal (USAN/INN); Alnovin (TN) |
(P) unclassified |
| D04206 |
Flufenisal (USAN/INN) |
(P) unclassified |
| D04273 |
Furaprofen (USAN/INN) |
(P) unclassified |
| D04277 |
Furobufen (USAN/INN) |
(P) unclassified |
| D04292 |
Galantamine (USAN/INN); Reminyl (TN) |
(P) Enzyme: CYP3A4 / Target: ACHE |
| D04479 |
Hyoscyamine hydrobromide (USP) |
(P) unclassified |
| D04490 |
Ibuprofen aluminum (USAN) |
(P) unclassified |
| D04530 |
Indoprofen (USAN/INN) |
(P) unclassified |
| D04638 |
Isoxepac (USAN/INN); Artil (TN) |
(P) unclassified |
| D04639 |
Isoxicam (USAN/INN); Maxicam (TN) |
(P) unclassified |
| D04641 |
Istradefylline (JAN/USAN/INN); Nourianz (TN); Nouriast (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D04666 |
Lanreotide acetate (JAN/USAN); Somatuline (TN) |
(P) unclassified |
| D04768 |
Lonafarnib (JAN/USAN/INN); Zokinvy (TN) |
(P) unclassified |
| D04863 |
Mavacoxib (USAN) |
(P) unclassified |
| D04868 |
Mebeverine hydrochloride (USAN) |
(P) unclassified |
| D04970 |
Methacholine chloride (JAN/USP/INN); Provocholine (TN) |
(P) unclassified |
| D05024 |
Mibefradil dihydrochloride (USAN); Posicor (TN) |
(P) unclassified |
| D05035 |
Milameline hydrochloride (USAN) |
(P) unclassified |
| D05121 |
Naproxol (USAN/INN) |
(P) unclassified |
| D05143 |
Nepafenac (JAN/USAN/INN); Nevanac (TN) |
(P) unclassified |
| D05152 |
Netupitant (USAN/INN) |
(P) unclassified |
| D05181 |
Aspirin aluminum (JP19) |
(P) unclassified |
| D05276 |
Pirenzepine hydrochloride hydrate (JP19); Gastrozepin (TN) |
(P) unclassified |
| D05319 |
Oxyphenbutazone hydrate; Tandearil (TN) |
(P) unclassified |
| D05351 |
Josamycin propionate (JP19); Josamy (TN) |
(P) CYP inhibition: CYP3A4 |
| D05404 |
Pemedolac (USAN/INN) |
(P) unclassified |
| D05451 |
Phenbutazone sodium glycerate (USAN) |
(P) unclassified |
| D05478 |
Pilocarpine nitrate (USP); Pilagan (TN) |
(P) unclassified |
| D05511 |
Piroxicam betadex (USAN) |
(P) unclassified |
| D05512 |
Piroxicam cinnamate (USAN) |
(P) unclassified |
| D05513 |
Piroxicam olamine (USAN) |
(P) unclassified |
| D05515 |
Pirprofen (USAN/INN) |
(P) unclassified |
| D05598 |
Pravadoline maleate (USAN) |
(P) unclassified |
| D05619 |
Prodolic acid (USAN/INN) |
(P) unclassified |
| D05699 |
Ranitidine bismuth citrate (USAN); Tritec (TN) |
(P) unclassified |
| D05775 |
Rufinamide (JAN/USP/INN); Banzel (TN) |
(P) unclassified |
| D05779 |
Sabcomeline hydrochloride (USAN) |
(P) unclassified |
| D05788 |
Salcolex (USAN); Salcolex tetrahydrate |
(P) unclassified |
| D05789 |
Salethamide maleate (USAN) |
(P) unclassified |
| D05791 |
Salicylate meglumine (USAN) |
(P) unclassified |
| D05793 |
Salnacedin (USAN/INN) |
(P) unclassified |
| D05830 |
Sermetacin (USAN/INN) |
(P) unclassified |
| D05928 |
Stiripentol (JAN/USAN/INN); Diacomit (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D05937 |
Sudoxicam (USAN/INN) |
(P) unclassified |
| D05995 |
Talmetacin (USAN/INN) |
(P) unclassified |
| D05998 |
Talosalate (USAN/INN) |
