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Drug interaction list


Query:
D00554  Ethinyl estradiol (USP); Ethinylestradiol (JP19/INN); Estinyl (TN)

Interactions: 867 hits    [ ATC classification | Therapeutic category ]

C06624  Oxytetracycline; Oxytetracycline anhydrous (P) unclassified
C07005  Flunisolide; Flunisolide anhydrous (P) unclassified
C07051  Indinavir (P) unclassified
C07370  Prednisone; 1,2-Dehydrocortisone; 17,21-Dihydroxypregna-1,4-diene-3,11,20-trione (P) unclassified
C07521  Thiopental (P) unclassified
C11752  Carfecillin; Carbenicillin phenyl (P) unclassified
D00085  Insulin (JAN/USP) (P) unclassified
D00088  Hydrocortisone (JP19/USP/INN); HC; Acticort (TN); Anusol HC (TN); Colocort (TN); Cortef (TN); Hytone (TN); Plenadren (TN) (P) unclassified
D00107  Tacrolimus (USP/INN); Tacrolimus hydrate (JP19); Prograf (TN); Protopic (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00109  Aspirin (JP19/USP); Aspalon (JAN); Acetylsalicylic acid; Easprin (TN); Durlaza (TN) (P) unclassified
D00130  Diflunisal (JAN/USP/INN); Dolobid (TN) (P) unclassified
D00136  Haloperidol (JP19/USP/INN); Haldol (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00165  Hydrocortisone acetate (JP19/USP); Cortifoam (TN); U-cort (TN) (P) unclassified
D00184  Cyclosporine (USP); Ciclosporin (JP19); Gengraf (TN); Neoral (TN); Restasis (TN); Sandimmune (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00201  Tetracycline (JAN/USP/INN); Sumycin (TN) (P) unclassified
D00204  Ampicillin (USP/INN); Anhydrous ampicillin (JP19); Omnipen (TN) (P) unclassified
D00205  Oxytetracycline (JAN/USP/INN); Oxytetracycline dihydrate; Terramycin (TN) (P) unclassified
D00211  Rifampin (USP); Rifampicin (JP19/INN); Rifadin (TN); Rimactane (TN) (P) CYP induction: CYP3A4
D00216  Acarbose (JAN/USAN/INN); Precose (TN) (P) unclassified
D00217  Acetaminophen (JP19/USP); Paracetamol (INN); Tylenol (TN) (P) unclassified
D00219  Acetohexamide (JP19/USP/INN); Dymelor (TN) (P) unclassified
D00228  Amoxapine (JP19/USP/INN); Asendin (TN) (P) unclassified
D00229  Amoxicillin (USP); Amoxicillin hydrate (JP19); Amoxicilline (INN); Amoxicillin trihydrate; Amoxil (TN); Dispermox (TN); Pasetocin (TN) (P) unclassified
D00244  Betamethasone (JP19/USP/INN); Celestone (TN); Rinderon (TN) (P) unclassified
D00246  Budesonide (JP19/USP/INN); Entocort EC (TN); Pulmicort (TN); Rhinocort (TN); Uceris (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00252  Carbamazepine (JP19/USP/INN); Equetro (TN); Tegretol (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D00271  Chlorpropamide (JP19/USP/INN); Diabinese (TN) (P) unclassified
D00283  Clozapine (JAN/USP/INN); Clozaril (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00290  Demeclocycline hydrochloride (USP); Demethylchlortetracycline hydrochloride (JP19); Declomycin (TN) (P) unclassified
D00292  Dexamethasone (JP19/USP/INN); Decadron (TN); Maxidex (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D00293  Diazepam (JP19/USP/INN); Diastat (TN); Valium (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00307  Doxycycline (USP); Doxycycline hydrate; Monodox (TN); Oracea (TN); Vibramycin (TN) (P) unclassified
D00320  Fentanyl (JAN/USP/INN); Duragesic (TN); Subsys (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00322  Fluconazole (JP19/USP/INN); Diflucan (TN) (P) CYP inhibition: CYP3A4
D00324  Flunisolide (JAN/USP); Aerospan (TN); Nasalide (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00325  Fluocinonide (JP19/USP/INN); Lidex (TN); Vanos (TN) (P) unclassified
D00328  Flurandrenolide (USP); Fludroxycortide (JAN/INN); Cordran (TN) (P) unclassified
D00335  Glipizide (USP/INN); Glucotrol (TN) (P) unclassified
D00336  Glyburide (USP); Glibenclamide (JP19/INN); Diabeta (TN); Glynase (TN); Micronase (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00354  Lamotrigine (JAN/USP/INN); Lamictal (TN) (P) unclassified
