| C00989 |
4-Hydroxybutanoic acid; 4-Hydroxybutanoate; 4-Hydroxybutyric acid |
(P) unclassified |
| C07051 |
Indinavir |
(P) unclassified |
| C07521 |
Thiopental |
(P) unclassified |
| C07546 |
Succinylcholine; Suxamethonium |
(P) unclassified |
| C07547 |
Tubocurarine |
(P) unclassified |
| C07548 |
Atracurium |
(P) unclassified |
| C07551 |
Pancuronium |
(P) unclassified |
| C07553 |
Vecuronium |
(P) unclassified |
| C17723 |
Metabutethamine |
(P) unclassified |
| D00033 |
Phenol (JP18/USP); Liquefied phenol (JP18); Phenol for disinfection (JP18); Phenol, liquefied; Paoscle (TN); Phenol (TN); Liquefied phenol (TN); Phenol for disinfection (TN) |
(P) unclassified |
| D00102 |
Nitrous oxide (JP18/USP); Nitrous oxide (TN) |
(P) unclassified |
| D00107 |
Tacrolimus (USP/INN); Tacrolimus hydrate (JP18); Prograf (TN); Protopic (TN) |
(P) Enzyme: CYP3A4 |
| D00110 |
Cocaine (USP); Cocaine (TN) |
(P) unclassified |
| D00184 |
Cyclosporine (USP); Ciclosporin (JP18); Gengraf (TN); Neoral (TN); Restasis (TN); Sandimmune (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D00197 |
Reserpine (JP18/USP/INN); Apoplon (TN); Serpalan (TN) |
(P) unclassified |
| D00198 |
Rescinnamine (JAN/INN); Tsuruselpi S (TN) |
(P) unclassified |
| D00199 |
Ajmaline (JP18); Ajimalin (TN) |
(P) unclassified |
| D00203 |
Amphotericin B (JP18/USP/INN); Ambisome (TN); Amphotec (TN); Fungizone (TN) |
(P) unclassified |
| D00211 |
Rifampin (USP); Rifampicin (JP18/INN); Rifadin (TN); Rimactane (TN) |
(P) CYP induction: CYP3A4 |
| D00235 |
Atenolol (JP18/USP/INN); Tenormin (TN) |
(P) unclassified |
| D00241 |
Baclofen (JP18/USP/INN); Kemstro (TN); Lioresal (TN) |
(P) unclassified |
| D00250 |
Capsaicin (JAN/USP); Zostrix (TN) |
(P) unclassified |
| D00252 |
Carbamazepine (JP18/USP/INN); Equetro (TN); Tegretol (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
| D00255 |
Carvedilol (JP18/USP/INN); Artist (TN); Coreg (TN) |
(P) Enzyme: CYP3A4 |
| D00268 |
Chlormezanone (JAN/INN); Trancopal (TN) |
(P) unclassified |
| D00276 |
Clarithromycin (JP18/USP/INN); Biaxin (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D00281 |
Clonidine (JAN/USP/INN); Catarpres-TTS (TN) |
(P) unclassified |
| D00292 |
Dexamethasone (JP18/USP/INN); Decadron (TN); Maxidex (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
| D00293 |
Diazepam (JP18/USP/INN); Diastat (TN); Valium (TN) |
(P) Enzyme: CYP3A4 |
| D00294 |
Diazoxide (JAN/USP/INN); Hyperstat (TN); Proglycem (TN) |
(P) unclassified |
| D00295 |
Cimetidine (JP18/USP/INN); Tagamet (TN) |
(P) CYP inhibition: CYP3A4 |
| D00297 |
Digitoxin (JAN/USP/INN); Crystodigin (TN) |
(P) unclassified |
| D00298 |
Digoxin (JP18/USP); Lanoxicaps (TN); Lanoxin (TN) |
(P) unclassified |
| D00303 |
Disopyramide (JP18/USAN/INN); Rythmodan P (TN) |
(P) Enzyme: CYP3A4 |
| D00319 |
Felodipine (JP18/USP/INN); Plendil (TN) |
(P) Enzyme: CYP3A4 / Target: CACNA1C CACNA1D CACNA1F CACNA1S |
| D00320 |
Fentanyl (JAN/USP/INN); Duragesic (TN); Subsys (TN) |
(P) Enzyme: CYP3A4 |
| D00322 |
Fluconazole (JP18/USP/INN); Diflucan (TN) |
(P) CYP inhibition: CYP3A4 |
| D00349 |
Isradipine (USP/INN); Dynacirc (TN) |
(P) Target: CACNA1C CACNA1D CACNA1F CACNA1S |
| D00358 |
Lidocaine (JP18/USP/INN); Dentipatch (TN); Xylocaine (TN) |
(P) Enzyme: CYP3A4 |
| D00371 |
Theophylline (JP18); Elixophyllin (TN); Quibron-t (TN); Theo-24 (TN); Theodur G (TN); Theolair (TN); Uniphyl (TN) |
(P) unclassified |
| D00378 |
Timolol (USAN); Timolol hemihydrate; Betimol (TN) |
(P) unclassified |
| D00387 |
Triazolam (JP18/USP/INN); Halcion (TN) |
(P) Enzyme: CYP3A4 |
| D00402 |
Methocarbamol (JAN/USP/INN); Delaxin (TN); Robaxin (TN) |
(P) unclassified |
| D00405 |
Methyldopa (USP); Methyldopa hydrate (JP18); Aldomet (TN) |
(P) unclassified |
| D00418 |
Minoxidil (JAN/USP/INN); Loniten (TN); Riup (TN); Rogaine (TN) |
(P) unclassified |
| D00420 |
Mitotane (JAN/USP/INN); Lysodren (TN) |
(P) unclassified |
| D00427 |
Ritonavir (JAN/USP/INN); Norvir (TN) |
(P) unclassified |
| D00429 |
Saquinavir (JAN/USP/INN); Fortovase (TN) |
(P) Enzyme: CYP3A4 |
| D00432 |
Nadolol (JP18/USP/INN); Corgard (TN) |
(P) unclassified |
| D00434 |
Simvastatin (JP18/USP/INN); MK-733; Zocor (TN) |
(P) Enzyme: CYP3A4 |
| D00435 |
Nevirapine (JAN/USP/INN); Viramune (TN) |
(P) Enzyme: CYP3A4 |
| D00437 |
Nifedipine (JP18/USP/INN); Adalat (TN); Afeditab CR (TN); Procardia (TN) |
(P) Enzyme: CYP3A4 / Target: CACNA1C CACNA1D CACNA1F CACNA1S |
| D00438 |
Nimodipine (USP/INN); Nimotop (TN); Nymalize (TN) |
(P) Enzyme: CYP3A4 / Target: CACNA1C CACNA1D CACNA1F CACNA1S |
| D00443 |
Spironolactone (JP18/USP/INN); Aldactone (TN) |
(P) unclassified |
| D00477 |
Procainamide hydrochloride (JP18/USP); Procan SR (TN); Procanbid (TN); Pronestyl (TN) |
(P) unclassified |
| D00480 |
Promethazine hydrochloride (JP18/USP); Phenergan (TN); Promethegan (TN) |
(P) unclassified |
| D00483 |
Propranolol hydrochloride (JP18/USP); Inderal (TN); Innopran XL (TN) |
(P) unclassified |
| D00492 |
Pancuronium bromide (JP18/USP/INN); Pavulon (TN) |
(P) unclassified |
| D00506 |
Phenobarbital (JP18/USP/INN); Luminal (TN) |
(P) unclassified |
| D00512 |
Phenytoin (JP18/USP/INN); Dilantin (TN) |
(P) unclassified |
| D00513 |
Pindolol (JP18/USP/INN); Blocklin-L (TN); Carvisken (TN); Visken (TN) |
(P) unclassified |
| D00515 |
Nitroglycerin (JP18/USP); Glyceryl trinitrate; Minitran (TN); Nitro-bid (TN); Nitro-dur (TN); Nitromist (TN); Transderm-nitro (TN) |
(P) unclassified |
| D00516 |
Isosorbide dinitrate (JP18/USP/INN); Dilatrate-sr (TN); Isordil (TN) |
(P) unclassified |
| D00517 |
Amyl nitrite (JP18/USP); Aspiral (TN); Vaporole (TN) |
(P) unclassified |
| D00542 |
Halothane (JP18/USP/INN); Fluothane (TN) |
(P) Enzyme: CYP3A4 |
| D00543 |
Enflurane (JP18/USP/INN); Ethrane (TN) |
(P) unclassified |
| D00544 |
Methoxyflurane (USP/INN); Penthrane (TN) |
(P) Enzyme: CYP3A4 |
| D00545 |
Isoflurane (JP18/USP/INN); Forane (TN) |
(P) unclassified |
| D00546 |
Desflurane (JAN/USP/INN); Suprane (TN) |
(P) unclassified |
| D00547 |
Sevoflurane (JP18/USAN/INN); Ultane (TN) |
(P) unclassified |
| D00548 |
Etomidate (USP/INN); Amidate (TN) |
(P) unclassified |
| D00549 |
Propofol (JAN/USP/INN); Diprivan (TN) |
(P) unclassified |
| D00550 |
Midazolam (JAN/USP/INN); Dormicum (TN); Buccolam (TN); Nayzilam (TN) |
(P) Enzyme: CYP3A4 |
| D00551 |
Tetracaine (USP/INN); Amethocaine; Amethocaine (TN) |
(P) unclassified |
| D00552 |
Benzocaine (USP/INN); Ethyl aminobenzoate (JP18); Parathesin (TN) |
(P) unclassified |
| D00553 |
Prilocaine (USP/INN); Propitocaine (JAN) |
(P) unclassified |
| D00570 |
Colchicine (JP18/USP); Colchicine (TN) |
(P) Enzyme: CYP3A4 |
| D00597 |
Acebutolol hydrochloride (JP18/USP); Sectral (TN) |
(P) unclassified |
| D00598 |
Betaxolol hydrochloride (JP18/USP); Betoptic (TN); Kerlone (TN) |
(P) unclassified |
| D00599 |
