| C06624 |
Oxytetracycline; Oxytetracycline anhydrous |
(P) unclassified |
| C07005 |
Flunisolide; Flunisolide anhydrous |
(P) unclassified |
| C07051 |
Indinavir |
(P) unclassified |
| C07370 |
Prednisone; 1,2-Dehydrocortisone; 17,21-Dihydroxypregna-1,4-diene-3,11,20-trione |
(P) unclassified |
| C07521 |
Thiopental |
(P) unclassified |
| C11752 |
Carfecillin; Carbenicillin phenyl |
(P) unclassified |
| D00085 |
Insulin (JAN/USP) |
(P) unclassified |
| D00088 |
Hydrocortisone (JP19/USP/INN); HC; Acticort (TN); Anusol HC (TN); Colocort (TN); Cortef (TN); Hytone (TN); Plenadren (TN) |
(P) unclassified |
| D00107 |
Tacrolimus (USP/INN); Tacrolimus hydrate (JP19); Prograf (TN); Protopic (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D00109 |
Aspirin (JP19/USP); Aspalon (JAN); Acetylsalicylic acid; Easprin (TN); Durlaza (TN) |
(P) unclassified |
| D00130 |
Diflunisal (JAN/USP/INN); Dolobid (TN) |
(P) unclassified |
| D00136 |
Haloperidol (JP19/USP/INN); Haldol (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D00165 |
Hydrocortisone acetate (JP19/USP); Cortifoam (TN); U-cort (TN) |
(P) unclassified |
| D00184 |
Cyclosporine (USP); Ciclosporin (JP19); Gengraf (TN); Neoral (TN); Restasis (TN); Sandimmune (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D00201 |
Tetracycline (JAN/USP/INN); Sumycin (TN) |
(P) unclassified |
| D00204 |
Ampicillin (USP/INN); Anhydrous ampicillin (JP19); Omnipen (TN) |
(P) unclassified |
| D00205 |
Oxytetracycline (JAN/USP/INN); Oxytetracycline dihydrate; Terramycin (TN) |
(P) unclassified |
| D00211 |
Rifampin (USP); Rifampicin (JP19/INN); Rifadin (TN); Rimactane (TN) |
(P) CYP induction: CYP3A4 |
| D00216 |
Acarbose (JAN/USAN/INN); Precose (TN) |
(P) unclassified |
| D00217 |
Acetaminophen (JP19/USP); Paracetamol (INN); Tylenol (TN) |
(P) unclassified |
| D00219 |
Acetohexamide (JP19/USP/INN); Dymelor (TN) |
(P) unclassified |
| D00228 |
Amoxapine (JP19/USP/INN); Asendin (TN) |
(P) unclassified |
| D00229 |
Amoxicillin (USP); Amoxicillin hydrate (JP19); Amoxicilline (INN); Amoxicillin trihydrate; Amoxil (TN); Dispermox (TN); Pasetocin (TN) |
(P) unclassified |
| D00244 |
Betamethasone (JP19/USP/INN); Celestone (TN); Rinderon (TN) |
(P) unclassified |
| D00246 |
Budesonide (JP19/USP/INN); Entocort EC (TN); Pulmicort (TN); Rhinocort (TN); Uceris (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D00252 |
Carbamazepine (JP19/USP/INN); Equetro (TN); Tegretol (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4 |
| D00271 |
Chlorpropamide (JP19/USP/INN); Diabinese (TN) |
(P) unclassified |
| D00283 |
Clozapine (JAN/USP/INN); Clozaril (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D00290 |
Demeclocycline hydrochloride (USP); Demethylchlortetracycline hydrochloride (JP19); Declomycin (TN) |
(P) unclassified |
| D00292 |
Dexamethasone (JP19/USP/INN); Decadron (TN); Maxidex (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4 |
| D00293 |
Diazepam (JP19/USP/INN); Diastat (TN); Valium (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D00307 |
Doxycycline (USP); Doxycycline hydrate; Monodox (TN); Oracea (TN); Vibramycin (TN) |
(P) unclassified |
| D00320 |
Fentanyl (JAN/USP/INN); Duragesic (TN); Subsys (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D00322 |
Fluconazole (JP19/USP/INN); Diflucan (TN) |
(P) CYP inhibition: CYP3A4 |
| D00324 |
Flunisolide (JAN/USP); Aerospan (TN); Nasalide (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D00325 |
Fluocinonide (JP19/USP/INN); Lidex (TN); Vanos (TN) |
(P) unclassified |
| D00328 |
Flurandrenolide (USP); Fludroxycortide (JAN/INN); Cordran (TN) |
(P) unclassified |
| D00335 |
Glipizide (USP/INN); Glucotrol (TN) |
(P) unclassified |
| D00336 |
Glyburide (USP); Glibenclamide (JP19/INN); Diabeta (TN); Glynase (TN); Micronase (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D00354 |
Lamotrigine (JAN/USP/INN); Lamictal (TN) |
(P) unclassified |
| D00371 |
Theophylline (JP19); Elixophyllin (TN); Quibron-t (TN); Theo-24 (TN); Theodur G (TN); Theolair (TN); Uniphyl (TN) |
(P) unclassified |
| D00375 |
Mephenytoin (USP/INN); Mesantoin (TN) |
(P) unclassified |
| D00377 |
Mesalamine (USP); Mesalazine (JP19/INN); Apriso (TN); Asacol (TN); Canasa (TN); Delzicol (TN); Lialda (TN); Mesalamine (TN); Pentasa (TN); Rowasa (TN); Sfrowasa (TN) |
(P) unclassified |
| D00379 |
Tolazamide (JAN/USP/INN); Tolinase (TN) |
(P) unclassified |
| D00380 |
Tolbutamide (JAN/USP/INN); Orinase (TN) |
(P) unclassified |
| D00385 |
Triamcinolone (JP19/USP/INN); Aristocort (TN); Kenacort (TN) |
(P) unclassified |
| D00394 |
Trimipramine (USAN/INN) |
(P) unclassified |
| D00395 |
Troglitazone (JAN/USAN/INN); Rezulin (TN) |
(P) unclassified |
| D00407 |
Methylprednisolone (JP19/USP/INN); Medrol (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D00420 |
Mitotane (JAN/USP/INN); Lysodren (TN) |
(P) unclassified |
| D00426 |
Risperidone (JP19/USP/INN); Risperdal (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D00427 |
Ritonavir (JAN/USP/INN); Norvir (TN) |
(P) unclassified |
| D00428 |
Salsalate (USP/INN); Sasapyrine (JAN); Disalcid (TN) |
(P) unclassified |
| D00429 |
Saquinavir (JAN/USP/INN); Fortovase (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D00430 |
Secobarbital (USP/INN); Seconal (TN) |
(P) unclassified |
| D00435 |
Nevirapine (JAN/USP/INN); Viramune (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D00448 |
Sulfasalazine (USP/INN); Salazosulfapyridine (JP19); Azulfidine (TN) |
(P) unclassified |
| D00455 |
Omeprazole (JP19/USP/INN); Prilosec (TN) |
(P) unclassified |
| D00458 |
Quetiapine fumarate (JP19/USP); Seroquel (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D00466 |
Piperacillin sodium (JP19/USP); Pentcillin (TN); Pipracil (TN) |
(P) unclassified |
| D00472 |
Prednisolone (JP19/USP/INN); Delta-cortef (TN) |
(P) unclassified |
| D00473 |
Prednisone (USP); Prednisone monohydrate; Deltasone (TN); Meticorten (TN); Rayos (TN) |
(P) unclassified |
| D00474 |
Primidone (JP19/USP/INN); Mysoline (TN) |
(P) unclassified |
| D00484 |
Protriptyline hydrochloride (USP); Vivactil (TN) |
(P) unclassified |
| D00491 |
Paclitaxel (JAN/USP/INN); Abraxane (TN); Taxol (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D00497 |
Penicillin V potassium (USP); Phenoxymethylpenicillin potassium (JAN); Veetids (TN) |
(P) unclassified |
| D00499 |
Pentobarbital (USP/INN); Nembutal (TN) |
(P) unclassified |
| D00500 |
Pentobarbital sodium (JAN/USP); Nembutal sodium (TN) |
(P) unclassified |
| D00506 |
Phenobarbital (JP19/USP/INN); Luminal (TN) |
(P) unclassified |
| D00512 |
Phenytoin (JP19/USP/INN); Dilantin (TN) |
(P) unclassified |
| D00537 |
Topiramate (JAN/USP/INN); Topamax (TN); Trokendi xr (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D00550 |
Midazolam (JAN/USP/INN); Dormicum (TN); Buccolam (TN); Nayzilam (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D00555 |
Amobarbital (JP19/INN); Isomytal (TN) |
(P) unclassified |
| D00563 |
Mirtazapine (JAN/USP/INN); Remeron (TN); Reflex (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D00566 |
Sodium salicylate (JP19/USP); Salsonin (TN) |
(P) unclassified |
| D00570 |
Colchicine (JP19/USP) |
(CI,P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D00573 |
Goserelin acetate (JP19/USP); Zoladex (TN) |
(P) unclassified |
| D00578 |
Voriconazole (JP19/USP/INN); Vfend (TN) |
(P) unclassified |
| D00593 |
Glimepiride (JP19/USP/INN); Amaryl (TN) |
(P) unclassified |
| D00594 |
Repaglinide (JAN/USP/INN); Prandin (TN); Surepost (TN) |
(P) unclassified |
| D00595 |
Buformin (USAN/INN) |
(P) unclassified |
| D00596 |
Rosiglitazone maleate (JAN/USP); Avandia (TN) |
(P) unclassified |
| D00606 |
Guanfacine hydrochloride (JAN/USP); Intuniv (TN); Tenex (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D00615 |
Amlodipine besylate (USP); Amlodipine besilate (JP19); Norvasc (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D00619 |
Verapamil hydrochloride (JP19/USP); Calan (TN); Covera-hs (TN); Vasolan (TN); Verelan (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D00625 |
Miglitol (JP19/USAN/INN); Glyset (TN) |
(P) unclassified |
| D00636 |
Amiodarone hydrochloride (JP19/USP); Ancaron (TN); Cordarone (TN); Nexterone (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D00660 |
Tazobactam (JP19/USP/INN) |
(P) unclassified |
| D00661 |
Cevimeline hydrochloride (USAN); Cevimeline hydrochloride hydrate (JAN); Evoxac (TN); Saligren (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D00670 |
Donepezil hydrochloride (JP19/USP); Aricept (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D00687 |
Salmeterol xinafoate (JAN/USP); Serevent (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D00689 |
Beclomethasone dipropionate (USP); Beclometasone dipropionate (JP19); Beclovent (TN); Qnasl (TN); Vanceril (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D00690 |
Mometasone furoate (JAN/USP); Asmanex (TN); Elocon (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D00698 |
Aprobarbital (INN); Alurate (TN) |
(P) unclassified |
| D00699 |
Butabarbital sodium (USP); Secbutabarbital sodium (INN); Butabarb (TN); Butisol sodium (TN) |
(P) unclassified |
| D00700 |
Mephobarbital (JAN/USP); Methylphenobarbital (INN); Mebaral (TN) |
(P) unclassified |
| D00701 |
Phenobarbital sodium (JAN/USP/INN); Luminal sodium (TN) |
(P) unclassified |
| D00708 |
Ethotoin (JAN/USP/INN); Accenon (TN); Peganone (TN) |
(P) unclassified |
| D00712 |
Methohexital sodium (USP); Brevital sodium (TN) |
(P) unclassified |
| D00713 |
Thiamylal sodium (JP19); Surital (TN) |
(P) unclassified |