D00371  Theophylline (JP19); Elixophyllin (TN); Quibron-t (TN); Theo-24 (TN); Theodur G (TN); Theolair (TN); Uniphyl (TN) (P) unclassified
D00375  Mephenytoin (USP/INN); Mesantoin (TN) (P) unclassified
D00377  Mesalamine (USP); Mesalazine (JP19/INN); Apriso (TN); Asacol (TN); Canasa (TN); Delzicol (TN); Lialda (TN); Mesalamine (TN); Pentasa (TN); Rowasa (TN); Sfrowasa (TN) (P) unclassified
D00379  Tolazamide (JAN/USP/INN); Tolinase (TN) (P) unclassified
D00380  Tolbutamide (JAN/USP/INN); Orinase (TN) (P) unclassified
D00385  Triamcinolone (JP19/USP/INN); Aristocort (TN); Kenacort (TN) (P) unclassified
D00394  Trimipramine (USAN/INN) (P) unclassified
D00395  Troglitazone (JAN/USAN/INN); Rezulin (TN) (P) unclassified
D00407  Methylprednisolone (JP19/USP/INN); Medrol (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00420  Mitotane (JAN/USP/INN); Lysodren (TN) (P) unclassified
D00426  Risperidone (JP19/USP/INN); Risperdal (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00427  Ritonavir (JAN/USP/INN); Norvir (TN) (P) unclassified
D00428  Salsalate (USP/INN); Sasapyrine (JAN); Disalcid (TN) (P) unclassified
D00429  Saquinavir (JAN/USP/INN); Fortovase (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00430  Secobarbital (USP/INN); Seconal (TN) (P) unclassified
D00435  Nevirapine (JAN/USP/INN); Viramune (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00448  Sulfasalazine (USP/INN); Salazosulfapyridine (JP19); Azulfidine (TN) (P) unclassified
D00455  Omeprazole (JP19/USP/INN); Prilosec (TN) (P) unclassified
D00458  Quetiapine fumarate (JP19/USP); Seroquel (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00466  Piperacillin sodium (JP19/USP); Pentcillin (TN); Pipracil (TN) (P) unclassified
D00472  Prednisolone (JP19/USP/INN); Delta-cortef (TN) (P) unclassified
D00473  Prednisone (USP); Prednisone monohydrate; Deltasone (TN); Meticorten (TN); Rayos (TN) (P) unclassified
D00474  Primidone (JP19/USP/INN); Mysoline (TN) (P) unclassified
D00484  Protriptyline hydrochloride (USP); Vivactil (TN) (P) unclassified
D00491  Paclitaxel (JAN/USP/INN); Abraxane (TN); Taxol (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00497  Penicillin V potassium (USP); Phenoxymethylpenicillin potassium (JAN); Veetids (TN) (P) unclassified
D00499  Pentobarbital (USP/INN); Nembutal (TN) (P) unclassified
D00500  Pentobarbital sodium (JAN/USP); Nembutal sodium (TN) (P) unclassified
D00506  Phenobarbital (JP19/USP/INN); Luminal (TN) (P) unclassified
D00512  Phenytoin (JP19/USP/INN); Dilantin (TN) (P) unclassified
D00537  Topiramate (JAN/USP/INN); Topamax (TN); Trokendi xr (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00550  Midazolam (JAN/USP/INN); Dormicum (TN); Buccolam (TN); Nayzilam (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00555  Amobarbital (JP19/INN); Isomytal (TN) (P) unclassified
D00563  Mirtazapine (JAN/USP/INN); Remeron (TN); Reflex (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00566  Sodium salicylate (JP19/USP); Salsonin (TN) (P) unclassified
D00570  Colchicine (JP19/USP) (CI,P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00573  Goserelin acetate (JP19/USP); Zoladex (TN) (P) unclassified
D00578  Voriconazole (JP19/USP/INN); Vfend (TN) (P) unclassified
D00593  Glimepiride (JP19/USP/INN); Amaryl (TN) (P) unclassified
D00594  Repaglinide (JAN/USP/INN); Prandin (TN); Surepost (TN) (P) unclassified
D00595  Buformin (USAN/INN) (P) unclassified
D00596  Rosiglitazone maleate (JAN/USP); Avandia (TN) (P) unclassified
