| C06174 |
Codeine; (5alpha,6alpha)-7,8-Didehydro-4,5-epoxy-3-methoxy-17-methylmorphinan-6-ol |
(P) unclassified |
| C07051 |
Indinavir |
(P) unclassified |
| D00020 |
Tryptophan (USP/INN); L-Tryptophan (JP19) |
(P) unclassified |
| D00058 |
gamma-Aminobutyric acid (JAN); Gammalon (TN) |
(P) unclassified |
| D00136 |
Haloperidol (JP19/USP/INN); Haldol (TN) |
(P) Enzyme: CYP3A4 |
| D00138 |
Scopolamine (INN); Transderm scop (TN) |
(P) unclassified |
| D00184 |
Cyclosporine (USP); Ciclosporin (JP19); Gengraf (TN); Neoral (TN); Restasis (TN); Sandimmune (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D00195 |
Codeine (USP); Codeine hydrate |
(P) unclassified |
| D00211 |
Rifampin (USP); Rifampicin (JP19/INN); Rifadin (TN); Rimactane (TN) |
(P) CYP induction: CYP3A4 |
| D00225 |
Alprazolam (JP19/USP/INN); Xanax (TN) |
(P) unclassified |
| D00228 |
Amoxapine (JP19/USP/INN); Asendin (TN) |
(P) unclassified |
| D00252 |
Carbamazepine (JP19/USP/INN); Equetro (TN); Tegretol (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
| D00265 |
Chloral hydrate (JP19/USP); Noctec (TN) |
(P) unclassified |
| D00267 |
Chlordiazepoxide (JP19/USP/INN); Libritabs (TN) |
(P) unclassified |
| D00270 |
Chlorpromazine (USP/INN); Thorazine (TN) |
(P) unclassified |
| D00276 |
Clarithromycin (JP19/USP/INN); Biaxin (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D00280 |
Clonazepam (JP19/USP/INN); Klonopin (TN) |
(P) unclassified |
| D00282 |
Clotrimazole (JP19/USP/INN); Lotrimin (TN); Mycelex (TN) |
(P) CYP inhibition: CYP3A4 |
| D00283 |
Clozapine (JAN/USP/INN); Clozaril (TN) |
(P) Enzyme: CYP3A4 |
| D00292 |
Dexamethasone (JP19/USP/INN); Decadron (TN); Maxidex (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
| D00293 |
Diazepam (JP19/USP/INN); Diastat (TN); Valium (TN) |
(P) Enzyme: CYP3A4 |
| D00295 |
Cimetidine (JP19/USP/INN); Tagamet (TN) |
(P) CYP inhibition: CYP3A4 |
| D00304 |
Divalproex sodium (USP); Valproate semisodium (INN); Depakote (TN) |
(P) unclassified |
| D00308 |
Droperidol (JP19/USP/INN); Droleptan (TN); Inapsine (TN) |
(P) unclassified |
| D00311 |
Estazolam (JP19/USP/INN); ProSom (TN) |
(P) unclassified |
| D00320 |
Fentanyl (JAN/USP/INN); Duragesic (TN); Subsys (TN) |
(P) Enzyme: CYP3A4 |
| D00322 |
Fluconazole (JP19/USP/INN); Diflucan (TN) |
(P) CYP inhibition: CYP3A4 |
| D00326 |
Fluoxetine (USAN/INN); Fluoxetine (TN) |
(P) unclassified |
| D00329 |
Flurazepam (JAN/INN); Insumin (TN) |
(P) unclassified |
| D00338 |
Halazepam (USAN/INN); Paxipam (TN) |
(P) unclassified |
| D00350 |
Itraconazole (JP19/USP); Itrizole (TN); Sporanox (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D00351 |
Ketoconazole (JP19/USP); Nizoral (TN); Xolegel (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D00354 |
Lamotrigine (JAN/USP/INN); Lamictal (TN) |
(P) unclassified |
| D00365 |
Lorazepam (JP19/USP/INN); Ativan (TN) |
(P) unclassified |
| D00370 |
Temazepam (USP/INN); Restoril (TN) |
(P) unclassified |
| D00373 |
Thioridazine (USP/INN); Mellaril-S (TN) |
(P) unclassified |
| D00374 |
Thiothixene (USP); Tiotixene (JAN); Navane (TN) |
(P) unclassified |
| D00375 |
Mephenytoin (USP/INN); Mesantoin (TN) |
(P) unclassified |
| D00376 |
Meprobamate (JAN/USP/INN); Equanil (TN); Miltown (TN) |
(P) unclassified |
| D00387 |
Triazolam (JP19/USP/INN); Halcion (TN) |
(P) Enzyme: CYP3A4 |
| D00388 |
Triclofos sodium (JP19/USAN); Tricloryl (TN) |
(P) unclassified |
| D00390 |
Triflupromazine (USP/INN); Vesprin (TN) |
(P) unclassified |
| D00392 |
Trimethadione (JP19/INN); Tridione (TN) |
(P) unclassified |
| D00394 |
Trimipramine (USAN/INN) |
(P) unclassified |
| D00399 |
Valproic acid (USP); Depakene (TN) |
(P) unclassified |
| D00403 |
Methotrimeprazine (USP); Levomepromazine (USAN/INN); Levoprome (TN) |
(P) unclassified |
| D00404 |
Methsuximide (USP); Mesuximide (INN); Celontin (TN) |
(P) unclassified |
| D00420 |
Mitotane (JAN/USP/INN); Lysodren (TN) |
(P) unclassified |
| D00426 |
Risperidone (JP19/USP/INN); Risperdal (TN) |
(P) Enzyme: CYP3A4 |
| D00427 |
Ritonavir (JAN/USP/INN); Norvir (TN) |
(P) unclassified |
| D00430 |
Secobarbital (USP/INN); Seconal (TN) |
(P) unclassified |
| D00435 |
Nevirapine (JAN/USP/INN); Viramune (TN) |
(P) Enzyme: CYP3A4 |
| D00437 |
Nifedipine (JP19/USP/INN); Adalat (TN); Afeditab CR (TN); Procardia (TN) |
(P) Enzyme: CYP3A4 |
| D00454 |
Olanzapine (JAN/USP/INN); Zyprexa (TN) |
(P) unclassified |
| D00457 |
Quazepam (JAN/USP/INN); Doral (TN) |
(P) Enzyme: CYP3A4 |
| D00458 |
Quetiapine fumarate (JP19/USP); Seroquel (TN) |
(P) Enzyme: CYP3A4 |
| D00464 |
Oxazepam (JAN/USP/INN); Serax (TN) |
(P) unclassified |
| D00470 |
Prazepam (JP19/USAN/INN); Centrax (TN) |
(P) unclassified |
| D00474 |
Primidone (JP19/USP/INN); Mysoline (TN) |
(P) unclassified |
| D00479 |
Prochlorperazine maleate (JP19/USP); Compazine (TN) |
(P) unclassified |
| D00482 |
Propoxyphene hydrochloride (USAN); Dextropropoxyphene hydrochloride; Darvon (TN) |
(P) unclassified |
| D00484 |
Protriptyline hydrochloride (USP); Vivactil (TN) |
(P) unclassified |
| D00493 |
Prochlorperazine (JAN/USP/INN); Compro (TN) |
(P) unclassified |
| D00495 |
Paramethadione (INN); Paradione (TN) |
(P) unclassified |
| D00498 |
Pentazocine (JP19/USP/INN); Fortral (TN) |
(P) Target: OPRK1 |
| D00499 |
Pentobarbital (USP/INN); Nembutal (TN) |
(P) unclassified |
| D00500 |
Pentobarbital sodium (JAN/USP); Nembutal sodium (TN) |
(P) unclassified |
| D00503 |
Perphenazine (JP19/USP/INN); Trilafon (TN) |
(P) unclassified |
| D00504 |
Phenacemide (JAN/INN); Phenurone (TN) |
(P) unclassified |
| D00505 |
Phenelzine sulfate (USP); Nardil (TN) |
(P) unclassified |
| D00506 |
Phenobarbital (JP19/USP/INN); Luminal (TN) |
(P) unclassified |
| D00508 |
Phensuximide (USP/INN); Milontin (TN) |
(P) unclassified |
| D00512 |
Phenytoin (JP19/USP/INN); Dilantin (TN) |
(P) unclassified |
| D00514 |
Dexmedetomidine (USAN/INN); Dexdor (TN); Precedex (TN) |
(P) unclassified |
| D00530 |
Zaleplon (JAN/USP/INN); Sonata (TN) |
(P) Enzyme: CYP3A4 |
| D00531 |
Nitrazepam (JP19/USAN/INN); Benzalin (TN); Nitrazepam (TN) |
(P) unclassified |
| D00532 |
Glutethimide (JAN/INN); Doriden (TN) |
(P) unclassified |
| D00533 |
Oxcarbazepine (JAN/USP/INN); Oxtellar (TN); Trileptal (TN) |
(P) unclassified |
| D00535 |
Vigabatrin (JAN/USP/INN); Sabril (TN) |
(P) unclassified |
| D00536 |
Felbamate (USPINN); Felbatol (TN) |
(P) unclassified |
| D00537 |
Topiramate (JAN/USP/INN); Topamax (TN); Trokendi xr (TN) |
(P) Enzyme: CYP3A4 |
| D00538 |
Zonisamide (JP19/USP/INN); Excegran (TN) |
(P) unclassified |
| D00539 |
Ethosuximide (JP19/USP/INN); Zarontin (TN) |
(P) Enzyme: CYP3A4 |
| D00550 |
Midazolam (JAN/USP/INN); Dormicum (TN); Buccolam (TN); Nayzilam (TN) |
(P) Enzyme: CYP3A4 |
| D00554 |
Ethinyl estradiol (USP); Ethinylestradiol (JP19/INN); Estinyl (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D00555 |
Amobarbital (JP19/INN); Isomytal (TN) |
(P) unclassified |