(P) unclassified |
| D06000 |
Talsaclidine fumarate (USAN) |
(P) unclassified |
| D06015 |
Tazomeline citrate (USAN) |
(P) unclassified |
| D06082 |
Tesicam (USAN) |
(P) unclassified |
| D06143 |
Tifurac sodium (USAN) |
(P) unclassified |
| D06156 |
Tiopinac (USAN/INN) |
(P) unclassified |
| D06273 |
Imidafenacin (JAN/INN); Uritos (TN); Staybla (TN) |
(P) Enzyme: CYP3A4 |
| D06288 |
Velnacrine maleate (USAN); Mentane (TN) |
(P) Target: ACHE |
| D06330 |
Xanomeline (USAN) |
(P) unclassified |
| D06331 |
Xanomeline tartrate (USAN) |
(P) unclassified |
| D06364 |
Zidometacin (USAN/INN) |
(P) unclassified |
| D06382 |
Zomepirac sodium (USAN); Zomepirac sodium dihydrate |
(P) unclassified |
| D06413 |
Nilotinib hydrochloride hydrate (JAN); Nilotinib monohydrochloride monohydrate; Tasigna (TN) |
(P) Enzyme: CYP3A4 |
| D06414 |
Dasatinib (USAN); Dasatinib hydrate (JAN); Sprycel (TN) |
(P) Enzyme: CYP3A4 |
| D06478 |
Darunavir ethanolate (JAN); Prezista (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D06597 |
Fosaprepitant dimeglumine (USAN); Fosaprepitant meglumine (JAN); Proemend (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4 |
| D06606 |
Ibuprofen lysine (USAN); Ibuprofen L-lysine (JAN); Solufenum; Neoprofen (TN) |
(P) unclassified |
| D07073 |
Dexamethasone cipecilate (JAN/INN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
| D07076 |
Camylofin (INN); Anafortan (TN) |
(P) unclassified |
| D07099 |
Cimetropium bromide (JAN/INN); Alginor (TN) |
(P) unclassified |
| D07141 |
Indobufen (INN) |
(P) unclassified |
| D07219 |
Flunoxaprofen (INN) |
(P) unclassified |
| D07226 |
Fesoterodine (INN) |
(P) Enzyme: CYP3A4 |
| D07262 |
Mofebutazone (INN); Monazone (TN) |
(P) unclassified |
| D07263 |
Clofezone (JAN/INN); Clofezone dihydrate |
(P) unclassified |
| D07264 |
Bumadizone (INN) |
(P) unclassified |
| D07265 |
Lonazolac (INN) |
(P) unclassified |
| D07266 |
Oxametacin (INN) |
(P) unclassified |
| D07267 |
Droxicam (INN) |
(P) unclassified |
| D07268 |
Ibuproxam (INN); Ibudros (TN) |
(P) unclassified |
| D07269 |
Dexketoprofen (INN) |
(P) unclassified |
| D07290 |
Dipyrocetyl (INN) |
(P) unclassified |
| D07291 |
Benorilate (INN); Benorylate |
(P) unclassified |
| D07292 |
Guacetisal (INN); Prontomucil (TN) |
(P) unclassified |
| D07293 |
Imidazole salicylate (INN); Selezen (TN) |
(P) unclassified |
| D07301 |
Phenglutarimide (INN) |
(P) unclassified |
| D07302 |
Bornaprine (INN) |
(P) unclassified |
| D07303 |
Tropatepine (INN) |
(P) unclassified |
| D07349 |
Choline alfoscerate (INN); Gliatilin (TN) |
(P) unclassified |
| D07406 |
Pimethixene (INN); Calmixene (TN) |
(P) unclassified |
| D07421 |
Aloxiprin (INN); Superpyrin (TN) |
(P) unclassified |
| D07443 |
Amfenac (INN) |
(P) unclassified |
| D07453 |
Amtolmetin guacil (INN); Artromed (TN) |
(P) unclassified |
| D07471 |
Atazanavir (INN); Reyataz (TN) |
(P) CYP inhibition: CYP3A4 |
| D07488 |
Balsalazide (INN) |
(P) unclassified |
| D07503 |