D00606  Guanfacine hydrochloride (JAN/USP); Intuniv (TN); Tenex (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00615  Amlodipine besylate (USP); Amlodipine besilate (JP19); Norvasc (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00619  Verapamil hydrochloride (JP19/USP); Calan (TN); Covera-hs (TN); Vasolan (TN); Verelan (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00625  Miglitol (JP19/USAN/INN); Glyset (TN) (P) unclassified
D00636  Amiodarone hydrochloride (JP19/USP); Ancaron (TN); Cordarone (TN); Nexterone (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00660  Tazobactam (JP19/USP/INN) (P) unclassified
D00661  Cevimeline hydrochloride (USAN); Cevimeline hydrochloride hydrate (JAN); Evoxac (TN); Saligren (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00670  Donepezil hydrochloride (JP19/USP); Aricept (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00687  Salmeterol xinafoate (JAN/USP); Serevent (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00689  Beclomethasone dipropionate (USP); Beclometasone dipropionate (JP19); Beclovent (TN); Qnasl (TN); Vanceril (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00690  Mometasone furoate (JAN/USP); Asmanex (TN); Elocon (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00698  Aprobarbital (INN); Alurate (TN) (P) unclassified
D00699  Butabarbital sodium (USP); Secbutabarbital sodium (INN); Butabarb (TN); Butisol sodium (TN) (P) unclassified
D00700  Mephobarbital (JAN/USP); Methylphenobarbital (INN); Mebaral (TN) (P) unclassified
D00701  Phenobarbital sodium (JAN/USP/INN); Luminal sodium (TN) (P) unclassified
D00708  Ethotoin (JAN/USP/INN); Accenon (TN); Peganone (TN) (P) unclassified
D00712  Methohexital sodium (USP); Brevital sodium (TN) (P) unclassified
D00713  Thiamylal sodium (JP19); Surital (TN) (P) unclassified
D00714  Thiopental sodium (JP19/USP/INN); Pentothal (TN) (P) unclassified
D00722  Oxybutynin chloride (USP); Oxybutynin hydrochloride (JP19); Ditropan (TN); Gelnique (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00727  Olsalazine sodium (USAN); Dipentum (TN) (P) unclassified
D00751  Methylprednisolone sodium succinate (JAN/USP); A-methapred (TN); Solu-medrol (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00785  Selegiline hydrochloride (JAN/USP); Eldepryl (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00809  Amitriptyline hydrochloride (JP19/USP); Elavil (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00810  Choline salicylate (JAN/USAN/INN); Arthropan (TN) (P) unclassified
D00811  Clomipramine hydrochloride (JP19/USP); Anafranil (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00812  Desipramine hydrochloride (JAN/USP); Norpramin (TN) (P) unclassified
D00814  Doxepin hydrochloride (USP); Sinequan (TN); Zonalon (TN) (P) unclassified
D00815  Imipramine hydrochloride (JP19/USP); Tofranil (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00816  Nortriptyline hydrochloride (JP19/USP/INN); Pamelor (TN) (P) unclassified
D00820  Trazodone hydrochloride (JAN/USP); Desyrel (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00821  Venlafaxine hydrochloride (JAN/USP); Effexor (TN) (P) unclassified
D00827  Magnesium salicylate (USP); Magnesium salicylate tetrahydrate; Magan (TN) (P) unclassified
D00831  Mefloquine hydrochloride (JP19/USP); Lariam (TN) (P) unclassified
D00836  Buprenorphine hydrochloride (JP19/USP); Buprenex (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00842  Morphine sulfate (USP); Morphine sulfate hydrate (JP19); Morphine sulfate pentahydrate; Astramor PH (TN); Avinza (TN); Depodur (TN); Kadian (TN); MS contin (TN) (P) unclassified
D00849  Methacycline hydrochloride (JAN/USP); Rondomycin (TN) (P) unclassified
D00850  Minocycline hydrochloride (JP19/USP); Arestin (TN); Dynacin (TN); Minocin (TN); Solodyn (TN) (P) unclassified
D00894  Amprenavir (JAN/USAN/INN); Agenerase (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00895  Delavirdine mesylate (USAN); Delavirdine mesilate (JAN); Rescriptor (TN) (P) unclassified