| D00557 |
Methaqualone (JAN/USAN/INN) |
(P) unclassified |
| D00560 |
Pimozide (JP19/USP/INN); Orap (TN) |
(P) Enzyme: CYP3A4 |
| D00561 |
Sertindole (USAN/INN); SerLect (TN) |
(P) unclassified |
| D00563 |
Mirtazapine (JAN/USP/INN); Remeron (TN); Reflex (TN) |
(P) Enzyme: CYP3A4 |
| D00619 |
Verapamil hydrochloride (JP19/USP); Calan (TN); Covera-hs (TN); Vasolan (TN); Verelan (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D00636 |
Amiodarone hydrochloride (JP19/USP); Ancaron (TN); Cordarone (TN); Nexterone (TN) |
(P) Enzyme: CYP3A4 |
| D00672 |
Hydroxyzine hydrochloride (JP19/USP); Hydroxyzine dihydrochloride; Atarax (TN); Vistaril (TN) |
(P) unclassified |
| D00693 |
Chlordiazepoxide hydrochloride (JAN/USP); Librium (TN) |
(P) unclassified |
| D00694 |
Clorazepate dipotassium (JP19/USP); Tranxene (TN) |
(P) unclassified |
| D00695 |
Flurazepam hydrochloride (USP); Flurazepam dihydrochloride; Dalmane (TN) |
(P) unclassified |
| D00696 |
Midazolam hydrochloride (USAN); Versed (TN) |
(P) Enzyme: CYP3A4 |
| D00698 |
Aprobarbital (INN); Alurate (TN) |
(P) unclassified |
| D00700 |
Mephobarbital (JAN/USP); Methylphenobarbital (INN); Mebaral (TN) |
(P) unclassified |
| D00701 |
Phenobarbital sodium (JAN/USP/INN); Luminal sodium (TN) |
(P) unclassified |
| D00702 |
Buspirone hydrochloride (USP); Buspar (TN) |
(P) unclassified |
| D00704 |
Ethchlorvynol (JAN/USP/INN); Placidyl (TN) |
(P) unclassified |
| D00705 |
Paraldehyde (USP); Paral (TN) |
(P) unclassified |
| D00706 |
Zolpidem tartrate (JP19/USP); Ambien (TN); Intermezzo (TN) |
(P) Enzyme: CYP3A4 |
| D00707 |
Fomepizole (JAN/USAN/INN); Antizol (TN) |
(P) CYP inhibition: CYP3A4 |
| D00708 |
Ethotoin (JAN/USP/INN); Accenon (TN); Peganone (TN) |
(P) unclassified |
| D00709 |
Levetiracetam (JP19/USP/INN); Keppra (TN); E keppra (TN) |
(P) unclassified |
| D00710 |
Valproate sodium (USAN); Sodium valproate (JP19); Depakene (TN); Selenica (TN) |
(P) unclassified |
| D00712 |
Methohexital sodium (USP); Brevital sodium (TN) |
(P) unclassified |
| D00714 |
Thiopental sodium (JP19/USP/INN); Pentothal (TN) |
(P) unclassified |
| D00753 |
Sirolimus (JAN/USAN/INN); Rapamune (TN); Rapamycin (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D00780 |
Bromocriptine mesylate (USP); Bromocriptine mesilate (JP19); Parlodel (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D00788 |
Acetophenazine maleate (USAN); Tindal (TN) |
(P) unclassified |
| D00789 |
Chlorpromazine hydrochloride (JP19/USP); Sonazine (TN) |
(P) unclassified |
| D00790 |
Chlorprothixene (JAN/USAN/INN); Taractan (TN) |
(P) unclassified |
| D00791 |
Fluphenazine hydrochloride (JAN/USP); Prolixin (TN) |
(P) unclassified |
| D00792 |
Fluphenazine enanthate (JP19/USP); Prolixin enanthate (TN) |
(P) unclassified |
| D00793 |
Fluphenazine decanoate (JAN/USP); Prolixin decanoate (TN) |
(P) unclassified |
| D00794 |
Loxapine succinate (USP); Loxitane (TN) |
(P) Enzyme: CYP3A4 |
| D00795 |
Mesoridazine besylate (USP); Serentil (TN) |
(P) unclassified |
| D00796 |
Molindone hydrochloride (USP); Moban (TN) |
(P) unclassified |
| D00797 |
Promazine hydrochloride (USP); Sparine (TN) |
(P) unclassified |
| D00798 |
Thioridazine hydrochloride (JP19/USP); Mellaril (TN) |
(P) unclassified |
| D00799 |
Trifluoperazine hydrochloride (JAN/USP); Stelazine (TN) |
(P) unclassified |
| D00800 |
Triflupromazine hydrochloride (JAN/USP); Vesprin (TN) |
(P) unclassified |
| D00801 |
Lithium carbonate (JP19/USP); Eskalith (TN); Lithobid (TN) |
(P) unclassified |
| D00809 |
Amitriptyline hydrochloride (JP19/USP); Elavil (TN) |
(P) Enzyme: CYP3A4 |
| D00811 |
Clomipramine hydrochloride (JP19/USP); Anafranil (TN) |
(P) Enzyme: CYP3A4 |
| D00812 |
Desipramine hydrochloride (JAN/USP); Norpramin (TN) |
(P) unclassified |
| D00814 |
Doxepin hydrochloride (USP); Sinequan (TN); Zonalon (TN) |
(P) unclassified |
| D00815 |
Imipramine hydrochloride (JP19/USP); Tofranil (TN) |
(P) Enzyme: CYP3A4 |
| D00816 |
Nortriptyline hydrochloride (JP19/USP/INN); Pamelor (TN) |
(P) unclassified |
| D00817 |
Bupropion hydrochloride (JAN/USP); Wellbutrin (TN); Zyban (TN) |
(P) unclassified |
| D00818 |
Maprotiline hydrochloride (JP19/USP); Ludiomil (TN) |
(P) unclassified |
| D00819 |
Nefazodone hydrochloride (USP); Serzone (TN) |
(P) unclassified |
| D00820 |
Trazodone hydrochloride (JAN/USP); Desyrel (TN) |
(P) Enzyme: CYP3A4 |
| D00821 |
Venlafaxine hydrochloride (JAN/USP); Effexor (TN) |
(P) unclassified |
| D00822 |
Citalopram hydrobromide (USP); Celexa (TN) |
(P) Enzyme: CYP3A4 |
| D00823 |
Fluoxetine hydrochloride (JAN/USP); Prozac (TN); Sarafem (TN) |
(P) unclassified |
| D00824 |
Fluvoxamine maleate (JP19/USP); Luvox (TN) |
(P) CYP inhibition: CYP3A4 |
| D00825 |
Sertraline hydrochloride (JAN/USP); Zoloft (TN) |
(P) Enzyme: CYP3A4 |
| D00826 |
Tranylcypromine sulfate (USP); Parnate (TN) |
(P) unclassified |
| D00831 |
Mefloquine hydrochloride (JP19/USP); Lariam (TN) |
(P) unclassified |
| D00835 |
Alfentanil hydrochloride (USP); Alfenta (TN) |
(P) unclassified |
| D00836 |
Buprenorphine hydrochloride (JP19/USP); Buprenex (TN) |
(P) Enzyme: CYP3A4 / Target: OPRK1 |
| D00837 |
Butorphanol tartrate (JAN/USP); Stadol (TN) |
(P) Target: OPRK1 |
| D00838 |
Dezocine (USAN); Dalgan (TN) |
(P) Target: OPRK1 |
| D00839 |
Hydromorphone hydrochloride (JAN/USP); Dilaudid (TN); Exalgo (TN); Palladone (TN) |
(P) unclassified |
| D00840 |
Levomethadyl acetate hydrochloride (USAN); Orlaam (TN) |
(P) Enzyme: CYP3A4 |
| D00841 |
Levorphanol tartrate (USP); Levorphanol tartrate dihydrate; Levo-dromoran (TN) |
(P) unclassified |
| D00842 |
Morphine sulfate (USP); Morphine sulfate hydrate (JP19); Morphine sulfate pentahydrate; Astramor PH (TN); Avinza (TN); Depodur (TN); Kadian (TN); MS contin (TN) |
(P) unclassified |
| D00843 |
Nalbuphine hydrochloride (USAN); Nubain (TN) |
(P) Target: OPRK1 |
| D00844 |
Oxymorphone hydrochloride (USP); Numorphan (TN); Opana (TN) |
(P) unclassified |
| D00845 |
Sufentanil citrate (USP); Dsuvia (TN); Sufenta (TN) |
(P) unclassified |
| D00847 |
Oxycodone hydrochloride (USP); Oxecta (TN); Oxycontin (TN); Roxicodone (TN) |
(P) Enzyme: CYP3A4 / Target: OPRK1 |
| D00854 |
Quinupristin and dalfopristin; Synercid (TN) |
(P) CYP inhibition: CYP3A4 |
| D00897 |
Indinavir sulfate (USP); Crixivan (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D00899 |
Nelfinavir mesylate (USAN/INN); Nelfinavir mesilate (JAN); Viracept (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D00960 |
Anastrozole (JP19/USP/INN); Arimidex (TN) |
(P) CYP inhibition: CYP3A4 |
| D00961 |
Bicalutamide (JP19/USP/INN); Casodex (TN) |
(P) CYP inhibition: CYP3A4 |
| D01044 |
Flupentixol (INN); Flupenthixol; Depixol (TN) |
(P) unclassified |
| D01071 |
Hexobarbital (JAN/INN) |
(P) unclassified |
| D01096 |
Hydroxyzine pamoate (JP19/USP); Atarax-P (TN); Vistaril pamoate (TN) |
(P) unclassified |
| D01101 |
Bromperidol (JAN/USAN/INN); Impromen (TN) |