Bendazac lysine (BAN); Bendalina (TN) |
(P) unclassified |
| D07511 |
Benzatropine (INN); Benztropine |
(P) unclassified |
| D07513 |
Benzetimide (INN); Spasmental [veterinary] (TN) |
(P) unclassified |
| D07516 |
Benzydamine (INN) |
(P) unclassified |
| D07517 |
Benzydamine salicylate; Fulgium (TN) |
(P) unclassified |
| D07541 |
Bromfenac (INN) |
(P) unclassified |
| D07549 |
Bumadizone calcium salt hemihydrate; Desflam (TN); Eumotol (TN) |
(P) unclassified |
| D07579 |
Aspirin calcium salt; Notras (TN) |
(P) unclassified |
| D07580 |
Aspirin DL-lysine (JAN); Aspirin lysine salt; Aspegic (TN) |
(P) unclassified |
| D07581 |
Aspirin magnesium salt; Mobidin (TN) |
(P) unclassified |
| D07582 |
Aspirin sodium; Sodium acetylsalicylate; Catalgine (TN) |
(P) unclassified |
| D07583 |
Phenytoin and phenobarbital; Aleviatin with phenobarbital (TN) |
(P) unclassified |
| D07595 |
Fosphenytoin sodium hydrate (JAN); Fostoin (TN) |
(P) CYP induction: CYP3A4 |
| D07612 |
Sodium salamidacetate; o-Carbamoylphenoxyacetic acid sodium salt; Clinit-n (TN) |
(P) unclassified |
| D07667 |
Cevimeline (INN) |
(P) Enzyme: CYP3A4 |
| D07710 |
Clarithromycin lactobionate; Klacid (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D07748 |
Conivaptan (INN) |
(P) unclassified |
| D07759 |
Cyclopentolate (INN); Bell Pentolate (TN) |
(P) unclassified |
| D07782 |
Delavirdine (INN) |
(P) unclassified |
| D07796 |
Dexamethasone 21-acetate; Dexamethasone acetate anhydrous; Decaject-L.A. (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
| D07797 |
Dexamethasone isonicotinate; Dexamethasone 21-isonicotinate; Voren [veterinary] (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
| D07798 |
Dexamethasone sodium hemisulfate; Dexamethasone 21-sodium sulfate |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
| D07799 |
Dexamethasone 21-tebutate; Dexamethasone tertiary butyl acetate; Dexamedium [veterinary] (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
| D07800 |
Dexamethasone 21-valerate; Voalla (TN); Zalucs (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
| D07801 |
Dexamethasone phenylpropionate; Dexafort [veterinary] (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
| D07802 |
Dexamethasone phosphate; Decadron-phosphate (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
| D07804 |
Dexetimide hydrochloride; Tremblex (TN) |
(P) unclassified |
| D07816 |
Diclofenac (USAN/INN); Solaraze (TN); Zorvolex (TN) |
(P) unclassified |
| D07817 |
Diclofenac diethylamine; Voltaren Emulgel (TN) |
(P) unclassified |
| D07818 |
Diclofenac epolamine; Diclofenac hydroxyethylpyrrolidine; Flector (TN) |
(P) unclassified |
| D07819 |
Diclofenac calcium; Voltaren Actingo Extra (TN) |
(P) unclassified |
| D07820 |
Dicycloverine (INN); Dicyclomine; Dicymine (TN) |
(P) unclassified |
| D07821 |
Dihexyverine (INN) |
(P) unclassified |
| D07824 |
Diethylamine salicylate; Algesal (TN) |
(P) unclassified |
| D07869 |
Donepezil (JAN/INN); Donaz (TN); Allydone (TN) |