D00896  Efavirenz (JAN/USP/INN); Sustiva (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D00897  Indinavir sulfate (USP); Crixivan (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00899  Nelfinavir mesylate (USAN/INN); Nelfinavir mesilate (JAN); Viracept (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00927  Bacampicillin hydrochloride (JP19/USAN); Spectrobid (TN) (P) unclassified
D00928  Nafcillin sodium (USP); Nafcillin sodium monohydrate; Unipen (TN) (P) unclassified
D00929  Oxacillin sodium (JAN/USP); Oxacillin sodium hydrate; Bactocill (TN) (P) unclassified
D00944  Metformin hydrochloride (JP19/USP); Glucophage (TN) (P) unclassified
D00945  Pioglitazone hydrochloride (JP19/USP); Actos (TN) (P) unclassified
D00951  Medroxyprogesterone acetate (JP19/USP); Depo-provera (TN); Depo-subq provera 104 (TN); Provera (TN) (CI,P) unclassified
D00961  Bicalutamide (JP19/USP/INN); Casodex (TN) (P) CYP inhibition: CYP3A4
D00964  Letrozole (JAN/USP/INN); Femara (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00971  Sodium thiosalicylate; Thiosalicylic acid sodium salt; Rexolate (TN) (P) unclassified
D00972  Betamethasone sodium phosphate (JP19/USP); Celestone (TN) (P) unclassified
D00973  Cortisone acetate (JP19/USP); Cortone acetate (TN) (P) unclassified
D00975  Dexamethasone sodium phosphate (JAN/USP); Dalalone (TN); Maxidex (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D00976  Hydrocortisone cypionate (P) unclassified
D00977  Hydrocortisone sodium phosphate (JP19/USP); Hydrocortone phosphate (TN) (P) unclassified
D00978  Hydrocortisone sodium succinate (JP19/USP); A-hydrocort (TN); Solu-cortef (TN) (P) unclassified
D00979  Methylprednisolone acetate (JAN/USP); Depo-medrol (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00980  Prednisolone acetate (JP19/USP/INN); Econopred (TN); Pred forte (TN) (P) unclassified
D00981  Prednisolone sodium phosphate (JP19/USP); Pediapred (TN) (P) unclassified
D00982  Prednisolone tebutate (JAN/USP); Hydeltra-TBA (TN) (P) unclassified
D00983  Triamcinolone acetonide (JP19/USP); Azmacort (TN); Kenalog (TN); Nasacort (TN) (P) unclassified
D00984  Triamcinolone diacetate (JAN/USP); Aristocort (TN) (P) unclassified
D00985  Triamcinolone hexacetonide (USP/INN); Aristospan (TN) (P) unclassified
D00986  Fludrocortisone acetate (JP19/USP); Florinef acetate (TN) (P) unclassified
D00988  Gonadorelin hydrochloride (USP); Factrel (TN) (P) unclassified
D00989  Leuprolide acetate (USP); Leuprorelin acetate (JP19); Lupron (TN); Lutrate (TN); Eligard (TN); Fensolvi (TN) (P) unclassified
D00990  Nafarelin acetate (USAN); Nafarelin acetate hydrate (JAN); Synarel (TN) (P) unclassified
D01010  Levothyroxine sodium (USP); Levothyroxine sodium hydrate (JP19); Levothroid (TN); Levoxyl (TN); Synthroid (TN) (P) unclassified
D01011  Liothyronine sodium (JP19/USP); Cytomel (TN); Triostat (TN) (P) unclassified
D01053  Penicillin G potassium (USP); Benzylpenicillin potassium (JP19); Pfizerpen (TN) (P) unclassified
D01055  Emivirine (USAN/INN); Coactinon (TN) (P) unclassified
D01061  Irinotecan hydrochloride (USP); Irinotecan hydrochloride hydrate (JP19); Irinotecan hydrochloride trihydrate; CPT 11; CPT-11; Campto (TN); Camptosar (TN); Onivyde (TN) (P) unclassified
D01071  Hexobarbital (JAN/INN) (P) unclassified
D01074  Hetacillin (USAN/INN); Versapen (TN) (P) unclassified
D01079  Tigecycline (JAN/USP); Tygacil (TN) (P) unclassified
D01087  Methyl salicylate (JP19/NF) (P) unclassified
D01110  Melitracen hydrochloride (JAN/USAN) (P) unclassified
D01111  Nateglinide (JP19/USP/INN); Starsis (TN) (P) unclassified
