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Drug interaction list


Query:
D06405  Nalfurafine hydrochloride (JAN/USAN)

Interactions: 711 hits    [ ATC classification | Therapeutic category ]

C06174  Codeine; (5alpha,6alpha)-7,8-Didehydro-4,5-epoxy-3-methoxy-17-methylmorphinan-6-ol (P) unclassified
C07051  Indinavir (P) unclassified
D00020  Tryptophan (USP/INN); L-Tryptophan (JP18) (P) unclassified
D00058  gamma-Aminobutyric acid (JAN); Gammalon (TN) (P) unclassified
D00136  Haloperidol (JP18/USP/INN); Haldol (TN) (P) Enzyme: CYP3A4
D00138  Scopolamine (INN); Transderm scop (TN) (P) unclassified
D00184  Cyclosporine (USP); Ciclosporin (JP18); Gengraf (TN); Neoral (TN); Restasis (TN); Sandimmune (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00195  Codeine (USP); Codeine hydrate (P) unclassified
D00211  Rifampin (USP); Rifampicin (JP18/INN); Rifadin (TN); Rimactane (TN) (P) CYP induction: CYP3A4
D00225  Alprazolam (JP18/USP/INN); Xanax (TN) (P) unclassified
D00228  Amoxapine (JP18/USP/INN); Asendin (TN) (P) unclassified
D00252  Carbamazepine (JP18/USP/INN); Equetro (TN); Tegretol (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00265  Chloral hydrate (JP18/USP); Noctec (TN) (P) unclassified
D00267  Chlordiazepoxide (JP18/USP/INN); Libritabs (TN) (P) unclassified
D00270  Chlorpromazine (USP/INN); Thorazine (TN) (P) unclassified
D00276  Clarithromycin (JP18/USP/INN); Biaxin (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00280  Clonazepam (JP18/USP/INN); Klonopin (TN) (P) unclassified
D00282  Clotrimazole (JP18/USP/INN); Lotrimin (TN); Mycelex (TN) (P) CYP inhibition: CYP3A4
D00283  Clozapine (JAN/USP/INN); Clozaril (TN) (P) Enzyme: CYP3A4
D00292  Dexamethasone (JP18/USP/INN); Decadron (TN); Maxidex (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00293  Diazepam (JP18/USP/INN); Diastat (TN); Valium (TN) (P) Enzyme: CYP3A4
D00295  Cimetidine (JP18/USP/INN); Tagamet (TN) (P) CYP inhibition: CYP3A4
D00304  Divalproex sodium (USP); Valproate semisodium (INN); Depakote (TN) (P) unclassified
D00308  Droperidol (JP18/USP/INN); Droleptan (TN); Inapsine (TN) (P) unclassified
D00311  Estazolam (JP18/USP/INN); ProSom (TN) (P) unclassified
D00320  Fentanyl (JAN/USP/INN); Duragesic (TN); Subsys (TN) (P) Enzyme: CYP3A4
D00322  Fluconazole (JP18/USP/INN); Diflucan (TN) (P) CYP inhibition: CYP3A4
D00326  Fluoxetine (USAN/INN); Fluoxetine (TN) (P) unclassified
D00329  Flurazepam (JAN/INN); Insumin (TN) (P) unclassified
D00338  Halazepam (USAN/INN); Paxipam (TN) (P) unclassified
D00350  Itraconazole (JP18/USP); Itrizole (TN); Sporanox (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00351  Ketoconazole (JP18/USP); Nizoral (TN); Xolegel (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00354  Lamotrigine (JAN/USP/INN); Lamictal (TN) (P) unclassified
D00365  Lorazepam (JP18/USP/INN); Ativan (TN) (P) unclassified
D00370  Temazepam (USP/INN); Restoril (TN) (P) unclassified
D00373  Thioridazine (USP/INN); Mellaril-S (TN) (P) unclassified
D00374  Thiothixene (USP); Tiotixene (JAN); Navane (TN) (P) unclassified
D00375  Mephenytoin (USP/INN); Mesantoin (TN) (P) unclassified
D00376  Meprobamate (JAN/USP/INN); Equanil (TN); Miltown (TN) (P) unclassified
D00387  Triazolam (JP18/USP/INN); Halcion (TN) (P) Enzyme: CYP3A4
D00388  Triclofos sodium (JP18/USAN); Tricloryl (TN) (P) unclassified
D00390  Triflupromazine (USP/INN); Vesprin (TN) (P) unclassified
D00392  Trimethadione (JP18/INN); Tridione (TN) (P) unclassified
D00394  Trimipramine (USAN/INN) (P) unclassified
D00399  Valproic acid (USP); Depakene (TN) (P) unclassified
D00403  Methotrimeprazine (USP); Levomepromazine (USAN/INN); Levoprome (TN) (P) unclassified
D00404  Methsuximide (USP); Mesuximide (INN); Celontin (TN) (P) unclassified
D00420  Mitotane (JAN/USP/INN); Lysodren (TN) (P) unclassified
D00426  Risperidone (JP18/USP/INN); Risperdal (TN) (P) Enzyme: CYP3A4
D00427  Ritonavir (JAN/USP/INN); Norvir (TN) (P) unclassified
D00430  Secobarbital (USP/INN); Seconal (TN) (P) unclassified
D00435  Nevirapine (JAN/USP/INN); Viramune (TN) (P) Enzyme: CYP3A4
D00437  Nifedipine (JP18/USP/INN); Adalat (TN); Afeditab CR (TN); Procardia (TN) (P) Enzyme: CYP3A4
D00454  Olanzapine (JAN/USP/INN); Zyprexa (TN) (P) unclassified
D00457  Quazepam (JAN/USP/INN); Doral (TN) (P) Enzyme: CYP3A4
D00458  Quetiapine fumarate (JP18/USP); Seroquel (TN) (P) Enzyme: CYP3A4
D00464  Oxazepam (JAN/USP/INN); Serax (TN) (P) unclassified
D00470  Prazepam (JP18/USAN/INN); Centrax (TN) (P) unclassified
D00474  Primidone (JP18/USP/INN); Mysoline (TN) (P) unclassified
D00479  Prochlorperazine maleate (JP18/USP); Compazine (TN) (P) unclassified
D00482  Propoxyphene hydrochloride (USAN); Dextropropoxyphene hydrochloride; Darvon (TN) (P) unclassified
D00484  Protriptyline hydrochloride (USP); Vivactil (TN) (P) unclassified
D00493  Prochlorperazine (JAN/USP/INN); Compro (TN) (P) unclassified
D00495  Paramethadione (INN); Paradione (TN) (P) unclassified
D00498  Pentazocine (JP18/USP/INN); Fortral (TN) (P) Target: OPRK1
D00499  Pentobarbital (USP/INN); Nembutal (TN) (P) unclassified
D00500  Pentobarbital sodium (JAN/USP); Nembutal sodium (TN) (P) unclassified
D00503  Perphenazine (JP18/USP/INN); Trilafon (TN) (P) unclassified
D00504  Phenacemide (JAN/INN); Phenurone (TN) (P) unclassified
D00505  Phenelzine sulfate (USP); Nardil (TN) (P) unclassified
D00506  Phenobarbital (JP18/USP/INN); Luminal (TN) (P) unclassified
D00508  Phensuximide (USP/INN); Milontin (TN) (P) unclassified
D00512  Phenytoin (JP18/USP/INN); Dilantin (TN) (P) unclassified
D00514  Dexmedetomidine (USAN/INN); Dexdor (TN); Precedex (TN) (P) unclassified
D00530  Zaleplon (JAN/USP/INN); Sonata (TN) (P) Enzyme: CYP3A4
D00531  Nitrazepam (JP18/USAN/INN); Benzalin (TN); Nitrazepam (TN) (P) unclassified
D00532  Glutethimide (JAN/INN); Doriden (TN) (P) unclassified
D00533  Oxcarbazepine (JAN/USP/INN); Oxtellar (TN); Trileptal (TN) (P) unclassified
D00535  Vigabatrin (JAN/USP/INN); Sabril (TN) (P) unclassified
D00536  Felbamate (USPINN); Felbatol (TN) (P) unclassified
D00537  Topiramate (JAN/USP/INN); Topamax (TN); Trokendi xr (TN) (P) Enzyme: CYP3A4
D00538  Zonisamide (JP18/USP/INN); Excegran (TN) (P) unclassified
D00539  Ethosuximide (JP18/USP/INN); Zarontin (TN) (P) Enzyme: CYP3A4