(P) Enzyme: CYP3A4 / Target: ACHE |
| D07888 |
Eltenac (INN); Telzenac (TN) |
(P) unclassified |
| D07909 |
Erythromycin thiocyanate; Erythrocin (TN) |
(P) unclassified |
| D07910 |
Erythromycin stinoprate (INN); Erysec (TN) |
(P) unclassified |
| D07928 |
Ethinylestradiol propanesulfonate; Turisteron (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D07951 |
Fentonium bromide (INN); Ulcesium (TN) |
(P) unclassified |
| D07984 |
Fluvoxamine (INN) |
(P) CYP inhibition: CYP3A4 |
| D07991 |
Fosfosal (INN); Aydolid (TN) |
(P) unclassified |
| D08021 |
Glucametacin (INN); Glucametan (TN) |
(P) unclassified |
| D08058 |
Ibuprofen arginine salt; Zafen (TN) |
(P) unclassified |
| D08059 |
Ibuprofen sodium; Ibuprofen sodium anhydrous; Esprenit (TN) |
(P) unclassified |
| D08094 |
Itopride (INN) |
(P) Target: ACHE |
| D08102 |
Ketoprofen lysine; Artrosilene (TN) |
(P) unclassified |
| D08103 |
Ketoprofen sodium; Orudis (TN) |
(P) unclassified |
| D08104 |
Ketorolac (INN); Toradol (TN) |
(P) unclassified |
| D08142 |
Lonazolac calcium salt; Argun (TN) |
(P) unclassified |
| D08149 |
Loxoprofen (INN) |
(P) unclassified |
| D08153 |
Mabuprofen (INN); Aldospray analgesico (TN) |
(P) unclassified |
| D08157 |
Mazaticol (INN) |
(P) unclassified |
| D08160 |
Mebeverine (INN); Arluy (TN) |
(P) unclassified |
| D08162 |
Meclofenamate sodium; Meclomen (TN) |
(P) unclassified |
| D08190 |
Dipyrone (BAN); Metamizole sodium; Vetalgin (TN) |
(P) unclassified |
| D08209 |
Metixene (INN) |
(P) unclassified |
| D08217 |
Mibefradil (INN) |
(P) unclassified |
| D08259 |
Nelfinavir (INN); Viracept (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D08261 |
Neostigmine (BAN); Prostigmin (TN) |
(P) Target: ACHE |
| D08275 |
Niflumic acid (INN); Niflugel (TN) |
(P) unclassified |
| D08287 |
Norfloxacin nicotinate; Quinabic soluble powder (TN) [veterinary] |
(P) unclassified |
| D08295 |
Olsalazine (INN) |
(P) unclassified |
| D08305 |
Orphenadrine (INN); Mialgin (TN) |
(P) unclassified |
| D08324 |
Oxyphenbutazone (INN); Reozon (TN) |
(P) unclassified |
| D08325 |
Oxyphencyclimine (INN) |
(P) unclassified |
| D08356 |
Phenobarbital diethylamine; Gratusminal (TN) |
(P) unclassified |
| D08363 |
Phenylbutazone calcium; Peralgin (TN) |
(P) unclassified |
| D08364 |
Phenylbutazone sodium; Ambene (TN) |
(P) unclassified |
| D08374 |
Piketoprofen (INN); Calmatel (TN) |
(P) unclassified |
| D08375 |
Piketoprofen hydrochloride; Triparsean (TN) |
(P) unclassified |
| D08376 |
Pilocarpine borate |
(P) unclassified |
| D08382 |
Piperidolate (INN) |
(P) unclassified |
| D08384 |
Pipethanate (INN); Piperilate |
(P) unclassified |
| D08389 |
Pirenzepine (USAN/INN) |
(P) unclassified |
| D08395 |
Piroheptine (INN) |
(P) unclassified |
| D08425 |
Procyclidine (INN) |
(P) unclassified |
| D08426 |
Profenamine (INN) |
(P) unclassified |
| D08427 |
Proglumetacin (INN); Bruxel (TN) |
(P) unclassified |
| D08441 |
Propiverine (INN) |
(P) Enzyme: CYP3A4 |