Carteolol hydrochloride (JP18/USP); Cartrol (TN); Ocupress (TN) |
(P) unclassified |
| D00600 |
Labetalol hydrochloride (JP18/USP); Normodyne (TN); Trandate (TN) |
(P) unclassified |
| D00601 |
Metoprolol tartrate (JP18/USP); Lopressor (TN) |
(P) unclassified |
| D00602 |
Penbutolol sulfate (JP18/USP); Levatol (TN) |
(P) unclassified |
| D00603 |
Timolol maleate (JP18/USP); Blocadren (TN); Istalol (TN); Timoptic (TN) |
(P) unclassified |
| D00604 |
Clonidine hydrochloride (JP18/USP); Nexiclon (TN); Kapvay (TN); Duraclon (TN); Catapres (TN) |
(P) unclassified |
| D00606 |
Guanfacine hydrochloride (JAN/USP); Intuniv (TN); Tenex (TN) |
(P) Enzyme: CYP3A4 |
| D00608 |
Doxazosin mesylate (USP); Doxazosin mesilate (JP18); Cardura (TN) |
(P) unclassified |
| D00609 |
Prazosin hydrochloride (JP18/USP); Minipress (TN) |
(P) unclassified |
| D00611 |
Mecamylamine hydrochloride (USP); Inversine (TN) |
(P) unclassified |
| D00612 |
Trimetaphan camsilate (JAN/INN); Trimetaphan camsylate; Arfonad (TN) |
(P) unclassified |
| D00614 |
Sodium nitroprusside (USP); Sodium nitroprusside hydrate (JAN); Nitropress (TN) |
(P) unclassified |
| D00615 |
Amlodipine besylate (USP); Amlodipine besilate (JP18); Norvasc (TN) |
(P) Enzyme: CYP3A4 / Target: CACNA1C CACNA1D CACNA1F CACNA1S |
| D00616 |
Diltiazem hydrochloride (JP18/USP); Cardizem (TN); Cartia XT (TN); Dilacor XR (TN); Dilt-CD (TN) |
(P) Enzyme: CYP3A4 / Target: CACNA1C CACNA1D CACNA1F CACNA1S |
| D00617 |
Nicardipine hydrochloride (JP18/USAN); Cardene (TN) |
(P) Enzyme: CYP3A4 / Target: CACNA1C CACNA1D CACNA1F CACNA1S |
| D00618 |
Nisoldipine (JAN/USAN/INN); Sular (TN) |
(P) Enzyme: CYP3A4 / Target: CACNA1C CACNA1D CACNA1F CACNA1S |
| D00619 |
Verapamil hydrochloride (JP18/USP); Calan (TN); Covera-hs (TN); Vasolan (TN); Verelan (TN) |
(P) Enzyme: CYP3A4 / Target: CACNA1C CACNA1D CACNA1F CACNA1S / CYP inhibition: CYP3A4 |
| D00629 |
Nitrendipine (JP18/USAN/INN); Baypress (TN) |
(P) Enzyme: CYP3A4 / Target: CACNA1C CACNA1D CACNA1F CACNA1S |
| D00630 |
Isosorbide mononitrate (JP18/USP/INN); Imdur (TN); Ismo (TN) |
(P) unclassified |
| D00631 |
Bepridil hydrochloride (USAN); Bepridil hydrochloride hydrate (JAN); Vascor (TN) |
(P) Enzyme: CYP3A4 / Target: CACNA1C CACNA1D CACNA1F CACNA1S |
| D00634 |
Bisoprolol fumarate (JP18/USP); Zebeta (TN) |
(P) unclassified |
| D00635 |
Metoprolol succinate (USP); Toprol XL (TN) |
(P) unclassified |
| D00636 |
Amiodarone hydrochloride (JP18/USP); Ancaron (TN); Cordarone (TN); Nexterone (TN) |
(P) Enzyme: CYP3A4 |
| D00637 |
Disopyramide phosphate (JAN/USP); Norpace (TN) |
(P) Enzyme: CYP3A4 |
| D00638 |
Flecainide acetate (JP18/USP); Tambocor (TN) |
(P) unclassified |
| D00639 |
Mexiletine hydrochloride (JP18/USP); Mexitil (TN) |
(P) unclassified |
| D00640 |
Propafenone hydrochloride (JP18/USP); Rythmol (TN) |
(P) Enzyme: CYP3A4 |
| D00642 |
Quinidine gluconate (USP); Quinaglute (TN) |
(P) unclassified |
| D00643 |
Quinidine polygalacturonate; Cardioquin (TN) |
(P) unclassified |
| D00644 |
Esmolol hydrochloride (JAN/USP); Brevibloc (TN) |
(P) unclassified |
| D00645 |
Bretylium tosylate (USP); Bretylium tosilate (INN); Bretylol (TN) |
(P) unclassified |
| D00647 |
Dofetilide (JAN/USP/INN); Tikosyn (TN) |
(P) unclassified |
| D00648 |
Ibutilide fumarate (USP); Corvert (TN) |
(P) unclassified |
| D00696 |
Midazolam hydrochloride (USAN); Versed (TN) |
(P) Enzyme: CYP3A4 |
| D00701 |
Phenobarbital sodium (JAN/USP/INN); Luminal sodium (TN) |
(P) unclassified |
| D00711 |
Ketamine hydrochloride (JP18/USP); Ketalar (TN) |
(P) unclassified |
| D00712 |
Methohexital sodium (USP); Brevital sodium (TN) |
(P) unclassified |
| D00713 |
Thiamylal sodium (JP18); Surital (TN) |
(P) unclassified |
| D00714 |
Thiopental sodium (JP18/USP/INN); Pentothal (TN) |
(P) unclassified |
| D00732 |
Chloroprocaine hydrochloride (USP); Clorotekal (TN); Iheezo (TN); Nesacaine (TN) |
(P) unclassified |
| D00733 |
Dibucaine (USP); Cinchocaine (INN); Nupercaine (TN) |
(P) unclassified |
| D00735 |
Dyclonine hydrochloride (USP); Dyclone (TN); Dyclopro (TN) |
(P) unclassified |
| D00737 |
Etidocaine hydrochloride; Duranest (TN) |
(P) unclassified |
| D00738 |
Mepivacaine hydrochloride (JP18/USP); Carbocaine (TN); Polocaine (TN); Scandonest plain (TN) |
(P) unclassified |
| D00740 |
Procaine hydrochloride (JP18/USP); Novocain (TN) |
(P) unclassified |
| D00741 |
Tetracaine hydrochloride (JP18/USP); Protocaine hydrochloride (TN) |
(P) unclassified |
| D00753 |
Sirolimus (JAN/USAN/INN); Rapamune (TN); Rapamycin (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D00755 |
Phenyramidol hydrochloride (USAN); Fenyramidol hydrochloride |
(P) unclassified |
| D00758 |
Atracurium besylate (USP); Atracurium besilate (INN); Tracrium (TN) |
(P) unclassified |
| D00759 |
Cisatracurium besylate (USP); Cisatracurium besilate (INN); Nimbex (TN) |
(P) unclassified |
| D00760 |
Doxacurium chloride (USAN/INN); Nuromax (TN) |
(P) unclassified |
| D00762 |
Metyrosine (USP); Metirosine (JAN/INN); Demser (TN) |
(P) unclassified |
| D00763 |
Mivacurium chloride (USAN/INN); Mivacron (TN) |
(P) unclassified |
| D00764 |
Pipecuronium bromide (JAN/USAN/INN); Arduan (TN) |
(P) unclassified |
| D00765 |
Rocuronium bromide (JAN/USP/INN); Zemuron (TN) |
(P) unclassified |
| D00766 |
Succinylcholine chloride (USP); Suxamethonium chloride (INN); Anectine (TN); Quelicin (TN) |
(P) unclassified |
| D00767 |
Vecuronium bromide (JAN/USP/INN); Norcuron (TN) |
(P) unclassified |
| D00768 |
Carisoprodol (JAN/USP/INN); Soma (TN) |
(P) unclassified |
| D00770 |
Chlorphenesin carbamate (JP18/USAN); Maolate (TN) |
(P) unclassified |
| D00771 |
Chlorzoxazone (JAN/USP/INN); Paraflex (TN) |
(P) unclassified |
| D00772 |
Cyclobenzaprine hydrochloride (USP); Flexeril (TN) |
(P) unclassified |
| D00774 |
Orphenadrine citrate (USP); Norflex (TN) |
(P) unclassified |
| D00776 |
Tizanidine hydrochloride (JP18/USP); Zanaflex (TN) |
(P) unclassified |
| D00783 |
Botulinum toxin type A (JAN); Botox (TN); Dysport (TN) |
(P) unclassified |
| D00785 |
Selegiline hydrochloride (JAN/USP); Eldepryl (TN) |
(P) Enzyme: CYP3A4 |
| D00809 |
Amitriptyline hydrochloride (JP18/USP); Elavil (TN) |
(P) Enzyme: CYP3A4 |
| D00811 |
Clomipramine hydrochloride (JP18/USP); Anafranil (TN) |
(P) Enzyme: CYP3A4 |
| D00815 |
Imipramine hydrochloride (JP18/USP); Tofranil (TN) |
(P) Enzyme: CYP3A4 |
| D00818 |
Maprotiline hydrochloride (JP18/USP); Ludiomil (TN) |
(P) unclassified |
| D00831 |
Mefloquine hydrochloride (JP18/USP); Lariam (TN) |
(P) unclassified |
| D00835 |
Alfentanil hydrochloride (USP); Alfenta (TN) |
(P) unclassified |
| D00845 |
Sufentanil citrate (USP); Dsuvia (TN); Sufenta (TN) |
(P) unclassified |
| D00894 |
Amprenavir (JAN/USAN/INN); Agenerase (TN) |
(P) Enzyme: CYP3A4 |
| D00897 |
Indinavir sulfate (USP); Crixivan (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D00899 |