D00550  Midazolam (JAN/USP/INN); Dormicum (TN); Buccolam (TN); Nayzilam (TN) (P) Enzyme: CYP3A4
D00554  Ethinyl estradiol (USP); Ethinylestradiol (JP18/INN); Estinyl (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00555  Amobarbital (JP18/INN); Isomytal (TN) (P) unclassified
D00557  Methaqualone (JAN/USAN/INN) (P) unclassified
D00560  Pimozide (JP18/USP/INN); Orap (TN) (P) Enzyme: CYP3A4
D00561  Sertindole (USAN/INN); SerLect (TN) (P) unclassified
D00563  Mirtazapine (JAN/USP/INN); Remeron (TN); Reflex (TN) (P) Enzyme: CYP3A4
D00619  Verapamil hydrochloride (JP18/USP); Calan (TN); Covera-hs (TN); Vasolan (TN); Verelan (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00636  Amiodarone hydrochloride (JP18/USP); Ancaron (TN); Cordarone (TN); Nexterone (TN) (P) Enzyme: CYP3A4
D00672  Hydroxyzine hydrochloride (JP18/USP); Hydroxyzine dihydrochloride; Atarax (TN); Vistaril (TN) (P) unclassified
D00693  Chlordiazepoxide hydrochloride (JAN/USP); Librium (TN) (P) unclassified
D00694  Clorazepate dipotassium (JP18/USP); Tranxene (TN) (P) unclassified
D00695  Flurazepam hydrochloride (USP); Flurazepam dihydrochloride; Dalmane (TN) (P) unclassified
D00696  Midazolam hydrochloride (USAN); Versed (TN) (P) Enzyme: CYP3A4
D00698  Aprobarbital (INN); Alurate (TN) (P) unclassified
D00700  Mephobarbital (JAN/USP); Methylphenobarbital (INN); Mebaral (TN) (P) unclassified
D00701  Phenobarbital sodium (JAN/USP/INN); Luminal sodium (TN) (P) unclassified
D00702  Buspirone hydrochloride (USP); Buspar (TN) (P) unclassified
D00704  Ethchlorvynol (JAN/USP/INN); Placidyl (TN) (P) unclassified
D00705  Paraldehyde (USP); Paral (TN) (P) unclassified
D00706  Zolpidem tartrate (JP18/USP); Ambien (TN); Intermezzo (TN) (P) Enzyme: CYP3A4
D00707  Fomepizole (JAN/USAN/INN); Antizol (TN) (P) CYP inhibition: CYP3A4
D00708  Ethotoin (JAN/USP/INN); Accenon (TN); Peganone (TN) (P) unclassified
D00709  Levetiracetam (JAN/USP/INN); Keppra (TN); E keppra (TN) (P) unclassified
D00710  Valproate sodium (USAN); Sodium valproate (JP18); Depakene (TN); Selenica (TN) (P) unclassified
D00712  Methohexital sodium (USP); Brevital sodium (TN) (P) unclassified
D00714  Thiopental sodium (JP18/USP/INN); Pentothal (TN) (P) unclassified
D00753  Sirolimus (JAN/USAN/INN); Rapamune (TN); Rapamycin (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00780  Bromocriptine mesylate (USP); Bromocriptine mesilate (JP18); Parlodel (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00788  Acetophenazine maleate (USAN); Tindal (TN) (P) unclassified
D00789  Chlorpromazine hydrochloride (JP18/USP); Sonazine (TN) (P) unclassified
D00790  Chlorprothixene (JAN/USAN/INN); Taractan (TN) (P) unclassified
D00791  Fluphenazine hydrochloride (JAN/USP); Prolixin (TN) (P) unclassified
D00792  Fluphenazine enanthate (JP18/USP); Prolixin enanthate (TN) (P) unclassified
D00793  Fluphenazine decanoate (JAN/USP); Prolixin decanoate (TN) (P) unclassified
D00794  Loxapine succinate (USP); Loxitane (TN) (P) Enzyme: CYP3A4
D00795  Mesoridazine besylate (USP); Serentil (TN) (P) unclassified
D00796  Molindone hydrochloride (USP); Moban (TN) (P) unclassified
D00797  Promazine hydrochloride (USP); Sparine (TN) (P) unclassified
D00798  Thioridazine hydrochloride (JP18/USP); Mellaril (TN) (P) unclassified
D00799  Trifluoperazine hydrochloride (JAN/USP); Stelazine (TN) (P) unclassified
D00800  Triflupromazine hydrochloride (JAN/USP); Vesprin (TN) (P) unclassified
D00801  Lithium carbonate (JP18/USP); Eskalith (TN); Lithobid (TN) (P) unclassified
D00809  Amitriptyline hydrochloride (JP18/USP); Elavil (TN) (P) Enzyme: CYP3A4
D00811  Clomipramine hydrochloride (JP18/USP); Anafranil (TN) (P) Enzyme: CYP3A4
D00812  Desipramine hydrochloride (JAN/USP); Norpramin (TN) (P) unclassified
D00814  Doxepin hydrochloride (USP); Sinequan (TN); Zonalon (TN) (P) unclassified
D00815  Imipramine hydrochloride (JP18/USP); Tofranil (TN) (P) Enzyme: CYP3A4
D00816  Nortriptyline hydrochloride (JP18/USP/INN); Pamelor (TN) (P) unclassified
D00817  Bupropion hydrochloride (JAN/USP); Wellbutrin (TN); Zyban (TN) (P) unclassified
D00818  Maprotiline hydrochloride (JP18/USP); Ludiomil (TN) (P) unclassified
D00819  Nefazodone hydrochloride (USP); Serzone (TN) (P) unclassified
D00820  Trazodone hydrochloride (JAN/USP); Desyrel (TN) (P) Enzyme: CYP3A4
D00821  Venlafaxine hydrochloride (JAN/USP); Effexor (TN) (P) unclassified
D00822  Citalopram hydrobromide (USP); Celexa (TN) (P) Enzyme: CYP3A4
D00823  Fluoxetine hydrochloride (JAN/USP); Prozac (TN); Sarafem (TN) (P) unclassified
D00824  Fluvoxamine maleate (JP18/USP); Luvox (TN) (P) CYP inhibition: CYP3A4
D00825  Sertraline hydrochloride (JAN/USP); Zoloft (TN) (P) Enzyme: CYP3A4
D00826  Tranylcypromine sulfate (USP); Parnate (TN) (P) unclassified
D00831  Mefloquine hydrochloride (JP18/USP); Lariam (TN) (P) unclassified
D00835  Alfentanil hydrochloride (USP); Alfenta (TN) (P) unclassified
D00836  Buprenorphine hydrochloride (JP18/USP); Buprenex (TN) (P) Enzyme: CYP3A4 / Target: OPRK1
D00837  Butorphanol tartrate (JAN/USP); Stadol (TN) (P) Target: OPRK1
D00838  Dezocine (USAN); Dalgan (TN) (P) Target: OPRK1
D00839  Hydromorphone hydrochloride (JAN/USP); Dilaudid (TN); Exalgo (TN); Palladone (TN) (P) unclassified
D00840  Levomethadyl acetate hydrochloride (USAN); Orlaam (TN) (P) Enzyme: CYP3A4
D00841  Levorphanol tartrate (USP); Levorphanol tartrate dihydrate; Levo-dromoran (TN) (P) unclassified
D00842  Morphine sulfate (USP); Morphine sulfate hydrate (JP18); Morphine sulfate pentahydrate; Astramor PH (TN); Avinza (TN); Depodur (TN); Kadian (TN); MS contin (TN) (P) unclassified
D00843  Nalbuphine hydrochloride (USAN); Nubain (TN) (P) Target: OPRK1
D00844  Oxymorphone hydrochloride (USP); Numorphan (TN); Opana (TN) (P) unclassified
D00845  Sufentanil citrate (USP); Dsuvia (TN); Sufenta (TN) (P) unclassified
D00847  Oxycodone hydrochloride (USP); Oxecta (TN); Oxycontin (TN); Roxicodone (TN) (P) Enzyme: CYP3A4 / Target: OPRK1
D00854  Quinupristin and dalfopristin; Synercid (TN) (P) CYP inhibition: CYP3A4
D00897  Indinavir sulfate (USP); Crixivan (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00899  Nelfinavir mesylate (USAN/INN); Nelfinavir mesilate (JAN); Viracept (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00960  Anastrozole (JP18/USP/INN); Arimidex (TN) (P) CYP inhibition: CYP3A4