(P) Enzyme: CYP3A4 |
| D01105 |
Moperone hydrochloride (JAN); Luvatren (TN) |
(P) unclassified |
| D01107 |
Milnacipran hydrochloride (JAN/USAN); Savella (TN); Toledomin (TN) |
(P) unclassified |
| D01110 |
Melitracen hydrochloride (JAN/USAN) |
(P) unclassified |
| D01150 |
Methyprylon (JAN/INN); Noludar (TN) |
(P) unclassified |
| D01164 |
Aripiprazole (JP19/USP/INN); Abilify (TN) |
(P) Enzyme: CYP3A4 |
| D01177 |
Remifentanil hydrochloride (JAN/USAN); Ultiva (TN) |
(P) unclassified |
| D01179 |
Duloxetine hydrochloride (JAN/USP); Cymbalta (TN); Yentreve (TN) |
(P) unclassified |
| D01190 |
Ethylphenacemide (JAN); Pheneturide (INN) |
(P) unclassified |
| D01205 |
Dexmedetomidine hydrochloride (JAN/USP); Igalmi (TN); Precedex (TN) |
(P) unclassified |
| D01219 |
Oxypertine (JAN/USAN/INN); Forit (TN) |
(P) unclassified |
| D01226 |
Sulpiride (JP19/USAN/INN); Dogmatyl (TN) |
(P) unclassified |
| D01230 |
Flunitrazepam (JP19/USAN/INN); Rohypnol (TN) |
(P) unclassified |
| D01235 |
Josamycin (JP19/USAN/INN); Leucomycin A3; JM |
(P) CYP inhibition: CYP3A4 |
| D01245 |
Bromazepam (JP19/USAN/INN); Lectopam (TN) |
(P) unclassified |
| D01253 |
Clobazam (JAN/USAN/INN); Mystan (TN); Onfi (TN) |
(P) Enzyme: CYP3A4 |
| D01254 |
Tofisopam (JP19/INN); Emandaxin (TN) |
(P) unclassified |
| D01268 |
Cloxazolam (JP19/INN); Sepazon (TN) |
(P) unclassified |
| D01276 |
Atazanavir sulfate (JAN/USAN); Reyataz (TN) |
(P) CYP inhibition: CYP3A4 |
| D01285 |
Lofepramine hydrochloride (JAN/USAN); Amplit (TN) |
(P) unclassified |
| D01292 |
Medazepam (JP19/INN); Pamnace (TN) |
(P) unclassified |
| D01293 |
Ethyl loflazepate (JP19/INN); Meilax (TN) |
(P) Enzyme: CYP3A4 |
| D01310 |
Secobarbital sodium (JAN/USP); Seconal sodium (TN) |
(P) unclassified |
| D01314 |
Dibenzepin hydrochloride (JAN/USAN) |
(P) unclassified |
| D01316 |
Mexazolam (JAN/INN); Melex (TN) |
(P) Enzyme: CYP3A4 |
| D01321 |
Zotepine (JAN/INN); Setous (TN) |
(P) unclassified |
| D01322 |
Troleandomycin (USAN/INN); Triacetyloleandomycin (JAN); TAO; Tao (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D01328 |
Clotiazepam (JP19/INN); Rize (TN) |
(P) unclassified |
| D01339 |
Midecamycin (JP19/INN); Medemycin (TN) |
(P) CYP inhibition: CYP3A4 |
| D01354 |
Fludiazepam (JP19/INN); Erispan (TN) |
(P) unclassified |
| D01355 |
Tramadol hydrochloride (JP19/USP); Ultram (TN) |
(P) Enzyme: CYP3A4 |
| D01358 |
Mianserin hydrochloride (JAN/USAN); Tetramide (TN) |
(P) Enzyme: CYP3A4 |
| D01372 |
Zopiclone (JP19/INN); Amoban (TN) |
(P) Enzyme: CYP3A4 |
| D01382 |
Metharbital (JAN/INN); Gemonil (TN) |
(P) unclassified |
| D01383 |
Meperidine hydrochloride (USP); Pethidine hydrochloride (JP19); Demerol (TN) |
(P) unclassified |
| D01391 |
Bromovalerylurea (JP19); Bromisoval (INN); Bromisovalum; Bromural (TN); Brovarin (TN) |
(P) unclassified |
| D01399 |
Fentanyl citrate (JP19/USP); Abstral (TN); Fentora (TN); Lazanda (TN); Oralet (TN) |
(P) Enzyme: CYP3A4 |
| D01408 |
Flurazepam hydrochloride (JP19); Flurazepam monohydrochloride; Dalmate (TN) |
(P) unclassified |
| D01412 |
Perazine maleate (JAN) |
(P) unclassified |
| D01429 |
Fosfluconazole (JAN/INN); Prodif (TN) |
(P) CYP inhibition: CYP3A4 |
| D01447 |
Thioproperazine mesilate (JAN); Thioproperazine mesylate |
(P) unclassified |
| D01448 |
Trifluoperazine maleate (JAN) |
(P) unclassified |
| D01477 |
Opipramol hydrochloride (JAN/USAN); Insidon (TN) |
(P) unclassified |
| D01481 |
Dihydrocodeine phosphate (JP19); Dihydro (TN) |
(P) unclassified |
| D01482 |
Pipamperone hydrochloride (JAN) |
(P) unclassified |
| D01485 |
Propericiazine (JAN); Periciazine; Neuleptil (TN) |
(P) unclassified |
| D01514 |
Etizolam (JP19/INN); Sedekopan (TN) |
(P) Enzyme: CYP3A4 |
| D01520 |
Levomepromazine hydrochloride (JAN/USAN); Nozinan (TN) |
(P) unclassified |
| D01522 |
Tiapride hydrochloride (JP19); Gramalil (TN) |
(P) unclassified |
| D01546 |
Dothiepin hydrochloride (USAN); Dosulepin hydrochloride (JAN); Prothiaden (TN) |
(P) unclassified |
| D01548 |
Mosapramine hydrochloride (JAN); Cremin (TN) |
(P) unclassified |
| D01593 |
Nimetazepam (JAN/INN); Erimin (TN) |
(P) unclassified |
| D01597 |
Clothiapine (USAN); Clotiapine (JAN/INN); Entumin (TN) |
(P) unclassified |
| D01636 |
Midecamycin acetate (JP19); Miocamycin; Miocamycin (TN) |
(P) CYP inhibition: CYP3A4 |
| D01657 |
Lormetazepam (JAN/USAN/INN); Loramet (TN) |
(P) unclassified |
| D01740 |
Barbital (JP19/INN) |
(P) unclassified |
| D01744 |
Brotizolam (JP19/USAN/INN); Lendormin (TN) |
(P) Enzyme: CYP3A4 |
| D01787 |
Sulthiame (USAN); Sultiame (JP19); Ospolot (TN) |
(P) unclassified |
| D01793 |
Bifemelane hydrochloride (JAN) |
(P) unclassified |
| D01807 |
Mebutamate (JAN/USAN); Capla (TN); Dormate (TN) |
(P) unclassified |
| D01860 |
Perazine dimalonate (JAN) |
(P) unclassified |
| D01879 |
Eptazocine hydrobromide (JAN); Sedapain (TN) |
(P) Target: OPRK1 |
| D01898 |
Haloperidol decanoate (JAN/USP); Halomonth (TN) |
(P) Enzyme: CYP3A4 |
| D01939 |
Ziprasidone hydrochloride (USP); Ziprasidone hydrochloride hydrate (JAN); Geodon (TN) |
(P) unclassified |
| D01980 |
Luliconazole (JAN/USAN/INN); Lulicon (TN); Luzu (TN) |
(P) CYP inhibition: CYP3A4 |
| D02022 |
Prochlorperazine mesilate (JAN); Prochlorperazine dimethanesulfonate; Novamin (TN) |
(P) unclassified |
| D02037 |
Perphenazine maleate (JP19); PZC (TN) |
(P) unclassified |
| D02071 |
Scopolamine hydrobromide (USP); Scopolamine hydrobromide hydrate (JP19); Scopolamine hydrobromide trihydrate; Hysco (TN); Isopto hyoscine (TN) |
(P) unclassified |
| D02096 |
Fosphenytoin sodium (USP); Cerebyx (TN); Sesquient (TN) |
(P) CYP induction: CYP3A4 |
| D02097 |
Tiagabine hydrochloride (USP); Gabitril (TN) |
(P) unclassified |
| D02100 |
Ziprasidone mesylate (USAN); Ziprasidone mesylate hydrate; Geodon (TN) |
(P) unclassified |
| D02101 |
Codeine phosphate (USP); Codeine phosphate hydrate (JP19) |
(P) unclassified |
| D02102 |
Methadone hydrochloride (JAN/USP); Dolophine hydrochloride (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
| D02103 |
Phenytoin sodium (USP); Phenytoin sodium for injection (JP19); Aleviatin (TN); Dilantin (TN) |
(P) unclassified |
| D02111 |
Pentazocine lactate (USP); Talwin (TN) |
(P) Target: OPRK1 |
| D02162 |
Chlorprothixene hydrochloride (JAN) |
(P) unclassified |
| D02163 |
Fluphenazine maleate (JAN); Flumezin (TN) |
(P) unclassified |
| D02175 |
Compound oxycodone (JP19); Pavinal (TN) |
(P) Enzyme: CYP3A4 |
| D02208 |
Sultopride hydrochloride (JAN); Sultopride monohydrochloride; Barnetil (TN) |
(P) unclassified |
| D02227 |
Pentazocine hydrochloride (JAN/USP); Sosegon (TN); Talacen (TN) |
(P) Target: OPRK1 |
| D02236 |
Flupentixol dihydrochloride (JAN) |
(P) unclassified |
| D02248 |
Levomepromazine maleate (JP19/USAN); Hirnamin (TN) |
(P) unclassified |
| D02252 |
Amobarbital sodium (JAN/USP); Amytal sodium (TN) |
(P) unclassified |
| D02253 |
Pentobarbital calcium (JP19); Ravona (TN) |