| D08479 |
Rifampicin sodium; Rifadine (TN) |
(P) CYP induction: CYP3A4 |
| D08501 |
Trolamine salicylate (USP); Salicylic acid trolamine; Salicylic acid triethanolamine; Arthricream (TN) |
(P) unclassified |
| D08522 |
Solifenacin (INN) |
(P) Enzyme: CYP3A4 |
| D08555 |
Tacrine (INN); Tacrinal (TN) |
(P) Target: ACHE |
| D08586 |
Thiosalicylic acid; Pirosal (TN); Thiocyl (TN) |
(P) unclassified |
| D08592 |
Tiaramide (INN) |
(P) unclassified |
| D08595 |
Tiemonium methylsulfate; Visceralgine (TN) |
(P) unclassified |
| D08616 |
Teneligliptin (INN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D08630 |
Tribuzone (prop.INN); Benetazon (TN) |
(P) unclassified |
| D08638 |
Trihexyphenidyl (INN); Apo-trihex (TN) |
(P) unclassified |
| D08653 |
Tropatepine hydrochloride; Lepticur (TN) |
(P) unclassified |
| D08657 |
Apricoxib (USAN/INN) |
(P) unclassified |
| D08774 |
Amoxicillin hydrate, clarithromycin and lansoprazole; Lansap (TN); Prevpac (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D08837 |
Aclidinium bromide (JAN/USAN/INN); Tudorza (TN); Eklira (TN) |
(P) CYP inhibition: CYP3A4 |
| D08838 |
Acotiamide hydrochloride (USAN); Acotiamide hydrochloride hydrate (JAN) |
(P) Target: ACHE |
| D08876 |
Boceprevir (INN/USAN); Victrelis (TN) |
(P) unclassified |
| D08923 |
Fesoterodine fumarate (JAN/USAN); Toviaz (TN) |
(P) Enzyme: CYP3A4 |
| D09012 |
Telaprevir (JAN/USAN/INN); Incivek (TN); Incivo (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D09017 |
Ticagrelor (JAN/USAN/INN); Brilinta (TN) |
(P) unclassified |
| D09347 |
Fostamatinib (USAN) |
(P) Enzyme: CYP3A4 |
| D09348 |
Fostamatinib disodium (USAN); Fostamatinib sodium hydrate (JAN); Fostamatinib disodium hexahydrate; Tavalisse (TN) |
(P) Enzyme: CYP3A4 |
| D09394 |
Fidaxomicin (JAN/USAN); Dificid (TN); Dificlir (TN) |
(P) CYP inhibition: CYP3A4 |
| D09402 |
Darotropium bromide (USAN/INN) |
(P) unclassified |
| D09535 |
Mirabegron (JAN/USAN/INN); Myrbetriq (TN) |
(P) Enzyme: CYP3A4 |
| D09568 |
Naproxcinod (USAN/INN) |
(P) unclassified |
| D09638 |
Lomitapide mesylate (USAN); Lomitapide mesilate (JAN); Juxtapid (TN); Lojuxta (TN) |
(P) Enzyme: CYP3A4 |
| D09701 |
Abiraterone acetate (JAN/USP); Zytiga (TN) |
(P) Enzyme: CYP3A4 |
| D09731 |
Crizotinib (JAN/USAN/INN); Xalkori (TN) |
(P) Enzyme: CYP3A4 |
| D09750 |
Ipidacrine hydrochloride hydrate (JAN) |
(P) Target: ACHE |
| D09752 |
Carpronium chloride hydrate (JAN); Furozin (TN) |
(P) unclassified |
| D09756 |
Teneligliptin hydrobromide hydrate (JAN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D09760 |
Ibuprofen sodium (USAN); Ibuprofen sodium hydrate |
(P) unclassified |
| D09799 |
Carotegrast methyl (JAN); Carogra (TN) |
(P) CYP inhibition: CYP3A4 |
| D09819 |
Chlorpromazine tannate (JAN) |
(P) unclassified |
| D09881 |
Cobicistat (JAN/USAN/INN); Tybost (TN) |
(P) Enzyme-Target: CYP3A4 |
| D09894 |
Eliglustat tartrate (JAN/USAN); Eliglustat hemitartrate; Cerdelga (TN) |
(P) unclassified |
| D09917 |