D00961  Bicalutamide (JP18/USP/INN); Casodex (TN) (P) CYP inhibition: CYP3A4
D01044  Flupentixol (INN); Flupenthixol; Depixol (TN) (P) unclassified
D01071  Hexobarbital (JAN/INN) (P) unclassified
D01096  Hydroxyzine pamoate (JP18/USP); Atarax-P (TN); Vistaril pamoate (TN) (P) unclassified
D01101  Bromperidol (JAN/USAN/INN); Impromen (TN) (P) Enzyme: CYP3A4
D01105  Moperone hydrochloride (JAN); Luvatren (TN) (P) unclassified
D01107  Milnacipran hydrochloride (JAN/USAN); Savella (TN); Toledomin (TN) (P) unclassified
D01110  Melitracen hydrochloride (JAN/USAN) (P) unclassified
D01150  Methyprylon (JAN/INN); Noludar (TN) (P) unclassified
D01164  Aripiprazole (JP18/USP/INN); Abilify (TN) (P) Enzyme: CYP3A4
D01177  Remifentanil hydrochloride (JAN/USAN); Ultiva (TN) (P) unclassified
D01179  Duloxetine hydrochloride (JAN/USP); Cymbalta (TN); Yentreve (TN) (P) unclassified
D01190  Ethylphenacemide (JAN); Pheneturide (INN) (P) unclassified
D01205  Dexmedetomidine hydrochloride (JAN/USP); Igalmi (TN); Precedex (TN) (P) unclassified
D01219  Oxypertine (JAN/USAN/INN); Forit (TN) (P) unclassified
D01226  Sulpiride (JP18/USAN/INN); Dogmatyl (TN) (P) unclassified
D01230  Flunitrazepam (JP18/USAN/INN); Rohypnol (TN) (P) unclassified
D01235  Josamycin (JP18/USAN/INN); Leucomycin A3; JM; Josamycin (TN) (P) CYP inhibition: CYP3A4
D01245  Bromazepam (JP18/USAN/INN); Lectopam (TN) (P) unclassified
D01253  Clobazam (JAN/USAN/INN); Mystan (TN); Onfi (TN) (P) Enzyme: CYP3A4
D01254  Tofisopam (JP18/INN); Emandaxin (TN) (P) unclassified
D01268  Cloxazolam (JP18/INN); Sepazon (TN) (P) unclassified
D01276  Atazanavir sulfate (JAN/USAN); Reyataz (TN) (P) CYP inhibition: CYP3A4
D01285  Lofepramine hydrochloride (JAN/USAN); Amplit (TN) (P) unclassified
D01292  Medazepam (JP18/INN); Pamnace (TN) (P) unclassified
D01293  Ethyl loflazepate (JP18/INN); Meilax (TN) (P) Enzyme: CYP3A4
D01310  Secobarbital sodium (JAN/USP); Seconal sodium (TN) (P) unclassified
D01314  Dibenzepin hydrochloride (JAN/USAN) (P) unclassified
D01316  Mexazolam (JAN/INN); Melex (TN) (P) Enzyme: CYP3A4
D01321  Zotepine (JAN/INN); Setous (TN) (P) unclassified
D01322  Troleandomycin (USAN/INN); Triacetyloleandomycin (JAN); TAO; Tao (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D01328  Clotiazepam (JP18/INN); Rize (TN) (P) unclassified
D01339  Midecamycin (JP18/INN); Medemycin (TN) (P) CYP inhibition: CYP3A4
D01354  Fludiazepam (JP18/INN); Erispan (TN) (P) unclassified
D01355  Tramadol hydrochloride (JP18/USP); Ultram (TN) (P) Enzyme: CYP3A4
D01358  Mianserin hydrochloride (JAN/USAN); Tetramide (TN) (P) Enzyme: CYP3A4
D01372  Zopiclone (JP18/INN); Amoban (TN); Zopiclone (TN) (P) Enzyme: CYP3A4
D01382  Metharbital (JAN/INN); Gemonil (TN) (P) unclassified
D01383  Meperidine hydrochloride (USP); Pethidine hydrochloride (JP18); Demerol (TN) (P) unclassified
D01391  Bromovalerylurea (JP18); Bromisoval (INN); Bromisovalum; Bromovalerylurea (TN); Bromural (TN); Brovarin (TN) (P) unclassified
D01399  Fentanyl citrate (JP18/USP); Abstral (TN); Fentora (TN); Lazanda (TN); Oralet (TN) (P) Enzyme: CYP3A4
D01408  Flurazepam hydrochloride (JP18); Flurazepam monohydrochloride; Dalmate (TN) (P) unclassified
D01412  Perazine maleate (JAN) (P) unclassified
D01429  Fosfluconazole (JAN/INN); Prodif (TN) (P) CYP inhibition: CYP3A4
D01447  Thioproperazine mesilate (JAN); Thioproperazine mesylate (P) unclassified
D01448  Trifluoperazine maleate (JAN); Trifluoperazine (TN) (P) unclassified
D01477  Opipramol hydrochloride (JAN/USAN); Insidon (TN) (P) unclassified
D01481  Dihydrocodeine phosphate (JP18); Dihydro (TN) (P) unclassified
D01482  Pipamperone hydrochloride (JAN) (P) unclassified
D01485  Propericiazine (JAN); Periciazine; Neuleptil (TN) (P) unclassified
D01514  Etizolam (JP18/INN); Sedekopan (TN) (P) Enzyme: CYP3A4
D01520  Levomepromazine hydrochloride (JAN/USAN); Nozinan (TN) (P) unclassified
D01522  Tiapride hydrochloride (JP18); Gramalil (TN) (P) unclassified
D01546  Dothiepin hydrochloride (USAN); Dosulepin hydrochloride (JAN); Dosulepin (TN) (P) unclassified
D01548  Mosapramine hydrochloride (JAN); Cremin (TN) (P) unclassified
D01593  Nimetazepam (JAN/INN); Erimin (TN) (P) unclassified
D01597  Clothiapine (USAN); Clotiapine (JAN/INN); Entumin (TN) (P) unclassified
D01636  Midecamycin acetate (JP18); Miocamycin; Miocamycin (TN) (P) CYP inhibition: CYP3A4
D01657  Lormetazepam (JAN/USAN/INN); Loramet (TN) (P) unclassified
D01740  Barbital (JP18/INN); Barbital (TN) (P) unclassified
D01744  Brotizolam (JP18/USAN/INN); Lendormin (TN) (P) Enzyme: CYP3A4
D01787  Sulthiame (USAN); Sultiame (JP18); Ospolot (TN) (P) unclassified
D01793  Bifemelane hydrochloride (JAN) (P) unclassified
D01807  Mebutamate (JAN/USAN); Capla (TN); Dormate (TN) (P) unclassified
D01860  Perazine dimalonate (JAN) (P) unclassified
D01879  Eptazocine hydrobromide (JAN); Sedapain (TN) (P) Target: OPRK1
D01898  Haloperidol decanoate (JAN/USP); Halomonth (TN) (P) Enzyme: CYP3A4
D01939  Ziprasidone hydrochloride (USP); Ziprasidone hydrochloride hydrate (JAN); Geodon (TN) (P) unclassified
D01980  Luliconazole (JAN/USAN/INN); Lulicon (TN); Luzu (TN) (P) CYP inhibition: CYP3A4
D02022  Prochlorperazine mesilate (JAN); Prochlorperazine dimethanesulfonate; Novamin (TN) (P) unclassified
D02037  Perphenazine maleate (JP18); PZC (TN) (P) unclassified
D02071  Scopolamine hydrobromide (USP); Scopolamine hydrobromide hydrate (JP18); Scopolamine hydrobromide trihydrate; Hysco (TN); Isopto hyoscine (TN) (P) unclassified
D02096  Fosphenytoin sodium (USP); Cerebyx (TN); Sesquient (TN) (P) CYP induction: CYP3A4
D02097  Tiagabine hydrochloride (USP); Gabitril (TN) (P) unclassified
D02100  Ziprasidone mesylate (USAN); Ziprasidone mesylate hydrate; Geodon (TN) (P) unclassified
D02101  Codeine phosphate (USP); Codeine phosphate hydrate (JP18); Codeine (TN) (P) unclassified
D02102  Methadone hydrochloride (JAN/USP); Dolophine hydrochloride (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D02103  Phenytoin sodium (USP); Phenytoin sodium for injection (JP18); Aleviatin (TN); Dilantin (TN) (P) unclassified
D02111  Pentazocine lactate (USP); Talwin (TN) (P) Target: OPRK1
D02162  Chlorprothixene hydrochloride (JAN) (P) unclassified
D02163  Fluphenazine maleate (JAN); Flumezin (TN) (P) unclassified
D02175  Compound oxycodone (JP18); Pavinal (TN) (P) Enzyme: CYP3A4