| D00714 |
Thiopental sodium (JP19/USP/INN); Pentothal (TN) |
(P) unclassified |
| D00722 |
Oxybutynin chloride (USP); Oxybutynin hydrochloride (JP19); Ditropan (TN); Gelnique (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D00727 |
Olsalazine sodium (USAN); Dipentum (TN) |
(P) unclassified |
| D00751 |
Methylprednisolone sodium succinate (JAN/USP); A-methapred (TN); Solu-medrol (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D00785 |
Selegiline hydrochloride (JAN/USP); Eldepryl (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D00809 |
Amitriptyline hydrochloride (JP19/USP); Elavil (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D00810 |
Choline salicylate (JAN/USAN/INN); Arthropan (TN) |
(P) unclassified |
| D00811 |
Clomipramine hydrochloride (JP19/USP); Anafranil (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D00812 |
Desipramine hydrochloride (JAN/USP); Norpramin (TN) |
(P) unclassified |
| D00814 |
Doxepin hydrochloride (USP); Sinequan (TN); Zonalon (TN) |
(P) unclassified |
| D00815 |
Imipramine hydrochloride (JP19/USP); Tofranil (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D00816 |
Nortriptyline hydrochloride (JP19/USP/INN); Pamelor (TN) |
(P) unclassified |
| D00820 |
Trazodone hydrochloride (JAN/USP); Desyrel (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D00821 |
Venlafaxine hydrochloride (JAN/USP); Effexor (TN) |
(P) unclassified |
| D00827 |
Magnesium salicylate (USP); Magnesium salicylate tetrahydrate; Magan (TN) |
(P) unclassified |
| D00831 |
Mefloquine hydrochloride (JP19/USP); Lariam (TN) |
(P) unclassified |
| D00836 |
Buprenorphine hydrochloride (JP19/USP); Buprenex (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D00842 |
Morphine sulfate (USP); Morphine sulfate hydrate (JP19); Morphine sulfate pentahydrate; Astramor PH (TN); Avinza (TN); Depodur (TN); Kadian (TN); MS contin (TN) |
(P) unclassified |
| D00849 |
Methacycline hydrochloride (JAN/USP); Rondomycin (TN) |
(P) unclassified |
| D00850 |
Minocycline hydrochloride (JP19/USP); Arestin (TN); Dynacin (TN); Minocin (TN); Solodyn (TN) |
(P) unclassified |
| D00894 |
Amprenavir (JAN/USAN/INN); Agenerase (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D00895 |
Delavirdine mesylate (USAN); Delavirdine mesilate (JAN); Rescriptor (TN) |
(P) unclassified |
| D00896 |
Efavirenz (JAN/USP/INN); Sustiva (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4 |
| D00897 |
Indinavir sulfate (USP); Crixivan (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D00899 |
Nelfinavir mesylate (USAN/INN); Nelfinavir mesilate (JAN); Viracept (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D00927 |
Bacampicillin hydrochloride (JP19/USAN); Spectrobid (TN) |
(P) unclassified |
| D00928 |
Nafcillin sodium (USP); Nafcillin sodium monohydrate; Unipen (TN) |
(P) unclassified |
| D00929 |
Oxacillin sodium (JAN/USP); Oxacillin sodium hydrate; Bactocill (TN) |
(P) unclassified |
| D00944 |
Metformin hydrochloride (JP19/USP); Glucophage (TN) |
(P) unclassified |
| D00945 |
Pioglitazone hydrochloride (JP19/USP); Actos (TN) |
(P) unclassified |
| D00951 |
Medroxyprogesterone acetate (JP19/USP); Depo-provera (TN); Depo-subq provera 104 (TN); Provera (TN) |
(CI,P) unclassified |
| D00961 |
Bicalutamide (JP19/USP/INN); Casodex (TN) |
(P) CYP inhibition: CYP3A4 |
| D00964 |
Letrozole (JAN/USP/INN); Femara (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D00971 |
Sodium thiosalicylate; Thiosalicylic acid sodium salt; Rexolate (TN) |
(P) unclassified |
| D00972 |
Betamethasone sodium phosphate (JP19/USP); Celestone (TN) |
(P) unclassified |
| D00973 |
Cortisone acetate (JP19/USP); Cortone acetate (TN) |
(P) unclassified |
| D00975 |
Dexamethasone sodium phosphate (JAN/USP); Dalalone (TN); Maxidex (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4 |
| D00976 |
Hydrocortisone cypionate |
(P) unclassified |
| D00977 |
Hydrocortisone sodium phosphate (JP19/USP); Hydrocortone phosphate (TN) |
(P) unclassified |
| D00978 |
Hydrocortisone sodium succinate (JP19/USP); A-hydrocort (TN); Solu-cortef (TN) |
(P) unclassified |
| D00979 |
Methylprednisolone acetate (JAN/USP); Depo-medrol (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D00980 |
Prednisolone acetate (JP19/USP/INN); Econopred (TN); Pred forte (TN) |
(P) unclassified |
| D00981 |
Prednisolone sodium phosphate (JP19/USP); Pediapred (TN) |
(P) unclassified |
| D00982 |
Prednisolone tebutate (JAN/USP); Hydeltra-TBA (TN) |
(P) unclassified |
| D00983 |
Triamcinolone acetonide (JP19/USP); Azmacort (TN); Kenalog (TN); Nasacort (TN) |
(P) unclassified |
| D00984 |
Triamcinolone diacetate (JAN/USP); Aristocort (TN) |
(P) unclassified |
| D00985 |
Triamcinolone hexacetonide (USP/INN); Aristospan (TN) |
(P) unclassified |
| D00986 |
Fludrocortisone acetate (JP19/USP); Florinef acetate (TN) |
(P) unclassified |
| D00988 |
Gonadorelin hydrochloride (USP); Factrel (TN) |
(P) unclassified |
| D00989 |
Leuprolide acetate (USP); Leuprorelin acetate (JP19); Lupron (TN); Lutrate (TN); Eligard (TN); Fensolvi (TN) |
(P) unclassified |
| D00990 |
Nafarelin acetate (USAN); Nafarelin acetate hydrate (JAN); Synarel (TN) |
(P) unclassified |
| D01010 |
Levothyroxine sodium (USP); Levothyroxine sodium hydrate (JP19); Levothroid (TN); Levoxyl (TN); Synthroid (TN) |
(P) unclassified |
| D01011 |
Liothyronine sodium (JP19/USP); Cytomel (TN); Triostat (TN) |
(P) unclassified |
| D01053 |
Penicillin G potassium (USP); Benzylpenicillin potassium (JP19); Pfizerpen (TN) |
(P) unclassified |
| D01055 |
Emivirine (USAN/INN); Coactinon (TN) |
(P) unclassified |
| D01061 |
Irinotecan hydrochloride (USP); Irinotecan hydrochloride hydrate (JP19); Irinotecan hydrochloride trihydrate; CPT 11; CPT-11; Campto (TN); Camptosar (TN); Onivyde (TN) |
(P) unclassified |
| D01071 |
Hexobarbital (JAN/INN) |
(P) unclassified |
| D01074 |
Hetacillin (USAN/INN); Versapen (TN) |
(P) unclassified |
| D01079 |
Tigecycline (JAN/USP); Tygacil (TN) |
(P) unclassified |
| D01087 |
Methyl salicylate (JP19/NF) |
(P) unclassified |
| D01110 |
Melitracen hydrochloride (JAN/USAN) |
(P) unclassified |
| D01111 |
Nateglinide (JP19/USP/INN); Starsis (TN) |
(P) unclassified |
| D01115 |
Eplerenone (JP19/USAN/INN); Inspra (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D01160 |
Saquinavir mesylate (USP); Saquinavir mesilate (JAN); Invirase (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D01164 |
Aripiprazole (JP19/USP/INN); Abilify (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D01176 |
Blonanserin (JP19/INN); AD 5423 |
(CI,P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D01178 |
Phenethicillin potassium (JP19); Pheneticillin potassium; Syncillin (TN); Synthepen (TN) |
(P) unclassified |
| D01207 |
Omeprazole sodium (USAN); Losec sodium (TN) |
(P) unclassified |
| D01213 |
Tolvaptan (JP19/USAN/INN); Samsca (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D01214 |
Tobicillin (JAN/INN) |
(P) unclassified |
| D01227 |
Bosentan (USAN); Bosentan hydrate (JAN); Tracleer (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4 |
| D01229 |
Paramethasone acetate (JAN/USAN); Haldrone (TN) |
(P) unclassified |
| D01239 |
Prednisolone sodium succinate (JP19/USP); Kohakusanin (TN) |
(P) unclassified |
| D01249 |
Flucloxacillin sodium (JAN); Flucloxacillin sodium hydrate; Floxapen (TN) |
(P) unclassified |
| D01251 |
Ampicillin hydrate (JP19); Ampicillin trihydrate; Amcill (TN) |
(P) unclassified |
| D01253 |
Clobazam (JAN/USAN/INN); Mystan (TN); Onfi (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D01266 |
Difluprednate (JAN/USAN/INN); Durezol (TN) |
(P) unclassified |
| D01272 |
Clobetasol propionate (JP19/USP); Clobex (TN); Cormax (TN); Olux (TN) |
(P) unclassified |
| D01273 |
Clobetasone butyrate (JAN/USAN); Kindavate (TN) |
(P) unclassified |
| D01276 |
Atazanavir sulfate (JAN/USAN); Reyataz (TN) |
(P) CYP inhibition: CYP3A4 |
| D01283 |
Carbenicillin indanyl sodium (USP); Carindacillin sodium (JAN); Geocillin (TN) |
(P) unclassified |
| D01285 |
Lofepramine hydrochloride (JAN/USAN); Amplit (TN) |
(P) unclassified |
| D01287 |
Levobupivacaine hydrochloride (JAN/USAN); Chirocaine (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D01308 |
Halcinonide (JAN/USP/INN); Halog (TN) |
(P) unclassified |
| D01310 |
Secobarbital sodium (JAN/USP); Seconal sodium (TN) |
(P) unclassified |
| D01314 |
Dibenzepin hydrochloride (JAN/USAN) |
(P) unclassified |
| D01327 |
Diflorasone diacetate (JP19/USP); Florone (TN); Psorcon (TN) |
(P) unclassified |
| D01334 |
Cyclacillin (USAN); Ciclacillin (JP19/INN); Cyclapen-W (TN); Vastcillin (TN) |
(P) unclassified |
| D01356 |
Glymidine sodium (JAN/USAN/INN) |
(P) unclassified |
| D01357 |
Betamethasone valerate (JP19/USP); Beta-Val (TN); Luxiq (TN); Rinderon-V (TN) |
(P) unclassified |
| D01367 |
Fluorometholone (JP19/USP/INN); NSC 33001; Fluor-op (TN); Fml (TN); Oxylone (TN) |
(P) unclassified |
| D01372 |
Zopiclone (JP19/INN); Amoban (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D01382 |
Metharbital (JAN/INN); Gemonil (TN) |
(P) unclassified |
| D01387 |
Amcinonide (JAN/USP/INN); Cyclocort (TN) |
(P) unclassified |
| D01399 |
Fentanyl citrate (JP19/USP); Abstral (TN); Fentora (TN); Lazanda (TN); Oralet (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D01402 |
Betamethasone acetate (JAN/USP) |
(P) unclassified |
| D01418 |
Tamibarotene (JAN/USAN/INN); Am 80; Amnoid (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D01425 |
Lopinavir (JAN/USP/INN) |
(P) unclassified |
| D01429 |
Fosfluconazole (JAN/INN); Prodif (TN) |
(P) CYP inhibition: CYP3A4 |