(P) unclassified |
| D02260 |
Paroxetine hydrochloride hemihydrate (USP); Paroxetine hydrochloride hydrate (JP19); Paxil (TN) |
(P) unclassified |
| D02271 |
Morphine hydrochloride hydrate (JP19); Morphine hydrochloride trihydrate; Anpec (TN) |
(P) unclassified |
| D02340 |
Loxapine (USAN/INN); Adasuve (TN) |
(P) Enzyme: CYP3A4 |
| D02356 |
Verapamil (USAN/INN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D02360 |
Sertraline (INN) |
(P) Enzyme: CYP3A4 |
| D02361 |
Propiomazine (USAN/INN) |
(P) unclassified |
| D02362 |
Paroxetine (USP/INN) |
(P) unclassified |
| D02372 |
Perospirone hydrochloride hydrate (JP19); Lullan (TN) |
(P) unclassified |
| D02408 |
Trimipramine maleate (JAN/USP); Surmontil (TN) |
(P) unclassified |
| D02484 |
Artemether and lumefantrine; Coartem (TN) |
(P) unclassified |
| D02497 |
Fosamprenavir (INN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D02555 |
Posaconazole (JAN/USAN/INN); Noxafil (TN) |
(P) CYP inhibition: CYP3A4 |
| D02559 |
Toloxatone (INN); Humoryl (TN) |
(P) unclassified |
| D02561 |
Moclobemide (USAN/INN); Aurorix (TN) |
(P) unclassified |
| D02565 |
Dimetacrine (INN) |
(P) unclassified |
| D02566 |
Maprotiline (USAN) |
(P) unclassified |
| D02567 |
Escitalopram oxalate (JAN/USP); Lexapro (TN) |
(P) Enzyme: CYP3A4 |
| D02570 |
Desvenlafaxine succinate (USAN); Desvenlafaxine succinate hydrate (JAN); Desvenlafaxine succinate monohydrate; Pristiq (TN) |
(P) Enzyme: CYP3A4 |
| D02572 |
Viloxazine hydrochloride (USAN); Qelbree (TN); Vivalan (TN) |
(P) unclassified |
| D02573 |
Reboxetine mesylate (USAN); Reboxetine mesilate; Vestra (TN) |
(P) unclassified |
| D02575 |
Tianeptine (INN); Stablon (TN) |
(P) unclassified |
| D02578 |
Agomelatine (INN); Valdoxan (TN) |
(P) unclassified |
| D02579 |
Iproniazid (INN) |
(P) unclassified |
| D02580 |
Isocarboxazid (INN); Marplan (TN) |
(P) unclassified |
| D02604 |
Acepromazine maleate (USP) |
(P) unclassified |
| D02608 |
Perazine fendizoate (JAN) |
(P) unclassified |
| D02609 |
Prochlorperazine edisylate (USP); Compazine syrup (TN) |
(P) unclassified |
| D02611 |
Phenoperidine (INN) |
(P) unclassified |
| D02612 |
Thiothixene hydrochloride (USP); Thiothixene dihydrochloride dihydrate; Tiotixene dihydrochloride |
(P) unclassified |
| D02613 |
Clopenthixol (USAN) |
(P) unclassified |
| D02615 |
Chlorpromazine hydrochloride, promethazine hydrochloride and phenobarbital; Vegetamin (TN) |
(P) unclassified |
| D02618 |
Butobarbital (BAN); Butethal; Neonal (TN) |
(P) unclassified |
| D02619 |
Carbromal (INN); Adalin (TN) |
(P) unclassified |
| D02621 |
Fluanisone (INN) |
(P) unclassified |
| D02622 |
Pipamperone (USAN/INN); Floropipamide |
(P) unclassified |
| D02623 |
Moperone (INN) |
(P) unclassified |
| D02624 |
Eszopiclone (JAN/USP/INN); Estorra (TN); Lunesta (TN) |
(P) Enzyme: CYP3A4 |
| D02625 |
Trifluperidol (USAN/INN); Triperidol (TN) |
(P) unclassified |
| D02626 |
Bromperidol decanoate (USAN) |
(P) Enzyme: CYP3A4 |
| D02627 |
Benperidol (USAN/INN); Anquil (TN) |
(P) unclassified |
| D02629 |
Fluspirilene (USAN/INN); Imap (TN) |
(P) unclassified |
| D02630 |
Penfluridol (USAN/INN); Semap (TN) |
(P) unclassified |
| D02642 |
Butaperazine (USAN) |
(P) unclassified |
| D02643 |
Butaperazine maleate (USAN) |
(P) unclassified |
| D02666 |
Iloperidone (USAN/INN); Fanapt (TN) |
(P) Enzyme: CYP3A4 |
| D02671 |
Mesoridazine (USAN/INN); Lidanar (TN) |
(P) unclassified |
| D02680 |
Pipotiazine palmitate (USAN); Piportil depot (TN) |
(P) unclassified |
| D02682 |
Remoxipride (USAN) |
(P) unclassified |
| D02683 |
Remoxipride hydrochloride (USAN) |
(P) unclassified |
| D02689 |
Ramelteon (JAN/USAN/INN); Rozerem (TN) |
(P) unclassified |
| D02691 |
Somatropin (USP/INN); Somatropin (genetical recombination) (JAN); Human growth hormone (JAN); Asellacrin (TN); Humatrope (TN); Nutropin (TN); Omnitrope (TN) |
(P) unclassified |
| D02717 |
Valnoctamide (USAN/INN); Axiquel (TN) |
(P) unclassified |
| D02732 |
Pranlukast hydrate (JP19); Onon (TN) |
(P) Enzyme: CYP3A4 |
| D02766 |
Valpromide (INN); Depamide (TN) |
(P) unclassified |
| D02770 |
Adinazolam (USAN/INN) |
(P) unclassified |
| D02771 |
Adinazolam mesylate (USAN) |
(P) unclassified |
| D02787 |
Alaproclate (USAN/INN) |
(P) unclassified |
| D02817 |
Allobarbital (USAN/INN) |
(P) unclassified |
| D02861 |
Indinavir sulfate ethanolate (JAN); Crixivan (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D02867 |
Fosamprenavir calcium hydrate (JAN); Lexiva (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D02941 |
Anileridine (USP/INN) |
(P) unclassified |
| D02942 |
Anileridine hydrochloride (USP); Leritine (TN) |
(P) unclassified |
| D02968 |
Aprepitant (JAN/USP/INN); Aponvie (TN); Emend (TN); Cinvanti (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4 |
| D02995 |
Asenapine maleate (JAN/USAN); Saphris (TN) |
(P) unclassified |
| D03083 |
Bentazepam (USAN/INN) |
(P) unclassified |
| D03089 |
Benzoctamine hydrochloride (USAN) |
(P) unclassified |
| D03106 |
Bexarotene (JAN/USAN/INN); Targretin (TN) |
(P) unclassified |
| D03156 |
Brifentanil hydrochloride (USAN) |
(P) unclassified |
| D03165 |
Bromocriptine (USAN/INN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D03197 |
Butorphanol (USAN/INN) |
(P) Target: OPRK1 |
| D03199 |
Butriptyline hydrochloride (USAN) |
(P) unclassified |
| D03274 |
Chlorpromazine hibenzate (JAN); Contomin (TN) |
(P) unclassified |
| D03405 |
Carfentanil citrate (USAN) |
(P) unclassified |
| D03444 |
Opium (USP); Opium, powdered (JP19); Diluted opium powder (JP19) |
(P) unclassified |
| D03445 |
Opium alkaloids hydrochlorides (JP19); Pan opin (TN) |
(P) unclassified |
| D03503 |
Cimetidine hydrochloride (USP) |
(P) CYP inhibition: CYP3A4 |
| D03556 |
Zuclopenthixol (INN); Clopixol (TN) |
(P) unclassified |
| D03562 |
Clorazepate monopotassium (USAN) |
(P) unclassified |
| D03579 |
Codeine polistirex (USAN) |
(P) unclassified |
| D03580 |
Codeine sulfate (USP); Codeine sulfate trihydrate |
(P) unclassified |
| D03618 |
Cyclazocine (USAN/INN) |
(P) Target: OPRK1 |
| D03656 |
Darunavir (USAN/INN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D03658 |
Dasatinib (JAN/INN) |
(P) Enzyme: CYP3A4 |
| D03669 |
Deferasirox (JAN/USAN/INN); Exjade (TN); Jadenu (TN) |
(P) CYP induction: CYP3A4 |
| D03783 |
Oxycodone terephthalate (USP) |
(P) Enzyme: CYP3A4 / Target: OPRK1 |
| D03785 |
Dichloralphenazone (USP) |
(P) unclassified |
| D03825 |
Dihydrocodeine bitartrate (USP) |
(P) unclassified |
| D03833 |
Indinavir (USAN); Indinavir hydrate |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D03835 |
Fosamprenavir calcium (USAN); Lexiva (TN); Telzir (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D03837 |
Fosamprenavir sodium (USAN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D03844 |
Phenytoin, phenobarbital and caffeine and sodium benzoate; Hydantol F (TN) |
(P) unclassified |
| D03852 |
Droperidol and fentanyl citrate; Innovar (TN) |