Nelfinavir mesylate (USAN/INN); Nelfinavir mesilate (JAN); Viracept (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D00961 |
Bicalutamide (JP18/USP/INN); Casodex (TN) |
(P) CYP inhibition: CYP3A4 |
| D01025 |
Levobunolol hydrochloride (JAN/USP); Betagan (TN) |
(P) unclassified |
| D01026 |
Sotalol hydrochloride (JAN/USP); Betapace (TN); Sorine (TN) |
(P) unclassified |
| D01041 |
Sparteine (INN) |
(P) unclassified |
| D01061 |
Irinotecan hydrochloride (USP); Irinotecan hydrochloride hydrate (JP18); Irinotecan hydrochloride trihydrate; CPT 11; CPT-11; Campto (TN); Camptosar (TN); Onivyde (TN) |
(P) unclassified |
| D01071 |
Hexobarbital (JAN/INN) |
(P) unclassified |
| D01104 |
Barnidipine hydrochloride (JAN); Hypoca (TN) |
(P) Enzyme: CYP3A4 / Target: CACNA1C CACNA1D CACNA1F CACNA1S |
| D01145 |
Azelnidipine (JP18/INN); Calblock (TN) |
(P) Enzyme: CYP3A4 / Target: CACNA1C CACNA1D CACNA1F CACNA1S |
| D01151 |
Lemildipine (JAN/INN) |
(P) Target: CACNA1C CACNA1D CACNA1F CACNA1S |
| D01152 |
Oxethazaine (JP18/USAN); Oxetacaine (INN); Strocain (TN) |
(P) unclassified |
| D01160 |
Saquinavir mesylate (USP); Saquinavir mesilate (JAN); Invirase (TN) |
(P) Enzyme: CYP3A4 |
| D01162 |
Verteporfin (JAN/USP/INN); Visudyne (TN) |
(P) unclassified |
| D01173 |
Cilnidipine (JP18/INN); Atelec (TN) |
(P) Enzyme: CYP3A4 / Target: CACNA1C CACNA1D CACNA1F CACNA1S |
| D01176 |
Blonanserin (JAN/INN); AD 5423 |
(P) Enzyme: CYP3A4 |
| D01177 |
Remifentanil hydrochloride (JAN/USAN); Ultiva (TN) |
(P) unclassified |
| D01179 |
Duloxetine hydrochloride (JAN/USP); Cymbalta (TN); Yentreve (TN) |
(P) unclassified |
| D01182 |
Alprenolol hydrochloride (JP18/USAN); Regletin (TN) |
(P) unclassified |
| D01215 |
Alcuronium chloride (JAN/USAN/INN); Alloferin (TN) |
(P) unclassified |
| D01227 |
Bosentan (USAN); Bosentan hydrate (JAN); Tracleer (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
| D01240 |
Deslanoside (JP18/USP/INN); Cedilanid-d (TN) |
(P) unclassified |
| D01243 |
Prilocaine hydrochloride (USP); Propitocaine hydrochloride (JAN); Citanest (TN) |
(P) unclassified |
| D01253 |
Clobazam (JAN/USAN/INN); Mystan (TN); Onfi (TN) |
(P) Enzyme: CYP3A4 |
| D01276 |
Atazanavir sulfate (JAN/USAN); Reyataz (TN) |
(P) CYP inhibition: CYP3A4 |
| D01280 |
Warfarin potassium (JP18); Athrombin-K (TN) |
(P) unclassified |
| D01287 |
Levobupivacaine hydrochloride (JAN/USAN); Chirocaine (TN) |
(P) Enzyme: CYP3A4 |
| D01302 |
Hydralazine hydrochloride (JP18/USP); Apresoline (TN) |
(P) unclassified |
| D01326 |
Aprindine hydrochloride (JP18/USAN); Aspenon (TN) |
(P) unclassified |
| D01333 |
Urapidil (JP18/INN); Ebrantil (TN) |
(P) unclassified |
| D01337 |
Epoprostenol sodium (JAN/USAN); Flolan (TN); Veletri (TN) |
(P) unclassified |
| D01369 |
Bevantolol hydrochloride (JAN/USAN); Calvan (TN); Vantol (TN) |
(P) Target: CACNA1C CACNA1D CACNA1F CACNA1S |
| D01399 |
Fentanyl citrate (JP18/USP); Abstral (TN); Fentora (TN); Lazanda (TN); Oralet (TN) |
(P) Enzyme: CYP3A4 |
| D01425 |
Lopinavir (JAN/USP/INN) |
(P) unclassified |
| D01429 |
Fosfluconazole (JAN/INN); Prodif (TN) |
(P) CYP inhibition: CYP3A4 |
| D01450 |
Bupivacaine hydrochloride (USP); Bupivacaine hydrochloride hydrate (JP18); Marcaine (TN) |
(P) Enzyme: CYP3A4 |
| D01454 |
Bupranolol hydrochloride (JP18) |
(P) unclassified |
| D01455 |
Cifenline succinate (USAN); Cibenzoline succinate (JP18); Cibenol (TN); Cipralan (TN) |
(P) Enzyme: CYP3A4 |
| D01469 |
Amosulalol hydrochloride (JP18); Lowgan (TN) |
(P) unclassified |
| D01471 |
Esatenolol (JAN/INN); (S)-Atenolol |
(P) unclassified |
| D01492 |
Bucumolol hydrochloride (JP18) |
(P) unclassified |
| D01504 |
Bufetolol hydrochloride (JP18); Adobiol (TN) |
(P) unclassified |
| D01507 |
Tolperisone hydrochloride (JP18); Muscalm (TN) |
(P) unclassified |
| D01512 |
Befunolol hydrochloride (JAN); Bentos (TN) |
(P) unclassified |
| D01553 |
Manidipine hydrochloride (JP18); Manidipine dihydrochloride; Calslot (TN) |
(P) Enzyme: CYP3A4 / Target: CACNA1C CACNA1D CACNA1F CACNA1S |
| D01554 |
Pilsicainide hydrochloride hydrate (JP18); Pilsicainide hydrochloride; SUN 1165 (TN); Sunrythm (TN) |
(P) unclassified |
| D01562 |
Aranidipine (JAN/INN); Sapresta (TN) |
(P) Enzyme: CYP3A4 / Target: CACNA1C CACNA1D CACNA1F CACNA1S |
| D01565 |
Indometacin farnesil (JAN); Infree (TN) |
(P) unclassified |
| D01603 |
Bethanidine sulfate (JAN/USAN); Tenathan (TN) |
(P) unclassified |
| D01604 |
Efonidipine hydrochloride ethanolate (JAN); Efonidipine hydrochloride ethanol; Efonidipine hydrochloride; NZ 105 ethanolate; Landel (TN) |
(P) Target: CACNA1C CACNA1D CACNA1F CACNA1S |
| D01638 |
Afloqualone (JP18/INN); Airomate (TN) |
(P) unclassified |
| D01659 |
Syrosingopine (JAN/INN); Siringina (TN) |
(P) unclassified |
| D01671 |
Eperisone hydrochloride (JP18); Epenard (TN) |
(P) unclassified |
| D01691 |
Nipradilol (JAN/INN); Hypadil (TN) |
(P) unclassified |
| D01712 |
Theophylline sodium acetate (JAN) |
(P) unclassified |
| D01721 |
Pentaerythritol tetranitrate (JAN); Pentaerithrityl tetranitrate (INN); Pentritol tempules (TN) |
(P) unclassified |
| D01741 |
Celiprolol hydrochloride (JAN/USAN); Selectol (TN) |
(P) unclassified |
| D01756 |
Trolnitrate phosphate (JAN); Nitretamin (TN) |
(P) unclassified |
| D01768 |
Benoxinate hydrochloride (USP); Oxybuprocaine hydrochloride (JP18); Benoxil (TN) |
(P) unclassified |
| D01772 |
Ether (JP18/USP); Diethyl ether |
(P) unclassified |
| D01785 |
Pirmenol hydrochloride hydrate (JAN); Pimenol (TN) |
(P) unclassified |
| D01794 |
Bopindolol malonate (JAN); Sandonorm (TN) |
(P) unclassified |
| D01795 |
Tilisolol hydrochloride (JAN); Selecal (TN) |
(P) unclassified |
| D01804 |
Cadralazine (JP18/INN); Cadral (TN) |
(P) unclassified |
| D01806 |
Oxprenolol hydrochloride (JP18/USP); Okuspurecol (TN) |
(P) unclassified |
| D01810 |
Nicorandil (JP18/USAN/INN); Sigmart (TN) |
(P) unclassified |
| D01824 |
Phenprobamate (JAN/INN); Spantol (TN) |
(P) unclassified |
| D01830 |
Arotinolol hydrochloride (JP18); Almarl (TN) |
(P) unclassified |
| D01847 |
Landiolol hydrochloride (JAN/USAN); ONO 1101 hydrochloride; Onoact (TN); Rapiblyk (TN) |
(P) unclassified |
| D01849 |
Lercanidipine hydrochloride (JAN/USAN); Cardiovasc (TN) |
(P) Target: CACNA1C CACNA1D CACNA1F CACNA1S |
| D01856 |
Nifekalant hydrochloride (JAN); MS 551; Shinbit (TN) |
(P) unclassified |
| D01878 |
Tolycaine hydrochloride (JAN) |
(P) unclassified |
| D01896 |
Cilostazol (JP18/USP/INN); Pletal (TN) |
(P) Enzyme: CYP3A4 |
| D01902 |
Fonazine mesylate (USAN); Dimetotiazine mesilate (JAN); Banistyl (TN) |
(P) unclassified |
| D01908 |
Nilvadipine (JP18/USAN/INN); Nivadil (TN) |
(P) Enzyme: CYP3A4 / Target: CACNA1C CACNA1D CACNA1F CACNA1S |
| D01933 |
Vatanidipine hydrochloride (JAN); AE 0047; Calbren (TN) |
(P) Target: CACNA1C CACNA1D CACNA1F CACNA1S |
| D01935 |