| D01434 |
Deprodone propionate (JAN); Allomidon (TN) |
(P) unclassified |
| D01442 |
Hydrocortisone succinate (JP19) |
(P) unclassified |
| D01464 |
Flumethasone pivalate (USP); Flumetasone pivalate (JAN/BAN); Locorten (TN) |
(P) unclassified |
| D01466 |
Ethenzamide (JP19/INN) |
(P) unclassified |
| D01477 |
Opipramol hydrochloride (JAN/USAN); Insidon (TN) |
(P) unclassified |
| D01486 |
Rolitetracycline nitrate (JAN/USAN) |
(P) unclassified |
| D01489 |
Sulbenicillin sodium (JP19); Lilacillin (TN) |
(P) unclassified |
| D01499 |
Pivmecillinam hydrochloride (JP19); Melysin (TN); Pivya (TN) |
(P) unclassified |
| D01510 |
Dexamethasone metasulfobenzoate sodium (JAN); Dexamethazone metasulfobenzoate sodium; Dexapos; Santeson (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4 |
| D01546 |
Dothiepin hydrochloride (USAN); Dosulepin hydrochloride (JAN); Prothiaden (TN) |
(P) unclassified |
| D01557 |
Glycol salicylate (JAN); Ethylene glycol salicylate; Norgesic (TN); Phlogont (TN) |
(P) unclassified |
| D01596 |
Oxytetracycline hydrochloride (JP19/USP); Terramycin (TN) |
(P) unclassified |
| D01599 |
Gliclazide (JP19/INN); Glimicron (TN) |
(P) unclassified |
| D01615 |
Dexamethasone palmitate (JAN); Dexamethasone 21-palmitate; Limethason (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4 |
| D01619 |
Hydrocortisone butyrate (JP19/USP); Locoid (TN) |
(P) unclassified |
| D01632 |
Dexamethasone dipropionate (USAN); Dexamethasone propionate (JAN); Hifmeta (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4 |
| D01637 |
Betamethasone dipropionate (JP19/USP); Diprolene (TN); Rinderon-DP (TN); Sernivo (TN) |
(P) unclassified |
| D01649 |
Propicillin potassium (JAN) |
(P) unclassified |
| D01665 |
Voglibose (JP19/USAN/INN); Basen (TN) |
(P) unclassified |
| D01668 |
Sultamicillin tosilate hydrate (JP19); Sultamicillin tosylate dihydrate; Unasyn (TN) |
(P) unclassified |
| D01689 |
Loteprednol etabonate (JAN/USAN); Lotemax (TN) |
(P) unclassified |
| D01696 |
Lenampicillin hydrochloride (JP19); Kbt 1585; Valacillin (TN) |
(P) unclassified |
| D01703 |
Ciclesonide (JAN/USAN/INN); Alvesco (TN); Omnaris (TN); Zetonna (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D01708 |
Fluticasone propionate (JAN/USP); Cutivate (TN); Flonase (TN); Flovent (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D01712 |
Theophylline sodium acetate (JAN) |
(P) unclassified |
| D01740 |
Barbital (JP19/INN) |
(P) unclassified |
| D01744 |
Brotizolam (JP19/USAN/INN); Lendormin (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D01745 |
Domperidone (JP19/USAN/INN); Motilium (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D01764 |
Diflucortolone valerate (JP19); Afusona (TN) |
(P) unclassified |
| D01799 |
Glyclopyramide (JAN/INN); Deamelin-S (TN) |
(P) unclassified |
| D01811 |
Salicylamide (JAN/USP/INN) |
(P) unclassified |
| D01820 |
Alclometasone dipropionate (JAN/USP); Aclovate (TN) |
(P) unclassified |
| D01825 |
Fluocinolone acetonide (JP19/USP/INN); Fluocet (TN); Retisert (TN); Synalar (TN) |
(P) unclassified |
| D01831 |
Buserelin acetate (JAN/USAN); Suprecur (TN) |
(P) unclassified |
| D01832 |
Modafinil (JAN/USP/INN); Provigil (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4 |
| D01854 |
Mitiglinide calcium hydrate (JP19); Mitiglinide calcium dihydrate; Glufast (TN) |
(P) unclassified |
| D01886 |
Hydrocortisone probutate (USAN); Hydrocortisone butyrate propionate (JAN); Hydrocortisone buteprate; Pandel (TN) |
(P) unclassified |
| D01896 |
Cilostazol (JP19/USP/INN); Pletal (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D01898 |
Haloperidol decanoate (JAN/USP); Halomonth (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D01948 |
Dexamethasone valerate (JAN); Dexamethasone 17-valerate; DV-17; Voalla ointment (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4 |
| D01977 |
Gefitinib (JP19/USAN/INN); Iressa (TN) |
(P) unclassified |
| D01998 |
Prednisolone farnesylate (JAN); PNF 21; Farnerate (TN) |
(P) unclassified |
| D02008 |
Tadalafil (JAN/USP/INN); Adcirca (TN); Cialis (TN); Zalutia (TN) |
(CI,P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D02032 |
Betamethasone butyrate propionate (JAN); Antebate (TN) |
(P) unclassified |
| D02096 |
Fosphenytoin sodium (USP); Cerebyx (TN); Sesquient (TN) |
(P) CYP induction: CYP3A4 |
| D02103 |
Phenytoin sodium (USP); Phenytoin sodium for injection (JP19); Aleviatin (TN); Dilantin (TN) |
(P) unclassified |
| D02116 |
Histrelin acetate; Vantas (TN); Supprelin (TN) |
(P) unclassified |
| D02119 |
Ampicillin sodium (JP19/USP); Omnipen-N (TN); Viccillin (TN) |
(P) unclassified |
| D02122 |
Tetracycline hydrochloride (JP19/USP); Bristacycline (TN) |
(P) unclassified |
| D02129 |
Doxycycline hyclate (USP); Doxycycline hydrochloride hydrate (JP19); Doryx (TN); Lymepak (TN); Periostat (TN); Vibra-tabs (TN) |
(P) unclassified |
| D02137 |
Dicloxacillin sodium (USP); Dicloxacillin sodium hydrate (JP19); Dycill (TN) |
(P) unclassified |
| D02156 |
Prednisolone hemisuccinate (USP); Prednisolone succinate (JP19) |
(P) unclassified |
| D02157 |
Penicillin G benzathine (USP); Benzylpenicillin benzathine hydrate (JP19); Bicillin L-A (TN); Permapen (TN); Wycillin (TN); Stelues (TN) |
(P) unclassified |
| D02174 |
Dexamethasone acetate (JAN/USP); Decadronal (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4 |
| D02190 |
Carbenicillin disodium (USP); Carbenicillin sodium (JAN); Geopen (TN) |
(P) unclassified |
| D02196 |
Methicillin sodium (USAN); Meticillin sodium (JAN); Methicillin sodium monohydrate; Staphcillin (TN) |
(P) unclassified |
| D02199 |
Carbenicillin phenyl sodium (USAN); Carfecillin sodium (JAN) |
(P) unclassified |
| D02201 |
Talampicillin hydrochloride (JP19/USAN); Aseocillin (TN) |
(P) unclassified |
| D02203 |
Hetacillin potassium (JAN/USAN); Hetacin-K (TN) |
(P) unclassified |
| D02206 |
Buformin hydrochloride (JP19); Dibetos-B (TN) |
(P) unclassified |
| D02219 |
Terbinafine hydrochloride (JP19/USP); Lamisil (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D02221 |
Mezlocillin sodium (JAN); Mezlocillin sodium monohydrate; Mezlin (TN) |
(P) unclassified |
| D02223 |
Sulbactam sodium (JP19/USP); SBT |
(P) unclassified |
| D02229 |
Sildenafil citrate (JAN/USP); Revatio (TN); Viagra (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D02231 |
Cloxacillin sodium (USP); Cloxacillin sodium hydrate (JP19); Cloxapen (TN); Tegopen (TN) |
(P) unclassified |
| D02241 |
Ticarcillin disodium (USP); Ticarcillin sodium (JAN); Ticar (TN) |
(P) unclassified |
| D02251 |
Piperacillin (USP); Piperacillin hydrate (JP19) |
(P) unclassified |
| D02252 |
Amobarbital sodium (JAN/USP); Amytal sodium (TN) |
(P) unclassified |
| D02253 |
Pentobarbital calcium (JP19); Ravona (TN) |
(P) unclassified |
| D02255 |
Chlortetracycline hydrochloride (JAN/USP); Aureomycin (TN) |
(P) unclassified |
| D02271 |
Morphine hydrochloride hydrate (JP19); Morphine hydrochloride trihydrate; Anpec (TN) |
(P) unclassified |
| D02282 |
Rolitetracycline (JAN/USAN/INN); Synterin (TN) |
(P) unclassified |
| D02286 |
Betamethasone benzoate (USP); Uticort (TN) |
(P) unclassified |
| D02287 |
Clocortolone pivalate (USP); Cloderm (TN) |
(P) unclassified |
| D02288 |
Hydrocortisone valerate (USP); Westcort (TN) |
(P) unclassified |
| D02289 |
Medrysone (USAN); HMS (TN) |
(P) unclassified |
| D02336 |
Benzylpenicillin (INN); Penicillin G |
(P) unclassified |
| D02339 |
Azlocillin (USAN/INN) |
(P) unclassified |
| D02348 |
Dicloxacillin (USAN/INN) |
(P) unclassified |
| D02369 |
Histrelin (USAN/INN); Vantas (TN) |
(P) unclassified |
| D02372 |
Perospirone hydrochloride hydrate (JP19); Lullan (TN) |
(P) unclassified |
| D02405 |
Penicillin V benzathine (USP) |
(P) unclassified |
| D02408 |
Trimipramine maleate (JAN/USP); Surmontil (TN) |
(P) unclassified |
| D02415 |
Apalcillin sodium (USAN) |
(P) unclassified |
| D02425 |
Carbutamide (INN); Invenol (TN) |
(P) unclassified |
| D02426 |
Glycyclamide (INN); Tolcyclamide |
(P) unclassified |
| D02427 |
Glibornuride (USAN/INN); Glutril (TN) |
(P) unclassified |
| D02428 |
Glisentide (INN); Glypentide; Staticum (TN) |
(P) unclassified |
| D02429 |
Glisolamide (INN); Glysolamide; Diabenor (TN) |
(P) unclassified |
| D02430 |
Gliquidone (INN); Glurenorm (TN) |
(P) unclassified |
| D02461 |
Penicillin G procaine (USP); Duracillin (TN) |
(P) unclassified |
| D02476 |
Meclocycline (USAN/INN) |
(P) unclassified |
| D02477 |
Meclocycline sulfosalicylate (USP); Meclan (TN) |
(P) unclassified |
| D02484 |
Artemether and lumefantrine; Coartem (TN) |
(P) unclassified |
| D02497 |
Fosamprenavir (INN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D02498 |
Lopinavir and ritonavir; Kaletra (TN) |
(P) unclassified |
| D02504 |
Aspoxicillin hydrate (JP19); ASPC; Doyle (TN) |
(P) unclassified |
| D02506 |
Phenoxymethylpenicillin benzathine (JAN); Penicillin V benzathine tetrahydrate |
(P) unclassified |
| D02508 |
Pivampicillin hydrochloride (USAN) |
(P) unclassified |
| D02554 |
Rifaximin (JAN/USAN/INN); Xifaxan (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4 |
| D02565 |
Dimetacrine (INN) |
(P) unclassified |
| D02591 |
Dexamethasone acefurate (USAN/INN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4 |
| D02592 |
Dexamethasone beloxil (USAN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4 |
| D02618 |
Butobarbital (BAN); Butethal; Neonal (TN) |
(P) unclassified |
| D02624 |
Eszopiclone (JAN/USP/INN); Estorra (TN); Lunesta (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D02689 |
Ramelteon (JAN/USAN/INN); Rozerem (TN) |