Latrepirdine (USAN/INN) |
(P) Target: ACHE |
| D09918 |
Latrepirdine dihydrochloride (USAN); Dimebolin; Dimebon |
(P) Target: ACHE |
| D09996 |
Vemurafenib (JAN/USAN/INN); Zelboraf (TN) |
(P) CYP induction: CYP3A4 |
| D10003 |
Hemin (JAN); Normosang (TN); Panhematin (TN) |
(P) CYP induction: CYP3A4 |
| D10017 |
Naproxen etemesil (USAN) |
(P) unclassified |
| D10065 |
Daclatasvir (USAN) |
(P) Enzyme: CYP3A4 |
| D10081 |
Simeprevir (JAN/USAN) |
(P) unclassified |
| D10104 |
Dabrafenib mesylate (USAN); Dabrafenib mesilate (JAN); Tafinlar (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
| D10105 |
Daclatasvir dihydrochloride (USAN); Daclatasvir hydrochloride (JAN); Daklinza (TN) |
(P) Enzyme: CYP3A4 |
| D10127 |
Glycerol phenylbutyrate (JAN/USAN); Ravicti (TN) |
(P) unclassified |
| D10161 |
Sarilumab (USAN); Sarilumab (genetical receombination) (JAN); Kevzara (TN) |
(P) unclassified |
| D10180 |
Umeclidinium (USAN) |
(P) unclassified |
| D10181 |
Umeclidinium bromide (JAN/USAN); Incruse ellipta (TN) |
(P) unclassified |
| D10218 |
Enzalutamide (JAN/USAN); Xtandi (TN) |
(P) unclassified |
| D10246 |
Omeprazole, clarithromycin and amoxicillin; Omeclamox-pak (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D10254 |
Esflurbiprofen (JAN/USAN) |
(P) unclassified |
| D10372 |
Palbociclib (JAN/USAN); Ibrance (TN) |
(P) unclassified |
| D10466 |
Vonoprazan fumarate (JAN/USAN); Takecab (TN); Voquezna (TN) |
(P) Enzyme: CYP3A4 |
| D10469 |
Simeprevir sodium (JAN); Olysio (TN); Sovriad (TN) |
(P) unclassified |
| D10513 |
Clopidogrel sulfate and aspirin; Clopidogrel and acetylsalicyclic acid; Complavin (TN) |
(P) Enzyme: CYP3A4 |
| D10519 |
Rabeprazole, amoxicillin and clarithromycin; Rabecure (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D10527 |
Acetylsalicylic acid and lansoprazole; Acetylsalicylic acid and lansoprazole; Takelda (TN) |
(P) Enzyme: CYP3A4 |
| D10551 |
Ceritinib (JAN/USAN/INN); Zykadia (TN) |
(P) unclassified |
| D10564 |
Amenamevir (JAN/INN); Amenalief (TN) |
(P) unclassified |
| D10566 |
Pasireotide pamoate (JAN); Signifor lar (TN) |
(P) unclassified |
| D10582 |
Dasabuvir, ombitasvir, paritaprevir and ritonavir; Viekira pak (TN) |
(P) CYP inhibition: CYP3A4 |
| D10633 |
Finerenone (JAN/USAN/INN); Kerendia (TN) |
(P) Enzyme: CYP3A4 |
| D10639 |
Grazoprevir (USAN); Grazoprevir hydrate (JAN); Grazyna (TN) |
(P) unclassified |
| D10643 |
Isavuconazonium sulfate (JAN/USAN); Cresemba (TN) |
(P) unclassified |
| D10644 |
Isavuconazonium (USAN) |
(P) unclassified |
| D10656 |
Polmacoxib (USAN/INN) |
(P) unclassified |
| D10689 |
Amifampridine phosphate (JAN/USAN); Firdapse (TN) |
(P) unclassified |
| D10745 |
Ombitasvir, paritaprevir and ritonavir; Technivie (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D10753 |
Atazanavir and cobicistat; Evotaz (TN) |
(P) Enzyme: CYP3A4 |
| D10755 |
Elvitegravir, cobicistat, emtricitabine and tenofovir alafenamide; Genvoya (TN) |
(P) unclassified |
| D10756 |
