| C07005 |
Flunisolide; Flunisolide anhydrous |
(P) unclassified |
| C07370 |
Prednisone; 1,2-Dehydrocortisone; 17,21-Dihydroxypregna-1,4-diene-3,11,20-trione |
(P) unclassified |
| D00088 |
Hydrocortisone (JP19/USP/INN); HC; Acticort (TN); Anusol HC (TN); Colocort (TN); Cortef (TN); Hytone (TN); Plenadren (TN) |
(P) Enzyme: CYP3A / CYP inhibition: CYP3A |
| D00105 |
Estradiol (JAN/USP/INN); Climara (TN); Divigel (TN); Estrace (TN); Estraderm (TN); Estrasorb (TN); Estring (TN); Estrogel (TN); Innofem (TN); Vagifem (TN); Vivelle (TN) |
(P) unclassified |
| D00107 |
Tacrolimus (USP/INN); Tacrolimus hydrate (JP19); Prograf (TN); Protopic (TN) |
(P) unclassified |
| D00165 |
Hydrocortisone acetate (JP19/USP); Cortifoam (TN); U-cort (TN) |
(P) Enzyme: CYP3A / CYP inhibition: CYP3A |
| D00184 |
Cyclosporine (USP); Ciclosporin (JP19); Gengraf (TN); Neoral (TN); Restasis (TN); Sandimmune (TN) |
(P) unclassified |
| D00211 |
Rifampin (USP); Rifampicin (JP19/INN); Rifadin (TN); Rimactane (TN) |
(P) unclassified |
| D00225 |
Alprazolam (JP19/USP/INN); Xanax (TN) |
(P) Enzyme: CYP3A / CYP inhibition: CYP3A |
| D00244 |
Betamethasone (JP19/USP/INN); Celestone (TN); Rinderon (TN) |
(P) unclassified |
| D00246 |
Budesonide (JP19/USP/INN); Entocort EC (TN); Pulmicort (TN); Rhinocort (TN); Uceris (TN) |
(P) unclassified |
| D00252 |
Carbamazepine (JP19/USP/INN); Equetro (TN); Tegretol (TN) |
(P) unclassified |
| D00277 |
Clindamycin (USAN/INN); Cleocin (TN) |
(CI,P) unclassified |
| D00283 |
Clozapine (JAN/USP/INN); Clozaril (TN) |
(P) unclassified |
| D00292 |
Dexamethasone (JP19/USP/INN); Decadron (TN); Maxidex (TN) |
(P) unclassified |
| D00293 |
Diazepam (JP19/USP/INN); Diastat (TN); Valium (TN) |
(P) unclassified |
| D00295 |
Cimetidine (JP19/USP/INN); Tagamet (TN) |
(P) unclassified |
| D00298 |
Digoxin (JP19/USP); Lanoxicaps (TN); Lanoxin (TN) |
(P) Transporter inhibition: ABCB1 |
| D00303 |
Disopyramide (JP19/USAN/INN); Rythmodan P (TN) |
(P) unclassified |
| D00319 |
Felodipine (JP19/USP/INN); Plendil (TN) |
(P) unclassified |
| D00322 |
Fluconazole (JP19/USP/INN); Diflucan (TN) |
(P) unclassified |
| D00324 |
Flunisolide (JAN/USP); Aerospan (TN); Nasalide (TN) |
(P) unclassified |
| D00325 |
Fluocinonide (JP19/USP/INN); Lidex (TN); Vanos (TN) |
(P) unclassified |
| D00328 |
Flurandrenolide (USP); Fludroxycortide (JAN/INN); Cordran (TN) |
(P) unclassified |
| D00350 |
Itraconazole (JP19/USP); Itrizole (TN); Sporanox (TN) |
(P) unclassified |
| D00364 |
Loratadine (JAN/USP/INN); Claritin (TN) |
(P) unclassified |
| D00371 |
Theophylline (JP19); Elixophyllin (TN); Quibron-t (TN); Theo-24 (TN); Theodur G (TN); Theolair (TN); Uniphyl (TN) |
(P) unclassified |
| D00385 |
Triamcinolone (JP19/USP/INN); Aristocort (TN); Kenacort (TN) |
(P) unclassified |
| D00387 |
Triazolam (JP19/USP/INN); Halcion (TN) |
(P) unclassified |
| D00407 |
Methylprednisolone (JP19/USP/INN); Medrol (TN) |
(P) unclassified |
| D00411 |
Zafirlukast (JAN/USAN/INN); Accolate (TN) |
(P) unclassified |
| D00424 |
Rifabutin (JAN/USP/INN); Mycobutin (TN) |
(P) CYP induction: CYP3A |
| D00427 |
Ritonavir (JAN/USP/INN); Norvir (TN) |
(P) Enzyme: CYP3A / CYP inhibition: CYP3A |
| D00434 |
Simvastatin (JP19/USP/INN); MK-733; Zocor (TN) |
(P) unclassified |
| D00435 |
Nevirapine (JAN/USP/INN); Viramune (TN) |
(P) unclassified |
| D00458 |
Quetiapine fumarate (JP19/USP); Seroquel (TN) |
(P) unclassified |
| D00472 |
Prednisolone (JP19/USP/INN); Delta-cortef (TN) |
(P) Enzyme: CYP3A / CYP inhibition: CYP3A |
| D00473 |
Prednisone (USP); Prednisone monohydrate; Deltasone (TN); Meticorten (TN); Rayos (TN) |
(P) unclassified |
| D00491 |
Paclitaxel (JAN/USP/INN); Abraxane (TN); Taxol (TN) |
(P) unclassified |
| D00506 |
Phenobarbital (JP19/USP/INN); Luminal (TN) |
(P) CYP induction: CYP3A |
| D00512 |
Phenytoin (JP19/USP/INN); Dilantin (TN) |
(P) CYP induction: CYP3A |
| D00528 |
Caffeine (USP); Anhydrous caffeine (JP19); Anhydrous caffeine (TN); Respia (TN) |
(P) unclassified |
| D00550 |
Midazolam (JAN/USP/INN); Dormicum (TN); Buccolam (TN); Nayzilam (TN) |
(P) unclassified |
| D00560 |
Pimozide (JP19/USP/INN); Orap (TN) |
(CI) unclassified |
| D00563 |
Mirtazapine (JAN/USP/INN); Remeron (TN); Reflex (TN) |
(P) unclassified |
| D00570 |
Colchicine (JP19/USP) |
(CI,P) Transporter inhibition: ABCB1 |
| D00615 |
Amlodipine besylate (USP); Amlodipine besilate (JP19); Norvasc (TN) |
(P) unclassified |
| D00619 |
Verapamil hydrochloride (JP19/USP); Calan (TN); Covera-hs (TN); Vasolan (TN); Verelan (TN) |
(P) Transporter inhibition: ABCB1 |
| D00636 |
Amiodarone hydrochloride (JP19/USP); Ancaron (TN); Cordarone (TN); Nexterone (TN) |
(CI) unclassified |
| D00637 |
Disopyramide phosphate (JAN/USP); Norpace (TN) |
(P) unclassified |
| D00661 |
Cevimeline hydrochloride (USAN); Cevimeline hydrochloride hydrate (JAN); Evoxac (TN); Saligren (TN) |
(P) unclassified |
| D00670 |
Donepezil hydrochloride (JP19/USP); Aricept (TN) |
(P) unclassified |
| D00671 |
Fexofenadine hydrochloride (JP19/USP); Allegra (TN) |
(P) unclassified |
| D00680 |