(P) unclassified |
| D02691 |
Somatropin (USP/INN); Somatropin (genetical recombination) (JAN); Human growth hormone (JAN); Asellacrin (TN); Humatrope (TN); Nutropin (TN); Omnitrope (TN) |
(P) unclassified |
| D02704 |
Tampramine fumarate (USAN) |
(P) unclassified |
| D02715 |
Balsalazide disodium (USP); Colazide (TN) |
(P) unclassified |
| D02732 |
Pranlukast hydrate (JP19); Onon (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D02797 |
Albutoin (USAN/INN); Euprax (TN) |
(P) unclassified |
| D02817 |
Allobarbital (USAN/INN) |
(P) unclassified |
| D02861 |
Indinavir sulfate ethanolate (JAN); Crixivan (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D02867 |
Fosamprenavir calcium hydrate (JAN); Lexiva (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D02888 |
Amdinocillin (USAN); Mecillinam (INN); Coactin (TN) |
(P) unclassified |
| D02889 |
Pivmecillinam (INN); Amdinocillin pivoxil; Coactabs (TN) |
(P) unclassified |
| D02899 |
Amicycline (USAN/INN) |
(P) unclassified |
| D02925 |
Amoxicillin sodium (USAN) |
(P) unclassified |
| D02968 |
Aprepitant (JAN/USP/INN); Aponvie (TN); Emend (TN); Cinvanti (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4 |
| D03001 |
Atevirdine mesylate (USAN) |
(P) unclassified |
| D03038 |
Azipramine hydrochloride (USAN) |
(P) unclassified |
| D03039 |
Azlocillin sodium; Azlin (TN) |
(P) unclassified |
| D03106 |
Bexarotene (JAN/USAN/INN); Targretin (TN) |
(P) unclassified |
| D03150 |
Bortezomib (JAN/USAN/INN); Velcade (TN) |
(P) unclassified |
| D03180 |
Butabarbital (USP); Secbutabarbital (BAN) |
(P) unclassified |
| D03182 |
Butalbital (USP/INN); Sandoptal (TN) |
(P) unclassified |
| D03199 |
Butriptyline hydrochloride (USAN) |
(P) unclassified |
| D03218 |
Axitinib (JAN/USAN); Inlyta (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D03230 |
Insulin human (USP/INN); Insulin human (genetical recombination) (JP19); Insulin human (biosynthesis) (JAN); Insulin human (synthesis) (JAN); Humulin (TN) |
(P) unclassified |
| D03250 |
Insulin glargine (USAN/INN); Insulin glargine (genetical recombination) (JP19); Insulin glargine (genetical recombination) [Insulin glargin biosimilar 1] (JAN); Insulin glargine (genetical recombination) [Insulin glargin biosimilar 2] (JAN); Insulin glargine-yfgn; Lantus (TN) |
(P) unclassified |
| D03253 |
Brecanavir (USAN) |
(P) unclassified |
| D03260 |
Vardenafil hydrochloride hydrate (JAN); Vardenafil monohydrochloride trihydrate; Levitra (TN); Staxyn (TN) |
(CI,P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D03267 |
Gonadorelin diacetate (JP19) |
(P) unclassified |
| D03301 |
Prednisolone valerate acetate (JAN); PDL; Spirazon (TN) |
(P) unclassified |
| D03325 |
Mometasone furoate hydrate (JAN); Mometasone furoate monohydrate; Nasonex (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D03371 |
Capravirine (USAN/INN) |
(P) unclassified |
| D03385 |
Carbaspirin calcium (USAN); Carbasalate calcium (INN) |
(P) unclassified |
| D03387 |
Carbenicillin potassium (USAN) |
(P) unclassified |
| D03451 |
Cetocycline hydrochloride (USAN) |
(P) unclassified |
| D03477 |
Chlortetracycline bisulfate (USP) |
(P) unclassified |
| D03491 |
Cidoxepin hydrochloride (USAN) |
(P) unclassified |
| D03541 |
Clocortolone acetate (USAN) |
(P) unclassified |
| D03561 |
Cloprednol (USAN/INN); Cloradryn (TN) |
(P) unclassified |
| D03571 |
Cloxacillin benzathine (USP) |
(P) unclassified |
| D03594 |
Cortivazol (USAN) |
(P) unclassified |
| D03656 |
Darunavir (USAN/INN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D03658 |
Dasatinib (JAN/INN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D03669 |
Deferasirox (JAN/USAN/INN); Exjade (TN); Jadenu (TN) |
(P) CYP induction: CYP3A4 |
| D03671 |
Deflazacort (USAN/INN); Emflaza (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D03680 |
Demeclocycline (USP); Demethylchlortetracycline (JAN) |
(P) unclassified |
| D03681 |
Demecycline (USAN/INN) |
(P) unclassified |
| D03694 |
Deslorelin (USAN/INN) |
(P) unclassified |
| D03696 |
Desonide (USP/INN); Desowen (TN); Verdeso (TN) |
(P) unclassified |
| D03697 |
Desoximetasone (USP/INN); Topicort (TN) |
(P) unclassified |
| D03705 |
Sulbactam benzathine (USAN) |
(P) unclassified |
| D03706 |
Sulbactam pivoxil (USAN) |
(P) unclassified |
| D03707 |
Tazobactam sodium (JAN/USAN) |
(P) unclassified |
| D03799 |
Dienogest (JAN/USAN/INN); Endometrion (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D03812 |
Diflucortolone (USAN) |
(P) unclassified |
| D03813 |
Diflucortolone pivalate (USAN) |
(P) unclassified |
| D03820 |
Dutasteride (JAN/USP/INN); Avodart (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D03833 |
Indinavir (USAN); Indinavir hydrate |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D03835 |
Fosamprenavir calcium (USAN); Lexiva (TN); Telzir (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D03837 |
Fosamprenavir sodium (USAN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D03839 |
Droxinavir hydrochloride (USAN) |
(P) unclassified |
| D03840 |
Palinavir (USAN/INN) |
(P) unclassified |
| D03842 |
Telinavir (USAN/INN) |
(P) unclassified |
| D03843 |
Tipranavir disodium (USAN) |
(P) unclassified |
| D03903 |
Doxycycline calcium (USP) |
(P) unclassified |
| D03904 |
Doxycycline fosfatex (USAN) |
(P) unclassified |
| D04020 |
Epicillin (USAN/INN); Dexacillin (TN) |
(P) unclassified |
| D04023 |
Erlotinib hydrochloride (JAN/USAN); Tarceva (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D04024 |
Lapatinib ditosylate (USAN); Lapatinib tosilate hydrate (JAN); Lapatinib ditosylate monohydrate; Tykerb (TN); Tyverb (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D04030 |
Epitetracycline hydrochloride (USP) |
(P) unclassified |
| D04077 |
Eterobarb (USAN/INN); Antilon (TN) |
(P) unclassified |
| D04103 |
Etoformin hydrochloride (USAN) |
(P) unclassified |
| D04112 |
Etravirine (JAN/USAN/INN); Intelence (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4 |
| D04121 |
Exenatide (JAN/USAN/INN); Byetta (TN) |
(P) unclassified |
| D04145 |
Fendosal (USAN/INN); Alnovin (TN) |
(P) unclassified |
| D04174 |
Fertirelin acetate (USAN) |
(P) unclassified |
| D04196 |
Floxacillin (USAN); Flucloxacillin (INN); Floxapen (TN) |
(P) unclassified |
| D04201 |
Flucloronide (USAN); Fluclorolone acetonide (INN) |
(P) unclassified |
| D04206 |
Flufenisal (USAN/INN) |
(P) unclassified |
| D04208 |
Flumethasone (USAN); Flumetasone (INN) |
(P) unclassified |
| D04214 |
Flunisolide acetate (USAN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D04217 |
Fluocortin butyl (USAN) |
(P) unclassified |
| D04218 |
Fluocortolone (USAN/INN) |
(P) unclassified |
| D04219 |
Fluocortolone caproate (USAN) |
(P) unclassified |
| D04221 |
Fluorometholone acetate (USP); Fluorometholone 17-acetate; Flarex (TN) |
(P) unclassified |
| D04225 |
Fluperolone acetate (USAN); Methral (TN) |
(P) unclassified |
| D04244 |
Formocortal (USAN/INN); Deflamene (TN) |
(P) unclassified |
| D04270 |
Fumoxicillin (USAN/INN) |
(P) unclassified |
| D04322 |
Gliamilide (USAN/INN) |
(P) unclassified |
| D04354 |
Glyhexamide (USAN/INN); Subose (TN) |
(P) unclassified |
| D04355 |
Glyoctamide (USAN/INN) |
(P) unclassified |
| D04356 |
Glyparamide (USAN) |
(P) unclassified |
| D04361 |
Gonadorelin acetate (USP); Luteinizing (TN) |
(P) unclassified |
| D04403 |
Guar gum (NF) |
(P) unclassified |
| D04405 |
Goserelin (USAN/INN) |
(P) unclassified |
| D04409 |
Halobetasol propionate (USP); Ulobetasol propionate; Ultravate (TN) |
(P) unclassified |
| D04467 |
Hydrocortisone hemisuccinate (USP) |
(P) unclassified |
| D04475 |
Insulin aspart (USP/INN); Insulin aspart (genetical recombination) (JP19); Insulin aspart (genetical recombination) [Insulin aspart biosimilar 1] (JAN); Insulin X 14; Insulin aspart-szjj; nsulin aspart-xjhz; Merilog (TN); NovoRapid (TN); Novolog (TN); Kirsty (TN) |
(P) unclassified |
| D04477 |
Insulin lispro (USP/INN); Insulin lispro (genetical recombination) (JAN); Insulin lispro (genetical recombination) [Insulin lispro Biosimilar 1] (JAN); Insulin lispro-aabc; Humalog (TN); Lyumjev (TN) |
(P) unclassified |
| D04539 |
Insulin detemir (USAN/INN); Insulin detemir (genetical recombination) (JAN); Levemir (TN) |
(P) unclassified |
| D04540 |
Insulin glulisine (USAN/INN); Insulin glulisine (genetical recombination) (JAN); Apidra (TN) |
(P) unclassified |
| D04541 |
Insulin human, isophane (USP) |
(P) unclassified |
| D04542 |
Insulin human zinc (USP) |
(P) unclassified |
| D04543 |
Insulin human zinc, extended (USP) |
(P) unclassified |
| D04547 |
Insulin, isophane (USP); Isophane insulin (aqueous suspension) (JAN); Humalog PEN (TN) |
(P) unclassified |
| D04550 |
Insulin zinc, prompt (USP); Semilente iletin (TN) |
(P) unclassified |
| D04551 |
Insulin zinc (USP); Lente iletin (TN) |
(P) unclassified |
| D04556 |
Intriptyline hydrochloride (USAN) |
(P) unclassified |
| D04605 |
Iprindole (USAN/INN) |
(P) unclassified |
| D04641 |
Istradefylline (JAN/USAN/INN); Nourianz (TN); Nouriast (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D04652 |
Ketipramine fumarate (USAN) |
(P) unclassified |
| D04666 |
Lanreotide acetate (JAN/USAN); Somatuline (TN) |
(P) unclassified |
| D04719 |
Levopropylcillin potassium (USAN) |
(P) unclassified |
| D04768 |
Lonafarnib (JAN/USAN/INN); Zokinvy (TN) |
(CI,P) unclassified |
| D04786 |
Loviride (USAN/INN) |
(P) unclassified |
| D04820 |
Lurasidone hydrochloride (JAN/USAN); SM 13496; Latuda (TN) |
(CI,P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D04823 |
Lutrelin acetate (USAN) |
(P) unclassified |
| D04966 |