D02208  Sultopride hydrochloride (JAN); Sultopride monohydrochloride; Barnetil (TN) (P) unclassified
D02227  Pentazocine hydrochloride (JAN/USP); Sosegon (TN); Talacen (TN) (P) Target: OPRK1
D02236  Flupentixol dihydrochloride (JAN) (P) unclassified
D02248  Levomepromazine maleate (JP18/USAN); Hirnamin (TN) (P) unclassified
D02252  Amobarbital sodium (JAN/USP); Amytal sodium (TN) (P) unclassified
D02253  Pentobarbital calcium (JP18); Ravona (TN) (P) unclassified
D02260  Paroxetine hydrochloride hemihydrate (USP); Paroxetine hydrochloride hydrate (JP18); Paxil (TN) (P) unclassified
D02271  Morphine hydrochloride hydrate (JP18); Morphine hydrochloride trihydrate; Anpec (TN) (P) unclassified
D02340  Loxapine (USAN/INN); Adasuve (TN) (P) Enzyme: CYP3A4
D02356  Verapamil (USAN/INN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D02360  Sertraline (INN) (P) Enzyme: CYP3A4
D02361  Propiomazine (USAN/INN) (P) unclassified
D02362  Paroxetine (USP/INN); Paroxetine (TN) (P) unclassified
D02372  Perospirone hydrochloride hydrate (JAN); Lullan (TN) (P) unclassified
D02408  Trimipramine maleate (JAN/USP); Surmontil (TN) (P) unclassified
D02484  Artemether and lumefantrine; Coartem (TN) (P) unclassified
D02497  Fosamprenavir (INN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D02555  Posaconazole (JAN/USAN/INN); Noxafil (TN) (P) CYP inhibition: CYP3A4
D02559  Toloxatone (INN); Humoryl (TN) (P) unclassified
D02561  Moclobemide (USAN/INN); Aurorix (TN) (P) unclassified
D02565  Dimetacrine (INN) (P) unclassified
D02566  Maprotiline (USAN) (P) unclassified
D02567  Escitalopram oxalate (JAN/USP); Lexapro (TN) (P) Enzyme: CYP3A4
D02570  Desvenlafaxine succinate (USAN); Desvenlafaxine succinate hydrate (JAN); Desvenlafaxine succinate monohydrate; Pristiq (TN) (P) Enzyme: CYP3A4
D02572  Viloxazine hydrochloride (USAN); Qelbree (TN); Vivalan (TN) (P) unclassified
D02573  Reboxetine mesylate (USAN); Reboxetine mesilate; Vestra (TN) (P) unclassified
D02575  Tianeptine (INN); Stablon (TN) (P) unclassified
D02578  Agomelatine (INN); Valdoxan (TN) (P) unclassified
D02579  Iproniazid (INN) (P) unclassified
D02580  Isocarboxazid (INN); Marplan (TN) (P) unclassified
D02604  Acepromazine maleate (USP) (P) unclassified
D02608  Perazine fendizoate (JAN) (P) unclassified
D02609  Prochlorperazine edisylate (USP); Compazine syrup (TN) (P) unclassified
D02611  Phenoperidine (INN) (P) unclassified
D02612  Thiothixene hydrochloride (USP); Thiothixene dihydrochloride dihydrate; Tiotixene dihydrochloride; Thiothixene hydrochloride (TN) (P) unclassified
D02613  Clopenthixol (USAN) (P) unclassified
D02615  Chlorpromazine hydrochloride, promethazine hydrochloride and phenobarbital; Vegetamin (TN) (P) unclassified
D02618  Butobarbital (BAN); Butethal; Neonal (TN) (P) unclassified
D02619  Carbromal (INN); Adalin (TN) (P) unclassified
D02621  Fluanisone (INN) (P) unclassified
D02622  Pipamperone (USAN/INN); Floropipamide (P) unclassified
D02623  Moperone (INN) (P) unclassified
D02624  Eszopiclone (JAN/USP/INN); Estorra (TN); Lunesta (TN) (P) Enzyme: CYP3A4
D02625  Trifluperidol (USAN/INN); Triperidol (TN) (P) unclassified
D02626  Bromperidol decanoate (USAN) (P) Enzyme: CYP3A4
D02627  Benperidol (USAN/INN); Anquil (TN) (P) unclassified
D02629  Fluspirilene (USAN/INN); Imap (TN) (P) unclassified
D02630  Penfluridol (USAN/INN); Semap (TN) (P) unclassified
D02642  Butaperazine (USAN) (P) unclassified
D02643  Butaperazine maleate (USAN) (P) unclassified
D02666  Iloperidone (USAN/INN); Fanapt (TN) (P) Enzyme: CYP3A4
D02671  Mesoridazine (USAN/INN); Lidanar (TN) (P) unclassified
D02680  Pipotiazine palmitate (USAN); Piportil depot (TN) (P) unclassified
D02682  Remoxipride (USAN) (P) unclassified
D02683  Remoxipride hydrochloride (USAN) (P) unclassified
D02689  Ramelteon (JAN/USAN/INN); Rozerem (TN) (P) unclassified
D02691  Somatropin (USP/INN); Somatropin (genetical recombination) (JAN); Human growth hormone (JAN); Asellacrin (TN); Humatrope (TN); Nutropin (TN); Omnitrope (TN) (P) unclassified
D02717  Valnoctamide (USAN/INN); Axiquel (TN) (P) unclassified
D02732  Pranlukast hydrate (JP18); Onon (TN) (P) Enzyme: CYP3A4
D02766  Valpromide (INN); Depamide (TN) (P) unclassified
D02770  Adinazolam (USAN/INN) (P) unclassified
D02771  Adinazolam mesylate (USAN) (P) unclassified
D02787  Alaproclate (USAN/INN) (P) unclassified
D02817  Allobarbital (USAN/INN) (P) unclassified
D02861  Indinavir sulfate ethanolate (JAN); Crixivan (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D02867  Fosamprenavir calcium hydrate (JAN); Lexiva (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D02941  Anileridine (USP/INN) (P) unclassified
D02942  Anileridine hydrochloride (USP); Leritine (TN) (P) unclassified
D02968  Aprepitant (JAN/USP/INN); Aponvie (TN); Emend (TN); Cinvanti (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D02995  Asenapine maleate (JAN/USAN); Saphris (TN) (P) unclassified
D03083  Bentazepam (USAN/INN) (P) unclassified
D03089  Benzoctamine hydrochloride (USAN) (P) unclassified
D03106  Bexarotene (JAN/USAN/INN); Targretin (TN) (P) unclassified
D03156  Brifentanil hydrochloride (USAN) (P) unclassified
D03165  Bromocriptine (USAN/INN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D03197  Butorphanol (USAN/INN) (P) Target: OPRK1
D03199  Butriptyline hydrochloride (USAN) (P) unclassified
D03274  Chlorpromazine hibenzate (JAN); Contomin (TN) (P) unclassified
D03405  Carfentanil citrate (USAN) (P) unclassified
D03444  Opium (USP); Opium, powdered (JP18); Diluted opium powder (JP18) (P) unclassified
D03445  Opium alkaloids hydrochlorides (JP18); Pan opin (TN) (P) unclassified
D03503  Cimetidine hydrochloride (USP); Cimetidine hydrochloride (TN) (P) CYP inhibition: CYP3A4
D03556  Zuclopenthixol (INN); Clopixol (TN) (P) unclassified
D03562  Clorazepate monopotassium (USAN) (P) unclassified
D03579  Codeine polistirex (USAN) (P) unclassified
D03580  Codeine sulfate (USP); Codeine sulfate trihydrate; Codeine sulfate (TN) (P) unclassified
D03618  Cyclazocine (USAN/INN) (P) Target: OPRK1
D03656  Darunavir (USAN/INN); Darunavir (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D03658  Dasatinib (JAN/INN) (P) Enzyme: CYP3A4
D03669  Deferasirox (JAN/USAN/INN); Exjade (TN); Jadenu (TN) (P) CYP induction: CYP3A4
D03783  Oxycodone terephthalate (USP) (P) Enzyme: CYP3A4 / Target: OPRK1