Methylergonovine maleate (USP); Methylergometrine maleate (JP19); Methergine (TN) |
(P) unclassified |
| D00689 |
Beclomethasone dipropionate (USP); Beclometasone dipropionate (JP19); Beclovent (TN); Qnasl (TN); Vanceril (TN) |
(P) unclassified |
| D00690 |
Mometasone furoate (JAN/USP); Asmanex (TN); Elocon (TN) |
(P) unclassified |
| D00696 |
Midazolam hydrochloride (USAN); Versed (TN) |
(P) unclassified |
| D00701 |
Phenobarbital sodium (JAN/USP/INN); Luminal sodium (TN) |
(P) CYP induction: CYP3A |
| D00710 |
Valproate sodium (USAN); Sodium valproate (JP19); Depakene (TN); Selenica (TN) |
(P) unclassified |
| D00751 |
Methylprednisolone sodium succinate (JAN/USP); A-methapred (TN); Solu-medrol (TN) |
(P) unclassified |
| D00753 |
Sirolimus (JAN/USAN/INN); Rapamune (TN); Rapamycin (TN) |
(P) Transporter inhibition: ABCB1 |
| D00780 |
Bromocriptine mesylate (USP); Bromocriptine mesilate (JP19); Parlodel (TN) |
(P) unclassified |
| D00785 |
Selegiline hydrochloride (JAN/USP); Eldepryl (TN) |
(P) unclassified |
| D00821 |
Venlafaxine hydrochloride (JAN/USP); Effexor (TN) |
(P) unclassified |
| D00836 |
Buprenorphine hydrochloride (JP19/USP); Buprenex (TN) |
(P) unclassified |
| D00874 |
Moxifloxacin hydrochloride (JAN/USP); Avelox (TN); Vigamox (TN) |
(P) unclassified |
| D00879 |
Rifapentine (USAN/INN); Priftin (TN) |
(P) unclassified |
| D00892 |
Fluvastatin sodium (JAN/USP); Lescol (TN) |
(P) unclassified |
| D00896 |
Efavirenz (JAN/USP/INN); Sustiva (TN) |
(P) unclassified |
| D00972 |
Betamethasone sodium phosphate (JP19/USP); Celestone (TN) |
(P) unclassified |
| D00973 |
Cortisone acetate (JP19/USP); Cortone acetate (TN) |
(P) unclassified |
| D00975 |
Dexamethasone sodium phosphate (JAN/USP); Dalalone (TN); Maxidex (TN) |
(P) unclassified |
| D00976 |
Hydrocortisone cypionate |
(P) Enzyme: CYP3A / CYP inhibition: CYP3A |
| D00977 |
Hydrocortisone sodium phosphate (JP19/USP); Hydrocortone phosphate (TN) |
(P) Enzyme: CYP3A / CYP inhibition: CYP3A |
| D00978 |
Hydrocortisone sodium succinate (JP19/USP); A-hydrocort (TN); Solu-cortef (TN) |
(P) Enzyme: CYP3A / CYP inhibition: CYP3A |
| D00979 |
Methylprednisolone acetate (JAN/USP); Depo-medrol (TN) |
(P) unclassified |
| D00980 |
Prednisolone acetate (JP19/USP/INN); Econopred (TN); Pred forte (TN) |
(P) unclassified |
| D00981 |
Prednisolone sodium phosphate (JP19/USP); Pediapred (TN) |
(P) unclassified |
| D00982 |
Prednisolone tebutate (JAN/USP); Hydeltra-TBA (TN) |
(P) unclassified |
| D00983 |
Triamcinolone acetonide (JP19/USP); Azmacort (TN); Kenalog (TN); Nasacort (TN) |
(P) unclassified |
| D00984 |
Triamcinolone diacetate (JAN/USP); Aristocort (TN) |
(P) unclassified |
| D00985 |
Triamcinolone hexacetonide (USP/INN); Aristospan (TN) |
(P) unclassified |
| D00986 |
Fludrocortisone acetate (JP19/USP); Florinef acetate (TN) |
(P) unclassified |
| D00987 |
Cabergoline (JP19/USP/INN); Cabaser (TN); Dostinex (TN) |
(P) unclassified |
| D01061 |
Irinotecan hydrochloride (USP); Irinotecan hydrochloride hydrate (JP19); Irinotecan hydrochloride trihydrate; CPT 11; CPT-11; Campto (TN); Camptosar (TN); Onivyde (TN) |
(P) unclassified |
| D01068 |
Vinblastine sulfate (JP19/USP); Exal (TN); Velban (TN) |
(P) unclassified |
| D01073 |
Clindamycin phosphate (JP19/USP); Cleocin (TN); Dalacin-S (TN); Evoclin (TN) |
(CI,P) unclassified |
| D01104 |
Barnidipine hydrochloride (JAN); Hypoca (TN) |
(P) unclassified |
| D01115 |
Eplerenone (JP19/USAN/INN); Inspra (TN) |
(P) unclassified |
| D01145 |
Azelnidipine (JP19/INN); Calblock (TN) |
(P) unclassified |
| D01160 |
Saquinavir mesylate (USP); Saquinavir mesilate (JAN); Invirase (TN) |
(P) Transporter inhibition: ABCB1 |
| D01176 |
Blonanserin (JP19/INN); AD 5423 |
(P) unclassified |
| D01213 |
Tolvaptan (JP19/USAN/INN); Samsca (TN) |
(P) Transporter inhibition: ABCB1 |
| D01227 |
Bosentan (USAN); Bosentan hydrate (JAN); Tracleer (TN) |
(P) unclassified |
| D01229 |
Paramethasone acetate (JAN/USAN); Haldrone (TN) |
(P) unclassified |
| D01239 |
Prednisolone sodium succinate (JP19/USP); Kohakusanin (TN) |
(P) unclassified |
| D01266 |
Difluprednate (JAN/USAN/INN); Durezol (TN) |
(P) unclassified |
| D01272 |
Clobetasol propionate (JP19/USP); Clobex (TN); Cormax (TN); Olux (TN) |
(P) unclassified |
| D01273 |
Clobetasone butyrate (JAN/USAN); Kindavate (TN) |
(P) unclassified |
| D01280 |
Warfarin potassium (JP19); Athrombin-K (TN) |
(P) unclassified |
| D01287 |
Levobupivacaine hydrochloride (JAN/USAN); Chirocaine (TN) |
(P) unclassified |
| D01308 |
Halcinonide (JAN/USP/INN); Halog (TN) |
(P) unclassified |
| D01327 |
Diflorasone diacetate (JP19/USP); Florone (TN); Psorcon (TN) |
(P) unclassified |
| D01357 |
Betamethasone valerate (JP19/USP); Beta-Val (TN); Luxiq (TN); Rinderon-V (TN) |
(P) unclassified |
| D01367 |
Fluorometholone (JP19/USP/INN); NSC 33001; Fluor-op (TN); Fml (TN); Oxylone (TN) |
(P) unclassified |
| D01372 |
Zopiclone (JP19/INN); Amoban (TN) |
(P) unclassified |
| D01387 |
Amcinonide (JAN/USP/INN); Cyclocort (TN) |
(P) unclassified |
| D01402 |
Betamethasone acetate (JAN/USP) |