Metformin (USAN/INN) |
(P) unclassified |
| D04972 |
Methacycline (USAN); Metacycline (INN) |
(P) unclassified |
| D04982 |
Methetoin (USAN/INN) |
(P) unclassified |
| D04985 |
Methohexital (USP/INN) |
(P) unclassified |
| D05000 |
Methylprednisolone hemisuccinate (USP); Methylprednisolone succinate (JP19) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D05001 |
Methylprednisolone sodium phosphate (USAN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D05002 |
Methylprednisolone suleptanate (USAN/INN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D05021 |
Mezlocillin (USAN/INN) |
(P) unclassified |
| D05022 |
Mezlocillin sodium (USP) |
(P) unclassified |
| D05045 |
Minocycline (USAN/INN) |
(P) unclassified |
| D05181 |
Aspirin aluminum (JP19) |
(P) unclassified |
| D05184 |
Nitrocycline (USAN/INN) |
(P) unclassified |
| D05231 |
Octriptyline phosphate (USAN) |
(P) unclassified |
| D05259 |
Omeprazole magnesium (USP); Prilosec OTC (TN) |
(P) unclassified |
| D05261 |
Omeprazole sodium injection (JAN); Omeprazole sodium hydrate; Omepral (TN) |
(P) unclassified |
| D05322 |
Oxytetracycline calcium (USP); Terramycin (TN) |
(P) unclassified |
| D05380 |
Pazopanib hydrochloride (JAN/USAN); Votrient (TN) |
(P) unclassified |
| D05406 |
Penamecillin (USAN/INN) |
(P) unclassified |
| D05408 |
Penicillin G sodium (USP); Benzylpenicillin sodium |
(P) unclassified |
| D05411 |
Penicillin V (USP); Phenoxymethylpenicillin (INN); V-Cillin (TN) |
(P) unclassified |
| D05413 |
Penicillin V hydrabamine (USP) |
(P) unclassified |
| D05462 |
Oxycodone hydrochloride hydrate (JP19) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D05494 |
Pirbenicillin sodium (USAN) |
(P) unclassified |
| D05496 |
Piridicillin sodium (USAN) |
(P) unclassified |
| D05520 |
Pivampicillin pamoate (USAN) |
(P) unclassified |
| D05521 |
Pivampicillin probenate (USAN) |
(P) unclassified |
| D05538 |
Mozenavir (INN) |
(P) unclassified |
| D05594 |
Pramlintide (USAN/INN) |
(P) unclassified |
| D05595 |
Pramlintide acetate (USAN); Symlin (TN) |
(P) unclassified |
| D05601 |
Prednicarbate (USP/INN); Dermatop (TN) |
(P) unclassified |
| D05622 |
Proinsulin human (USAN) |
(P) unclassified |
| D05719 |
Resocortol butyrate (USAN) |
(P) unclassified |
| D05729 |
Rimexolone (USP/INN); Vexol (TN) |
(P) unclassified |
| D05775 |
Rufinamide (JAN/USP/INN); Banzel (TN) |
(P) unclassified |
| D05788 |
Salcolex (USAN); Salcolex tetrahydrate |
(P) unclassified |
| D05789 |
Salethamide maleate (USAN) |
(P) unclassified |
| D05791 |
Salicylate meglumine (USAN) |
(P) unclassified |
| D05793 |
Salnacedin (USAN/INN) |
(P) unclassified |
| D05796 |
Sancycline (USAN/INN); Bonomycin (TN) |
(P) unclassified |
| D05805 |
Sarmoxicillin (USAN/INN) |
(P) unclassified |
| D05806 |
Sarpicillin (USAN) |
(P) unclassified |
| D05972 |
Sultamicillin (USAN/INN) |
(P) unclassified |
| D05974 |
Suncillin sodium (USAN) |
(P) unclassified |
| D05998 |
Talosalate (USAN/INN) |
(P) unclassified |
| D06064 |
Temocillin (USAN) |
(P) unclassified |
| D06068 |
Temsirolimus (JAN/USAN/INN); Torisel (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D06098 |
Tetracycline metaphosphate (JAN); Tetracycline phosphate complex; Tetrax (TN) |
(P) unclassified |
| D06103 |
Theophylline (USP); Theophylline monohydrate; Accurbron (TN) |
(P) unclassified |
| D06104 |
Theophylline sodium glycinate (USP); Asbron (TN) |
(P) unclassified |
| D06106 |
Thiamylal |
(P) unclassified |
| D06113 |
Thiphencillin potassium (USAN) |
(P) unclassified |
| D06137 |
Ticarcillin cresyl sodium (USAN) |
(P) unclassified |
| D06138 |
Ticarcillin monosodium (USP); Ticarcillin monosodium hydrate |
(P) unclassified |
| D06171 |
Tixocortol pivalate (USAN) |
(P) unclassified |
| D06177 |
Tolbutamide sodium, sterile |
(P) unclassified |
| D06186 |
Tolpyrramide (USAN/INN) |
(P) unclassified |
| D06199 |
Trabectedin (JAN/USAN/INN); Yondelis (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D06216 |
Triamcinolone acetonide sodium phosphate (USAN) |
(P) unclassified |
| D06247 |
Triptorelin (USAN/INN) |
(P) unclassified |
| D06248 |
Triptorelin pamoate (USAN); Trelstar (TN); Triptodur (TN) |
(P) unclassified |
| D06273 |
Imidafenacin (JAN/INN); Uritos (TN); Staybla (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D06315 |
Fluticasone furoate (JAN/USAN/INN); Veramyst (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D06402 |
Sunitinib malate (JAN/USAN); Sutent (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D06404 |
Liraglutide (USAN/INN); Liraglutide (genetical recombination) (JAN); Victoza (TN) |
(P) unclassified |
| D06405 |
Nalfurafine hydrochloride (JAN/USAN); Remitch (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D06413 |
Nilotinib hydrochloride hydrate (JAN); Nilotinib monohydrochloride monohydrate; Tasigna (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D06414 |
Dasatinib (USAN); Dasatinib hydrate (JAN); Sprycel (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D06478 |
Darunavir ethanolate (JAN); Prezista (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D06553 |
Alogliptin benzoate (JAN/USAN); Vipidia (TN); Nesina (TN) |
(P) unclassified |
| D06597 |
Fosaprepitant dimeglumine (USAN); Fosaprepitant meglumine (JAN); Proemend (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4 |
| D06637 |
Romidepsin (JAN/USAN/INN); Istodax (TN) |
(P) unclassified |
| D06645 |
Sitagliptin phosphate (USAN); Sitagliptin phosphate hydrate (JP19); Sitagliptin phosphate monohydrate; Januvia (TN) |
(P) unclassified |
| D06673 |
Meprednisone (USP/INN) |
(P) unclassified |
| D06876 |
Hydrocortisone aceponate (INN); Efficort (TN) |
(P) unclassified |
| D06884 |
Lymecycline (INN) |
(P) unclassified |
| D06885 |
Clomocycline (INN) |
(P) unclassified |
| D06887 |
Talbutal (INN); Lotusate (TN) |
(P) unclassified |
| D07073 |
Dexamethasone cipecilate (JAN/INN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4 |
| D07080 |
Vildagliptin (JAN/USAN/INN); Equa (TN); Galvus (TN) |
(P) unclassified |
| D07116 |
Alclometasone (INN) |
(P) unclassified |
| D07117 |
Metahexamide (INN) |
(P) unclassified |
| D07118 |
Glisoxepide (INN) |
(P) unclassified |
| D07192 |
Benfluorex (INN/BAN); Mediaxal (TN) |
(P) unclassified |
| D07201 |
Fluprednidene (INN) |
(P) unclassified |
| D07202 |
Halometasone (INN) |
(P) unclassified |
| D07203 |
Methylprednisolone aceponate (INN); Advantan (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D07230 |
Prednylidene (INN) |
(P) unclassified |
| D07234 |
Metampicillin (INN) |
(P) unclassified |
| D07235 |
Azidocillin (INN) |
(P) unclassified |
| D07236 |
Clometocillin (INN) |
(P) unclassified |
| D07259 |
Buserelin (INN); Tiloryth (TN) |
(P) unclassified |
| D07290 |
Dipyrocetyl (INN) |
(P) unclassified |
| D07291 |
Benorilate (INN); Benorylate |
(P) unclassified |
| D07292 |
Guacetisal (INN); Prontomucil (TN) |
(P) unclassified |
| D07293 |
Imidazole salicylate (INN); Selezen (TN) |
(P) unclassified |
| D07298 |
Barbexaclone (INN); Maliasin (TN) |
(P) unclassified |
| D07321 |
Vinylbital (INN); Vinylbitone |
(P) unclassified |
| D07322 |
Vinbarbital (INN) |
(P) unclassified |
| D07323 |
Cyclobarbital (INN) |
(P) unclassified |
| D07324 |
Proxibarbal (INN); Centralgol (TN) |
(P) unclassified |
| D07334 |
Imipraminoxide (INN) |
(P) unclassified |
| D07335 |
Amineptine (INN); Survector (TN) |
(P) unclassified |
| D07336 |
Quinupramine (INN) |
(P) unclassified |
| D07421 |
Aloxiprin (INN); Superpyrin (TN) |
(P) unclassified |
| D07448 |
Amitriptyline (INN); Laroxyl (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D07452 |
Amoxicillin (INN); AMPC |
(P) unclassified |
| D07464 |
Paramethasone (INN); Dillar (TN) |
(P) unclassified |
| D07469 |
Aspoxicillin (JAN/INN); ASPC; Doyle (TN) |
(P) unclassified |
| D07471 |
Atazanavir (INN); Reyataz (TN) |
(P) CYP inhibition: CYP3A4 |
| D07484 |
Azidocillin sodium salt; InfectoBicillin H-Tabletten (TN); Longatren (TN) |
(P) unclassified |
| D07487 |
Bacampicillin (INN); Penglobe (TN) |
(P) unclassified |
| D07488 |
Balsalazide (INN) |
(P) unclassified |
| D07495 |
Beclometasone (INN) |
(P) unclassified |
| D07508 |
Benfluorex hydrochloride; Mediator (TN) |
(P) unclassified |
| D07538 |
Bosentan (INN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4 |
| D07569 |
Candesartan cilexetil and anmlodipine besylate (JP19); Unisia (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D07570 |
Ampicillin benzathine; Durapen (TN) |
(P) unclassified |
| D07579 |
Aspirin calcium salt; Notras (TN) |
(P) unclassified |
| D07580 |
Aspirin DL-lysine (JAN); Aspirin lysine salt; Aspegic (TN) |
(P) unclassified |
| D07581 |
Aspirin magnesium salt; Mobidin (TN) |
(P) unclassified |
| D07582 |
Aspirin sodium; Sodium acetylsalicylate; Catalgine (TN) |
(P) unclassified |
| D07583 |
Phenytoin and phenobarbital; Aleviatin with phenobarbital (TN) |
(P) unclassified |
| D07595 |
Fosphenytoin sodium hydrate (JAN); Fostoin (TN) |
(P) CYP induction: CYP3A4 |
| D07601 |
Butriptyline (INN); Evadyne (TN) |
(P) unclassified |
| D07612 |
Sodium salamidacetate; o-Carbamoylphenoxyacetic acid sodium salt; Clinit-n (TN) |
(P) unclassified |
| D07614 |
Carbenicillin (INN) |
(P) unclassified |
| D07621 |
Carindacillin (INN); Carbenicillin indanyl |
(P) unclassified |
| D07689 |
Chlortetracycline (INN); Aureomycin (TN) |
(P) unclassified |
| D07712 |
Clemizole penicillin (INN) |
(P) unclassified |
| D07715 |
Clobetasol (INN); Clobecort Amex (TN) |
(P) unclassified |
| D07717 |
Clobetasone (INN) |
(P) unclassified |
| D07719 |
Clocortolone (INN) |
(P) unclassified |
| D07727 |