Vinorelbine tartrate (USP); Vinorelbine ditartrate (JAN); KW 2307; Navelbine (TN) |
(P) Enzyme: CYP3A4 |
| D01943 |
Canrenoate potassium (USAN); Potassium canrenoate (JP18); Soldactone (TN) |
(P) unclassified |
| D01950 |
Dimethylaminoethyl reserpilinate dihydrochloride (JAN); Paratensiol |
(P) unclassified |
| D01958 |
Indenolol hydrochloride (JP18) |
(P) unclassified |
| D01967 |
p-Butylaminobenzoyldiethylaminoethyl hydrochloride (USAN); Diethylaminoethyl p-butylaminobenzoate hydrochloride (JAN); Calvital liquid (TN); T cain (TN) |
(P) unclassified |
| D01969 |
Gallopamil hydrochloride (JAN) |
(P) Target: CACNA1C CACNA1D CACNA1F CACNA1S |
| D01972 |
Lanatoside C (JAN/INN); Digilanogen C (TN) |
(P) unclassified |
| D01973 |
Eletriptan hydrobromide (JAN/USAN); Relpax (TN) |
(P) Enzyme: CYP3A4 |
| D01977 |
Gefitinib (JP18/USAN/INN); Iressa (TN) |
(P) unclassified |
| D01992 |
Tandospirone citrate (JAN/USAN); SM 3997; Sediel (TN) |
(P) unclassified |
| D02008 |
Tadalafil (JAN/USP/INN); Adcirca (TN); Cialis (TN); Zalutia (TN) |
(P) Enzyme: CYP3A4 |
| D02019 |
Magnesium sulfate hydrate and glucose; Magnesol (TN) |
(P) unclassified |
| D02045 |
Benidipine hydrochloride (JP18); KW 3049; Coniel (TN) |
(P) Enzyme: CYP3A4 / Target: CACNA1C CACNA1D CACNA1F CACNA1S |
| D02064 |
Pridinol mesilate (JAN); Pridinol methanesulfonate; Konlax (TN) |
(P) unclassified |
| D02081 |
Metipranolol hydrochloride; Optipranolol (TN) |
(P) unclassified |
| D02086 |
Lidocaine hydrochloride (JAN/USP); Dalcaine (TN); Xylocaine (TN) |
(P) Enzyme: CYP3A4 |
| D02087 |
Moricizine hydrochloride (USP); Ethmozine (TN) |
(P) unclassified |
| D02088 |
Tocainide hydrochloride (USP); Tonocard (TN) |
(P) unclassified |
| D02098 |
Proparacaine hydrochloride (USP); Alcaine (TN); Ophthetic (TN) |
(P) unclassified |
| D02102 |
Methadone hydrochloride (JAN/USP); Dolophine hydrochloride (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
| D02103 |
Phenytoin sodium (USP); Phenytoin sodium for injection (JP18); Aleviatin (TN); Dilantin (TN) |
(P) unclassified |
| D02106 |
Arsenic trioxide (JP18/USAN); Trisenox (TN) |
(P) unclassified |
| D02182 |
Cocaine hydrochloride (JP18/USP); Cocaine hydrochloride (TN) |
(P) unclassified |
| D02204 |
Hexamethonium bromide (JAN/INN); Hexamethonium bromide (TN) |
(P) unclassified |
| D02207 |
Tubocurarine chloride (USP); Tubocurarine chloride hydrate (JAN); Tubocurarine chloride (TN) |
(P) unclassified |
| D02220 |
Dibucaine hydrochloride (JP18/USP); Nupercaine hydrochloride (TN); Percamin (TN) |
(P) unclassified |
| D02237 |
Guanethidine sulfate (USAN) |
(P) unclassified |
| D02239 |
Sparteine sulfate (JAN/USAN); Sparteine sulfate pentahydrate |
(P) unclassified |
| D02260 |
Paroxetine hydrochloride hemihydrate (USP); Paroxetine hydrochloride hydrate (JP18); Paxil (TN) |
(P) unclassified |
| D02272 |
Quinidine sulfate (USP); Quinidine sulfate hydrate (JP18); Quinidex (TN) |
(P) unclassified |
| D02274 |
Dantrolene sodium (USP); Dantrolene sodium hydrate (JP18); Dantrium (TN); Ryanodex (TN) |
(P) unclassified |
| D02275 |
Suxamethonium chloride hydrate (JP18); Suxamethonium chloride dihydrate; Succin (TN) |
(P) unclassified |
| D02292 |
Gallamine triethiodide (USP); Flaxedil (TN) |
(P) unclassified |
| D02338 |
Acebutolol (USAN/INN) |
(P) unclassified |
| D02342 |
Bisoprolol (JAN/USAN/INN) |
(P) unclassified |
| D02347 |
Dantrolene (USAN/INN) |
(P) unclassified |
| D02356 |
Verapamil (USAN/INN) |
(P) Enzyme: CYP3A4 / Target: CACNA1C CACNA1D CACNA1F CACNA1S / CYP inhibition: CYP3A4 |
| D02358 |
Metoprolol (USAN/INN) |
(P) unclassified |
| D02363 |
Ketanserin (USAN/INN) |
(P) unclassified |
| D02372 |
Perospirone hydrochloride hydrate (JAN); Lullan (TN) |
(P) unclassified |
| D02374 |
Metipranolol (USAN/INN) |
(P) unclassified |
| D02389 |
Primidolol (USAN/INN) |
(P) unclassified |
| D02456 |
Aminobenzoic acid (USP); p-Aminobenzoic acid; RVPaba lipstick (TN) |
(P) unclassified |
| D02484 |
Artemether and lumefantrine; Coartem (TN) |
(P) unclassified |
| D02497 |
Fosamprenavir (INN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D02498 |
Lopinavir and ritonavir; Kaletra (TN) |
(P) unclassified |
| D02537 |
Dronedarone (INN) |
(P) Target: CACNA1C CACNA1D CACNA1F CACNA1S |
| D02555 |
Posaconazole (JAN/USAN/INN); Noxafil (TN) |
(P) CYP inhibition: CYP3A4 |
| D02564 |
Pargyline hydrochloride (USAN); Eutonyl (TN) |
(P) unclassified |
| D02567 |
Escitalopram oxalate (JAN/USP); Lexapro (TN) |
(P) Enzyme: CYP3A4 |
| D02587 |
Metildigoxin (JP18); Lanirapid (TN) |
(P) unclassified |
| D02595 |
Mephenesin (INN); Tolserol (TN) |
(P) unclassified |
| D02599 |
Orphenadrine hydrochloride; Disipal (TN) |
(P) unclassified |
| D02611 |
Phenoperidine (INN) |
(P) unclassified |
| D02691 |
Somatropin (USP/INN); Somatropin (genetical recombination) (JAN); Human growth hormone (JAN); Asellacrin (TN); Humatrope (TN); Nutropin (TN); Omnitrope (TN) |
(P) unclassified |
| D02714 |
Everolimus (JAN/USAN/INN); Afinitor (TN); Votubia (TN); Zortress (TN) |
(P) Enzyme: CYP3A4 |
| D02732 |
Pranlukast hydrate (JP18); Onon (TN) |
(P) Enzyme: CYP3A4 |
| D02735 |
Rimabotulinumtoxin B (USAN); Botulinum toxin type B (JAN); Myobloc (TN) |
(P) unclassified |
| D02746 |
Acecainide hydrochloride (USAN) |
(P) unclassified |
| D02763 |
Actodigin (USAN/INN) |
(P) unclassified |
| D02765 |
Adaprolol maleate (USAN) |
(P) unclassified |
| D02812 |
Aliflurane (USAN/INN) |
(P) unclassified |
| D02834 |
Alprenoxime hydrochloride (USAN) |
(P) unclassified |
| D02861 |
Indinavir sulfate ethanolate (JAN); Crixivan (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D02867 |
Fosamprenavir calcium hydrate (JAN); Lexiva (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D02906 |
Aminobenzoate potassium (USP); Potaba (TN) |
(P) unclassified |
| D02907 |
Aminobenzoate sodium (USP); Sodium aminobenzoate |
(P) unclassified |
| D02910 |
Amiodarone (USAN/INN) |
(P) Enzyme: CYP3A4 |
| D02914 |
Amlodipine maleate (USAN); Amvaz (TN) |
(P) Enzyme: CYP3A4 / Target: CACNA1C CACNA1D CACNA1F CACNA1S |
| D02941 |
Anileridine (USP/INN) |
(P) unclassified |
| D02942 |
Anileridine hydrochloride (USP); Leritine (TN) |
(P) unclassified |
| D02968 |
Aprepitant (JAN/USP/INN); Aponvie (TN); Emend (TN); Cinvanti (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4 |
| D02969 |
Aprindine (USAN/INN) |
(P) unclassified |
| D02991 |
Articaine hydrochloride (JAN/USP) |
(P) unclassified |
| D03037 |
Azimilide dihydrochloride (USAN) |
(P) unclassified |
| D03106 |
Bexarotene (JAN/USAN/INN); Targretin (TN) |
(P) unclassified |
| D03170 |
Bucindolol hydrochloride (USAN) |
(P) unclassified |
| D03177 |
Bunolol hydrochloride (USAN) |
(P) unclassified |
| D03198 |
Butoxamine hydrochloride (USAN) |
(P) unclassified |
| D03213 |
Apixaban (JAN/USAN/INN); Eliquis (TN) |
(P) Enzyme: CYP3A4 |
| D03253 |
Brecanavir (USAN) |
(P) unclassified |
| D03290 |