(P) unclassified |
| D01429 |
Fosfluconazole (JAN/INN); Prodif (TN) |
(P) unclassified |
| D01434 |
Deprodone propionate (JAN); Allomidon (TN) |
(P) unclassified |
| D01441 |
Imatinib mesylate (USAN); Imatinib mesilate (JAN); Gleevec (TN); Glivec (TN) |
(P) unclassified |
| D01442 |
Hydrocortisone succinate (JP19) |
(P) Enzyme: CYP3A / CYP inhibition: CYP3A |
| D01464 |
Flumethasone pivalate (USP); Flumetasone pivalate (JAN/BAN); Locorten (TN) |
(P) unclassified |
| D01478 |
Ebastine (JP19/USAN/INN); Kestine (TN) |
(P) unclassified |
| D01510 |
Dexamethasone metasulfobenzoate sodium (JAN); Dexamethazone metasulfobenzoate sodium; Dexapos; Santeson (TN) |
(P) unclassified |
| D01615 |
Dexamethasone palmitate (JAN); Dexamethasone 21-palmitate; Limethason (TN) |
(P) unclassified |
| D01619 |
Hydrocortisone butyrate (JP19/USP); Locoid (TN) |
(P) Enzyme: CYP3A / CYP inhibition: CYP3A |
| D01632 |
Dexamethasone dipropionate (USAN); Dexamethasone propionate (JAN); Hifmeta (TN) |
(P) unclassified |
| D01637 |
Betamethasone dipropionate (JP19/USP); Diprolene (TN); Rinderon-DP (TN); Sernivo (TN) |
(P) unclassified |
| D01689 |
Loteprednol etabonate (JAN/USAN); Lotemax (TN) |
(P) unclassified |
| D01703 |
Ciclesonide (JAN/USAN/INN); Alvesco (TN); Omnaris (TN); Zetonna (TN) |
(P) unclassified |
| D01708 |
Fluticasone propionate (JAN/USP); Cutivate (TN); Flonase (TN); Flovent (TN) |
(P) unclassified |
| D01712 |
Theophylline sodium acetate (JAN) |
(P) unclassified |
| D01745 |
Domperidone (JP19/USAN/INN); Motilium (TN) |
(P) unclassified |
| D01764 |
Diflucortolone valerate (JP19); Afusona (TN) |
(P) unclassified |
| D01769 |
Vindesine sulfate (JAN/USAN); Fildesin (TN) |
(P) Enzyme: CYP3A / CYP inhibition: CYP3A |
| D01820 |
Alclometasone dipropionate (JAN/USP); Aclovate (TN) |
(P) unclassified |
| D01825 |
Fluocinolone acetonide (JP19/USP/INN); Fluocet (TN); Retisert (TN); Synalar (TN) |
(P) unclassified |
| D01832 |
Modafinil (JAN/USP/INN); Provigil (TN) |
(P) unclassified |
| D01886 |
Hydrocortisone probutate (USAN); Hydrocortisone butyrate propionate (JAN); Hydrocortisone buteprate; Pandel (TN) |
(P) Enzyme: CYP3A / CYP inhibition: CYP3A |
| D01896 |
Cilostazol (JP19/USP/INN); Pletal (TN) |
(P) unclassified |
| D01915 |
Rosuvastatin calcium (JP19/USP); ZD 4522; Crestor (TN) |
(P) unclassified |
| D01935 |
Vinorelbine tartrate (USP); Vinorelbine ditartrate (JAN); KW 2307; Navelbine (TN) |
(P) unclassified |
| D01948 |
Dexamethasone valerate (JAN); Dexamethasone 17-valerate; DV-17; Voalla ointment (TN) |
(P) unclassified |
| D01973 |
Eletriptan hydrobromide (JAN/USAN); Relpax (TN) |
(P) unclassified |
| D01977 |
Gefitinib (JP19/USAN/INN); Iressa (TN) |
(P) unclassified |
| D01990 |
Clindamycin palmitate hydrochloride (JAN/USP); Cleocin (TN) |
(CI,P) unclassified |
| D01998 |
Prednisolone farnesylate (JAN); PNF 21; Farnerate (TN) |
(P) unclassified |
| D02008 |
Tadalafil (JAN/USP/INN); Adcirca (TN); Cialis (TN); Zalutia (TN) |
(CI,P) unclassified |
| D02032 |
Betamethasone butyrate propionate (JAN); Antebate (TN) |
(P) unclassified |
| D02096 |
Fosphenytoin sodium (USP); Cerebyx (TN); Sesquient (TN) |
(P) unclassified |
| D02102 |
Methadone hydrochloride (JAN/USP); Dolophine hydrochloride (TN) |
(P) Transporter inhibition: ABCB1 |
| D02103 |
Phenytoin sodium (USP); Phenytoin sodium for injection (JP19); Aleviatin (TN); Dilantin (TN) |
(P) CYP induction: CYP3A |
| D02106 |
Arsenic trioxide (JP19/USAN); Trisenox (TN) |
(P) unclassified |
| D02126 |
Primaquine phosphate (JAN/USP) |
(P) unclassified |
| D02132 |
Clindamycin hydrochloride (JP19/USP); Cleocin hydrochloride (TN); Dalacin (TN) |
(CI,P) unclassified |
| D02156 |
Prednisolone hemisuccinate (USP); Prednisolone succinate (JP19) |
(P) unclassified |
| D02165 |
Docetaxel (USP); Docetaxel hydrate (JP19); Docetaxel trihydrate; Taxotere (TN) |
(P) unclassified |
| D02173 |
Galantamine hydrobromide (JAN/USP); Razadyne (TN); Reminyl (TN) |
(P) unclassified |
| D02174 |
Dexamethasone acetate (JAN/USP); Decadronal (TN) |
(P) unclassified |
| D02197 |
Vincristine sulfate (JP19/USP); VCR; Marqibo (TN); Oncovin (TN); Vincasar (TN); Vincrex (TN) |
(P) Enzyme: CYP3A / CYP inhibition: CYP3A |
| D02211 |
Dihydroergotamine mesylate (USP); Dihydroergotamine mesilate (JP19); Migranal (TN); Trudhesa (TN) |
(CI) unclassified |
| D02229 |
Sildenafil citrate (JAN/USP); Revatio (TN); Viagra (TN) |
(P) unclassified |
| D02258 |
Atorvastatin calcium (USP); Atorvastatin calcium hydrate (JP19); Atorvastatin calcium trihydrate; Atorvaliq (TN); Lipitor (TN) |
(P) Transporter inhibition: ABCB1 |
| D02272 |
Quinidine sulfate (USP); Quinidine sulfate hydrate (JP19); Quinidex (TN) |
(P) unclassified |
| D02286 |
Betamethasone benzoate (USP); Uticort (TN) |
(P) unclassified |
| D02287 |
Clocortolone pivalate (USP); Cloderm (TN) |
(P) unclassified |
| D02288 |
Hydrocortisone valerate (USP); Westcort (TN) |
(P) Enzyme: CYP3A / CYP inhibition: CYP3A |
| D02289 |
Medrysone (USAN); HMS (TN) |
(P) unclassified |
| D02346 |
Lincomycin hydrochloride hydrate (JP19/USP); LCM; Lincocin (TN) |