(P) Enzyme: CYP3A4 |
| D03855 |
Pethidine hydrochloride and levallorphan tartrate; Pethilorfan (TN) |
(P) unclassified |
| D03863 |
Opium alkaloids and atropine (JP19); Opium alkaloids hydrochloride and atropine sulfate hydrate; Opiato (TN) |
(P) unclassified |
| D03866 |
Opium alkaloids and scopolamine (JP19); Weak opium alkaloids and scopolamine (JP19); Opium alkaloids hydrochloride and scopolamine hydrobromide hydrate; Opisco (TN) |
(P) unclassified |
| D03975 |
Allylisopropylacetylurea; Apronal; Apronalide |
(P) unclassified |
| D04024 |
Lapatinib ditosylate (USAN); Lapatinib tosilate hydrate (JAN); Lapatinib ditosylate monohydrate; Tykerb (TN); Tyverb (TN) |
(P) Enzyme: CYP3A4 |
| D04034 |
Chlorpromazine phenolphthalinate (JAN); Wintermin (TN) |
(P) unclassified |
| D04038 |
Perphenazine fendizoate (JAN); PZC (TN) |
(P) unclassified |
| D04105 |
Etoperidone hydrochloride (USAN); Etonin (TN) |
(P) unclassified |
| D04148 |
Fenfluramine hydrochloride (JAN/USAN); Fintepla (TN); Pondimin (TN) |
(P) Enzyme: CYP3A4 |
| D04300 |
Ganaxolone (USAN/INN); Ztalmy (TN) |
(P) Enzyme: CYP3A4 |
| D04314 |
Gepirone hydrochloride (USAN); Exxua (TN) |
(P) Enzyme: CYP3A4 |
| D04605 |
Iprindole (USAN/INN) |
(P) unclassified |
| D04641 |
Istradefylline (JAN/USAN/INN); Nourianz (TN); Nouriast (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D04649 |
Ketazocine (USAN/INN); Ketocyclazocine |
(P) Target: OPRK1 |
| D04650 |
Ketazolam (USAN/INN) |
(P) unclassified |
| D04666 |
Lanreotide acetate (JAN/USAN); Somatuline (TN) |
(P) unclassified |
| D04716 |
Levomethadyl acetate (USAN); Levacetylmethadol (INN) |
(P) Enzyme: CYP3A4 |
| D04749 |
Lithium citrate (USP); Lithonate (TN) |
(P) unclassified |
| D04750 |
Lithium hydroxide (USP) |
(P) unclassified |
| D04764 |
Lofentanil oxalate (USAN) |
(P) unclassified |
| D04820 |
Lurasidone hydrochloride (JAN/USAN); SM 13496; Latuda (TN) |
(P) Enzyme: CYP3A4 |
| D04882 |
Medazepam hydrochloride (USAN); Nobrium (TN) |
(P) unclassified |
| D04924 |
Meptazinol hydrochloride (USAN) |
(P) unclassified |
| D04965 |
Perphenazine hydrochloride; Perphenazine dihydrochloride; PZC (TN) |
(P) unclassified |
| D04973 |
Methadyl acetate (USAN); Acetylmethadol (INN) |
(P) unclassified |
| D04985 |
Methohexital (USP/INN) |
(P) unclassified |
| D05028 |
Midazolam maleate (USAN) |
(P) Enzyme: CYP3A4 |
| D05039 |
Minaprine (USAN/INN); Cantor (TN) |
(P) unclassified |
| D05040 |
Minaprine hydrochloride (USAN) |
(P) unclassified |
| D05048 |
Mirfentanil hydrochloride (USAN) |
(P) unclassified |
| D05154 |
Nexeridine hydrochloride (USAN) |
(P) unclassified |
| D05200 |
Nomifensine maleate (USAN); Merital (TN) |
(P) unclassified |
| D05217 |
Ocfentanil hydrochloride (USAN) |
(P) unclassified |
| D05312 |
Oxycodone (USAN/INN) |
(P) Enzyme: CYP3A4 / Target: OPRK1 |
| D05339 |
Paliperidone (JAN/USP/INN); Invega (TN) |
(P) unclassified |
| D05340 |
Paliperidone palmitate (JAN/USAN); Xeplion (TN); Trevicta (TN); Invega sustenna (TN); Invega trinza (TN) |
(P) unclassified |
| D05351 |
Josamycin propionate (JP19); Josamy (TN) |
(P) CYP inhibition: CYP3A4 |
| D05374 |
Paroxetine hydrochloride (USP); Paxil (TN) |
(P) unclassified |
| D05375 |
Paroxetine mesylate (USAN); Brisdelle (TN); Pexeva (TN) |
(P) unclassified |
| D05462 |
Oxycodone hydrochloride hydrate (JP19) |
(P) Enzyme: CYP3A4 / Target: OPRK1 |
| D05621 |
Progabide (USAN/INN); Gabren (TN) |
(P) unclassified |
| D05632 |
Propoxyphene napsylate (USAN); Darvon-N (TN) |
(P) unclassified |
| D05775 |
Rufinamide (JAN/USP/INN); Banzel (TN) |
(P) unclassified |
| D05928 |
Stiripentol (JAN/USAN/INN); Diacomit (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D05938 |
Sufentanil (USAN/INN) |
(P) unclassified |
| D06007 |
Tapentadol (USAN/INN) |
(P) unclassified |
| D06147 |
Tilidine hydrochloride (USAN); Valoron (TN) |
(P) unclassified |
| D06208 |
Trefentanil hydrochloride (USAN) |
(P) unclassified |
| D06268 |
Trimeperidine (INN) |
(P) unclassified |
| D06342 |
Xorphanol mesylate (USAN) |
(P) Target: OPRK1 |
| D06367 |
Zimeldine hydrochloride (USAN); Zimeldine hydrochloride hydrate |
(P) unclassified |
| D06413 |
Nilotinib hydrochloride hydrate (JAN); Nilotinib monohydrochloride monohydrate; Tasigna (TN) |
(P) Enzyme: CYP3A4 |
| D06414 |
Dasatinib (USAN); Dasatinib hydrate (JAN); Sprycel (TN) |
(P) Enzyme: CYP3A4 |
| D06478 |
Darunavir ethanolate (JAN); Prezista (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D06499 |
Opium tincture (JP19) |
(P) unclassified |
| D06573 |
Carisbamate (USAN) |
(P) unclassified |
| D06597 |
Fosaprepitant dimeglumine (USAN); Fosaprepitant meglumine (JAN); Proemend (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4 |
| D06623 |
Olanzapine pamoate (USAN); Olanzapine pamoate monohydrate; Zyprexa (TN) |
(P) unclassified |
| D06699 |
Japanese valerian (JP19); Powdered japanese valerian (JP19) |
(P) unclassified |
| D06887 |
Talbutal (INN); Lotusate (TN) |
(P) unclassified |
| D07065 |
Acepromazine (INN); Concentrat vo34 (TN) |
(P) unclassified |
| D07122 |
Alfentanil (INN); Rapifen (TN) |
(P) unclassified |
| D07132 |
Buprenorphine (JAN/INN); Temgesic (TN) |
(P) Enzyme: CYP3A4 / Target: OPRK1 |
| D07283 |
Esketamine (USAN/INN) |
(P) Enzyme: CYP3A4 |
| D07285 |
Nicomorphine (INN) |
(P) unclassified |
| D07286 |
Diamorphine (BAN); Heroin; Diacetylmorphine |
(P) unclassified |
| D07287 |
Dextromoramide (BAN) |
(P) unclassified |
| D07288 |
Piritramide (INN); Dipidolor (TN) |
(P) unclassified |
| D07289 |
Bezitramide (INN); Burgodin (TN) |
(P) unclassified |
| D07298 |
Barbexaclone (INN); Maliasin (TN) |
(P) unclassified |
| D07299 |
Lacosamide (JAN/USAN/INN); Erlosamide; Vimpat (TN) |
(P) Enzyme: CYP3A4 |
| D07300 |
Beclamide (INN) |
(P) unclassified |
| D07307 |
Cyamemazine (INN); Tercian (TN) |
(P) unclassified |
| D07308 |
Chlorproethazine (INN) |
(P) unclassified |
| D07309 |
Melperone (INN); Bunil (TN) |
(P) unclassified |
| D07310 |
Amisulpride (INN); Barhemsys (TN); Deniban (TN); Solian (TN) |
(P) unclassified |
| D07311 |
Veralipride (INN); Agreal (TN) |
(P) unclassified |
| D07312 |
Levosulpiride (INN); Levopraid (TN) |
(P) unclassified |
| D07313 |
Prothipendyl (INN) |
(P) unclassified |
| D07314 |
Pinazepam (INN); Domar (TN) |
(P) unclassified |
| D07315 |
Camazepam (INN) |
(P) unclassified |
| D07316 |
Captodiame (BAN) |
(P) unclassified |
| D07317 |
Emylcamate (INN) |
(P) unclassified |
| D07318 |
Mephenoxalone (INN); Dorsiflex (TN) |
(P) unclassified |
| D07319 |
Gedocarnil (INN) |
(P) unclassified |
| D07320 |
Etifoxine (INN/BAN) |
(P) unclassified |
| D07321 |
Vinylbital (INN); Vinylbitone |
(P) unclassified |
| D07322 |
Vinbarbital (INN) |
(P) unclassified |
| D07323 |
Cyclobarbital (INN) |
(P) unclassified |
| D07324 |
Proxibarbal (INN); Centralgol (TN) |
(P) unclassified |
| D07325 |
Chloralodol (INN); Chlorhexadol |
(P) unclassified |
| D07326 |
Loprazolam (INN); Dormonoct (TN) |