Promethazine methylenedisalicylate (JAN); Pyrethia (TN) |
(P) unclassified |
| D03449 |
Cetamolol hydrochloride (USAN) |
(P) unclassified |
| D03490 |
Cicloprolol hydrochloride (USAN) |
(P) unclassified |
| D03492 |
Cifenline (USAN); Cibenzoline (INN) |
(P) Enzyme: CYP3A4 |
| D03503 |
Cimetidine hydrochloride (USP); Cimetidine hydrochloride (TN) |
(P) CYP inhibition: CYP3A4 |
| D03553 |
Clonitrate (USAN/INN) |
(P) unclassified |
| D03655 |
Darodipine (USAN/INN) |
(P) Target: CACNA1C CACNA1D CACNA1F CACNA1S |
| D03656 |
Darunavir (USAN/INN); Darunavir (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D03658 |
Dasatinib (JAN/INN) |
(P) Enzyme: CYP3A4 |
| D03664 |
Debrisoquin sulfate (USAN); Declinax (TN) |
(P) unclassified |
| D03669 |
Deferasirox (JAN/USAN/INN); Exjade (TN); Jadenu (TN) |
(P) CYP induction: CYP3A4 |
| D03719 |
Dexivacaine (USAN/INN) |
(P) unclassified |
| D03729 |
Dexpropranolol hydrochloride (USAN) |
(P) unclassified |
| D03732 |
Dexsotalol hydrochloride (USAN) |
(P) unclassified |
| D03759 |
Diacetolol hydrochloride (USAN) |
(P) unclassified |
| D03819 |
Digitalis (USP); Digiglusin (TN) |
(P) unclassified |
| D03830 |
Diltiazem malate (USAN); Tiamate (TN) |
(P) Enzyme: CYP3A4 / Target: CACNA1C CACNA1D CACNA1F CACNA1S |
| D03833 |
Indinavir (USAN); Indinavir hydrate |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D03835 |
Fosamprenavir calcium (USAN); Lexiva (TN); Telzir (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D03837 |
Fosamprenavir sodium (USAN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D03839 |
Droxinavir hydrochloride (USAN) |
(P) unclassified |
| D03840 |
Palinavir (USAN/INN) |
(P) unclassified |
| D03841 |
Nitrous oxide and oxygen; Anesoxyn (TN) |
(P) unclassified |
| D03842 |
Telinavir (USAN/INN) |
(P) unclassified |
| D03843 |
Tipranavir disodium (USAN) |
(P) unclassified |
| D03852 |
Droperidol and fentanyl citrate; Innovar (TN) |
(P) Enzyme: CYP3A4 |
| D03914 |
Dronedarone hydrochloride (USP); Multaq (TN) |
(P) Target: CACNA1C CACNA1D CACNA1F CACNA1S |
| D03991 |
Encainide hydrochloride (USAN) |
(P) unclassified |
| D03994 |
Endralazine mesylate (USAN); Endralazine monomethanesulfonate; Migranal (TN) |
(P) unclassified |
| D04024 |
Lapatinib ditosylate (USAN); Lapatinib tosilate hydrate (JAN); Lapatinib ditosylate monohydrate; Tykerb (TN); Tyverb (TN) |
(P) Enzyme: CYP3A4 |
| D04046 |
Salicylamide, acetaminophen, anhydrous caffeine and promethazine methylenedisalicylate; PL (TN) |
(P) unclassified |
| D04048 |
Ropivacaine hydrochloride (USP); Ropivacaine hydrochloride hydrate (JAN); Anapeine (TN) |
(P) Enzyme: CYP3A4 |
| D04051 |
Erythrityl tetranitrate (USAN); Eritrityl tetranitrate (INN); Cardilate (TN) |
(P) unclassified |
| D04088 |
Ethyl chloride (USP) |
(P) unclassified |
| D04095 |
Etidocaine (USAN/INN) |
(P) unclassified |
| D04187 |
Fingolimod hydrochloride (JAN/USAN); Gilenya (TN) |
(P) unclassified |
| D04190 |
Flestolol sulfate (USAN) |
(P) unclassified |
| D04193 |
Flordipine (USAN/INN) |
(P) Target: CACNA1C CACNA1D CACNA1F CACNA1S |
| D04237 |
Fluroxene (USAN); Fluoromar (TN) |
(P) unclassified |
| D04257 |
Fospropofol disodium (USAN); Aquavan (TN); Lusedra (TN) |
(P) unclassified |
| D04265 |
Reserpine, hydralazine hydrochloride and hydrochlorothiazide |
(P) unclassified |
| D04266 |
Benzylhydrochlorothiazide, Reserpine and Carbazochrome; Behyd RA (TN) |
(P) unclassified |
| D04382 |
Guanethidine monosulfate (USP); Guanethidine sulfate (JP18); Ismelin (TN) |
(P) unclassified |
| D04386 |
Guanoclor sulfate (USAN); Vatensol (TN) |
(P) unclassified |
| D04398 |
Guanoxabenz (USAN/INN) |
(P) unclassified |
| D04399 |
Guanoxan sulfate (USAN); Envacar (TN) |
(P) unclassified |
| D04435 |
Hexafluorenium bromide (USAN); Hexafluronium bromide (INN); Mylaxen (TN) |
(P) unclassified |
| D04458 |
Hydralazine polistirex (USAN) |
(P) unclassified |
| D04531 |
Indoramin (USAN/INN) |
(P) unclassified |
| D04532 |
Indoramin hydrochloride (USAN) |
(P) unclassified |
| D04641 |
Istradefylline (JAN/USAN/INN); Nourianz (TN); Nouriast (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D04657 |
Lacidipine (USAN/INN); Motens (TN) |
(P) Target: CACNA1C CACNA1D CACNA1F CACNA1S |
| D04666 |
Lanreotide acetate (JAN/USAN); Somatuline (TN) |
(P) unclassified |
| D04710 |
Levobetaxolol hydrochloride (USAN); Betaxon (TN) |
(P) unclassified |
| D04768 |
Lonafarnib (JAN/USAN/INN); Zokinvy (TN) |
(P) unclassified |
| D04774 |
Lorajmine hydrochloride (USAN) |
(P) unclassified |
| D04777 |
Lorbamate (USAN/INN) |
(P) unclassified |
| D04778 |
Lorcainide hydrochloride (USAN) |
(P) unclassified |
| D04820 |
Lurasidone hydrochloride (JAN/USAN); SM 13496; Latuda (TN) |
(P) Enzyme: CYP3A4 |
| D04888 |
Medroxalol (USAN/INN) |
(P) unclassified |
| D04889 |
Medroxalol hydrochloride (USAN) |
(P) unclassified |
| D04955 |
Sematilide hydrochloride (USAN) |
(P) unclassified |
| D04985 |
Methohexital (USP/INN) |
(P) unclassified |
| D05011 |
Metoprolol fumarate (USP); Lopressor (TN) |
(P) unclassified |
| D05028 |
Midazolam maleate (USAN) |
(P) Enzyme: CYP3A4 |
| D05077 |
Moricizine (USAN); Moracizine (INN) |
(P) unclassified |
| D05087 |
Moxonidine (USAN/INN); Cynt (TN) |
(P) unclassified |
| D05127 |
Nebivolol (USAN/INN) |
(P) unclassified |
| D05208 |
Norflurane (USAN/INN) |
(P) unclassified |
| D05277 |
Formoterol fumarate hydrate (JP18); Formoterol fumarate dihydrate; Atock (TN); Foradil (TN) |
(P) unclassified |
| D05345 |
Pamatolol sulfate (USAN) |
(P) unclassified |
| D05380 |
Pazopanib hydrochloride (JAN/USAN); Votrient (TN) |
(P) unclassified |
| D05429 |
Aminophylline hydrate (JP18) |
(P) unclassified |
| D05430 |
Pentrinitrol (USAN); Petrin (TN) |
(P) unclassified |
| D05482 |
Pinacidil (USAN); Pinacidil hydrate; Pindac (TN) |
(P) unclassified |
| D05538 |
Mozenavir (INN) |
(P) unclassified |
| D05587 |
Practolol (USAN) |
(P) unclassified |
| D05626 |
Propanidid (USAN/INN); Epontol (TN) |
(P) unclassified |
| D05627 |
Propatyl nitrate (USAN); Propatylnitrate (INN); Etrynit (TN) |
(P) unclassified |
| D05665 |
Pyrrocaine (USAN/INN) |
(P) unclassified |
| D05703 |
Rapacuronium bromide (USAN/INN); Raplon (TN) |
(P) unclassified |
| D05705 |
Rauwolfia serpentina (USP); Rauwolfia extract; Himolfia (TN) |
(P) unclassified |
| D05743 |
Rodocaine (USAN) |
(P) unclassified |
| D05745 |
Roflurane (USAN/INN) |
(P) unclassified |
| D05775 |
Rufinamide (JAN/USP/INN); Banzel (TN) |
(P) unclassified |
| D05866 |
Sodium oxybate (USAN); Sodium gammahydroxybutyrate; Xyrem (TN) |
(P) unclassified |
| D05928 |
Stiripentol (JAN/USAN/INN); Diacomit (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D05938 |
Sufentanil (USAN/INN) |
(P) unclassified |
| D06055 |
Teflurane (USAN/INN) |
(P) unclassified |
| D06060 |
Teludipine hydrochloride (USAN) |
(P) unclassified |
| D06103 |
Theophylline (USP); Theophylline monohydrate; Accurbron (TN) |