(CI) unclassified |
| D02484 |
Artemether and lumefantrine; Coartem (TN) |
(P) Enzyme: CYP3A / CYP inhibition: CYP3A |
| D02554 |
Rifaximin (JAN/USAN/INN); Xifaxan (TN) |
(P) Transporter inhibition: ABCB1 |
| D02587 |
Metildigoxin (JP19); Lanirapid (TN) |
(P) Transporter inhibition: ABCB1 |
| D02591 |
Dexamethasone acefurate (USAN/INN) |
(P) unclassified |
| D02592 |
Dexamethasone beloxil (USAN) |
(P) unclassified |
| D02691 |
Somatropin (USP/INN); Somatropin (genetical recombination) (JAN); Human growth hormone (JAN); Asellacrin (TN); Humatrope (TN); Nutropin (TN); Omnitrope (TN) |
(P) unclassified |
| D02714 |
Everolimus (JAN/USAN/INN); Afinitor (TN); Votubia (TN); Zortress (TN) |
(P) Transporter inhibition: ABCB1 |
| D02732 |
Pranlukast hydrate (JP19); Onon (TN) |
(P) unclassified |
| D02968 |
Aprepitant (JAN/USP/INN); Aponvie (TN); Emend (TN); Cinvanti (TN) |
(P) unclassified |
| D03106 |
Bexarotene (JAN/USAN/INN); Targretin (TN) |
(P) CYP induction: CYP3A |
| D03213 |
Apixaban (JAN/USAN/INN); Eliquis (TN) |
(P) Transporter inhibition: ABCB1 |
| D03259 |
Gemtuzumab ozogamicin (USAN); Gemtuzumab ozogamicin (genetical recombination) (JAN); Gemtuzumab (INN); Mylotarg (TN) |
(P) unclassified |
| D03260 |
Vardenafil hydrochloride hydrate (JAN); Vardenafil monohydrochloride trihydrate; Levitra (TN); Staxyn (TN) |
(P) unclassified |
| D03301 |
Prednisolone valerate acetate (JAN); PDL; Spirazon (TN) |
(P) unclassified |
| D03325 |
Mometasone furoate hydrate (JAN); Mometasone furoate monohydrate; Nasonex (TN) |
(P) unclassified |
| D03503 |
Cimetidine hydrochloride (USP) |
(P) unclassified |
| D03505 |
Cinacalcet hydrochloride (JAN/USAN); Sensipar (TN); Mimpara (TN) |
(P) unclassified |
| D03541 |
Clocortolone acetate (USAN) |
(P) unclassified |
| D03561 |
Cloprednol (USAN/INN); Cloradryn (TN) |
(P) unclassified |
| D03594 |
Cortivazol (USAN) |
(P) unclassified |
| D03658 |
Dasatinib (JAN/INN) |
(P) unclassified |
| D03669 |
Deferasirox (JAN/USAN/INN); Exjade (TN); Jadenu (TN) |
(P) unclassified |
| D03671 |
Deflazacort (USAN/INN); Emflaza (TN) |
(P) Transporter inhibition: ABCB1 |
| D03693 |
Desloratadine (JAN/USP/INN); Clarinex (TN) |
(P) unclassified |
| D03696 |
Desonide (USP/INN); Desowen (TN); Verdeso (TN) |
(P) unclassified |
| D03697 |
Desoximetasone (USP/INN); Topicort (TN) |
(P) unclassified |
| D03799 |
Dienogest (JAN/USAN/INN); Endometrion (TN) |
(P) unclassified |
| D03812 |
Diflucortolone (USAN) |
(P) unclassified |
| D03813 |
Diflucortolone pivalate (USAN) |
(P) unclassified |
| D04024 |
Lapatinib ditosylate (USAN); Lapatinib tosilate hydrate (JAN); Lapatinib ditosylate monohydrate; Tykerb (TN); Tyverb (TN) |
(P) Transporter inhibition: ABCB1 |
| D04112 |
Etravirine (JAN/USAN/INN); Intelence (TN) |
(P) unclassified |
| D04201 |
Flucloronide (USAN); Fluclorolone acetonide (INN) |
(P) unclassified |
| D04208 |
Flumethasone (USAN); Flumetasone (INN) |
(P) unclassified |
| D04214 |
Flunisolide acetate (USAN) |
(P) unclassified |
| D04217 |
Fluocortin butyl (USAN) |
(P) unclassified |
| D04218 |
Fluocortolone (USAN/INN) |
(P) unclassified |
| D04219 |
Fluocortolone caproate (USAN) |
(P) unclassified |
| D04221 |
Fluorometholone acetate (USP); Fluorometholone 17-acetate; Flarex (TN) |
(P) unclassified |
| D04225 |
Fluperolone acetate (USAN); Methral (TN) |
(P) unclassified |
| D04244 |
Formocortal (USAN/INN); Deflamene (TN) |
(P) unclassified |
| D04409 |
Halobetasol propionate (USP); Ulobetasol propionate; Ultravate (TN) |
(P) unclassified |
| D04446 |
Betamethasone acetate and betamethasone sodium phosphate; Celestone soluspan (TN); Rinderon (TN) |
(P) unclassified |
| D04447 |
Betamethasone and d-chlorpheniramine maleate; Celestamine (TN) |
(P) unclassified |
| D04467 |
Hydrocortisone hemisuccinate (USP) |
(P) Enzyme: CYP3A / CYP inhibition: CYP3A |
| D04641 |
Istradefylline (JAN/USAN/INN); Nourianz (TN); Nouriast (TN) |
(P) unclassified |
| D04768 |
Lonafarnib (JAN/USAN/INN); Zokinvy (TN) |
(CI,P) Enzyme: CYP3A / CYP inhibition: CYP3A / Transporter inhibition: ABCB1 |
| D04820 |
Lurasidone hydrochloride (JAN/USAN); SM 13496; Latuda (TN) |
(P) unclassified |
| D05000 |
Methylprednisolone hemisuccinate (USP); Methylprednisolone succinate (JP19) |
(P) unclassified |
| D05001 |
Methylprednisolone sodium phosphate (USAN) |
(P) unclassified |
| D05002 |
Methylprednisolone suleptanate (USAN/INN) |
(P) unclassified |
| D05028 |
Midazolam maleate (USAN) |
(P) unclassified |
| D05333 |
Paclitaxel poliglumex (USAN/INN) |
(P) unclassified |
| D05429 |
Aminophylline hydrate (JP19) |
(P) unclassified |
| D05601 |
Prednicarbate (USP/INN); Dermatop (TN) |
(P) unclassified |
| D05719 |
Resocortol butyrate (USAN) |
(P) unclassified |
| D05729 |
Rimexolone (USP/INN); Vexol (TN) |
(P) unclassified |
| D05775 |
Rufinamide (JAN/USP/INN); Banzel (TN) |
(P) unclassified |
| D05928 |
Stiripentol (JAN/USAN/INN); Diacomit (TN) |
(P) unclassified |
| D06068 |
Temsirolimus (JAN/USAN/INN); Torisel (TN) |
(P) unclassified |
| D06103 |
Theophylline (USP); Theophylline monohydrate; Accurbron (TN) |