(P) unclassified |
| D07327 |
Doxefazepam (INN) |
(P) unclassified |
| D07328 |
Cinolazepam (INN); Gerodorm (TN) |
(P) unclassified |
| D07329 |
Pyrithyldione (INN) |
(P) unclassified |
| D07330 |
Clomethiazole (INN); Distraneurine (TN) |
(P) unclassified |
| D07331 |
Hexapropymate (INN); Merinax (TN) |
(P) unclassified |
| D07332 |
Methylpentynol (INN); Meparfynol; Methylparafynol; Atemorin (TN) |
(P) unclassified |
| D07333 |
Niaprazine (INN); Nopron (TN) |
(P) unclassified |
| D07335 |
Amineptine (INN); Survector (TN) |
(P) unclassified |
| D07336 |
Quinupramine (INN) |
(P) unclassified |
| D07337 |
Nialamide (INN); Niamid (TN) |
(P) unclassified |
| D07338 |
Iproclozide (INN) |
(P) unclassified |
| D07339 |
Oxitriptan (INN); Levothym (TN) |
(P) unclassified |
| D07340 |
Oxaflozane (INN) |
(P) unclassified |
| D07341 |
Medifoxamine (INN) |
(P) unclassified |
| D07342 |
Pivagabine (INN) |
(P) unclassified |
| D07435 |
Papaveretum (BAN); Omnopon (TN) |
(P) unclassified |
| D07448 |
Amitriptyline (INN); Laroxyl (TN) |
(P) Enzyme: CYP3A4 |
| D07471 |
Atazanavir (INN); Reyataz (TN) |
(P) CYP inhibition: CYP3A4 |
| D07528 |
Bifemelane (INN) |
(P) unclassified |
| D07583 |
Phenytoin and phenobarbital; Aleviatin with phenobarbital (TN) |
(P) unclassified |
| D07591 |
Bupropion (INN) |
(P) unclassified |
| D07593 |
Buspirone (INN); Gen-Buspirone (TN) |
(P) unclassified |
| D07595 |
Fosphenytoin sodium hydrate (JAN); Fostoin (TN) |
(P) CYP induction: CYP3A4 |
| D07601 |
Butriptyline (INN); Evadyne (TN) |
(P) unclassified |
| D07620 |
Carfentanil (INN) |
(P) unclassified |
| D07685 |
Chlorproethazine hydrochloride; Neuriplege (TN) |
(P) unclassified |
| D07686 |
Chlorprothixene acetate; Truxal (TN) |
(P) unclassified |
| D07687 |
Chlorprothixene citrate; Truxal (TN) |
(P) unclassified |
| D07704 |
Citalopram (USP/INN); Citadur (TN) |
(P) Enzyme: CYP3A4 |
| D07705 |
Citalopram hydrochloride; Seropram (TN) |
(P) Enzyme: CYP3A4 |
| D07710 |
Clarithromycin lactobionate; Klacid (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D07725 |
Clomethiazole edisilate; Heminevrin (TN) |
(P) unclassified |
| D07727 |
Clomipramine (INN); Anafranil (TN) |
(P) Enzyme: CYP3A4 |
| D07740 |
Codeine hydrochloride; Bisoltus (TN) |
(P) unclassified |
| D07756 |
Cyamemazine tartrate; Tercian (TN) |
(P) unclassified |
| D07757 |
Cyclobarbital calcium (BAN); Phanodorn calcium (TN) |
(P) unclassified |
| D07791 |
Desipramine (INN) |
(P) unclassified |
| D07793 |
Desvenlafaxine (INN); Khedezla (TN) |
(P) Enzyme: CYP3A4 |
| D07808 |
Dextromoramide tartrate; Palfium (TN) |
(P) unclassified |
| D07809 |
Dextropropoxyphene (INN); Propoxypene |
(P) unclassified |
| D07810 |
Diacetylmorphine hydrochloride; Diamorphine hydrochloride; Heroin hydrochloride |
(P) unclassified |
| D07812 |
Dibenzepin (INN) |
(P) unclassified |
| D07831 |
Dihydrocodeine (INN); Remedacen (TN) |
(P) unclassified |
| D07832 |
Dihydrocodeine thiocyanate; Paracodin (TN) |
(P) unclassified |
| D07865 |
Dixyrazine; Esucos (TN) |
(P) unclassified |
| D07872 |
Dosulepin (INN); Dothiepin; Dothep (TN) |
(P) unclassified |
| D07875 |
Doxepin (INN); Sinequan (TN) |
(P) unclassified |
| D07880 |
Duloxetine (INN); Yentreve (TN) |
(P) unclassified |
| D07904 |
Eptazocine (INN) |
(P) Target: OPRK1 |
| D07913 |
Escitalopram (INN); Esertia (TN) |
(P) Enzyme: CYP3A4 |
| D07928 |
Ethinylestradiol propanesulfonate; Turisteron (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D07930 |
Etifoxine hydrochloride; Stresam (TN) |
(P) unclassified |
| D07937 |
Etorphine (INN) |
(P) Target: OPRK1 |
| D07938 |
Bupropion hydrobromide (USAN); Aplenzin (TN) |
(P) unclassified |
| D07945 |
Fenfluramine (INN); Ponderax (TN) |
(P) Enzyme: CYP3A4 |
| D07976 |
Flupentixol decanoate; Fluanxol depot (TN) |
(P) unclassified |
| D07977 |
Fluphenazine (INN); Moditen (TN) |
(P) unclassified |
| D07984 |
Fluvoxamine (INN) |
(P) CYP inhibition: CYP3A4 |
| D07993 |
Fosphenytoin (INN) |
(P) CYP induction: CYP3A4 |
| D08035 |
Haloperidol lactate; Haldol (TN) |
(P) Enzyme: CYP3A4 |
| D08047 |
Hydromorphone (INN) |
(P) unclassified |
| D08054 |
Hydroxyzine (INN); Marex (TN) |
(P) unclassified |
| D08070 |
Imipramine (INN); Tofranil (TN) |
(P) Enzyme: CYP3A4 |
| D08071 |
Imipramine pamoate (USP); Imipramine embonate; Tofranil-pm (TN) |
(P) Enzyme: CYP3A4 |
| D08085 |
Iproniazid phosphate; Marsilid (TN) |
(P) unclassified |
| D08100 |
Ketobemidone (INN) |
(P) Target: OPRK1 |
| D08101 |
Ketobemidone hydrochloride; Ketogan (TN) |
(P) Target: OPRK1 |
| D08121 |
Levomethadone (INN) |
(P) unclassified |
| D08122 |
Levomethadone hydrochloride; L-polamidon (TN) |
(P) unclassified |
| D08123 |
Levorphanol (INN) |
(P) unclassified |
| D08133 |
Lithium; Normothymin-E (TN) |
(P) unclassified |
| D08134 |
Lithium acetate; Quilonorm (TN) |
(P) unclassified |
| D08135 |
Lithium bromide |
(P) unclassified |
| D08136 |
Lithium gluconate; Lithioderm (TN) |
(P) unclassified |
| D08137 |
Lithium sulfate; Lithionit (TN) |
(P) unclassified |
| D08140 |
Lofepramine (INN) |
(P) unclassified |
| D08145 |
Loprazolam mesilate; Loprazolam mesylate; Loprazolam methanesulfonate; Havlane (TN) |
(P) unclassified |
| D08148 |
Loxapine hydrochloride; Desconex (TN) |
(P) Enzyme: CYP3A4 |
| D08170 |
Melatonin (JAN); Melatonina (TN); Melatobel (TN) |
(P) unclassified |
| D08171 |
Melitracen (INN); Adelax (TN) |
(P) unclassified |
| D08172 |
Melperone hydrochloride; Buronil (TN) |
(P) unclassified |
| D08182 |
Meptazinol (INN) |
(P) unclassified |
| D08195 |
Methadone (BAN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
| D08216 |
Mianserin (INN); Tolvon (TN) |
(P) Enzyme: CYP3A4 |
| D08222 |
Milnacipran (INN) |
(P) unclassified |
| D08226 |
Molindone (INN) |
(P) unclassified |
| D08233 |
Morphine (BAN); Substitol (TN) |
(P) unclassified |
| D08234 |
Morphine tartrate |
(P) unclassified |
| D08235 |
Mosapramine (INN) |
(P) unclassified |
| D08246 |
Nalbuphine (INN); Intapan (TN) |
(P) Target: OPRK1 |
| D08257 |
Nefazodone (INN) |
(P) unclassified |
| D08259 |
Nelfinavir (INN); Viracept (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D08273 |
Nicomorphine hydrochloride; Vilan (TN) |
(P) unclassified |
| D08283 |
Nordazepam (INN); Calmday (TN) |
(P) Enzyme: CYP3A4 |
| D08288 |
Nortriptyline (INN); Nortrilen (TN) |
(P) unclassified |
| D08297 |
Opipramol (INN) |
(P) unclassified |
| D08323 |
Oxymorphone (INN) |
(P) unclassified |
| D08341 |
Perphenazine decanoate; Trilafon dekanoat (TN) |
(P) unclassified |
| D08342 |
Perphenazine enantate; Perphenazine enanthate; Trilafon (TN) |
(P) unclassified |
| D08343 |
Pethidine (INN); Meperidine |
(P) unclassified |
| D08349 |
Phenelzine (BAN) |
(P) unclassified |
| D08356 |
Phenobarbital diethylamine; Gratusminal (TN) |
(P) unclassified |
| D08385 |
Pipotiazine (INN); Piportil (TN) |
(P) unclassified |
| D08430 |
Promazine (INN); Combelen [veterinary] (TN) |
(P) unclassified |
| D08439 |