D03785  Dichloralphenazone (USP) (P) unclassified
D03825  Dihydrocodeine bitartrate (USP) (P) unclassified
D03833  Indinavir (USAN); Indinavir hydrate (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D03835  Fosamprenavir calcium (USAN); Lexiva (TN); Telzir (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D03837  Fosamprenavir sodium (USAN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D03844  Phenytoin, phenobarbital and caffeine and sodium benzoate; Hydantol F (TN) (P) unclassified
D03852  Droperidol and fentanyl citrate; Innovar (TN) (P) Enzyme: CYP3A4
D03855  Pethidine hydrochloride and levallorphan tartrate; Pethilorfan (TN) (P) unclassified
D03863  Opium alkaloids and atropine (JP18); Opium alkaloids hydrochloride and atropine sulfate hydrate; Opiato (TN) (P) unclassified
D03866  Opium alkaloids and scopolamine (JP18); Weak opium alkaloids and scopolamine (JP18); Opium alkaloids hydrochloride and scopolamine hydrobromide hydrate; Opisco (TN) (P) unclassified
D03975  Allylisopropylacetylurea; Apronal; Apronalide (P) unclassified
D04024  Lapatinib ditosylate (USAN); Lapatinib tosilate hydrate (JAN); Lapatinib ditosylate monohydrate; Tykerb (TN); Tyverb (TN) (P) Enzyme: CYP3A4
D04034  Chlorpromazine phenolphthalinate (JAN); Wintermin (TN) (P) unclassified
D04038  Perphenazine fendizoate (JAN); PZC (TN) (P) unclassified
D04105  Etoperidone hydrochloride (USAN); Etonin (TN) (P) unclassified
D04148  Fenfluramine hydrochloride (JAN/USAN); Fintepla (TN); Pondimin (TN) (P) Enzyme: CYP3A4
D04300  Ganaxolone (USAN/INN); Ztalmy (TN) (P) Enzyme: CYP3A4
D04314  Gepirone hydrochloride (USAN); Exxua (TN) (P) Enzyme: CYP3A4
D04605  Iprindole (USAN/INN) (P) unclassified
D04641  Istradefylline (JAN/USAN/INN); Nourianz (TN); Nouriast (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D04649  Ketazocine (USAN/INN); Ketocyclazocine (P) Target: OPRK1
D04650  Ketazolam (USAN/INN) (P) unclassified
D04666  Lanreotide acetate (JAN/USAN); Somatuline (TN) (P) unclassified
D04716  Levomethadyl acetate (USAN); Levacetylmethadol (INN) (P) Enzyme: CYP3A4
D04749  Lithium citrate (USP); Lithonate (TN) (P) unclassified
D04750  Lithium hydroxide (USP) (P) unclassified
D04764  Lofentanil oxalate (USAN) (P) unclassified
D04820  Lurasidone hydrochloride (JAN/USAN); SM 13496; Latuda (TN) (P) Enzyme: CYP3A4
D04882  Medazepam hydrochloride (USAN); Nobrium (TN) (P) unclassified
D04924  Meptazinol hydrochloride (USAN) (P) unclassified
D04965  Perphenazine hydrochloride; Perphenazine dihydrochloride; PZC intramuscular injection (TN) (P) unclassified
D04973  Methadyl acetate (USAN); Acetylmethadol (INN) (P) unclassified
D04985  Methohexital (USP/INN) (P) unclassified
D05028  Midazolam maleate (USAN) (P) Enzyme: CYP3A4
D05039  Minaprine (USAN/INN); Cantor (TN) (P) unclassified
D05040  Minaprine hydrochloride (USAN) (P) unclassified
D05048  Mirfentanil hydrochloride (USAN) (P) unclassified
D05154  Nexeridine hydrochloride (USAN) (P) unclassified
D05200  Nomifensine maleate (USAN); Merital (TN) (P) unclassified
D05217  Ocfentanil hydrochloride (USAN) (P) unclassified
D05312  Oxycodone (USAN/INN) (P) Enzyme: CYP3A4 / Target: OPRK1
D05339  Paliperidone (JAN/USP/INN); Invega (TN) (P) unclassified
D05340  Paliperidone palmitate (JAN/USAN); Xeplion (TN); Trevicta (TN); Invega sustenna (TN); Invega trinza (TN) (P) unclassified
D05351  Josamycin propionate (JP18); Josamy (TN) (P) CYP inhibition: CYP3A4
D05374  Paroxetine hydrochloride (USP); Paxil (TN) (P) unclassified
D05375  Paroxetine mesylate (USAN); Brisdelle (TN); Pexeva (TN) (P) unclassified
D05462  Oxycodone hydrochloride hydrate (JP18) (P) Enzyme: CYP3A4 / Target: OPRK1
D05621  Progabide (USAN/INN); Gabren (TN) (P) unclassified
D05632  Propoxyphene napsylate (USAN); Darvon-N (TN) (P) unclassified
D05775  Rufinamide (JAN/USP/INN); Banzel (TN) (P) unclassified
D05928  Stiripentol (JAN/USAN/INN); Diacomit (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D05938  Sufentanil (USAN/INN) (P) unclassified
D06007  Tapentadol (USAN/INN) (P) unclassified
D06147  Tilidine hydrochloride (USAN); Valoron (TN) (P) unclassified
D06208  Trefentanil hydrochloride (USAN) (P) unclassified
D06268  Trimeperidine (INN) (P) unclassified
D06342  Xorphanol mesylate (USAN) (P) Target: OPRK1
D06367  Zimeldine hydrochloride (USAN); Zimeldine hydrochloride hydrate (P) unclassified
D06413  Nilotinib hydrochloride hydrate (JAN); Nilotinib monohydrochloride monohydrate; Tasigna (TN) (P) Enzyme: CYP3A4
D06414  Dasatinib (USAN); Dasatinib hydrate (JAN); Sprycel (TN) (P) Enzyme: CYP3A4
D06478  Darunavir ethanolate (JAN); Prezista (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D06499  Opium tincture (JP18); Opium tincture (TN) (P) unclassified
D06573  Carisbamate (USAN) (P) unclassified
D06597  Fosaprepitant dimeglumine (USAN); Fosaprepitant meglumine (JAN); Proemend (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D06623  Olanzapine pamoate (USAN); Olanzapine pamoate monohydrate; Zyprexa (TN) (P) unclassified
D06699  Japanese valerian (JP18); Powdered japanese valerian (JP18); Valerianae radix (TN) (P) unclassified
D06887  Talbutal (INN); Lotusate (TN) (P) unclassified
D07065  Acepromazine (INN); Concentrat vo34 (TN) (P) unclassified
D07122  Alfentanil (INN); Rapifen (TN) (P) unclassified
D07132  Buprenorphine (JAN/INN); Temgesic (TN) (P) Enzyme: CYP3A4 / Target: OPRK1
D07283  Esketamine (USAN/INN) (P) Enzyme: CYP3A4
D07285  Nicomorphine (INN) (P) unclassified
D07286  Diamorphine (BAN); Heroin; Diacetylmorphine (P) unclassified
D07287  Dextromoramide (BAN) (P) unclassified
D07288  Piritramide (INN); Dipidolor (TN) (P) unclassified
D07289  Bezitramide (INN); Burgodin (TN) (P) unclassified
D07298  Barbexaclone (INN); Maliasin (TN) (P) unclassified
D07299  Lacosamide (JAN/USAN/INN); Erlosamide; Vimpat (TN) (P) Enzyme: CYP3A4
D07300  Beclamide (INN) (P) unclassified
D07307  Cyamemazine (INN); Tercian (TN) (P) unclassified
D07308  Chlorproethazine (INN) (P) unclassified
D07309  Melperone (INN); Bunil (TN) (P) unclassified
D07310  Amisulpride (INN); Barhemsys (TN); Deniban (TN); Solian (TN) (P) unclassified
D07311  Veralipride (INN); Agreal (TN) (P) unclassified
D07312  Levosulpiride (INN); Levopraid (TN) (P) unclassified
D07313  Prothipendyl (INN) (P) unclassified