(P) unclassified |
| D06104 |
Theophylline sodium glycinate (USP); Asbron (TN) |
(P) unclassified |
| D06171 |
Tixocortol pivalate (USAN) |
(P) unclassified |
| D06199 |
Trabectedin (JAN/USAN/INN); Yondelis (TN) |
(P) unclassified |
| D06216 |
Triamcinolone acetonide sodium phosphate (USAN) |
(P) unclassified |
| D06273 |
Imidafenacin (JAN/INN); Uritos (TN); Staybla (TN) |
(P) unclassified |
| D06304 |
Vindesine (USAN/INN) |
(P) Enzyme: CYP3A / CYP inhibition: CYP3A |
| D06305 |
Vinepidine sulfate (USAN) |
(P) unclassified |
| D06306 |
Vinglycinate sulfate (USAN) |
(P) unclassified |
| D06307 |
Vinleurosine sulfate (USAN) |
(P) unclassified |
| D06308 |
Vinrosidine sulfate (USAN) |
(P) unclassified |
| D06309 |
Vinzolidine sulfate (USAN) |
(P) unclassified |
| D06315 |
Fluticasone furoate (JAN/USAN/INN); Veramyst (TN) |
(P) unclassified |
| D06412 |
Aliskiren fumarate (JAN/USAN); Aliskiren hemifumarate; Tekturna (TN) |
(P) Transporter inhibition: ABCB1 |
| D06414 |
Dasatinib (USAN); Dasatinib hydrate (JAN); Sprycel (TN) |
(P) unclassified |
| D06466 |
Freeze-dried BCG for intravesical use; Immunobladder (TN); Tice BCG (TN) |
(P) unclassified |
| D06597 |
Fosaprepitant dimeglumine (USAN); Fosaprepitant meglumine (JAN); Proemend (TN) |
(P) unclassified |
| D06637 |
Romidepsin (JAN/USAN/INN); Istodax (TN) |
(P) Enzyme: CYP3A / CYP inhibition: CYP3A |
| D06673 |
Meprednisone (USP/INN) |
(P) unclassified |
| D06876 |
Hydrocortisone aceponate (INN); Efficort (TN) |
(P) Enzyme: CYP3A / CYP inhibition: CYP3A |
| D07073 |
Dexamethasone cipecilate (JAN/INN) |
(P) unclassified |
| D07082 |
Dabigatran etexilate mesylate (USAN); Dabigatran etexilate methanesulfonate (JAN); Dabigatran etexilate mesilate; Pradaxa (TN) |
(CI,P) Transporter inhibition: ABCB1 |
| D07086 |
Rivaroxaban (JAN/USAN/INN); Xarelto (TN) |
(P) Transporter inhibition: ABCB1 |
| D07116 |
Alclometasone (INN) |
(P) unclassified |
| D07201 |
Fluprednidene (INN) |
(P) unclassified |
| D07202 |
Halometasone (INN) |
(P) unclassified |
| D07203 |
Methylprednisolone aceponate (INN); Advantan (TN) |
(P) unclassified |
| D07230 |
Prednylidene (INN) |
(P) unclassified |
| D07464 |
Paramethasone (INN); Dillar (TN) |
(P) unclassified |
| D07495 |
Beclometasone (INN) |
(P) unclassified |
| D07538 |
Bosentan (INN) |
(P) unclassified |
| D07569 |
Candesartan cilexetil and anmlodipine besylate (JP19); Unisia (TN) |
(P) unclassified |
| D07583 |
Phenytoin and phenobarbital; Aleviatin with phenobarbital (TN) |
(P) CYP induction: CYP3A |
| D07585 |
Isopropylantipyrine, ergotamine tartrate and anhydrous caffeine; Cleamine A (TN) |
(CI) unclassified |
| D07595 |
Fosphenytoin sodium hydrate (JAN); Fostoin (TN) |
(P) unclassified |
| D07715 |
Clobetasol (INN); Clobecort Amex (TN) |
(P) unclassified |
| D07717 |
Clobetasone (INN) |
(P) unclassified |
| D07719 |
Clocortolone (INN) |
(P) unclassified |
| D07749 |
Cortisone (INN) |
(P) unclassified |
| D07796 |
Dexamethasone 21-acetate; Dexamethasone acetate anhydrous; Decaject-L.A. (TN) |
(P) unclassified |
| D07797 |
Dexamethasone isonicotinate; Dexamethasone 21-isonicotinate; Voren [veterinary] (TN) |
(P) unclassified |
| D07798 |
Dexamethasone sodium hemisulfate; Dexamethasone 21-sodium sulfate |
(P) unclassified |
| D07799 |
Dexamethasone 21-tebutate; Dexamethasone tertiary butyl acetate; Dexamedium [veterinary] (TN) |
(P) unclassified |
| D07800 |
Dexamethasone 21-valerate; Voalla (TN); Zalucs (TN) |
(P) unclassified |
| D07801 |
Dexamethasone phenylpropionate; Dexafort [veterinary] (TN) |
(P) unclassified |
| D07802 |
Dexamethasone phosphate; Decadron-phosphate (TN) |
(P) unclassified |
| D07827 |
Diflorasone (INN); Murode (TN) |
(P) unclassified |
| D07866 |
Docetaxel (JAN/INN); Taxotere (TN) |
(P) unclassified |
| D07868 |
Domperidone maleate |
(P) unclassified |
| D07869 |
Donepezil (JAN/INN); Donaz (TN); Allydone (TN) |
(P) unclassified |
| D07967 |
Fludrocortisone (INN); Astonin-H (TN) |
(P) unclassified |
| D07972 |
Fluocortin (INN) |
(P) unclassified |
| D07973 |
Fluocortolone 21-pivalate; Fluocortolone pivalate; Ultradil (TN) |
(P) unclassified |
| D07980 |
Fluprednidene acetate; Fluprednidene 21-acetate; Decoderm (TN) |
(P) unclassified |
| D07981 |
Fluticasone (INN); Fluticaps (TN) |
(P) unclassified |
| D07993 |
Fosphenytoin (INN) |
(P) unclassified |
| D08095 |
Ivabradine hydrochloride (JAN/USAN); Ivabrandine hydrochloride; Corlanor (TN); Corlentor (TN); Coralan (TN) |
(P) unclassified |
| D08147 |
Loteprednol (INN) |
(P) unclassified |
| D08195 |
Methadone (BAN) |
(P) Transporter inhibition: ABCB1 |
| D08227 |
Mometasone (INN) |
(P) unclassified |
| D08356 |
Phenobarbital diethylamine; Gratusminal (TN) |
(P) CYP induction: CYP3A |
| D08412 |
Prednisolone pivalate; Prednisolone 21-pivalate; Ultracortenol (TN) |
(P) unclassified |
| D08413 |
Prednisolone sodium metazoate (USAN); Prednisolone metasulfobenzoate sodium; Prednisolone 21-(sodium 3-sulfobenzoate); Predenema (TN) |
(P) unclassified |
| D08414 |
Prednisolone 21-(sodium tetrahydrophthalate); Prednisolone sodium tetrahydrophthalate; Fenicort (TN) |