Clomipramine (INN); Anafranil (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D07733 |
Cloxacillin (INN); Orbenin (TN) |
(P) unclassified |
| D07735 |
Clometocillin potassium; Rixapen (TN) |
(P) unclassified |
| D07749 |
Cortisone (INN) |
(P) unclassified |
| D07757 |
Cyclobarbital calcium (BAN); Phanodorn calcium (TN) |
(P) unclassified |
| D07782 |
Delavirdine (INN) |
(P) unclassified |
| D07791 |
Desipramine (INN) |
(P) unclassified |
| D07796 |
Dexamethasone 21-acetate; Dexamethasone acetate anhydrous; Decaject-L.A. (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4 |
| D07797 |
Dexamethasone isonicotinate; Dexamethasone 21-isonicotinate; Voren [veterinary] (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4 |
| D07798 |
Dexamethasone sodium hemisulfate; Dexamethasone 21-sodium sulfate |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4 |
| D07799 |
Dexamethasone 21-tebutate; Dexamethasone tertiary butyl acetate; Dexamedium [veterinary] (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4 |
| D07800 |
Dexamethasone 21-valerate; Voalla (TN); Zalucs (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4 |
| D07801 |
Dexamethasone phenylpropionate; Dexafort [veterinary] (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4 |
| D07802 |
Dexamethasone phosphate; Decadron-phosphate (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4 |
| D07812 |
Dibenzepin (INN) |
(P) unclassified |
| D07824 |
Diethylamine salicylate; Algesal (TN) |
(P) unclassified |
| D07827 |
Diflorasone (INN); Murode (TN) |
(P) unclassified |
| D07869 |
Donepezil (JAN/INN); Donaz (TN); Allydone (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D07872 |
Dosulepin (INN); Dothiepin; Dothep (TN) |
(P) unclassified |
| D07875 |
Doxepin (INN); Sinequan (TN) |
(P) unclassified |
| D07876 |
Doxycycline (INN); Doxychel (TN) |
(P) unclassified |
| D07877 |
Doxycycline hydrochloride; Vibramycin (TN) |
(P) unclassified |
| D07957 |
Fertirelin (INN) |
(P) unclassified |
| D07965 |
Flucloxacillin sodium salt; Floxapen (TN) |
(P) unclassified |
| D07967 |
Fludrocortisone (INN); Astonin-H (TN) |
(P) unclassified |
| D07972 |
Fluocortin (INN) |
(P) unclassified |
| D07973 |
Fluocortolone 21-pivalate; Fluocortolone pivalate; Ultradil (TN) |
(P) unclassified |
| D07980 |
Fluprednidene acetate; Fluprednidene 21-acetate; Decoderm (TN) |
(P) unclassified |
| D07981 |
Fluticasone (INN); Fluticaps (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D07991 |
Fosfosal (INN); Aydolid (TN) |
(P) unclassified |
| D07993 |
Fosphenytoin (INN) |
(P) CYP induction: CYP3A4 |
| D08017 |
Flucloxacillin magnesium; Floxapen (TN) |
(P) unclassified |
| D08027 |
Gonadorelin (INN); Fertagyl (TN) |
(P) unclassified |
| D08070 |
Imipramine (INN); Tofranil (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D08071 |
Imipramine pamoate (USP); Imipramine embonate; Tofranil-pm (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D08072 |
Imipraminoxide hydrochloride; Elepsin (TN) |
(P) unclassified |
| D08080 |
Insulin injection, biphasic isophane (BAN); Biphasic isophane insuline human (genetical recombination) injectable aqueous suspension (JP19); Insulin Humacart (TN) |
(P) unclassified |
| D08095 |
Ivabradine hydrochloride (JAN/USAN); Ivabrandine hydrochloride; Corlanor (TN); Corlentor (TN); Coralan (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D08110 |
Lenampicillin (INN) |
(P) unclassified |
| D08113 |
Leuprolide (USAN); Leuprorelin (INN); Enantone (TN) |
(P) unclassified |
| D08140 |
Lofepramine (INN) |
(P) unclassified |
| D08147 |
Loteprednol (INN) |
(P) unclassified |
| D08171 |
Melitracen (INN); Adelax (TN) |
(P) unclassified |
| D08191 |
Metampicillin sodium; Serfabiotic (TN) |
(P) unclassified |
| D08227 |
Mometasone (INN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D08233 |
Morphine (BAN); Substitol (TN) |
(P) unclassified |
| D08234 |
Morphine tartrate |
(P) unclassified |
| D08241 |
Nafarelin (INN) |
(P) unclassified |
| D08242 |
Nafcillin (INN) |
(P) unclassified |
| D08259 |
Nelfinavir (INN); Viracept (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D08288 |
Nortriptyline (INN); Nortrilen (TN) |
(P) unclassified |
| D08295 |
Olsalazine (INN) |
(P) unclassified |
| D08297 |
Opipramol (INN) |
(P) unclassified |
| D08307 |
Oxacillin (INN) |
(P) unclassified |
| D08329 |
Penethamate hydriodide (BAN); Mamyzin [veterinary] (TN) |
(P) unclassified |
| D08350 |
Pheneticillin (INN); Phenethicillin |
(P) unclassified |
| D08351 |
Phenformin (BAN) |
(P) unclassified |
| D08352 |
Phenformin hydrochloride; Debei (TN) |
(P) unclassified |
| D08356 |
Phenobarbital diethylamine; Gratusminal (TN) |
(P) unclassified |
| D08360 |
Phenoxymethylpenicillin calcium; Calcipen (TN) |
(P) unclassified |
| D08378 |
Pioglitazone (INN); Actos (TN) |
(P) unclassified |
| D08380 |
Piperacillin (INN); Peracin (TN) |
(P) unclassified |
| D08396 |
Pivampicillin (INN); Pondocillin (TN) |
(P) unclassified |
| D08412 |
Prednisolone pivalate; Prednisolone 21-pivalate; Ultracortenol (TN) |
(P) unclassified |
| D08413 |
Prednisolone sodium metazoate (USAN); Prednisolone metasulfobenzoate sodium; Prednisolone 21-(sodium 3-sulfobenzoate); Predenema (TN) |
(P) unclassified |
| D08414 |
Prednisolone 21-(sodium tetrahydrophthalate); Prednisolone sodium tetrahydrophthalate; Fenicort (TN) |
(P) unclassified |
| D08415 |
Prednisolone steaglate (BAN); Prednisolone 21-steaglate; Sintisone (TN) |
(P) unclassified |
| D08416 |
Prednisone acetate; Prednisone 21-acetate |
(P) unclassified |
| D08438 |
Propicillin (BAN) |
(P) unclassified |
| D08447 |
Protriptyline (INN) |
(P) unclassified |
| D08476 |
Resocortol (INN) |
(P) unclassified |
| D08479 |
Rifampicin sodium; Rifadine (TN) |
(P) CYP induction: CYP3A4 |
| D08488 |
Amlodipine besilate and atorvastatin calcium; Caduet (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D08491 |
Rosiglitazone (INN); Gaudil (TN) |
(P) unclassified |
| D08497 |
Rupatadine fumarate (JAN/USAN); Rinialer (TN); Rupafin (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D08501 |
Trolamine salicylate (USP); Salicylic acid trolamine; Salicylic acid triethanolamine; Arthricream (TN) |
(P) unclassified |
| D08516 |
Sitagliptin (USAN/INN) |
(P) unclassified |
| D08533 |
Sulbactam (INN) |
(P) unclassified |
| D08534 |
Sulbenicillin (INN) |
(P) unclassified |
| D08557 |
Talampicillin (INN) |
(P) unclassified |
| D08567 |
Temocillin disodium salt; Negaban (TN) |
(P) unclassified |
| D08586 |
Thiosalicylic acid; Pirosal (TN); Thiocyl (TN) |
(P) unclassified |
| D08593 |
Ticarcillin (INN); Ticillin [veterinary] (TN) |
(P) unclassified |
| D08605 |
Tipranavir (INN); Aptivus (TN) |
(P) unclassified |
| D08610 |
Tixocortol (INN) |
(P) unclassified |
| D08616 |
Teneligliptin (INN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D08649 |
Triptorelin acetate; Decapeptyl (TN) |
(P) unclassified |
| D08660 |
Ulobetasol (INN); Halobetasol |
(P) unclassified |
| D08699 |
Salmeterol xinafoate and fluticasone propionate; Adoair diskus (TN); Aerivio Spiromax (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D08843 |
Albiglutide (USAN); Albiglutide (genetical recombination) (JAN); Tanzeum (TN) |
(P) unclassified |
| D08856 |
Anamorelin hydrochloride (JAN/USAN); Adlumiz (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D08897 |
Dapagliflozin (JAN/USAN/INN); Forxiga (TN) |
(P) unclassified |
| D08923 |
Fesoterodine fumarate (JAN/USAN); Toviaz (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D08964 |
Perampanel (JAN/USAN); Fycompa (TN) |
(P) unclassified |
| D08976 |
Pomalidomide (JAN/USAN/INN); Pomalyst (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D08996 |
Saxagliptin (USAN/INN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D09017 |
Ticagrelor (JAN/USAN/INN); Brilinta (TN) |
(CI,P) unclassified |
| D09033 |
Voclosporin (JAN/USAN/INN); Lupkynis (TN) |
(CI,P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D09319 |
Indacaterol maleate (JAN/USAN); Arcapta (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D09348 |
Fostamatinib disodium (USAN); Fostamatinib sodium hydrate (JAN); Fostamatinib disodium hexahydrate; Tavalisse (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D09365 |
Palovarotene (JAN/USAN/INN); Sohonos (TN) |
(CI,P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D09566 |
Linagliptin (JAN/USAN/INN); Tradjenta (TN) |
(P) unclassified |
| D09572 |
Riociguat (JAN/USAN/INN); Adempas (TN) |
(P) unclassified |
| D09587 |
Brentuximab vedotin (USAN/INN); Brentuximab vedotin (genetical recombination) (JAN); Adcetris (TN) |
(P) unclassified |
| D09592 |
Canagliflozin (USAN/INN); Canagliflozin hydrate (JAN); Invokana (TN) |
(P) unclassified |
| D09595 |
Budesonide and formoterol fumarate dihydrate; Symbicort (TN); Budeforu (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D09634 |
Lersivirine (USAN/INN) |
(P) unclassified |
| D09638 |
Lomitapide mesylate (USAN); Lomitapide mesilate (JAN); Juxtapid (TN); Lojuxta (TN) |
(CI,P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D09647 |
Omadacycline (USAN) |
(P) unclassified |
| D09720 |
Rilpivirine (JAN/USAN/INN); Rekambys (TN) |
(P) unclassified |
| D09727 |
Insulin degludec (USAN/INN); Insulin degludec (genetical recombination) (JAN); Tresiba (TN) |
(P) unclassified |
| D09728 |
Bosutinib hydrate (JAN); Bosutinib monohydrate; Bosulif (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D09729 |
Lixisenatide (JAN/USAN/INN); Adlyxin (TN); Lyxumia (TN) |
(P) unclassified |
| D09730 |
Olaparib (JAN/USAN/INN); Lynparza (TN) |
(P) unclassified |
| D09731 |