D07314  Pinazepam (INN); Domar (TN) (P) unclassified
D07315  Camazepam (INN) (P) unclassified
D07316  Captodiame (BAN) (P) unclassified
D07317  Emylcamate (INN) (P) unclassified
D07318  Mephenoxalone (INN); Dorsiflex (TN) (P) unclassified
D07319  Gedocarnil (INN) (P) unclassified
D07320  Etifoxine (INN/BAN) (P) unclassified
D07321  Vinylbital (INN); Vinylbitone (P) unclassified
D07322  Vinbarbital (INN) (P) unclassified
D07323  Cyclobarbital (INN); Ciclobarbital (TN) (P) unclassified
D07324  Proxibarbal (INN); Centralgol (TN) (P) unclassified
D07325  Chloralodol (INN); Chlorhexadol (P) unclassified
D07326  Loprazolam (INN); Dormonoct (TN) (P) unclassified
D07327  Doxefazepam (INN) (P) unclassified
D07328  Cinolazepam (INN); Gerodorm (TN) (P) unclassified
D07329  Pyrithyldione (INN) (P) unclassified
D07330  Clomethiazole (INN); Distraneurine (TN) (P) unclassified
D07331  Hexapropymate (INN); Merinax (TN) (P) unclassified
D07332  Methylpentynol (INN); Meparfynol; Methylparafynol; Atemorin (TN) (P) unclassified
D07333  Niaprazine (INN); Nopron (TN) (P) unclassified
D07335  Amineptine (INN); Survector (TN) (P) unclassified
D07336  Quinupramine (INN) (P) unclassified
D07337  Nialamide (INN); Niamid (TN) (P) unclassified
D07338  Iproclozide (INN); Iproclozide (TN) (P) unclassified
D07339  Oxitriptan (INN); Levothym (TN) (P) unclassified
D07340  Oxaflozane (INN) (P) unclassified
D07341  Medifoxamine (INN) (P) unclassified
D07342  Pivagabine (INN) (P) unclassified
D07435  Papaveretum (BAN); Omnopon (TN) (P) unclassified
D07448  Amitriptyline (INN); Laroxyl (TN) (P) Enzyme: CYP3A4
D07471  Atazanavir (INN); Reyataz (TN) (P) CYP inhibition: CYP3A4
D07528  Bifemelane (INN) (P) unclassified
D07583  Phenytoin and phenobarbital; Aleviatin with phenobarbital (TN) (P) unclassified
D07591  Bupropion (INN) (P) unclassified
D07593  Buspirone (INN); Gen-Buspirone (TN) (P) unclassified
D07595  Fosphenytoin sodium hydrate (JAN); Fostoin (TN) (P) CYP induction: CYP3A4
D07601  Butriptyline (INN); Evadyne (TN) (P) unclassified
D07620  Carfentanil (INN) (P) unclassified
D07685  Chlorproethazine hydrochloride; Neuriplege (TN) (P) unclassified
D07686  Chlorprothixene acetate; Truxal (TN) (P) unclassified
D07687  Chlorprothixene citrate; Truxal (TN) (P) unclassified
D07704  Citalopram (USP/INN); Citadur (TN) (P) Enzyme: CYP3A4
D07705  Citalopram hydrochloride; Seropram (TN) (P) Enzyme: CYP3A4
D07710  Clarithromycin lactobionate; Klacid (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D07725  Clomethiazole edisilate; Heminevrin (TN) (P) unclassified
D07727  Clomipramine (INN); Anafranil (TN) (P) Enzyme: CYP3A4
D07740  Codeine hydrochloride; Bisoltus (TN) (P) unclassified
D07756  Cyamemazine tartrate; Tercian (TN) (P) unclassified
D07757  Cyclobarbital calcium (BAN); Phanodorn calcium (TN) (P) unclassified
D07791  Desipramine (INN) (P) unclassified
D07793  Desvenlafaxine (INN); Khedezla (TN) (P) Enzyme: CYP3A4
D07808  Dextromoramide tartrate; Palfium (TN) (P) unclassified
D07809  Dextropropoxyphene (INN); Propoxypene (P) unclassified
D07810  Diacetylmorphine hydrochloride; Diamorphine hydrochloride; Heroin hydrochloride; Diamorphine (TN) (P) unclassified
D07812  Dibenzepin (INN) (P) unclassified
D07831  Dihydrocodeine (INN); Remedacen (TN) (P) unclassified
D07832  Dihydrocodeine thiocyanate; Paracodin (TN) (P) unclassified
D07865  Dixyrazine; Esucos (TN) (P) unclassified
D07872  Dosulepin (INN); Dothiepin; Dothep (TN) (P) unclassified
D07875  Doxepin (INN); Sinequan (TN) (P) unclassified
D07880  Duloxetine (INN); Yentreve (TN) (P) unclassified
D07904  Eptazocine (INN) (P) Target: OPRK1
D07913  Escitalopram (INN); Esertia (TN) (P) Enzyme: CYP3A4
D07928  Ethinylestradiol propanesulfonate; Turisteron (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D07930  Etifoxine hydrochloride; Stresam (TN) (P) unclassified
D07937  Etorphine (INN) (P) Target: OPRK1
D07938  Bupropion hydrobromide (USAN); Aplenzin (TN) (P) unclassified
D07945  Fenfluramine (INN); Ponderax (TN) (P) Enzyme: CYP3A4
D07976  Flupentixol decanoate; Fluanxol depot (TN) (P) unclassified
D07977  Fluphenazine (INN); Moditen (TN) (P) unclassified
D07984  Fluvoxamine (INN) (P) CYP inhibition: CYP3A4
D07993  Fosphenytoin (INN) (P) CYP induction: CYP3A4
D08035  Haloperidol lactate; Haldol (TN) (P) Enzyme: CYP3A4
D08047  Hydromorphone (INN) (P) unclassified
D08054  Hydroxyzine (INN); Marex (TN) (P) unclassified
D08070  Imipramine (INN); Tofranil (TN) (P) Enzyme: CYP3A4
D08071  Imipramine pamoate (USP); Imipramine embonate; Tofranil-pm (TN) (P) Enzyme: CYP3A4
D08085  Iproniazid phosphate; Marsilid (TN) (P) unclassified
D08100  Ketobemidone (INN) (P) Target: OPRK1
D08101  Ketobemidone hydrochloride; Ketogan (TN) (P) Target: OPRK1
D08121  Levomethadone (INN) (P) unclassified
D08122  Levomethadone hydrochloride; L-polamidon (TN) (P) unclassified
D08123  Levorphanol (INN) (P) unclassified
D08133  Lithium; Normothymin-E (TN) (P) unclassified
D08134  Lithium acetate; Quilonorm (TN) (P) unclassified
D08135  Lithium bromide; Lithium Microsol (TN) (P) unclassified
D08136  Lithium gluconate; Lithioderm (TN) (P) unclassified
D08137  Lithium sulfate; Lithionit (TN) (P) unclassified
D08140  Lofepramine (INN) (P) unclassified
D08145  Loprazolam mesilate; Loprazolam mesylate; Loprazolam methanesulfonate; Havlane (TN) (P) unclassified
D08148  Loxapine hydrochloride; Desconex (TN) (P) Enzyme: CYP3A4
D08170  Melatonin (JAN); Melatonina (TN); Melatobel (TN) (P) unclassified
D08171  Melitracen (INN); Adelax (TN) (P) unclassified
D08172  Melperone hydrochloride; Buronil (TN) (P) unclassified
D08182  Meptazinol (INN) (P) unclassified
D08195  Methadone (BAN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D08216  Mianserin (INN); Tolvon (TN) (P) Enzyme: CYP3A4
D08222  Milnacipran (INN) (P) unclassified
D08226  Molindone (INN) (P) unclassified
D08233  Morphine (BAN); Morfina Dosa (TN); Substitol (TN) (P) unclassified
D08234  Morphine tartrate; Morphine Tartrate (TN) (P) unclassified
D08235  Mosapramine (INN) (P) unclassified
D08246  Nalbuphine (INN); Intapan (TN) (P) Target: OPRK1
D08257  Nefazodone (INN) (P) unclassified
D08259  Nelfinavir (INN); Viracept (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D08273  Nicomorphine hydrochloride; Vilan (TN) (P) unclassified
D08283  Nordazepam (INN); Calmday (TN) (P) Enzyme: CYP3A4