(P) unclassified |
| D08415 |
Prednisolone steaglate (BAN); Prednisolone 21-steaglate; Sintisone (TN) |
(P) unclassified |
| D08416 |
Prednisone acetate; Prednisone 21-acetate |
(P) unclassified |
| D08476 |
Resocortol (INN) |
(P) unclassified |
| D08479 |
Rifampicin sodium; Rifadine (TN) |
(P) unclassified |
| D08488 |
Amlodipine besilate and atorvastatin calcium; Caduet (TN) |
(P) unclassified |
| D08497 |
Rupatadine fumarate (JAN/USAN); Rinialer (TN); Rupafin (TN) |
(P) unclassified |
| D08610 |
Tixocortol (INN) |
(P) unclassified |
| D08660 |
Ulobetasol (INN); Halobetasol |
(P) unclassified |
| D08675 |
Vinblastine (INN) |
(P) unclassified |
| D08679 |
Vincristine (INN); Tecnocris (TN) |
(P) Enzyme: CYP3A / CYP inhibition: CYP3A |
| D08680 |
Vinorelbine (INN); Navelbine (TN) |
(P) unclassified |
| D08856 |
Anamorelin hydrochloride (JAN/USAN); Adlumiz (TN) |
(P) unclassified |
| D08964 |
Perampanel (JAN/USAN); Fycompa (TN) |
(P) Enzyme: CYP3A / CYP inhibition: CYP3A |
| D09017 |
Ticagrelor (JAN/USAN/INN); Brilinta (TN) |
(CI,P) Enzyme: CYP3A / CYP inhibition: CYP3A / Transporter inhibition: ABCB1 |
| D09032 |
Vinflunine ditartrate (USAN); Javlor (TN) |
(P) unclassified |
| D09187 |
Estradiol and levonorgestrel; Wellnara (TN); Climara pro (TN) |
(P) unclassified |
| D09215 |
Eslicarbazepine (USAN/INN) |
(P) unclassified |
| D09319 |
Indacaterol maleate (JAN/USAN); Arcapta (TN) |
(P) Transporter inhibition: ABCB1 |
| D09348 |
Fostamatinib disodium (USAN); Fostamatinib sodium hydrate (JAN); Fostamatinib disodium hexahydrate; Tavalisse (TN) |
(P) CYP inhibition: CYP3A |
| D09365 |
Palovarotene (JAN/USAN/INN); Sohonos (TN) |
(CI,P) unclassified |
| D09546 |
Edoxaban tosilate hydrate (JAN); Edoxaban tosylate monohydrate; Lixiana (TN); Savaysa (TN) |
(P) Transporter inhibition: ABCB1 |
| D09570 |
Bilastine (JAN/INN); Bilanoa (TN) |
(P) unclassified |
| D09572 |
Riociguat (JAN/USAN/INN); Adempas (TN) |
(P) Enzyme: CYP3A / CYP inhibition: CYP3A / Transporter inhibition: ABCB1 |
| D09594 |
Olmesartan medoxomil and azelnidipine; Rezaltas (TN) |
(P) unclassified |
| D09612 |
Eslicarbazepine acetate (USAN); Zebinix (TN); Aptiom (TN) |
(P) unclassified |
| D09638 |
Lomitapide mesylate (USAN); Lomitapide mesilate (JAN); Juxtapid (TN); Lojuxta (TN) |
(CI,P) unclassified |
| D09720 |
Rilpivirine (JAN/USAN/INN); Rekambys (TN) |
(P) Enzyme: CYP3A / CYP inhibition: CYP3A |
| D09728 |
Bosutinib hydrate (JAN); Bosutinib monohydrate; Bosulif (TN) |
(P) unclassified |
| D09730 |
Olaparib (JAN/USAN/INN); Lynparza (TN) |
(P) Enzyme: CYP3A / CYP inhibition: CYP3A |
| D09731 |
Crizotinib (JAN/USAN/INN); Xalkori (TN) |
(P) CYP inhibition: CYP3A |
| D09733 |
Afatinib dimaleate (USAN); Afatinib maleate (JAN); Gilotrif (TN); Giotrif (TN) |
(P) Transporter inhibition: ABCB1 |
| D09743 |
Telmisartan and amlodipine besilate (JP19); Telmisartan and amlodipine besylate; Micamlo (TN); Twynsta (TN) |
(P) unclassified |
| D09745 |
Valsartan and amlodipine besilate; Exforge (TN) |
(P) unclassified |
| D09783 |
Tofacitinib citrate (JAN/USAN); Tasocitinib citrate; Xeljanz (TN) |
(P) unclassified |
| D09785 |
Delamanid (JAN/USAN); Deltyba (TN) |
(P) unclassified |
| D09796 |
Hydrocortisone caproate (JAN) |
(P) Enzyme: CYP3A / CYP inhibition: CYP3A |
| D09894 |
Eliglustat tartrate (JAN/USAN); Eliglustat hemitartrate; Cerdelga (TN) |
(CI,P) Transporter inhibition: ABCB1 |
| D09920 |
Lenvatinib mesylate (USAN); Lenvatinib mesilate (JAN); Lenvima (TN) |
(P) Enzyme: CYP3A / CYP inhibition: CYP3A / Transporter inhibition: ABCB1 |
| D09951 |
Ponatinib hydrochloride (JAN/USAN); Iclusig (TN) |
(P) Enzyme: CYP3A / CYP inhibition: CYP3A |
| D09956 |
Quizartinib dihydrochloride (USAN); Quizartinib hydrochloride (JAN); Vanflyta (TN) |
(P) Enzyme: CYP3A / CYP inhibition: CYP3A |
| D09958 |
Rilpivirine hydrochloride (JAN/USAN); Edurant (TN) |
(P) Enzyme: CYP3A / CYP inhibition: CYP3A |
| D09960 |
Ruxolitinib phosphate (JAN/USAN); Jakafi (TN); Jakavi (TN); Opzelura (TN) |
(P) unclassified |
| D09996 |
Vemurafenib (JAN/USAN/INN); Zelboraf (TN) |
(P) unclassified |
| D10003 |
Hemin (JAN); Normosang (TN); Panhematin (TN) |
(P) unclassified |
| D10024 |
Selumetinib sulfate (JAN/USAN); Koselugo (TN) |
(P) unclassified |
| D10064 |
Dabrafenib (USAN) |
(P) unclassified |
| D10082 |
Suvorexant (JAN/USAN); MK-4305; Belsomra (TN) |
(P) Enzyme: CYP3A / CYP inhibition: CYP3A |
| D10093 |
Asunaprevir (JAN/USAN); Sunvepra (TN) |
(P) Enzyme: CYP3A / CYP inhibition: CYP3A / Transporter inhibition: ABCB1 |
| D10095 |
Cabozantinib s-malate (USAN); Cabozantinib malate (JAN); Cometriq (TN); Cabometyx (TN) |
(P) unclassified |
| D10104 |
Dabrafenib mesylate (USAN); Dabrafenib mesilate (JAN); Tafinlar (TN) |
(P) unclassified |
| D10127 |
Glycerol phenylbutyrate (JAN/USAN); Ravicti (TN) |
(P) CYP induction: CYP3A |
| D10223 |
Ibrutinib (JAN/USAN); Imbruvica (TN) |
(P) Enzyme: CYP3A / CYP inhibition: CYP3A |
| D10226 |
Sacubitril valsartan sodium hydrate (JAN); Sacubitril mixture with valsartan; Entresto (TN) |
(P) unclassified |
| D10243 |