(P) unclassified |
| D06104 |
Theophylline sodium glycinate (USP); Asbron (TN) |
(P) unclassified |
| D06106 |
Thiamylal |
(P) unclassified |
| D06129 |
Tiapamil hydrochloride (USAN) |
(P) Target: CACNA1C CACNA1D CACNA1F CACNA1S |
| D06162 |
Tiprenolol hydrochloride (USAN) |
(P) unclassified |
| D06172 |
Tocainide (USAN/INN) |
(P) unclassified |
| D06176 |
Tolamolol (USAN/INN) |
(P) unclassified |
| D06213 |
Treprostinil (JAN/USAN/INN); Remodulin (TN) |
(P) unclassified |
| D06234 |
Trimazosin hydrochloride (USAN); Trimazosin hydrochloride monohydrate |
(P) unclassified |
| D06402 |
Sunitinib malate (JAN/USAN); Sutent (TN) |
(P) Enzyme: CYP3A4 |
| D06407 |
Vandetanib (JAN/USAN/INN); Caprelsa (TN) |
(P) Enzyme: CYP3A4 |
| D06413 |
Nilotinib hydrochloride hydrate (JAN); Nilotinib monohydrochloride monohydrate; Tasigna (TN) |
(P) Enzyme: CYP3A4 |
| D06414 |
Dasatinib (USAN); Dasatinib hydrate (JAN); Sprycel (TN) |
(P) Enzyme: CYP3A4 |
| D06478 |
Darunavir ethanolate (JAN); Prezista (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D06517 |
Pirmenol hydrochloride (USAN); Pirmavar (TN) |
(P) unclassified |
| D06534 |
Phenolated water (JP18); Phenolated water for disinfection (JP18); Phenol hydrate; Phenol water (TN); Phenolated water for disinfection (TN) |
(P) unclassified |
| D06597 |
Fosaprepitant dimeglumine (USAN); Fosaprepitant meglumine (JAN); Proemend (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4 |
| D06622 |
Nebivolol hydrochloride (USAN); Bystolic (TN) |
(P) unclassified |
| D06637 |
Romidepsin (JAN/USAN/INN); Istodax (TN) |
(P) unclassified |
| D06646 |
Epanolol (USAN/INN) |
(P) unclassified |
| D06652 |
Tedisamil (USAN) |
(P) unclassified |
| D06653 |
Tedisamil sesquifumarate (USAN) |
(P) unclassified |
| D06665 |
Vernakalant hydrochloride (USAN) |
(P) unclassified |
| D06881 |
Acetyldigitoxin (INN); Acylanid (TN) |
(P) unclassified |
| D07077 |
Ambrisentan (JAN/INN); Letairis (TN); Volibris (TN) |
(P) unclassified |
| D07122 |
Alfentanil (INN); Rapifen (TN) |
(P) unclassified |
| D07147 |
Gitoformate (INN) |
(P) unclassified |
| D07156 |
Alprenolol (INN) |
(P) unclassified |
| D07166 |
Methoserpidine (INN) |
(P) unclassified |
| D07167 |
Bietaserpine (prop.INN) |
(P) unclassified |
| D07168 |
Tolonidine (INN) |
(P) unclassified |
| D07169 |
Guanazodine (INN) |
(P) unclassified |
| D07170 |
Dihydralazine (INN) |
(P) unclassified |
| D07171 |
Sitaxentan (USAN/INN) |
(P) unclassified |
| D07181 |
Mepindolol (INN) |
(P) unclassified |
| D07182 |
Tertatolol (INN) |
(P) unclassified |
| D07183 |
Cloranolol (INN) |
(P) unclassified |
| D07184 |
Talinolol (INN) |
(P) unclassified |
| D07185 |
Fendiline (INN) |
(P) Target: CACNA1C CACNA1D CACNA1F CACNA1S |
| D07274 |
Styramate (INN) |
(P) unclassified |
| D07275 |
Febarbamate (INN) |
(P) unclassified |
| D07276 |
Thiocolchicoside (INN); Coltramyl (TN) |
(P) unclassified |
| D07277 |
Tetrazepam (INN); Myolastan (TN) |
(P) unclassified |
| D07282 |
Alfaxalone (INN) |
(P) unclassified |
| D07284 |
Butanilicaine (INN) |
(P) unclassified |
| D07428 |
Bunaftine (INN) |
(P) unclassified |
| D07450 |
Amlodipine (USP/INN); Norvasc (TN) |
(P) Enzyme: CYP3A4 / Target: CACNA1C CACNA1D CACNA1F CACNA1S |
| D07465 |
Arotinolol (INN) |
(P) unclassified |
| D07468 |
Articaine (INN); Carticaine |
(P) unclassified |
| D07471 |
Atazanavir (INN); Reyataz (TN) |
(P) CYP inhibition: CYP3A4 |
| D07494 |
Barnidipine (INN); Vasexten (TN) |
(P) Enzyme: CYP3A4 / Target: CACNA1C CACNA1D CACNA1F CACNA1S |
| D07496 |
Befunolol (INN) |
(P) unclassified |
| D07505 |
Latanoprost and timolol maleate; Xalacom (TN) |
(P) unclassified |
| D07509 |
Benidipine (INN) |
(P) Enzyme: CYP3A4 / Target: CACNA1C CACNA1D CACNA1F CACNA1S |
| D07520 |
Bepridil (INN); Bepadin (TN) |
(P) Enzyme: CYP3A4 / Target: CACNA1C CACNA1D CACNA1F CACNA1S |
| D07526 |
Betaxolol (INN); Betaxolol (TN) |
(P) unclassified |
| D07537 |
Bopindolol (INN); Sandonorm (TN) |
(P) unclassified |
| D07538 |
Bosentan (INN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
| D07552 |
Bupivacaine (USAN/INN); Bucaine (TN); Exparel (TN) |
(P) Enzyme: CYP3A4 |
| D07555 |
Acetyldigoxin; Cedigossima (TN) |
(P) unclassified |
| D07556 |
beta-Acetyldigoxin; Acetyldigoxin beta isomer; Corotal (TN) |
(P) unclassified |
| D07569 |
Candesartan cilexetil and anmlodipine besylate (JP18); Unisia (TN) |
(P) Enzyme: CYP3A4 |
| D07583 |
Phenytoin and phenobarbital; Aleviatin with phenobarbital (TN) |
(P) unclassified |
| D07590 |
Bupranolol (INN) |
(P) unclassified |
| D07595 |
Fosphenytoin sodium hydrate (JAN); Fostoin (TN) |
(P) CYP induction: CYP3A4 |
| D07608 |
Carazolol (INN); Conducton (TN); Suacron [veterinary] (TN) |
(P) unclassified |
| D07624 |
Carteolol (INN) |
(P) unclassified |
| D07660 |
Celiprolol (INN); Celiprolol PCH (TN) |
(P) unclassified |
| D07678 |
Chloroprocaine (INN) |
(P) unclassified |
| D07758 |
Cyclobenzaprine (INN) |
(P) unclassified |
| D07830 |
Dihydralazine sulfate; Dihydralazine hydrogen sulfate; Nepresol (TN) |
(P) unclassified |
| D07845 |
Diltiazem (INN); Surazem (TN) |
(P) Enzyme: CYP3A4 / Target: CACNA1C CACNA1D CACNA1F CACNA1S |
| D07874 |
Doxazosin (INN); Cardura XL (TN) |
(P) unclassified |
| D07881 |
Dyclonine (INN) |
(P) unclassified |
| D07886 |
Efonidipine (INN) |
(P) Target: CACNA1C CACNA1D CACNA1F CACNA1S |
| D07894 |
Encainide (INN) |
(P) unclassified |
| D07898 |
Eperisone (INN) |
(P) unclassified |
| D07916 |
Esmolol (INN) |
(P) unclassified |
| D07943 |
Fendiline hydrochloride; Sensit (TN) |
(P) Target: CACNA1C CACNA1D CACNA1F CACNA1S |
| D07953 |
Fenyramidol (INN) |
(P) unclassified |
| D07962 |
Flecainide (INN) |
(P) unclassified |
| D08009 |
Gallopamil (INN) |
(P) Target: CACNA1C CACNA1D CACNA1F CACNA1S |
| D08020 |
Lorcainide (INN) |
(P) unclassified |
| D08030 |
Guanethidine (INN) |
(P) unclassified |
| D08031 |
Guanfacine (INN); Estulic (TN) |
(P) Enzyme: CYP3A4 |
| D08044 |
Hydralazine (INN); Hidral (TN) |
(P) unclassified |
| D08048 |
Hydroquinidine (DCF); Dihydroquinidine |
(P) unclassified |
| D08049 |
Hydroquinidine hydrochloride; Idrochinidine (TN); Serecor (TN) |
(P) unclassified |
| D08060 |
Ibutilide (INN) |
(P) unclassified |
| D08074 |
Penbutolol (INN) |
(P) unclassified |
| D08078 |
Indenolol (INN) |
(P) unclassified |
| D08095 |
Ivabradine hydrochloride (JAN/USAN); Ivabrandine hydrochloride; Corlanor (TN); Corlentor (TN); Coralan (TN) |
(CI) Enzyme: CYP3A4 |
| D08098 |
Ketamine (INN); Tekam (TN) |
(P) unclassified |
| D08099 |
Ketanserin tartrate; Sufrexal (TN) |
(P) unclassified |
| D08111 |
Lercanidipine (INN); Lercanil (TN) |
(P) Target: CACNA1C CACNA1D CACNA1F CACNA1S |
| D08115 |
Levobunolol (INN) |
(P) unclassified |
| D08116 |
Levobupivacaine (INN); Novabupi (TN) |
(P) Enzyme: CYP3A4 |
| D08127 |
Lidocaine hydrochloride monohydrate; Lidocaine (TN); Zingo (TN) |
(P) Enzyme: CYP3A4 |