D08288  Nortriptyline (INN); Nortrilen (TN) (P) unclassified
D08297  Opipramol (INN); Opipramol dura (TN) (P) unclassified
D08323  Oxymorphone (INN) (P) unclassified
D08341  Perphenazine decanoate; Trilafon dekanoat (TN) (P) unclassified
D08342  Perphenazine enantate; Perphenazine enanthate; Trilafon (TN) (P) unclassified
D08343  Pethidine (INN); Meperidine; Pethidine DBL (TN) (P) unclassified
D08349  Phenelzine (BAN) (P) unclassified
D08356  Phenobarbital diethylamine; Gratusminal (TN) (P) unclassified
D08385  Pipotiazine (INN); Piportil (TN) (P) unclassified
D08430  Promazine (INN); Combelen [veterinary] (TN) (P) unclassified
D08439  Propiomazine maleate; Propavan (TN) (P) unclassified
D08446  Prothipendyl hydrochloride; Dominal (TN) (P) unclassified
D08447  Protriptyline (INN) (P) unclassified
D08456  Quetiapine (INN); Norsic (TN) (P) Enzyme: CYP3A4
D08472  Reboxetine (INN); Edronax (TN) (P) unclassified
D08473  Remifentanil (INN); Ultiva (TN) (P) unclassified
D08549  Sultopride (INN) (P) unclassified
D08585  Thioproperazine (INN) (P) unclassified
D08588  Tiagabine (INN); Gabitril (TN) (P) unclassified
D08589  Tianeptine sodium; Stablon (TN) (P) unclassified
D08590  Tiapride (INN); Tiapridal (TN) (P) unclassified
D08597  Tilidine (INN) (P) unclassified
D08616  Teneligliptin (INN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D08623  Tramadol (INN); Amanda (TN) (P) Enzyme: CYP3A4
D08625  Tranylcypromine (INN); Parnate (TN) (P) unclassified
D08626  Trazodone (INN); Trittico (TN) (P) Enzyme: CYP3A4
D08634  Triclofos (INN); Neguvon [veterinary] (TN) (P) unclassified
D08636  Trifluoperazine (INN); Apo-trifluoperazine (TN) (P) unclassified
D08637  Trifluperidol hydrochloride; Triperidol (TN) (P) unclassified
D08667  Calcium valproate; Valproic acid calcium salt; Convulsofin (TN) (P) unclassified
D08670  Venlafaxine (INN); Efectin (TN) (P) unclassified
D08673  Viloxazine (INN) (P) unclassified
D08687  Ziprasidone (INN); Zipradon (TN) (P) unclassified
D08690  Zolpidem (INN); Sanval (TN) (P) Enzyme: CYP3A4
D08691  Zuclopenthixol acetate; Cisordinol-acutard (TN) (P) unclassified
D08692  Zuclopenthixol decanoate; Clopixol depot (TN) (P) unclassified
D08693  Zuclopenthixol dihydrochloride; Clopixol (TN) (P) unclassified
D08774  Amoxicillin hydrate, clarithromycin and lansoprazole; Lansap (TN); Prevpac (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D08837  Aclidinium bromide (JAN/USAN/INN); Tudorza pressair (TN); Eklira genuair (TN) (P) CYP inhibition: CYP3A4
D08879  Brivaracetam (JAN/USAN/INN); Briviact (TN) (P) unclassified
D08964  Perampanel (JAN/USAN); Fycompa (TN) (P) unclassified
D08969  Pimavanserin tartrate (USAN); Nuplazide (TN) (P) Enzyme: CYP3A4
D09012  Telaprevir (JAN/USAN/INN); Incivek (TN); Incivo (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D09215  Eslicarbazepine (USAN/INN) (P) CYP induction: CYP3A4
D09216  Thiopropazate (INN) (P) unclassified
D09388  Tasimelteon (USAN/INN); Hetlioz (TN) (P) Enzyme: CYP3A4
D09394  Fidaxomicin (JAN/USAN); Dificid (TN); Dificlir (TN) (P) CYP inhibition: CYP3A4
D09569  Ezogabine (USAN); Retigabine (INN); Potiga (TN) (P) unclassified
D09612  Eslicarbazepine acetate (USAN); Zebinix (TN); Aptiom (TN) (P) CYP induction: CYP3A4
D09638  Lomitapide mesylate (USAN); Lomitapide mesilate (JAN); Juxtapid (TN); Lojuxta (TN) (P) Enzyme: CYP3A4
D09698  Vilazodone (USAN/INN) (P) Enzyme: CYP3A4
D09699  Vilazodone hydrochloride (USAN); Viibryd (TN) (P) Enzyme: CYP3A4
D09731  Crizotinib (JAN/USAN/INN); Xalkori (TN) (P) Enzyme: CYP3A4
D09756  Teneligliptin hydrobromide hydrate (JAN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D09799  Carotegrast methyl (JAN); Carogra (TN) (P) CYP inhibition: CYP3A4
D09819  Chlorpromazine tannate (JAN) (P) unclassified
D09876  Cariprazine hydrochloride (JAN/USAN); Vraylar (TN) (P) Enzyme: CYP3A4
D09996  Vemurafenib (JAN/USAN/INN); Zelboraf (TN) (P) CYP induction: CYP3A4
D09997  Cariprazine (USAN/INN) (P) Enzyme: CYP3A4
D09999  Tramadol hydrochloride and acetaminophen; Tramcet (TN) (P) Enzyme: CYP3A4
D10003  Hemin (JAN); Normosang (TN); Panhematin (TN) (P) CYP induction: CYP3A4
D10072  Levomilnacipran (USAN/INN) (P) unclassified
D10082  Suvorexant (JAN/USAN); MK-4305; Belsomra (TN) (P) unclassified
D10104  Dabrafenib mesylate (USAN); Dabrafenib mesilate (JAN); Tafinlar (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D10133  Levomilnacipran hydrochloride (USAN); Fetzima (TN) (P) unclassified
D10161  Sarilumab (USAN); Sarilumab (genetical receombination) (JAN); Kevzara (TN) (P) unclassified
D10184  Vortioxetine (USAN); Brintellix (TN) (P) unclassified
D10185  Vortioxetine hydrobromide (JAN/USAN); Brintellix (TN); Trintellix (TN) (P) unclassified
D10194  Remimazolam besylate (USAN); Remimazolam besilate (JAN); Anerem (TN); Byfavo (TN) (P) unclassified
D10199  Tapentadol hydrochloride (JAN); Nucynta (TN) (P) unclassified
D10218  Enzalutamide (JAN/USAN); Xtandi (TN) (P) unclassified
D10246  Omeprazole, clarithromycin and amoxicillin; Omeclamox-pak (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D10309  Brexpiprazole (JAN/USAN/INN); Rexulti (TN) (P) Enzyme: CYP3A4
D10355  Aripiprazole cavoxil (USAN) (P) Enzyme: CYP3A4
D10364  Aripiprazole lauroxil (USAN); Aristada (TN) (P) Enzyme: CYP3A4
D10372  Palbociclib (JAN/USAN); Ibrance (TN) (P) unclassified
D10466  Vonoprazan fumarate (JAN/USAN); Takecab (TN); Voquezna (TN) (P) Enzyme: CYP3A4
D10516  Aripiprazole hydrate (JAN); Aripiprazole monohydrate; Abilify maintena (TN) (P) Enzyme: CYP3A4
D10519  Rabeprazole, amoxicillin and clarithromycin; Rabecure (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D10551  Ceritinib (JAN/USAN/INN); Zykadia (TN) (P) unclassified
D10561  Fabomotizole (INN) (P) unclassified
D10564  Amenamevir (JAN/INN); Amenalief (TN) (P) unclassified
D10566  Pasireotide pamoate (JAN); Signifor lar (TN) (P) unclassified
D10582  Dasabuvir, ombitasvir, paritaprevir and ritonavir; Viekira pak (TN) (P) CYP inhibition: CYP3A4
D10627  Esketamine hydrochloride (JAN/USAN); Spravato (TN) (P) Enzyme: CYP3A4
D10643  Isavuconazonium sulfate (JAN/USAN); Cresemba (TN) (P) unclassified
D10745  Ombitasvir, paritaprevir and ritonavir; Technivie (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D10762  Fosravuconazole L-lysine ethanolate (JAN) (P) unclassified