Irbesartan and amlodipine besilate (JP19); Aimix (TN) |
(P) unclassified |
| D10252 |
Fexofenadine hydrochloride and pseudoephedrine hydrochloride; Allegra-d (TN) |
(P) unclassified |
| D10309 |
Brexpiprazole (JAN/USAN/INN); Rexulti (TN) |
(P) unclassified |
| D10372 |
Palbociclib (JAN/USAN); Ibrance (TN) |
(P) unclassified |
| D10385 |
Ezetimibe and atorvastatin; Atozet (TN); Liptruzet (TN) |
(P) unclassified |
| D10396 |
Nintedanib esylate (USAN); Nintedanib ethanesulfonate (JAN); Ofev (TN) |
(P) Transporter inhibition: ABCB1 |
| D10434 |
Vintafolide (USAN/INN) |
(P) unclassified |
| D10450 |
Alectinib hydrochloride (JAN); Alecensa (TN) |
(P) unclassified |
| D10452 |
Cabazitaxel acetonate (JAN); Cabazitaxel acetone; Jevtana (TN) |
(P) Enzyme: CYP3A / CYP inhibition: CYP3A |
| D10478 |
Naldemedine tosylate (JAN/USAN); Naldemedine tosilate; Symproic (TN) |
(P) unclassified |
| D10501 |
Fluticasone furoate and vilanterol trifenatate; Breo ellipta (TN); Relvar ellipita (TN) |
(P) unclassified |
| D10505 |
Glycopyrronium bromide and indacaterol maleate; Ultibro (TN) |
(P) Transporter inhibition: ABCB1 |
| D10524 |
Azilsartan and amlodipine besilate; Zacras (TN) |
(P) unclassified |
| D10528 |
Aldosterone (INN) |
(P) unclassified |
| D10531 |
Clindamycin phosphate hydrate (JAN) |
(CI,P) unclassified |
| D10533 |
Umeclidinium bromide and vilanterol; Anoro (TN) |
(P) unclassified |
| D10551 |
Ceritinib (JAN/USAN/INN); Zykadia (TN) |
(P) Enzyme: CYP3A / CYP inhibition: CYP3A |
| D10564 |
Amenamevir (JAN/INN); Amenalief (TN) |
(P) Enzyme: CYP3A / CYP inhibition: CYP3A / CYP induction: CYP3A |
| D10568 |
Pitavastatin calcium hydrate (JP19); Pitabastatin calcium pentahydrate; Livalo (TN) |
(P) unclassified |
| D10602 |
Clindamycin phosphate and benzoyl peroxide; Duac (TN); Onexton (TN) |
(P) unclassified |
| D10633 |
Finerenone (JAN/USAN/INN); Kerendia (TN) |
(P) unclassified |
| D10643 |
Isavuconazonium sulfate (JAN/USAN); Cresemba (TN) |
(P) Enzyme: CYP3A / CYP inhibition: CYP3A |
| D10663 |
Rimegepant sulfate (USAN); Rimegepant sulfate hydrate (JAN); Nurtec odt (TN); Vydura (TN) |
(P) unclassified |
| D10679 |
Venetoclax (JAN/USAN/INN); Venclexta (TN) |
(CI,P) unclassified |
| D10688 |
Abemaciclib (JAN/USAN/INN); Verzenio (TN) |
(P) Enzyme: CYP3A / CYP inhibition: CYP3A |
| D10733 |
Talazoparib tosylate (USAN); Talazoparib tosilate (JAN); Talzenna (TN) |
(P) unclassified |
| D10761 |
Polatuzumab vedotin (USAN); Polatuzumab vedotin (genetical recombination) (JAN); Polatuzumab vedotin-piiq; Polivy (TN) |
(P) Enzyme: CYP3A / CYP inhibition: CYP3A |
| D10762 |
Fosravuconazole L-lysine ethanolate (JAN) |
(P) CYP inhibition: CYP3A |
| D10780 |
Perampanel hydrate (JAN); Fycompa (TN) |
(P) Enzyme: CYP3A / CYP inhibition: CYP3A |
| D10800 |
Gilteritinib fumarate (JAN/USAN); Xospata (TN) |
(P) Transporter inhibition: ABCB1 |
| D10801 |
Letermovir (JAN/USAN/INN); Prevymis (TN) |
(P) CYP inhibition: CYP3A |
| D10805 |
Telmisartan, amlodipine and hydrochlorothiazide; Micatrio (TN) |
(P) unclassified |
| D10832 |
Darunavir and cobicistat; Prezcobix (TN); Rezolsta (TN) |
(P) Enzyme: CYP3A / CYP inhibition: CYP3A |
| D10836 |
Emtricitabine, rilpivirine and tenofovir alafenamide; Odefsey (TN) |
(P) Enzyme: CYP3A / CYP inhibition: CYP3A / Transporter inhibition: ABCB1 |
| D10866 |
Brigatinib (JAN/USAN); Alunbrig (TN) |
(P) unclassified |
| D10882 |
Daclatasvir, asunaprevir and beclabuvir; Ximency (TN) |
(P) Enzyme: CYP3A / CYP inhibition: CYP3A / Transporter inhibition: ABCB1 |
| D10888 |
Relugolix (JAN/USAN/INN); Orgovyx (TN) |
(P) Transporter inhibition: ABCB1 |
| D10891 |
Capmatinib hydrochloride (USAN); Capmatinib hydrochloride hydrate (JAN); Tabrecta (TN) |
(P) unclassified |
| D10892 |
Esaxerenone (JAN/INN) |
(P) Enzyme: CYP3A / CYP inhibition: CYP3A |
| D10893 |
Acalabrutinib (JAN/USAN/INN); Calquence (TN) |
(P) Enzyme: CYP3A / CYP inhibition: CYP3A |
| D10895 |
Fosaprepitant (INN) |
(P) unclassified |
| D10926 |
Entrectinib (JAN/USAN/INN); Rozlytrek (TN) |
(P) CYP inhibition: CYP3A |
| D10927 |
Erdafitinib (JAN/USAN/INN); Balversa (TN) |
(P) Transporter inhibition: ABCB1 |
| D10931 |
Etrasimod arginine (USAN); Etrasimod L-arginine (JAN); Velsipity (TN) |
(P) unclassified |
| D10990 |
Somatrogon (USAN/INN); Somatrogon (genetical recombination) (JAN); Somatrogon-ghla; Ngenla (TN) |
(P) unclassified |
| D10993 |
Tucidinostat (JAN/USAN/INN); Hiyasta (TN) |
(P) unclassified |
| D10999 |
Valbenazine tosylate (USAN); Valbenazine tosilate (JAN); Valbenazine ditosylate; Ingrezza (TN); Dysval (TN) |
(P) unclassified |
| D11000 |
Vamorolone (USAN/INN); Agamree (TN) |
(P) unclassified |
| D11012 |
Lorlatinib (JAN/USAN/INN); Lorbrena (TN) |
(P) Enzyme: CYP3A / CYP inhibition: CYP3A / CYP induction: CYP3A |
| D11022 |
Lemborexant (JAN/USAN/INN); Dayvigo (TN) |
(P) unclassified |
| D11035 |
Fluticasone furoate, umeclidinium bromide and vilanterol; Trelegy ellipta (TN) |
(P) unclassified |
| D11040 |
Apalutamide (JAN/INN); Erleada (TN) |
(P) unclassified |
| D11048 |
Upadacitinib hydrate (JAN); Upadacitinib hemihydrate; Rinvoq (TN) |