| D08155 |
Manidipine (INN); Manidipine 6300; Artedil (TN) |
(P) Enzyme: CYP3A4 / Target: CACNA1C CACNA1D CACNA1F CACNA1S |
| D08181 |
Mepivacaine (INN); Carboplyin Dental (TN) |
(P) unclassified |
| D08194 |
Deserpidine (INN); Halmonyl (TN) |
(P) unclassified |
| D08205 |
Methyldopa (INN); Aldomet (TN) |
(P) unclassified |
| D08212 |
Trimazosin (INN) |
(P) unclassified |
| D08215 |
Mexiletine (INN) |
(P) unclassified |
| D08254 |
Endralazine (INN) |
(P) unclassified |
| D08259 |
Nelfinavir (INN); Viracept (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D08270 |
Nicardipine (INN); Cardene (TN) |
(P) Enzyme: CYP3A4 / Target: CACNA1C CACNA1D CACNA1F CACNA1S |
| D08305 |
Orphenadrine (INN); Mialgin (TN) |
(P) unclassified |
| D08311 |
Oxetacaine hydrochloride; Emoren (TN) |
(P) unclassified |
| D08318 |
Oxprenolol (INN); Oxprenolol (TN) |
(P) unclassified |
| D08319 |
Oxybuprocaine (INN); Monofree oxybuprocaine (TN) |
(P) unclassified |
| D08377 |
Pilsicainide (INN) |
(P) unclassified |
| D08394 |
Pirmenol (INN) |
(P) unclassified |
| D08411 |
Prazosin (INN); Minipress (TN) |
(P) unclassified |
| D08418 |
Pridinol (INN) |
(P) unclassified |
| D08419 |
Pridinol hydrochloride; Pridinol (TN) |
(P) unclassified |
| D08421 |
Procainamide (INN) |
(P) unclassified |
| D08422 |
Procaine (INN); Solution of novocain (TN) |
(P) unclassified |
| D08435 |
Propafenone (INN); Propafenon hexal (TN) |
(P) Enzyme: CYP3A4 |
| D08443 |
Propranolol (INN); Propranolol (TN) |
(P) unclassified |
| D08448 |
Proxymetacaine (INN); Proparacaine |
(P) unclassified |
| D08453 |
Pargyline (INN) |
(P) unclassified |
| D08458 |
Quinidine (BAN); Kinidin (TN) |
(P) unclassified |
| D08459 |
Quinidine phenylethylbarbiturate; Quinidine 5-ethyl 5-phenyl barbiturate; Natisedine (TN) |
(P) unclassified |
| D08473 |
Remifentanil (INN); Ultiva (TN) |
(P) unclassified |
| D08479 |
Rifampicin sodium; Rifadine (TN) |
(P) CYP induction: CYP3A4 |
| D08482 |
Rilmenidine (INN); Hyperium (TN) |
(P) unclassified |
| D08488 |
Amlodipine besilate and atorvastatin calcium; Caduet (TN) |
(P) Enzyme: CYP3A4 |
| D08490 |
Ropivacaine (INN); Naropin (TN) |
(P) Enzyme: CYP3A4 |
| D08493 |
Dorzolamide hydrochloride and timolol maleate (JP18); Cosopt (TN) |
(P) Enzyme: CYP3A4 |
| D08517 |
Sitaxentan sodium (USAN); Thelin (TN) |
(P) unclassified |
| D08525 |
Sotalol (INN); Darob mite (TN) |
(P) unclassified |
| D08553 |
Suxethonium chloride (INN); Curacit (TN) |
(P) unclassified |
| D08572 |
Tertatolol hydrochloride; Artex (TN) |
(P) unclassified |
| D08598 |
Tilisolol (INN) |
(P) unclassified |
| D08600 |
Timolol (INN); Timolol (TN); Betimol (TN) |
(P) unclassified |
| D08605 |
Tipranavir (INN); Aptivus (TN) |
(P) unclassified |
| D08611 |
Tizanidine (INN); Sirdalud (TN) |
(P) unclassified |
| D08617 |
Tolperisone (INN); Musclex (TN) |
(P) unclassified |
| D08640 |
Trimecaine (INN); Mesidicain; Mesocain |
(P) unclassified |
| D08641 |
Trimecaine hydrochloride; Mesocain (TN) |
(P) unclassified |
| D08655 |
Tubocurarine chloride (INN); Tubaine (TN); Tubocurarine Chloride (TN) |
(P) unclassified |
| D08662 |
Urapidil hydrochloride; Ebrantil (TN) |
(P) unclassified |
| D08768 |
Promethazine hibenzate; Hiberna (TN) |
(P) unclassified |
| D08856 |
Anamorelin hydrochloride (JAN/USAN); Adlumiz (TN) |
(P) Enzyme: CYP3A4 |
| D08892 |
Clevidipine (USAN/INN); Clevidipine butyrate; Cleviprex (TN) |
(P) Target: CACNA1C CACNA1D CACNA1F CACNA1S |
| D08941 |
Levamlodipine malate (USAN) |
(P) Target: CACNA1C CACNA1D CACNA1F CACNA1S |
| D09017 |
Ticagrelor (JAN/USAN/INN); Brilinta (TN) |
(P) unclassified |
| D09033 |
Voclosporin (JAN/USAN/INN); Lupkynis (TN) |
(P) Enzyme: CYP3A4 |
| D09546 |
Edoxaban tosilate hydrate (JAN); Edoxaban tosylate monohydrate; Lixiana (TN); Savaysa (TN) |
(P) unclassified |
| D09570 |
Bilastine (JAN/INN); Bilanoa (TN) |
(P) unclassified |
| D09572 |
Riociguat (JAN/USAN/INN); Adempas (TN) |
(P) unclassified |
| D09595 |
Budesonide and formoterol fumarate dihydrate; Symbicort (TN); Budeforu (TN) |
(P) Enzyme: CYP3A4 |
| D09638 |
Lomitapide mesylate (USAN); Lomitapide mesilate (JAN); Juxtapid (TN); Lojuxta (TN) |
(CI,P) Enzyme: CYP3A4 |
| D09670 |
Sotatercept (USAN/INN); Sotatercept (genetical recombination) (JAN); sotatercept-csrk; Winrevair (TN); Airwin (TN) |
(P) unclassified |
| D09728 |
Bosutinib hydrate (JAN); Bosutinib monohydrate; Bosulif (TN) |
(P) Enzyme: CYP3A4 |
| D09730 |
Olaparib (JAN/USAN/INN); Lynparza (TN) |
(P) unclassified |
| D09731 |
Crizotinib (JAN/USAN/INN); Xalkori (TN) |
(P) Enzyme: CYP3A4 |
| D09743 |
Telmisartan and amlodipine besilate (JP18); Telmisartan and amlodipine besylate; Micamlo (TN); Twynsta (TN) |
(P) Enzyme: CYP3A4 |
| D09745 |
Valsartan and amlodipine besilate; Exforge (TN) |
(P) Enzyme: CYP3A4 |
| D09783 |
Tofacitinib citrate (JAN/USAN); Tasocitinib citrate; Xeljanz (TN) |
(P) Enzyme: CYP3A4 |
| D09789 |
Kirenidipine hydrochloride (JAN) |
(P) Target: CACNA1C CACNA1D CACNA1F CACNA1S |
| D09799 |
Carotegrast methyl (JAN); Carogra (TN) |
(P) CYP inhibition: CYP3A4 |
| D09815 |
Travoprost and timolol maleate; Duotrav (TN) |
(P) unclassified |
| D09843 |
Beradilol monoethyl maleate (JAN); TZC-5665 |
(P) unclassified |
| D09847 |
Metildigoxin (INN); Medigoxin (BAN) |
(P) unclassified |
| D09951 |
Ponatinib hydrochloride (JAN/USAN); Iclusig (TN) |
(P) unclassified |
| D09960 |
Ruxolitinib phosphate (JAN/USAN); Jakafi (TN); Jakavi (TN); Opzelura (TN) |
(P) Enzyme: CYP3A4 |
| D09994 |
Selexipag (JAN/USAN/INN); Uptravi (TN) |
(P) Enzyme: CYP3A4 |
| D09996 |
Vemurafenib (JAN/USAN/INN); Zelboraf (TN) |
(P) CYP induction: CYP3A4 |
| D10003 |
Hemin (JAN); Normosang (TN); Panhematin (TN) |
(P) CYP induction: CYP3A4 |
| D10082 |
Suvorexant (JAN/USAN); MK-4305; Belsomra (TN) |
(P) unclassified |
| D10093 |
Asunaprevir (JAN/USAN); Sunvepra (TN) |
(CI) CYP induction: CYP3A4 |
| D10104 |
Dabrafenib mesylate (USAN); Dabrafenib mesilate (JAN); Tafinlar (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
| D10105 |
Daclatasvir dihydrochloride (USAN); Daclatasvir hydrochloride (JAN); Daklinza (TN) |
(CI) Enzyme: CYP3A4 |
| D10135 |
Macitentan (JAN/USAN); Opsumit (TN) |
(P) Enzyme: CYP3A4 |
| D10161 |
Sarilumab (USAN); Sarilumab (genetical receombination) (JAN); Kevzara (TN) |
(P) unclassified |
| D10218 |
Enzalutamide (JAN/USAN); Xtandi (TN) |
(P) unclassified |
| D10223 |
Ibrutinib (JAN/USAN); Imbruvica (TN) |
(P) unclassified |
| D10243 |
Irbesartan and amlodipine besilate (JP18); Aimix (TN) |
(P) Enzyme: CYP3A4 |
| D10255 |
Anagrelide hydrochloride hydrate (JAN); Anagrelide hydrochloride monohydrate; Agrylin (TN) |
(P) unclassified |
| D10267 |
Methyldopa and hydrochlorothiazide; Methyldopa and hydrochlorothiazide (TN) |
(P) unclassified |
| D10298 |
Brimonidine tartrate and timolol maleate; Combigan (TN); Aibeta (TN) |
(P) unclassified |
| D10372 |