Propiomazine maleate; Propavan (TN) |
(P) unclassified |
| D08446 |
Prothipendyl hydrochloride; Dominal (TN) |
(P) unclassified |
| D08447 |
Protriptyline (INN) |
(P) unclassified |
| D08456 |
Quetiapine (INN); Norsic (TN) |
(P) Enzyme: CYP3A4 |
| D08472 |
Reboxetine (INN); Edronax (TN) |
(P) unclassified |
| D08473 |
Remifentanil (INN); Ultiva (TN) |
(P) unclassified |
| D08549 |
Sultopride (INN) |
(P) unclassified |
| D08585 |
Thioproperazine (INN) |
(P) unclassified |
| D08588 |
Tiagabine (INN); Gabitril (TN) |
(P) unclassified |
| D08589 |
Tianeptine sodium; Stablon (TN) |
(P) unclassified |
| D08590 |
Tiapride (INN); Tiapridal (TN) |
(P) unclassified |
| D08597 |
Tilidine (INN) |
(P) unclassified |
| D08616 |
Teneligliptin (INN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D08623 |
Tramadol (INN); Amanda (TN) |
(P) Enzyme: CYP3A4 |
| D08625 |
Tranylcypromine (INN); Parnate (TN) |
(P) unclassified |
| D08626 |
Trazodone (INN); Trittico (TN) |
(P) Enzyme: CYP3A4 |
| D08634 |
Triclofos (INN); Neguvon [veterinary] (TN) |
(P) unclassified |
| D08636 |
Trifluoperazine (INN) |
(P) unclassified |
| D08637 |
Trifluperidol hydrochloride; Triperidol (TN) |
(P) unclassified |
| D08667 |
Calcium valproate; Valproic acid calcium salt; Convulsofin (TN) |
(P) unclassified |
| D08670 |
Venlafaxine (INN); Efectin (TN) |
(P) unclassified |
| D08673 |
Viloxazine (INN) |
(P) unclassified |
| D08687 |
Ziprasidone (INN); Zipradon (TN) |
(P) unclassified |
| D08690 |
Zolpidem (INN); Sanval (TN) |
(P) Enzyme: CYP3A4 |
| D08691 |
Zuclopenthixol acetate; Cisordinol-acutard (TN) |
(P) unclassified |
| D08692 |
Zuclopenthixol decanoate; Clopixol depot (TN) |
(P) unclassified |
| D08693 |
Zuclopenthixol dihydrochloride; Clopixol (TN) |
(P) unclassified |
| D08774 |
Amoxicillin hydrate, clarithromycin and lansoprazole; Lansap (TN); Prevpac (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D08837 |
Aclidinium bromide (JAN/USAN/INN); Tudorza (TN); Eklira (TN) |
(P) CYP inhibition: CYP3A4 |
| D08879 |
Brivaracetam (JAN/USAN/INN); Briviact (TN) |
(P) unclassified |
| D08964 |
Perampanel (JAN/USAN); Fycompa (TN) |
(P) unclassified |
| D08969 |
Pimavanserin tartrate (USAN); Nuplazide (TN) |
(P) Enzyme: CYP3A4 |
| D09012 |
Telaprevir (JAN/USAN/INN); Incivek (TN); Incivo (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D09215 |
Eslicarbazepine (USAN/INN) |
(P) CYP induction: CYP3A4 |
| D09216 |
Thiopropazate (INN) |
(P) unclassified |
| D09388 |
Tasimelteon (USAN/INN); Hetlioz (TN) |
(P) Enzyme: CYP3A4 |
| D09394 |
Fidaxomicin (JAN/USAN); Dificid (TN); Dificlir (TN) |
(P) CYP inhibition: CYP3A4 |
| D09569 |
Ezogabine (USAN); Retigabine (INN); Potiga (TN) |
(P) unclassified |
| D09612 |
Eslicarbazepine acetate (USAN); Zebinix (TN); Aptiom (TN) |
(P) CYP induction: CYP3A4 |
| D09638 |
Lomitapide mesylate (USAN); Lomitapide mesilate (JAN); Juxtapid (TN); Lojuxta (TN) |
(P) Enzyme: CYP3A4 |
| D09698 |
Vilazodone (USAN/INN) |
(P) Enzyme: CYP3A4 |
| D09699 |
Vilazodone hydrochloride (USAN); Viibryd (TN) |
(P) Enzyme: CYP3A4 |
| D09731 |
Crizotinib (JAN/USAN/INN); Xalkori (TN) |
(P) Enzyme: CYP3A4 |
| D09756 |
Teneligliptin hydrobromide hydrate (JAN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D09799 |
Carotegrast methyl (JAN); Carogra (TN) |
(P) CYP inhibition: CYP3A4 |
| D09819 |
Chlorpromazine tannate (JAN) |
(P) unclassified |
| D09876 |
Cariprazine hydrochloride (JAN/USAN); Vraylar (TN) |
(P) Enzyme: CYP3A4 |
| D09996 |
Vemurafenib (JAN/USAN/INN); Zelboraf (TN) |
(P) CYP induction: CYP3A4 |
| D09997 |
Cariprazine (USAN/INN) |
(P) Enzyme: CYP3A4 |
| D09999 |
Tramadol hydrochloride and acetaminophen; Tramcet (TN) |
(P) Enzyme: CYP3A4 |
| D10003 |
Hemin (JAN); Normosang (TN); Panhematin (TN) |
(P) CYP induction: CYP3A4 |
| D10072 |
Levomilnacipran (USAN/INN) |
(P) unclassified |
| D10082 |
Suvorexant (JAN/USAN); MK-4305; Belsomra (TN) |
(P) unclassified |
| D10104 |
Dabrafenib mesylate (USAN); Dabrafenib mesilate (JAN); Tafinlar (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
| D10127 |
Glycerol phenylbutyrate (JAN/USAN); Ravicti (TN) |
(P) unclassified |
| D10133 |
Levomilnacipran hydrochloride (USAN); Fetzima (TN) |
(P) unclassified |
| D10161 |
Sarilumab (USAN); Sarilumab (genetical receombination) (JAN); Kevzara (TN) |
(P) unclassified |
| D10184 |
Vortioxetine (USAN); Brintellix (TN) |
(P) unclassified |
| D10185 |
Vortioxetine hydrobromide (JAN/USAN); Brintellix (TN); Trintellix (TN) |
(P) unclassified |
| D10194 |
Remimazolam besylate (USAN); Remimazolam besilate (JAN); Anerem (TN); Byfavo (TN) |
(P) unclassified |
| D10199 |
Tapentadol hydrochloride (JAN); Nucynta (TN) |
(P) unclassified |
| D10218 |
Enzalutamide (JAN/USAN); Xtandi (TN) |
(P) unclassified |
| D10246 |
Omeprazole, clarithromycin and amoxicillin; Omeclamox-pak (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D10309 |
Brexpiprazole (JAN/USAN/INN); Rexulti (TN) |
(P) Enzyme: CYP3A4 |
| D10355 |
Aripiprazole cavoxil (USAN) |
(P) Enzyme: CYP3A4 |
| D10364 |
Aripiprazole lauroxil (USAN); Aristada (TN) |
(P) Enzyme: CYP3A4 |
| D10372 |
Palbociclib (JAN/USAN); Ibrance (TN) |
(P) unclassified |
| D10466 |
Vonoprazan fumarate (JAN/USAN); Takecab (TN); Voquezna (TN) |
(P) Enzyme: CYP3A4 |
| D10516 |
Aripiprazole hydrate (JAN); Aripiprazole monohydrate; Abilify maintena (TN) |
(P) Enzyme: CYP3A4 |
| D10519 |
Rabeprazole, amoxicillin and clarithromycin; Rabecure (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D10551 |
Ceritinib (JAN/USAN/INN); Zykadia (TN) |
(P) unclassified |
| D10561 |
Fabomotizole (INN) |
(P) unclassified |
| D10564 |
Amenamevir (JAN/INN); Amenalief (TN) |
(P) unclassified |
| D10566 |
Pasireotide pamoate (JAN); Signifor lar (TN) |
(P) unclassified |
| D10582 |
Dasabuvir, ombitasvir, paritaprevir and ritonavir; Viekira pak (TN) |
(P) CYP inhibition: CYP3A4 |
| D10627 |
Esketamine hydrochloride (JAN/USAN); Spravato (TN) |
(P) Enzyme: CYP3A4 |
| D10633 |
Finerenone (JAN/USAN/INN); Kerendia (TN) |
(P) Enzyme: CYP3A4 |
| D10643 |
Isavuconazonium sulfate (JAN/USAN); Cresemba (TN) |
(P) unclassified |
| D10745 |
Ombitasvir, paritaprevir and ritonavir; Technivie (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D10762 |
Fosravuconazole L-lysine ethanolate (JAN) |
(P) unclassified |
| D10774 |
Vonoprazan, amoxicillin and metronidazole; Vonopion (TN) |
(P) Enzyme: CYP3A4 |
| D10775 |
Vonoprazan, amoxicillin and clarithromycin; Vonosap (TN); Voquenza (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D10780 |
Perampanel hydrate (JAN); Fycompa (TN) |
(P) unclassified |
| D10801 |
Letermovir (JAN/USAN/INN); Prevymis (TN) |
(P) unclassified |
| D10811 |
Fentanyl hydrochloride (JAN); Ionsys (TN) |
(P) Enzyme: CYP3A4 |
| D10895 |
Fosaprepitant (INN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4 |
| D10915 |
Cannabidiol (JAN/USAN/INN); CBD; Epidiolex (TN) |
(P) Enzyme: CYP3A4 |
| D10926 |
Entrectinib (JAN/USAN/INN); Rozlytrek (TN) |