(P) unclassified |
| D11053 |
Encorafenib (JAN/USAN/INN); Braftovi (TN) |
(P) unclassified |
| D11070 |
Tirabrutinib hydrochloride (JAN/USAN); Velexbru (TN) |
(P) unclassified |
| D11090 |
Ivosidenib (JAN/USAN/INN); Tibsovo (TN) |
(P) unclassified |
| D11138 |
Larotrectinib sulfate (JAN/USAN); Vitrakvi (TN) |
(P) Enzyme: CYP3A / CYP inhibition: CYP3A |
| D11159 |
Leniolisib phosphate (JAN/USAN); Joenja (TN) |
(P) unclassified |
| D11194 |
Somapacitan (USAN/INN); Somapacitan (genetical recombination) (JAN); Somapacitan-beco; Sogroya (TN) |
(P) unclassified |
| D11208 |
Elafibranor (USAN); Iqirvo (TN) |
(P) unclassified |
| D11282 |
Dolutegravir sodium and rilpivirine hydrochloride; Juluca (TN) |
(P) Enzyme: CYP3A / CYP inhibition: CYP3A |
| D11296 |
Fedratinib hydrochloride (USAN); Fedratinib hydrochloride hydrate (JAN); Fedratinib dihydrochloride monohydrate; Inrebic (TN) |
(P) unclassified |
| D11370 |
Fosnetupitant chloride hydrochloride (JAN/USAN); Arokaris (TN) |
(P) unclassified |
| D11371 |
Capivasertib (JAN/USAN); Truqap (TN) |
(P) Enzyme: CYP3A / CYP inhibition: CYP3A |
| D11382 |
Darunavir, cobicistat, emtricitabine and tenofovir alafenamide; Symtuza (TN) |
(P) Enzyme: CYP3A / CYP inhibition: CYP3A / Transporter inhibition: ABCB1 |
| D11417 |
Pemigatinib (JAN/USAN/INN); Pemazyre (TN) |
(P) unclassified |
| D11422 |
Zanubrutinib (JAN/USAN/INN); Brukinsa (TN) |
(P) Enzyme: CYP3A / CYP inhibition: CYP3A |
| D11454 |
Repotrectinib (JAN/USAN); Augtyro (TN) |
(P) unclassified |
| D11485 |
Tazemetostat hydrobromide (JAN/USAN); Tazverik (TN) |
(P) Transporter inhibition: ABCB1 |
| D11520 |
Ezetimibe and rosuvastatin; Roszet (TN); Rosuzet (TN) |
(P) unclassified |
| D11525 |
Enfortumab vedotin (USAN); Enfortumab vedotin (genetical recombination) (JAN); Enfortumab vedotin-ejfv; Padcev (TN) |
(P) unclassified |
| D11572 |
Beclomethasone dipropionate monohydrate; Beconase aq (TN) |
(P) unclassified |
| D11659 |
Tolvaptan sodium phosphate (JAN); Samtasu (TN) |
(P) unclassified |
| D11662 |
Valemetostat tosilate (JAN); Valemetostat tosylate; Ezharmia (TN) |
(P) unclassified |
| D11713 |
Selpercatinib (JAN/USAN/INN); Retevmo (TN) |
(P) unclassified |
| D11725 |
Futibatinib (JAN/USAN/INN); Lytgobi (TN) |
(P) unclassified |
| D11793 |
Zuranolone (JAN/USAN/INN); Zurzuvae (TN) |
(P) unclassified |
| D11814 |
Tisotumab vedotin (USAN/INN); Tisotumab vedotin (genetical recombination) (JAN); Tisotumab vedotin-tftv; Tivdak (TN) |
(P) unclassified |
| D11816 |
Belumosudil mesylate (USAN); Belumosudil mesilate (JAN); Rezurock (TN) |
(P) CYP inhibition: CYP3A |
| D11835 |
Vorasidenib citrate (USAN); Vorasidenib citric acid hydrate (JAN); Voranigo (TN) |
(P) Enzyme: CYP3A / CYP inhibition: CYP3A |
| D11861 |
Indacaterol acetate, glycopyrronium bromide and mometasone furoate; Enerzair (TN) |
(P) unclassified |
| D11862 |
Indacaterol and mometasone furoate; Atectura (TN) |
(P) unclassified |
| D11887 |
Daridorexant hydrochloride (JAN/USAN); Quviviq (TN) |
(P) Enzyme: CYP3A / CYP inhibition: CYP3A |
| D11920 |
Pimitespib (JAN); Jeselhy (TN) |
(P) CYP inhibition: CYP3A |
| D11954 |
Belzutifan (JAN/USAN/INN); Welireg (TN) |
(P) CYP induction: CYP3A |
| D11970 |
Ritlecitinib tosylate (USAN); Ritlecitinib tosilate (JAN); Litfulo (TN) |
(P) CYP inhibition: CYP3A |
| D12015 |
St. John's wort; SJW |
(P) unclassified |
| D12050 |
Pirtobrutinib (JAN/USAN); Jaypirca (TN) |
(P) CYP inhibition: CYP3A |
| D12055 |
Sotorasib (JAN/USAN); Lumakras (TN) |
(P) Enzyme: CYP3A / CYP inhibition: CYP3A |
| D12217 |
Imlunestrant tosylate (USAN); Imlunestrant tosilate (JAN); Inluriyo (TN) |
(P) unclassified |
| D12245 |
Lazertinib mesylate (USAN); Lazertinib mesilate hydrate (JAN); Lazcluze (TN) |
(P) unclassified |
| D12251 |
Iptacopan (USAN/INN) |
(P) unclassified |
| D12252 |
Iptacopan hydrochloride (USAN); Iptacopan hydrochloride hydrate (JAN); Iptacopan hydrochloride monohydrate; Fabhalta (TN) |
(P) unclassified |
| D12265 |
Mavacamten (JAN/USAN/INN); Camzyos (TN) |
(P) unclassified |
| D12269 |
Nirmatrelvir and ritonavir; Paxlovid (TN) |
(P) CYP inhibition: CYP3A |
| D12364 |
Taletrectinib adipate (JAN/USAN); Ibtrozi (TN) |
(P) Enzyme: CYP3A / CYP inhibition: CYP3A |
| D12396 |
Sebetralstat (JAN/USAN/INN); Ekterly (TN) |
(P) unclassified |
| D12438 |
Pitavastatin calcium and ezetimibe; Livazebe (TN) |
(P) unclassified |
| D12442 |
Tucatinib ethanolate (JAN); Tucatinib hemiethanolate; Tukysa (TN) |
(P) unclassified |
| D12586 |
Mifepristone and misoprostol; Mefeego (TN) |
(P) Enzyme: CYP3A / CYP inhibition: CYP3A |
| D12611 |
Vornorexant hydrate (JAN) |
(P) unclassified |
| D12704 |
Acalabrutinib maleate hydrate (JAN); Acalabrutinib maleate monohydrate; Calquence (TN) |
(P) Enzyme: CYP3A / CYP inhibition: CYP3A |
| D12837 |
Risovalisib mesilate hydrate (JAN); Risovalisib mesylate dihydrate; Haizexin (TN) |
(P) CYP induction: CYP3A |
| D12963 |
Macitentan and tadalafil; Opsynvi (TN); Yuvanci (TN) |
(P) Enzyme: CYP3A / CYP inhibition: CYP3A |
| D13026 |
Atogepant hydrate (JAN); Aquipta (TN) |
(P) unclassified |