Palbociclib (JAN/USAN); Ibrance (TN) |
(P) unclassified |
| D10466 |
Vonoprazan fumarate (JAN/USAN); Takecab (TN); Voquezna (TN) |
(P) Enzyme: CYP3A4 |
| D10501 |
Fluticasone furoate and vilanterol trifenatate; Breo ellipta (TN); Relvar ellipita (TN) |
(P) Enzyme: CYP3A4 |
| D10503 |
Ethacizine |
(P) unclassified |
| D10506 |
Fluticasone propionate and formoterol fumarate hydrate; Flutiform (TN) |
(P) Enzyme: CYP3A4 |
| D10512 |
Brinzolamide and timolol maleate; Azorga (TN) |
(P) Enzyme: CYP3A4 |
| D10519 |
Rabeprazole, amoxicillin and clarithromycin; Rabecure (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D10524 |
Azilsartan and amlodipine besilate; Zacras (TN) |
(P) Enzyme: CYP3A4 |
| D10533 |
Umeclidinium bromide and vilanterol; Anoro (TN) |
(P) Enzyme: CYP3A4 |
| D10551 |
Ceritinib (JAN/USAN/INN); Zykadia (TN) |
(P) unclassified |
| D10564 |
Amenamevir (JAN/INN); Amenalief (TN) |
(P) unclassified |
| D10566 |
Pasireotide pamoate (JAN); Signifor lar (TN) |
(P) unclassified |
| D10569 |
Tafluprost and timolol maleate; Tapcom (TN) |
(P) unclassified |
| D10591 |
Clonidine and chlorthalidone; Clorpres (TN) |
(P) unclassified |
| D10643 |
Isavuconazonium sulfate (JAN/USAN); Cresemba (TN) |
(P) unclassified |
| D10679 |
Venetoclax (JAN/USAN/INN); Venclexta (TN) |
(P) unclassified |
| D10688 |
Abemaciclib (JAN/USAN/INN); Verzenio (TN) |
(P) unclassified |
| D10755 |
Elvitegravir, cobicistat, emtricitabine and tenofovir alafenamide; Genvoya (TN) |
(P) unclassified |
| D10762 |
Fosravuconazole L-lysine ethanolate (JAN) |
(P) unclassified |
| D10774 |
Vonoprazan, amoxicillin and metronidazole; Vonopion (TN) |
(P) Enzyme: CYP3A4 |
| D10775 |
Vonoprazan, amoxicillin and clarithromycin; Vonosap (TN); Voquenza (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D10801 |
Letermovir (JAN/USAN/INN); Prevymis (TN) |
(P) unclassified |
| D10804 |
Carteolol and latanoprost; Mikeluna (TN) |
(P) unclassified |
| D10805 |
Telmisartan, amlodipine and hydrochlorothiazide; Micatrio (TN) |
(P) Enzyme: CYP3A4 |
| D10811 |
Fentanyl hydrochloride (JAN); Ionsys (TN) |
(P) Enzyme: CYP3A4 |
| D10832 |
Darunavir and cobicistat; Prezcobix (TN); Rezolsta (TN) |
(P) unclassified |
| D10866 |
Brigatinib (JAN/USAN); Alunbrig (TN) |
(P) Enzyme: CYP3A4 |
| D10882 |
Daclatasvir, asunaprevir and beclabuvir; Ximency (TN) |
(CI) CYP induction: CYP3A4 |
| D10926 |
Entrectinib (JAN/USAN/INN); Rozlytrek (TN) |
(P) Enzyme: CYP3A4 |
| D10931 |
Etrasimod arginine (USAN); Etrasimod L-arginine (JAN); Velsipity (TN) |
(P) Enzyme: CYP3A4 |
| D10967 |
Ozanimod hydrochloride (JAN/USAN); Zeposia (TN) |
(P) unclassified |
| D10990 |
Somatrogon (USAN/INN); Somatrogon (genetical recombination) (JAN); Somatrogon-ghla; Ngenla (TN) |
(P) unclassified |
| D10993 |
Tucidinostat (JAN/USAN/INN); Hiyasta (TN) |
(P) unclassified |
| D11012 |
Lorlatinib (JAN/USAN/INN); Lorbrena (TN) |
(P) unclassified |
| D11035 |
Fluticasone furoate, umeclidinium bromide and vilanterol; Trelegy ellipta (TN) |
(P) unclassified |
| D11036 |
Glycopyrrolate and formoterol; Bevespi (TN) |
(P) unclassified |
| D11040 |
Apalutamide (JAN/INN); Erleada (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
| D11053 |
Encorafenib (JAN/USAN/INN); Braftovi (TN) |
(P) Enzyme: CYP3A4 |
| D11062 |
Osilodrostat phosphate (JAN/USAN); Isturisa (TN) |
(P) Enzyme: CYP3A4 |
| D11072 |
Siponimod fumarate (USAN); Siponimod fumaric acid (JAN); Mayzent (TN) |
(P) unclassified |
| D11090 |
Ivosidenib (JAN/USAN/INN); Tibsovo (TN) |
(P) unclassified |
| D11138 |
Larotrectinib sulfate (JAN/USAN); Vitrakvi (TN) |
(P) unclassified |
| D11190 |
Vosoritide (USAN/INN); Vosoritide (genetical recombination) (JAN); Voxzogo (TN) |
(P) unclassified |
| D11194 |
Somapacitan (USAN/INN); Somapacitan (genetical recombination) (JAN); Somapacitan-beco; Sogroya (TN) |
(P) unclassified |
| D11296 |
Fedratinib hydrochloride (USAN); Fedratinib hydrochloride hydrate (JAN); Fedratinib dihydrochloride monohydrate; Inrebic (TN) |
(P) Enzyme: CYP3A4 |
| D11370 |
Fosnetupitant chloride hydrochloride (JAN/USAN); Arokaris (TN) |
(P) unclassified |
| D11371 |
Capivasertib (JAN/USAN); Truqap (TN) |
(P) Enzyme: CYP3A4 |
| D11382 |
Darunavir, cobicistat, emtricitabine and tenofovir alafenamide; Symtuza (TN) |
(P) unclassified |
| D11405 |
Prabotulinumtoxin A (USAN); PrabotulinumtoxinA-xvfs; Jeuveau (TN) |
(P) unclassified |
| D11422 |
Zanubrutinib (JAN/USAN/INN); Brukinsa (TN) |
(P) unclassified |
| D11441 |
Aprocitentan (USAN/INN); Tryvio (TN) |
(P) unclassified |
| D11454 |
Repotrectinib (JAN/USAN); Augtyro (TN) |
(P) Enzyme: CYP3A4 |
| D11485 |
Tazemetostat hydrobromide (JAN/USAN); Tazverik (TN) |
(P) unclassified |
| D11557 |
Tecovirimat hydrate (JAN); Tecovirimat monohydrate; Tpoxx (TN); Tepoxx (TN) |
(P) unclassified |
| D11584 |
Budesonide, glycopyrronium bromide and formoterol fumarate; Budesonide, glycopyrrolate and formoterol fumarate; Breztri (TN) |
(P) unclassified |
| D11662 |
Valemetostat tosilate (JAN); Valemetostat tosylate; Ezharmia (TN) |
(P) unclassified |
| D11674 |
Berotralstat hydrochloride (JAN/USAN); Orladeyo (TN) |
(P) CYP inhibition: CYP3A4 |
| D11713 |
Selpercatinib (JAN/USAN/INN); Retevmo (TN) |
(P) Enzyme: CYP3A4 |
| D11804 |
Aspirin and vonoprazan; Cabpirin (TN) |
(P) unclassified |
| D11816 |
Belumosudil mesylate (USAN); Belumosudil mesilate (JAN); Rezurock (TN) |
(P) unclassified |
| D11881 |
Amlodipine benzoate; Katerzia (TN) |
(P) Enzyme: CYP3A4 / Target: CACNA1C CACNA1D CACNA1F CACNA1S |
| D11887 |
Daridorexant hydrochloride (JAN/USAN); Quviviq (TN) |
(P) unclassified |
| D11920 |
Pimitespib (JAN); Jeselhy (TN) |
(P) unclassified |
| D11954 |
Belzutifan (JAN/USAN/INN); Welireg (TN) |
(P) unclassified |
| D11970 |
Ritlecitinib tosylate (USAN); Ritlecitinib tosilate (JAN); Litfulo (TN) |
(P) unclassified |
| D12050 |
Pirtobrutinib (JAN/USAN); Jaypirca (TN) |
(P) Enzyme: CYP3A4 |
| D12055 |
Sotorasib (JAN/USAN); Lumakras (TN) |
(P) unclassified |
| D12245 |
Lazertinib mesylate (USAN); Lazertinib mesilate hydrate (JAN); Lazcluze (TN) |
(P) Enzyme: CYP3A4 |
| D12252 |
Iptacopan hydrochloride (USAN); Iptacopan hydrochloride hydrate (JAN); Iptacopan hydrochloride monohydrate; Fabhalta (TN) |
(P) unclassified |
| D12265 |
Mavacamten (JAN/USAN/INN); Camzyos (TN) |
(P) unclassified |
| D12269 |
Nirmatrelvir and ritonavir; Paxlovid (TN) |
(P) Enzyme: CYP3A4 |
| D12353 |
Ensitrelvir fumarate (USAN); Ensitrelvir fumaric acid (JAN); Xocova (TN) |
(P) unclassified |
| D12410 |
Landiolol (USAN/INN) |
(P) unclassified |
| D12586 |
Mifepristone and misoprostol; Mefeego (TN) |
(P) unclassified |
| D12637 |
Darunavir hydrate |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D12752 |
Darunavir propylene glycolate |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D12963 |
Macitentan and tadalafil; Opsynvi (TN); Yuvanci (TN) |
(P) unclassified |