(P) Enzyme: CYP3A4 |
| D10990 |
Somatrogon (USAN/INN); Somatrogon (genetical recombination) (JAN); Somatrogon-ghla; Ngenla (TN) |
(P) unclassified |
| D11012 |
Lorlatinib (JAN/USAN/INN); Lorbrena (TN) |
(P) unclassified |
| D11022 |
Lemborexant (JAN/USAN/INN); Dayvigo (TN) |
(P) Enzyme: CYP3A4 |
| D11040 |
Apalutamide (JAN/INN); Erleada (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
| D11053 |
Encorafenib (JAN/USAN/INN); Braftovi (TN) |
(P) Enzyme: CYP3A4 |
| D11056 |
Mirtazapine hydrate (JAN) |
(P) Enzyme: CYP3A4 |
| D11090 |
Ivosidenib (JAN/USAN/INN); Tibsovo (TN) |
(P) unclassified |
| D11138 |
Larotrectinib sulfate (JAN/USAN); Vitrakvi (TN) |
(P) unclassified |
| D11149 |
Brexanolone (USAN/INN); Zulresso (TN) |
(P) unclassified |
| D11150 |
Cenobamate (JAN/USAN/INN); Xcopri (TN) |
(P) Enzyme: CYP3A4 |
| D11169 |
Lumateperone (USAN/INN) |
(P) unclassified |
| D11170 |
Lumateperone tosylate (USAN); Caplyta (TN) |
(P) unclassified |
| D11194 |
Somapacitan (USAN/INN); Somapacitan (genetical recombination) (JAN); Somapacitan-beco; Sogroya (TN) |
(P) unclassified |
| D11214 |
Oliceridine (USAN/INN); Olinvyk (TN) |
(P) unclassified |
| D11296 |
Fedratinib hydrochloride (USAN); Fedratinib hydrochloride hydrate (JAN); Fedratinib dihydrochloride monohydrate; Inrebic (TN) |
(P) Enzyme: CYP3A4 |
| D11370 |
Fosnetupitant chloride hydrochloride (JAN/USAN); Arokaris (TN) |
(P) unclassified |
| D11371 |
Capivasertib (JAN/USAN); Truqap (TN) |
(P) unclassified |
| D11422 |
Zanubrutinib (JAN/USAN/INN); Brukinsa (TN) |
(P) unclassified |
| D11454 |
Repotrectinib (JAN/USAN); Augtyro (TN) |
(P) Enzyme: CYP3A4 |
| D11485 |
Tazemetostat hydrobromide (JAN/USAN); Tazverik (TN) |
(P) unclassified |
| D11557 |
Tecovirimat hydrate (JAN); Tecovirimat monohydrate; Tpoxx (TN); Tepoxx (TN) |
(P) unclassified |
| D11619 |
Desvenlafaxine succinate anhydrous |
(P) unclassified |
| D11673 |
Berotralstat (USAN/INN) |
(P) CYP inhibition: CYP3A4 |
| D11674 |
Berotralstat hydrochloride (JAN/USAN); Orladeyo (TN) |
(P) CYP inhibition: CYP3A4 |
| D11713 |
Selpercatinib (JAN/USAN/INN); Retevmo (TN) |
(P) Enzyme: CYP3A4 |
| D11769 |
Asenapine (INN); Secuado (TN) |
(P) unclassified |
| D11788 |
Remimazolam (USAN/INN); Byfavo (TN) |
(P) unclassified |
| D11793 |
Zuranolone (JAN/USAN/INN); Zurzuvae (TN) |
(P) Enzyme: CYP3A4 |
| D11804 |
Aspirin and vonoprazan; Cabpirin (TN) |
(P) unclassified |
| D11816 |
Belumosudil mesylate (USAN); Belumosudil mesilate (JAN); Rezurock (TN) |
(P) Enzyme: CYP3A4 |
| D11835 |
Vorasidenib citrate (USAN); Vorasidenib citric acid hydrate (JAN); Voranigo (TN) |
(P) unclassified |
| D11886 |
Daridorexant (USAN/INN) |
(P) unclassified |
| D11887 |
Daridorexant hydrochloride (JAN/USAN); Quviviq (TN) |
(P) unclassified |
| D11920 |
Pimitespib (JAN); Jeselhy (TN) |
(P) unclassified |
| D11954 |
Belzutifan (JAN/USAN/INN); Welireg (TN) |
(P) unclassified |
| D11968 |
Teneligliptin hydrobromide (JAN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D11970 |
Ritlecitinib tosylate (USAN); Ritlecitinib tosilate (JAN); Litfulo (TN) |
(P) unclassified |
| D12015 |
St. John's wort; SJW |
(P) unclassified |
| D12050 |
Pirtobrutinib (JAN/USAN); Jaypirca (TN) |
(P) Enzyme: CYP3A4 |
| D12055 |
Sotorasib (JAN/USAN); Lumakras (TN) |
(P) unclassified |
| D12117 |
Olanzapine and samidorphan; Lybalvi (TN) |
(P) unclassified |
| D12245 |
Lazertinib mesylate (USAN); Lazertinib mesilate hydrate (JAN); Lazcluze (TN) |
(P) Enzyme: CYP3A4 |
| D12252 |
Iptacopan hydrochloride (USAN); Iptacopan hydrochloride hydrate (JAN); Iptacopan hydrochloride monohydrate; Fabhalta (TN) |
(P) CYP induction: CYP3A4 |
| D12403 |
Venlafaxine besylate monohydrate; Venlafaxine besylate (TN) |
(P) unclassified |
| D12442 |
Tucatinib ethanolate (JAN); Tucatinib hemiethanolate; Tukysa (TN) |
(P) unclassified |
| D12444 |
Nilotinib hydrochloride dihydrate (JAN) |
(P) Enzyme: CYP3A4 |
| D12493 |
Dextromethorphan hydrobromide and bupropion hydrochloride; Auvelity (TN) |
(P) unclassified |
| D12544 |
Vortioxetine hemihydrobromide (USAN) |
(P) unclassified |
| D12586 |
Mifepristone and misoprostol; Mefeego (TN) |
(P) unclassified |
| D12637 |
Darunavir hydrate |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D12660 |
Alphacetylmethadol (INN) |
(P) unclassified |
| D12661 |
Betacetylmethadol (INN) |
(P) unclassified |
| D12662 |
Allylprodine (INN) |
(P) unclassified |
| D12663 |
Ethylmethylthiambutene (INN) |
(P) unclassified |
| D12664 |
Diethylthiambutene (INN) |
(P) unclassified |
| D12665 |
Dimethylthiambutene (INN) |
(P) unclassified |
| D12666 |
Alphameprodine (INN); alpha-Meprodine |
(P) unclassified |
| D12667 |
Betameprodine (INN); beta-Meprodine |
(P) unclassified |
| D12668 |
Clonitazene (INN) |
(P) unclassified |
| D12669 |
Etonitazene (INN) |
(P) unclassified |
| D12670 |
Desomorphine (INN) |
(P) unclassified |
| D12671 |
Dipipanone (BAN) |
(P) unclassified |
| D12672 |
Dimenoxadol (INN) |
(P) unclassified |
| D12673 |
Dimepheptanol (INN) |
(P) unclassified |
| D12674 |
Alphamethadol (INN) |
(P) unclassified |
| D12675 |
Betamethadol (INN) |
(P) unclassified |
| D12676 |
Isomethadone (INN) |
(P) unclassified |
| D12677 |
Proheptazine (INN) |
(P) unclassified |
| D12678 |
Alphaprodine (INN) |
(P) unclassified |
| D12679 |
Betaprodine (INN) |
(P) unclassified |
| D12680 |
Etoxeridine (INN) |
(P) unclassified |
| D12681 |
Hydroxypethidine (INN); Bemidone |
(P) unclassified |
| D12682 |
Furethidine (INN) |
(P) unclassified |
| D12683 |
Piminodine (INN) |
(P) unclassified |
| D12685 |
Benzethidine (INN) |
(P) unclassified |
| D12686 |
Hydromorphinol (INN) |
(P) unclassified |
| D12687 |
Levophenacylmorphan (INN) |
(P) unclassified |
| D12688 |
Phenomorphan (INN) |
(P) unclassified |
| D12689 |
Methyldihydromorphine (INN) |
(P) unclassified |
| D12690 |
Metopon (BAN); Methyldihydromorphinone |
(P) unclassified |
| D12691 |
Methyldesorphine (INN) |
(P) unclassified |
| D12692 |
Norlevorphanol (INN) |
(P) unclassified |
| D12693 |
Phenampromide (INN) |
(P) unclassified |
| D12694 |
Diampromide (INN) |
(P) unclassified |
| D12695 |
Levomoramide (INN) |
(P) unclassified |
| D12696 |
Levomethorphan (INN) |
(P) unclassified |
| D12697 |
Morpheridin (INN) |
(P) unclassified |
| D12698 |
Phenadoxone (INN) |
(P) unclassified |
| D12699 |
Dioxaphetyl butyrate (INN) |
(P) unclassified |
| D12700 |
Acetorphine (INN) |
(P) Target: OPRK1 |
| D12701 |
Norpipanone (INN) |
(P) unclassified |
| D12752 |
Darunavir propylene glycolate |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D12837 |
Risovalisib mesilate hydrate (JAN); Risovalisib mesylate dihydrate; Haizexin (TN) |
(P) unclassified |
| D12968 |
Xanomeline and trospium chloride; Cobenfy (TN) |
(P) unclassified |
| D13025 |
Properidine (INN); Ipropethidine |
(P) unclassified |
| D13183 |
Brexpiprazole fumarate hydrate (JAN) |
(P) Enzyme: CYP3A4 |
| D13231 |
Dimdazenil (INN) |
(P) unclassified |