Crizotinib (JAN/USAN/INN); Xalkori (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D09743 |
Telmisartan and amlodipine besilate (JP19); Telmisartan and amlodipine besylate; Micamlo (TN); Twynsta (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D09744 |
Pioglitazone hydrochloride and metformin hydrochloride (JP19); Pioglitazone and metformin; Metact (TN) |
(P) unclassified |
| D09745 |
Valsartan and amlodipine besilate; Exforge (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D09753 |
Saxagliptin hydrate (JAN); Onglyza (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D09756 |
Teneligliptin hydrobromide hydrate (JAN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D09763 |
Dapagliflozin propanediol (USAN); Dapagliflozin propylene glycolate hydrate (JP19); Dapagliflozin propandiol monohydrate; Forxiga (TN); Farxiga (TN) |
(P) unclassified |
| D09783 |
Tofacitinib citrate (JAN/USAN); Tasocitinib citrate; Xeljanz (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D09796 |
Hydrocortisone caproate (JAN) |
(P) unclassified |
| D09799 |
Carotegrast methyl (JAN); Carogra (TN) |
(P) CYP inhibition: CYP3A4 |
| D09848 |
Pioglitazone hydrochloride and glimepiride tablets (JP19); Pioglitazone and glimepiride; Duetact (TN); Sonias (TN) |
(P) unclassified |
| D09889 |
Dulaglutide (USAN/INN); Dulaglutide (genetical recombination) (JAN); Trulicity (TN) |
(P) unclassified |
| D09894 |
Eliglustat tartrate (JAN/USAN); Eliglustat hemitartrate; Cerdelga (TN) |
(CI,P) unclassified |
| D09906 |
Fosdevirine (USAN/INN) |
(P) unclassified |
| D09940 |
Omadacycline tosylate (USAN); Nuzyra (TN) |
(P) unclassified |
| D09951 |
Ponatinib hydrochloride (JAN/USAN); Iclusig (TN) |
(P) unclassified |
| D09956 |
Quizartinib dihydrochloride (USAN); Quizartinib hydrochloride (JAN); Vanflyta (TN) |
(P) unclassified |
| D09958 |
Rilpivirine hydrochloride (JAN/USAN); Edurant (TN) |
(P) unclassified |
| D09960 |
Ruxolitinib phosphate (JAN/USAN); Jakafi (TN); Jakavi (TN); Opzelura (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D09996 |
Vemurafenib (JAN/USAN/INN); Zelboraf (TN) |
(P) CYP induction: CYP3A4 |
| D09999 |
Tramadol hydrochloride and acetaminophen; Tramcet (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D10003 |
Hemin (JAN); Normosang (TN); Panhematin (TN) |
(P) CYP induction: CYP3A4 |
| D10024 |
Selumetinib sulfate (JAN/USAN); Koselugo (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D10025 |
Semaglutide (USAN/INN); Semaglutide (genetical recombination) (JAN); Ozempic (TN) |
(P) unclassified |
| D10082 |
Suvorexant (JAN/USAN); MK-4305; Belsomra (TN) |
(P) unclassified |
| D10095 |
Cabozantinib s-malate (USAN); Cabozantinib malate (JAN); Cometriq (TN); Cabometyx (TN) |
(P) unclassified |
| D10104 |
Dabrafenib mesylate (USAN); Dabrafenib mesilate (JAN); Tafinlar (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4 |
| D10127 |
Glycerol phenylbutyrate (JAN/USAN); Ravicti (TN) |
(P) unclassified |
| D10135 |
Macitentan (JAN/USAN); Opsumit (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D10137 |
Regorafenib hydrate (JAN); Stivarga (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D10159 |
Alogliptin benzoate and pioglitazone hydrochloride; Liovel (TN); Oseni (TN); Incresync (TN) |
(P) unclassified |
| D10160 |
Mitiglinide calcium hydrate and voglibose; Glubes (TN) |
(P) unclassified |
| D10161 |
Sarilumab (USAN); Sarilumab (genetical receombination) (JAN); Kevzara (TN) |
(P) unclassified |
| D10195 |
Luseogliflozin hydrate (JAN); Lusefi (TN) |
(P) unclassified |
| D10196 |
Ipragliflozin (INN) |
(P) unclassified |
| D10200 |
Ipragliflozin L-proline (JAN); Suglat (TN) |
(P) unclassified |
| D10218 |
Enzalutamide (JAN/USAN); Xtandi (TN) |
(P) unclassified |
| D10223 |
Ibrutinib (JAN/USAN); Imbruvica (TN) |
(P) unclassified |
| D10243 |
Irbesartan and amlodipine besilate (JP19); Aimix (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D10244 |
Metformin hydrochloride and rosiglitazone maleate; Avandamet (TN) |
(P) unclassified |
| D10251 |
Glimepiride and rosiglitazone maleate; Avandaryl (TN) |
(P) unclassified |
| D10253 |
Alogliptin benzoate and metformin hydrochloride; Kazano (TN); Vipdomet (TN) |
(P) unclassified |
| D10258 |
Simvastatin and sitagliptin phosphate; Juvisync (TN) |
(P) unclassified |
| D10261 |
Metformin hydrochloride and sitagliptin phosphate; Janumet (TN) |
(P) unclassified |
| D10262 |
Saxagliptin hydrochloride; Onglyza (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D10263 |
Metformin hydrochloride and saxagliptin hydrochloride; Kombiglyze (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D10264 |
Linagliptin and metformin hydrochloride; Jentaduet (TN) |
(P) unclassified |
| D10265 |
Glipizide and metformin hydrochloride; Metaglip (TN) |
(P) unclassified |
| D10266 |
Glyburide and metformin hydrochloride; Glibenclamide and metformin hydrochloride; Glucovance (TN) |
(P) unclassified |
| D10307 |
Avatrombopag maleate (JAN/USAN); Doptelet (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D10309 |
Brexpiprazole (JAN/USAN/INN); Rexulti (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D10313 |
Ertugliflozin (USAN/INN) |
(P) unclassified |
| D10369 |
Eravacycline (USAN/INN) |
(P) unclassified |
| D10372 |
Palbociclib (JAN/USAN); Ibrance (TN) |
(P) unclassified |
| D10421 |
Eravacycline dihydrochloride (USAN); Xerava (TN) |
(P) unclassified |
| D10450 |
Alectinib hydrochloride (JAN); Alecensa (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D10452 |
Cabazitaxel acetonate (JAN); Cabazitaxel acetone; Jevtana (TN) |
(P) unclassified |
| D10459 |
Empagliflozin (JAN/USAN/INN); Jardiance (TN) |
(P) unclassified |
| D10466 |
Vonoprazan fumarate (JAN/USAN); Takecab (TN); Voquezna (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D10473 |
Insulin peglispro (USAN/INN) |
(P) unclassified |
| D10478 |
Naldemedine tosylate (JAN/USAN); Naldemedine tosilate; Symproic (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D10500 |
Metformin hydrochloride and repaglinide; Prandimet (TN) |
(P) unclassified |
| D10501 |
Fluticasone furoate and vilanterol trifenatate; Breo ellipta (TN); Relvar ellipita (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D10502 |
Gemigliptin (INN) |
(P) unclassified |
| D10505 |
Glycopyrronium bromide and indacaterol maleate; Ultibro (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D10506 |
Fluticasone propionate and formoterol fumarate hydrate; Flutiform (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D10516 |
Aripiprazole hydrate (JAN); Aripiprazole monohydrate; Abilify maintena (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D10524 |
Azilsartan and amlodipine besilate; Zacras (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D10528 |
Aldosterone (INN) |
(P) unclassified |
| D10533 |
Umeclidinium bromide and vilanterol; Anoro (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D10551 |
Ceritinib (JAN/USAN/INN); Zykadia (TN) |
(P) unclassified |
| D10564 |
Amenamevir (JAN/INN); Amenalief (TN) |
(P) unclassified |
| D10566 |
Pasireotide pamoate (JAN); Signifor lar (TN) |
(P) unclassified |
| D10570 |
Insulin degludec (genetical recombination) and insulin aspart (genetical recombination); Ryzodeg (TN) |
(P) unclassified |
| D10586 |
Dapagliflozin and metformin; Xigduo xr (TN) |
(P) unclassified |
| D10587 |
Canagliflozin and metformin; Invokamet (TN) |
(P) unclassified |
| D10588 |
Empagliflozin and linagliptin; Glyxambi (TN) |
(P) unclassified |
| D10624 |
Doravirine (JAN/USAN/INN); Pifeltro (TN) |
(P) unclassified |
| D10633 |
Finerenone (JAN/USAN/INN); Kerendia (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D10643 |
Isavuconazonium sulfate (JAN/USAN); Cresemba (TN) |
(P) unclassified |
| D10663 |
Rimegepant sulfate (USAN); Rimegepant sulfate hydrate (JAN); Nurtec odt (TN); Vydura (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D10666 |
Sarecycline (USAN/INN) |
(P) unclassified |
| D10667 |
Sarecycline hydrochloride (USAN); Seysara (TN) |
(P) unclassified |
| D10669 |
Sotagliflozin (USAN/INN); Inpefa (TN) |
(P) unclassified |
| D10679 |
Venetoclax (JAN/USAN/INN); Venclexta (TN) |
(CI,P) unclassified |
| D10688 |
Abemaciclib (JAN/USAN/INN); Verzenio (TN) |
(P) unclassified |
| D10743 |
Vildagliptin and metformin hydrochloride |
(P) unclassified |
| D10752 |
Empagliflozin and metformin; Synjardy (TN) |
(P) unclassified |
| D10755 |
Elvitegravir, cobicistat, emtricitabine and tenofovir alafenamide; Genvoya (TN) |
(P) unclassified |
| D10761 |
Polatuzumab vedotin (USAN); Polatuzumab vedotin (genetical recombination) (JAN); Polatuzumab vedotin-piiq; Polivy (TN) |
(P) unclassified |
| D10762 |
Fosravuconazole L-lysine ethanolate (JAN) |
(P) unclassified |
| D10774 |
Vonoprazan, amoxicillin and metronidazole; Vonopion (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D10775 |
Vonoprazan, amoxicillin and clarithromycin; Vonosap (TN); Voquenza (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D10780 |
Perampanel hydrate (JAN); Fycompa (TN) |
(P) unclassified |
| D10800 |
Gilteritinib fumarate (JAN/USAN); Xospata (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D10801 |
Letermovir (JAN/USAN/INN); Prevymis (TN) |
(P) unclassified |
| D10805 |
Telmisartan, amlodipine and hydrochlorothiazide; Micatrio (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D10826 |
Saxagliptin and dapagliflozin; Qtern (TN) |
(P) unclassified |
| D10832 |
Darunavir and cobicistat; Prezcobix (TN); Rezolsta (TN) |
(P) unclassified |
| D10865 |
Bexagliflozin (USAN); Brenzavvy (TN) |
(P) unclassified |
| D10866 |