Elvitegravir, cobicistat, emtricitabine and tenofovir disoproxil; Stribild (TN) |
(P) unclassified |
| D10762 |
Fosravuconazole L-lysine ethanolate (JAN) |
(P) unclassified |
| D10774 |
Vonoprazan, amoxicillin and metronidazole; Vonopion (TN) |
(P) Enzyme: CYP3A4 |
| D10775 |
Vonoprazan, amoxicillin and clarithromycin; Vonosap (TN); Voquenza (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D10801 |
Letermovir (JAN/USAN/INN); Prevymis (TN) |
(P) unclassified |
| D10832 |
Darunavir and cobicistat; Prezcobix (TN); Rezolsta (TN) |
(P) unclassified |
| D10895 |
Fosaprepitant (INN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4 |
| D10926 |
Entrectinib (JAN/USAN/INN); Rozlytrek (TN) |
(P) Enzyme: CYP3A4 |
| D10938 |
Glycopyrronium (USAN) |
(P) unclassified |
| D10939 |
Glycopyrronium tosylate (USAN); Glycopyrronium tosilate hydrate (JAN); Glycopyrronium tosylate monohydrate; Qbrexza (TN); Rapifort (TN) |
(P) unclassified |
| D10989 |
Sofpironium bromide (JAN/USAN/INN); Ecclock (TN); Sofdra (TN) |
(P) Enzyme: CYP3A4 |
| D10990 |
Somatrogon (USAN/INN); Somatrogon (genetical recombination) (JAN); Somatrogon-ghla; Ngenla (TN) |
(P) unclassified |
| D11012 |
Lorlatinib (JAN/USAN/INN); Lorbrena (TN) |
(P) unclassified |
| D11027 |
Ropeginterferon alfa-2b (INN); Ropeginterferon alfa-2b (genetical recombination) (JAN); Ropeginterferon alfa-2b-njft; Besremi (TN) |
(P) unclassified |
| D11040 |
Apalutamide (JAN/INN); Erleada (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
| D11053 |
Encorafenib (JAN/USAN/INN); Braftovi (TN) |
(P) Enzyme: CYP3A4 |
| D11090 |
Ivosidenib (JAN/USAN/INN); Tibsovo (TN) |
(P) unclassified |
| D11138 |
Larotrectinib sulfate (JAN/USAN); Vitrakvi (TN) |
(P) unclassified |
| D11194 |
Somapacitan (USAN/INN); Somapacitan (genetical recombination) (JAN); Somapacitan-beco; Sogroya (TN) |
(P) unclassified |
| D11296 |
Fedratinib hydrochloride (USAN); Fedratinib hydrochloride hydrate (JAN); Fedratinib dihydrochloride monohydrate; Inrebic (TN) |
(P) Enzyme: CYP3A4 |
| D11370 |
Fosnetupitant chloride hydrochloride (JAN/USAN); Arokaris (TN) |
(P) unclassified |
| D11371 |
Capivasertib (JAN/USAN); Truqap (TN) |
(P) unclassified |
| D11382 |
Darunavir, cobicistat, emtricitabine and tenofovir alafenamide; Symtuza (TN) |
(P) unclassified |
| D11422 |
Zanubrutinib (JAN/USAN/INN); Brukinsa (TN) |
(P) unclassified |
| D11454 |
Repotrectinib (JAN/USAN); Augtyro (TN) |
(P) Enzyme: CYP3A4 |
| D11485 |
Tazemetostat hydrobromide (JAN/USAN); Tazverik (TN) |
(P) unclassified |
| D11557 |
Tecovirimat hydrate (JAN); Tecovirimat monohydrate; Tpoxx (TN); Tepoxx (TN) |
(P) unclassified |
| D11565 |
Grazoprevir (USAN/INN); Grazoprevir anhydrous |
(P) unclassified |
| D11673 |
Berotralstat (USAN/INN) |
(P) CYP inhibition: CYP3A4 |
| D11674 |
Berotralstat hydrochloride (JAN/USAN); Orladeyo (TN) |
(P) CYP inhibition: CYP3A4 |
| D11708 |
Givosiran sodium (JAN); Givlaari (TN) |
(P) unclassified |
| D11713 |
Selpercatinib (JAN/USAN/INN); Retevmo (TN) |