D10774  Vonoprazan, amoxicillin and metronidazole; Vonopion (TN) (P) Enzyme: CYP3A4
D10775  Vonoprazan, amoxicillin and clarithromycin; Vonosap (TN); Voquenza (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D10780  Perampanel hydrate (JAN); Fycompa (TN) (P) unclassified
D10801  Letermovir (JAN/USAN/INN); Prevymis (TN) (P) unclassified
D10811  Fentanyl hydrochloride (JAN); Ionsys (TN) (P) Enzyme: CYP3A4
D10895  Fosaprepitant (INN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D10915  Cannabidiol (JAN/USAN/INN); CBD; Epidiolex (TN) (P) Enzyme: CYP3A4
D10926  Entrectinib (JAN/USAN/INN); Rozlytrek (TN) (P) Enzyme: CYP3A4
D10990  Somatrogon (USAN/INN); Somatrogon (genetical recombination) (JAN); Somatrogon-ghla; Ngenla (TN) (P) unclassified
D11012  Lorlatinib (JAN/USAN/INN); Lorbrena (TN) (P) unclassified
D11022  Lemborexant (JAN/USAN/INN); Dayvigo (TN) (P) Enzyme: CYP3A4
D11040  Apalutamide (JAN/INN); Erleada (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D11053  Encorafenib (JAN/USAN/INN); Braftovi (TN) (P) Enzyme: CYP3A4
D11056  Mirtazapine hydrate (JAN) (P) Enzyme: CYP3A4
D11090  Ivosidenib (JAN/USAN/INN); Tibsovo (TN) (P) unclassified
D11138  Larotrectinib sulfate (JAN/USAN); Vitrakvi (TN) (P) unclassified
D11149  Brexanolone (USAN/INN); Zulresso (TN) (P) unclassified
D11150  Cenobamate (JAN/USAN/INN); Xcopri (TN) (P) Enzyme: CYP3A4
D11169  Lumateperone (USAN/INN) (P) unclassified
D11170  Lumateperone tosylate (USAN); Caplyta (TN) (P) unclassified
D11194  Somapacitan (USAN/INN); Somapacitan (genetical recombination) (JAN); Somapacitan-beco; Sogroya (TN) (P) unclassified
D11214  Oliceridine (USAN/INN); Olinvyk (TN) (P) unclassified
D11296  Fedratinib hydrochloride (USAN); Fedratinib hydrochloride hydrate (JAN); Fedratinib dihydrochloride monohydrate; Inrebic (TN) (P) Enzyme: CYP3A4
D11370  Fosnetupitant chloride hydrochloride (JAN/USAN); Arokaris (TN) (P) unclassified
D11371  Capivasertib (JAN/USAN); Truqap (TN) (P) Enzyme: CYP3A4
D11422  Zanubrutinib (JAN/USAN/INN); Brukinsa (TN) (P) unclassified
D11454  Repotrectinib (JAN/USAN); Augtyro (TN) (P) Enzyme: CYP3A4
D11485  Tazemetostat hydrobromide (JAN/USAN); Tazverik (TN) (P) unclassified
D11557  Tecovirimat hydrate (JAN); Tecovirimat monohydrate; Tpoxx (TN); Tepoxx (TN) (P) unclassified
D11619  Desvenlafaxine succinate anhydrous; Desvenlafaxine succinate (TN) (P) unclassified
D11673  Berotralstat (USAN/INN) (P) CYP inhibition: CYP3A4
D11674  Berotralstat hydrochloride (JAN/USAN); Orladeyo (TN) (P) CYP inhibition: CYP3A4
D11713  Selpercatinib (JAN/USAN/INN); Retevmo (TN) (P) Enzyme: CYP3A4
D11769  Asenapine (INN); Secuado (TN) (P) unclassified
D11788  Remimazolam (USAN/INN); Byfavo (TN) (P) unclassified
D11793  Zuranolone (JAN/USAN/INN); Zurzuvae (TN) (P) Enzyme: CYP3A4
D11804  Aspirin and vonoprazan; Cabpirin (TN) (P) unclassified
D11816  Belumosudil mesylate (USAN); Belumosudil mesilate (JAN); Rezurock (TN) (P) unclassified
D11886  Daridorexant (USAN/INN) (P) unclassified
D11887  Daridorexant hydrochloride (JAN/USAN); Quviviq (TN) (P) unclassified
D11920  Pimitespib (JAN); Jeselhy (TN) (P) unclassified
D11954  Belzutifan (JAN/USAN/INN); Welireg (TN) (P) unclassified
D11968  Teneligliptin hydrobromide (JAN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D11970  Ritlecitinib tosylate (USAN); Ritlecitinib tosilate (JAN); Litfulo (TN) (P) unclassified
D12015  St. John's wort; SJW (P) unclassified
D12050  Pirtobrutinib (JAN/USAN); Jaypirca (TN) (P) Enzyme: CYP3A4
D12055  Sotorasib (JAN/USAN); Lumakras (TN) (P) unclassified
D12117  Olanzapine and samidorphan; Lybalvi (TN) (P) unclassified
D12245  Lazertinib mesylate (USAN); Lazertinib mesilate hydrate (JAN); Lazcluze (TN) (P) Enzyme: CYP3A4
D12252  Iptacopan hydrochloride (USAN); Iptacopan hydrochloride hydrate (JAN); Iptacopan hydrochloride monohydrate; Fabhalta (TN) (P) unclassified
D12403  Venlafaxine besylate monohydrate; Venlafaxine besylate (TN) (P) unclassified
D12493  Dextromethorphan hydrobromide and bupropion hydrochloride; Auvelity (TN) (P) unclassified
D12544  Vortioxetine hemihydrobromide (USAN) (P) unclassified
D12586  Mifepristone and misoprostol; Mefeego (TN) (P) unclassified
D12637  Darunavir hydrate (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D12660  Alphacetylmethadol (INN) (P) unclassified
D12661  Betacetylmethadol (INN) (P) unclassified
D12662  Allylprodine (INN) (P) unclassified
D12663  Ethylmethylthiambutene (INN) (P) unclassified
D12664  Diethylthiambutene (INN) (P) unclassified
D12665  Dimethylthiambutene (INN) (P) unclassified
D12666  Alphameprodine (INN); alpha-Meprodine (P) unclassified
D12667  Betameprodine (INN); beta-Meprodine (P) unclassified
D12668  Clonitazene (INN) (P) unclassified
D12669  Etonitazene (INN) (P) unclassified
D12670  Desomorphine (INN) (P) unclassified
D12671  Dipipanone (BAN) (P) unclassified
D12672  Dimenoxadol (INN) (P) unclassified
D12673  Dimepheptanol (INN) (P) unclassified
D12674  Alphamethadol (INN) (P) unclassified
D12675  Betamethadol (INN) (P) unclassified
D12676  Isomethadone (INN) (P) unclassified
D12677  Proheptazine (INN) (P) unclassified
D12678  Alphaprodine (INN) (P) unclassified
D12679  Betaprodine (INN) (P) unclassified
D12680  Etoxeridine (INN) (P) unclassified
D12681  Hydroxypethidine (INN); Bemidone (P) unclassified
D12682  Furethidine (INN) (P) unclassified
D12683  Piminodine (INN) (P) unclassified
D12685  Benzethidine (INN) (P) unclassified
D12686  Hydromorphinol (INN) (P) unclassified
D12687  Levophenacylmorphan (INN) (P) unclassified
D12688  Phenomorphan (INN) (P) unclassified
D12689  Methyldihydromorphine (INN) (P) unclassified
D12690  Metopon (BAN); Methyldihydromorphinone (P) unclassified
D12691  Methyldesorphine (INN) (P) unclassified
D12692  Norlevorphanol (INN) (P) unclassified
D12693  Phenampromide (INN) (P) unclassified
D12694  Diampromide (INN) (P) unclassified
D12695  Levomoramide (INN) (P) unclassified
D12696  Levomethorphan (INN) (P) unclassified
D12697  Morpheridin (INN) (P) unclassified
D12698  Phenadoxone (INN) (P) unclassified
D12699  Dioxaphetyl butyrate (INN) (P) unclassified
D12700  Acetorphine (INN) (P) Target: OPRK1
D12701  Norpipanone (INN) (P) unclassified
D12752  Darunavir propylene glycolate (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D13025  Properidine (INN); Ipropethidine (P) unclassified