Brigatinib (JAN/USAN); Alunbrig (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D10891 |
Capmatinib hydrochloride (USAN); Capmatinib hydrochloride hydrate (JAN); Tabrecta (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D10892 |
Esaxerenone (JAN/INN) |
(P) unclassified |
| D10893 |
Acalabrutinib (JAN/USAN/INN); Calquence (TN) |
(P) unclassified |
| D10926 |
Entrectinib (JAN/USAN/INN); Rozlytrek (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D10927 |
Erdafitinib (JAN/USAN/INN); Balversa (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D10931 |
Etrasimod arginine (USAN); Etrasimod L-arginine (JAN); Velsipity (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D10990 |
Somatrogon (USAN/INN); Somatrogon (genetical recombination) (JAN); Somatrogon-ghla; Ngenla (TN) |
(P) unclassified |
| D10993 |
Tucidinostat (JAN/USAN/INN); Hiyasta (TN) |
(P) unclassified |
| D10999 |
Valbenazine tosylate (USAN); Valbenazine tosilate (JAN); Valbenazine ditosylate; Ingrezza (TN); Dysval (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D11000 |
Vamorolone (USAN/INN); Agamree (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D11012 |
Lorlatinib (JAN/USAN/INN); Lorbrena (TN) |
(P) unclassified |
| D11014 |
Glecaprevir and pibrentasvir; Mavyret (TN) |
(P) unclassified |
| D11022 |
Lemborexant (JAN/USAN/INN); Dayvigo (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D11023 |
Evogliptin (INN) |
(P) unclassified |
| D11034 |
Insulin glargine and lixisenatide; Insulin glargine (genetical recombination) and lixisenatide; Soliqua (TN) |
(P) unclassified |
| D11035 |
Fluticasone furoate, umeclidinium bromide and vilanterol; Trelegy ellipta (TN) |
(P) unclassified |
| D11040 |
Apalutamide (JAN/INN); Erleada (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4 |
| D11043 |
Ertugliflozin pidolate; Ertugliflozin L-pyroglutamic acid; Steglatro (TN) |
(P) unclassified |
| D11048 |
Upadacitinib hydrate (JAN); Upadacitinib hemihydrate; Rinvoq (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D11053 |
Encorafenib (JAN/USAN/INN); Braftovi (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D11066 |
Ertugliflozin and sitagliptin; Steglujan (TN) |
(P) unclassified |
| D11067 |
Ertugliflozin and metformin; Segluromet (TN) |
(P) unclassified |
| D11070 |
Tirabrutinib hydrochloride (JAN/USAN); Velexbru (TN) |
(P) unclassified |
| D11090 |
Ivosidenib (JAN/USAN/INN); Tibsovo (TN) |
(P) unclassified |
| D11093 |
Avacopan (JAN/USAN/INN); Tavneos (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D11109 |
Anagliptin and Metformin hydrochloride |
(P) unclassified |
| D11138 |
Larotrectinib sulfate (JAN/USAN); Vitrakvi (TN) |
(P) unclassified |
| D11159 |
Leniolisib phosphate (JAN/USAN); Joenja (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D11194 |
Somapacitan (USAN/INN); Somapacitan (genetical recombination) (JAN); Somapacitan-beco; Sogroya (TN) |
(P) unclassified |
| D11246 |
Dapivirine (USAN/INN) |
(P) unclassified |
| D11296 |
Fedratinib hydrochloride (USAN); Fedratinib hydrochloride hydrate (JAN); Fedratinib dihydrochloride monohydrate; Inrebic (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D11342 |
Dorzagliatin (USAN) |
(P) unclassified |
| D11360 |
Tirzepatide (JAN/USAN); Mounjaro (TN); Zepbound (TN) |
(P) unclassified |
| D11370 |
Fosnetupitant chloride hydrochloride (JAN/USAN); Arokaris (TN) |
(P) unclassified |
| D11371 |
Capivasertib (JAN/USAN); Truqap (TN) |
(P) unclassified |
| D11382 |
Darunavir, cobicistat, emtricitabine and tenofovir alafenamide; Symtuza (TN) |
(P) unclassified |
| D11417 |
Pemigatinib (JAN/USAN/INN); Pemazyre (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D11422 |
Zanubrutinib (JAN/USAN/INN); Brukinsa (TN) |
(P) unclassified |
| D11454 |
Repotrectinib (JAN/USAN); Augtyro (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D11485 |
Tazemetostat hydrobromide (JAN/USAN); Tazverik (TN) |
(P) unclassified |
| D11525 |
Enfortumab vedotin (USAN); Enfortumab vedotin (genetical recombination) (JAN); Enfortumab vedotin-ejfv; Padcev (TN) |
(P) unclassified |
| D11557 |
Tecovirimat hydrate (JAN); Tecovirimat monohydrate; Tpoxx (TN); Tepoxx (TN) |
(P) unclassified |
| D11567 |
Insulin degludec and liraglutide; Xultophy (TN) |
(P) unclassified |
| D11572 |
Beclomethasone dipropionate monohydrate; Beconase aq (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D11584 |
Budesonide, glycopyrronium bromide and formoterol fumarate; Budesonide, glycopyrrolate and formoterol fumarate; Breztri (TN) |
(P) unclassified |
| D11659 |
Tolvaptan sodium phosphate (JAN); Samtasu (TN) |
(P) unclassified |
| D11662 |
Valemetostat tosilate (JAN); Valemetostat tosylate; Ezharmia (TN) |
(P) unclassified |
| D11674 |
Berotralstat hydrochloride (JAN/USAN); Orladeyo (TN) |
(P) CYP inhibition: CYP3A4 |
| D11711 |
Dapagliflozin, metformin and saxagliptin; Qternmet xr (TN) |
(P) unclassified |
| D11713 |
Selpercatinib (JAN/USAN/INN); Retevmo (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D11725 |
Futibatinib (JAN/USAN/INN); Lytgobi (TN) |
(P) unclassified |
| D11793 |
Zuranolone (JAN/USAN/INN); Zurzuvae (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D11804 |
Aspirin and vonoprazan; Cabpirin (TN) |
(P) unclassified |
| D11807 |
Imeglimin hydrochloride (JAN); Twymeeg (TN) |
(P) unclassified |
| D11814 |
Tisotumab vedotin (USAN/INN); Tisotumab vedotin (genetical recombination) (JAN); Tisotumab vedotin-tftv; Tivdak (TN) |
(P) unclassified |
| D11816 |
Belumosudil mesylate (USAN); Belumosudil mesilate (JAN); Rezurock (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D11835 |
Vorasidenib citrate (USAN); Vorasidenib citric acid hydrate (JAN); Voranigo (TN) |
(P) unclassified |
| D11856 |
Empagliflozin, linagliptin and metformin hydrochloride; Trijardy xr (TN) |
(P) unclassified |
| D11861 |
Indacaterol acetate, glycopyrronium bromide and mometasone furoate; Enerzair (TN) |
(P) unclassified |
| D11862 |
Indacaterol and mometasone furoate; Atectura (TN) |
(P) unclassified |
| D11887 |
Daridorexant hydrochloride (JAN/USAN); Quviviq (TN) |
(P) unclassified |
| D11920 |
Pimitespib (JAN); Jeselhy (TN) |
(P) unclassified |
| D11923 |
Lobeglitazone (INN) |
(P) unclassified |
| D11924 |
Beinaglutide (INN) |
(P) unclassified |
| D11954 |
Belzutifan (JAN/USAN/INN); Welireg (TN) |
(P) unclassified |
| D11968 |
Teneligliptin hydrobromide (JAN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D11970 |
Ritlecitinib tosylate (USAN); Ritlecitinib tosilate (JAN); Litfulo (TN) |
(P) unclassified |
| D12015 |
St. John's wort; SJW |
(P) unclassified |
| D12050 |
Pirtobrutinib (JAN/USAN); Jaypirca (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D12055 |
Sotorasib (JAN/USAN); Lumakras (TN) |
(P) unclassified |
| D12217 |
Imlunestrant tosylate (USAN); Imlunestrant tosilate (JAN); Inluriyo (TN) |
(P) Enzyme: CYP3A4 / Target: ESR1 / CYP inhibition: CYP3A4 |
| D12245 |
Lazertinib mesylate (USAN); Lazertinib mesilate hydrate (JAN); Lazcluze (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D12252 |
Iptacopan hydrochloride (USAN); Iptacopan hydrochloride hydrate (JAN); Iptacopan hydrochloride monohydrate; Fabhalta (TN) |
(P) CYP induction: CYP3A4 |
| D12265 |
Mavacamten (JAN/USAN/INN); Camzyos (TN) |
(P) unclassified |
| D12269 |
Nirmatrelvir and ritonavir; Paxlovid (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D12294 |
Sitagliptin phosphate (JAN) |
(P) unclassified |
| D12311 |
Bortezomib hydrate (JAN) |
(P) unclassified |
| D12337 |
Leuprolide mesylate (USAN); Leuprorelin mesylate; Leuprorelin mesilate; Camcevi (TN) |
(P) unclassified |
| D12358 |
Insulin icodec (USAN/INN); Insulin icodec (genetical recombination) (JAN); Insulin icodec-abae; Awiqli (TN) |
(P) unclassified |
| D12364 |
Taletrectinib adipate (JAN/USAN); Ibtrozi (TN) |
(P) unclassified |
| D12396 |
Sebetralstat (JAN/USAN/INN); Ekterly (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D12442 |
Tucatinib ethanolate (JAN); Tucatinib hemiethanolate; Tukysa (TN) |
(P) unclassified |
| D12444 |
Nilotinib hydrochloride dihydrate (JAN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D12484 |
Carfloglitazar (INN) |
(P) unclassified |
| D12586 |
Mifepristone and misoprostol; Mefeego (TN) |
(P) unclassified |
| D12595 |
Aspirin trelamine (USAN) |
(P) unclassified |
| D12596 |
Aspirin trelamine hydrochloride (USAN) |
(P) unclassified |
| D12611 |
Vornorexant hydrate (JAN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D12637 |
Darunavir hydrate |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D12703 |
Linagliptin hydrate (JAN); Linagliptin hemihydrate |
(P) unclassified |
| D12704 |
Acalabrutinib maleate hydrate (JAN); Acalabrutinib maleate monohydrate; Calquence (TN) |
(P) unclassified |
| D12752 |
Darunavir propylene glycolate |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D12837 |
Risovalisib mesilate hydrate (JAN); Risovalisib mesylate dihydrate; Haizexin (TN) |
(P) unclassified |
| D12963 |
Macitentan and tadalafil; Opsynvi (TN); Yuvanci (TN) |
(CI,P) unclassified |
| D13015 |
Enavogliflozin (INN) |
(P) unclassified |
| D13018 |
Elsulfavirine (INN) |
(P) unclassified |
| D13026 |
Atogepant hydrate (JAN); Aquipta (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 |
| D13028 |
Insulin efsitora alfa (INN); Insulin efsitora alfa (genetical recombination) (JAN) |
(P) unclassified |
| D13055 |
Sitagliptin hydrochloride; Sitagliptin monohydrochloride monohydrate; Brynovin (TN) |
(P) unclassified |
| D13245 |
Insulin icodec (genetical recombination) and semaglutide (genetical recombination); Kyinsu (TN) |
(P) unclassified |