(P) Enzyme: CYP3A4 |
| D11804 |
Aspirin and vonoprazan; Cabpirin (TN) |
(P) unclassified |
| D11815 |
Belumosudil (USAN) |
(P) Enzyme: CYP3A4 |
| D11816 |
Belumosudil mesylate (USAN); Belumosudil mesilate (JAN); Rezurock (TN) |
(P) Enzyme: CYP3A4 |
| D11835 |
Vorasidenib citrate (USAN); Vorasidenib citric acid hydrate (JAN); Voranigo (TN) |
(P) unclassified |
| D11887 |
Daridorexant hydrochloride (JAN/USAN); Quviviq (TN) |
(P) unclassified |
| D11920 |
Pimitespib (JAN); Jeselhy (TN) |
(P) unclassified |
| D11954 |
Belzutifan (JAN/USAN/INN); Welireg (TN) |
(P) unclassified |
| D11968 |
Teneligliptin hydrobromide (JAN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D11970 |
Ritlecitinib tosylate (USAN); Ritlecitinib tosilate (JAN); Litfulo (TN) |
(P) unclassified |
| D12050 |
Pirtobrutinib (JAN/USAN); Jaypirca (TN) |
(P) Enzyme: CYP3A4 |
| D12055 |
Sotorasib (JAN/USAN); Lumakras (TN) |
(P) unclassified |
| D12217 |
Imlunestrant tosylate (USAN); Imlunestrant tosilate (JAN); Inluriyo (TN) |
(P) Enzyme: CYP3A4 |
| D12245 |
Lazertinib mesylate (USAN); Lazertinib mesilate hydrate (JAN); Lazcluze (TN) |
(P) Enzyme: CYP3A4 |
| D12252 |
Iptacopan hydrochloride (USAN); Iptacopan hydrochloride hydrate (JAN); Iptacopan hydrochloride monohydrate; Fabhalta (TN) |
(P) CYP induction: CYP3A4 |
| D12269 |
Nirmatrelvir and ritonavir; Paxlovid (TN) |
(P) Enzyme: CYP3A4 |
| D12318 |
Buntanetap (USAN) |
(P) Target: ACHE |
| D12319 |
Buntanetap tartrate (USAN) |
(P) Target: ACHE |
| D12353 |
Ensitrelvir fumarate (USAN); Ensitrelvir fumaric acid (JAN); Xocova (TN) |
(P) unclassified |
| D12364 |
Taletrectinib adipate (JAN/USAN); Ibtrozi (TN) |
(P) unclassified |
| D12442 |
Tucatinib ethanolate (JAN); Tucatinib hemiethanolate; Tukysa (TN) |
(P) unclassified |
| D12444 |
Nilotinib hydrochloride dihydrate (JAN) |
(P) Enzyme: CYP3A4 |
| D12586 |
Mifepristone and misoprostol; Mefeego (TN) |
(P) unclassified |
| D12595 |
Aspirin trelamine (USAN) |
(P) unclassified |
| D12596 |
Aspirin trelamine hydrochloride (USAN) |
(P) unclassified |
| D12597 |
Ibuprofen trelamine (USAN); Ibuprofen diethylaminoethyl ester |
(P) unclassified |
| D12598 |
Ibuprofen trelamine hydrochloride (USAN) |
(P) unclassified |
| D12619 |
Ensitrelvir (USAN/INN) |
(P) unclassified |
| D12637 |
Darunavir hydrate |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D12752 |
Darunavir propylene glycolate |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D12837 |
Risovalisib mesilate hydrate (JAN); Risovalisib mesylate dihydrate; Haizexin (TN) |
(P) unclassified |
| D12930 |
Benzgalantamine (USAN/INN) |
(P) Target: ACHE |
| D12931 |
Benzgalantamine gluconate (USAN); Zunveyl (TN) |
(P) Target: ACHE |
| D13152 |
Aceclidine hydrochloride; Vizz (TN) |
(P) unclassified |
| D13221 |
Direclidine (USAN/INN) |
(P) unclassified |
| D13222 |
Direclidine citrate (USAN); Direclidine citrate monohydrate |
(P) unclassified |
| D13252 |
Betovumeline (USAN/INN) |
(P) unclassified |