D01115  Eplerenone (JP19/USAN/INN); Inspra (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D01160  Saquinavir mesylate (USP); Saquinavir mesilate (JAN); Invirase (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D01164  Aripiprazole (JP19/USP/INN); Abilify (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D01176  Blonanserin (JP19/INN); AD 5423 (CI,P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D01178  Phenethicillin potassium (JP19); Pheneticillin potassium; Syncillin (TN); Synthepen (TN) (P) unclassified
D01207  Omeprazole sodium (USAN); Losec sodium (TN) (P) unclassified
D01213  Tolvaptan (JP19/USAN/INN); Samsca (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D01214  Tobicillin (JAN/INN) (P) unclassified
D01227  Bosentan (USAN); Bosentan hydrate (JAN); Tracleer (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D01229  Paramethasone acetate (JAN/USAN); Haldrone (TN) (P) unclassified
D01239  Prednisolone sodium succinate (JP19/USP); Kohakusanin (TN) (P) unclassified
D01249  Flucloxacillin sodium (JAN); Flucloxacillin sodium hydrate; Floxapen (TN) (P) unclassified
D01251  Ampicillin hydrate (JP19); Ampicillin trihydrate; Amcill (TN) (P) unclassified
D01253  Clobazam (JAN/USAN/INN); Mystan (TN); Onfi (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D01266  Difluprednate (JAN/USAN/INN); Durezol (TN) (P) unclassified
D01272  Clobetasol propionate (JP19/USP); Clobex (TN); Cormax (TN); Olux (TN) (P) unclassified
D01273  Clobetasone butyrate (JAN/USAN); Kindavate (TN) (P) unclassified
D01276  Atazanavir sulfate (JAN/USAN); Reyataz (TN) (P) CYP inhibition: CYP3A4
D01283  Carbenicillin indanyl sodium (USP); Carindacillin sodium (JAN); Geocillin (TN) (P) unclassified
D01285  Lofepramine hydrochloride (JAN/USAN); Amplit (TN) (P) unclassified
D01287  Levobupivacaine hydrochloride (JAN/USAN); Chirocaine (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D01308  Halcinonide (JAN/USP/INN); Halog (TN) (P) unclassified
D01310  Secobarbital sodium (JAN/USP); Seconal sodium (TN) (P) unclassified
D01314  Dibenzepin hydrochloride (JAN/USAN) (P) unclassified
D01327  Diflorasone diacetate (JP19/USP); Florone (TN); Psorcon (TN) (P) unclassified
D01334  Cyclacillin (USAN); Ciclacillin (JP19/INN); Cyclapen-W (TN); Vastcillin (TN) (P) unclassified
D01356  Glymidine sodium (JAN/USAN/INN) (P) unclassified
D01357  Betamethasone valerate (JP19/USP); Beta-Val (TN); Luxiq (TN); Rinderon-V (TN) (P) unclassified
D01367  Fluorometholone (JP19/USP/INN); NSC 33001; Fluor-op (TN); Fml (TN); Oxylone (TN) (P) unclassified
D01372  Zopiclone (JP19/INN); Amoban (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D01382  Metharbital (JAN/INN); Gemonil (TN) (P) unclassified
D01387  Amcinonide (JAN/USP/INN); Cyclocort (TN) (P) unclassified
D01399  Fentanyl citrate (JP19/USP); Abstral (TN); Fentora (TN); Lazanda (TN); Oralet (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D01402  Betamethasone acetate (JAN/USP) (P) unclassified
D01418  Tamibarotene (JAN/USAN/INN); Am 80; Amnoid (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D01425  Lopinavir (JAN/USP/INN) (P) unclassified
D01429  Fosfluconazole (JAN/INN); Prodif (TN) (P) CYP inhibition: CYP3A4
D01434  Deprodone propionate (JAN); Allomidon (TN) (P) unclassified
D01442  Hydrocortisone succinate (JP19) (P) unclassified
D01464  Flumethasone pivalate (USP); Flumetasone pivalate (JAN/BAN); Locorten (TN) (P) unclassified
D01466  Ethenzamide (JP19/INN) (P) unclassified
D01477  Opipramol hydrochloride (JAN/USAN); Insidon (TN) (P) unclassified
D01486  Rolitetracycline nitrate (JAN/USAN) (P) unclassified
D01489  Sulbenicillin sodium (JP19); Lilacillin (TN) (P) unclassified
D01499  Pivmecillinam hydrochloride (JP19); Melysin (TN); Pivya (TN) (P) unclassified
D01510  Dexamethasone metasulfobenzoate sodium (JAN); Dexamethazone metasulfobenzoate sodium; Dexapos; Santeson (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D01546  Dothiepin hydrochloride (USAN); Dosulepin hydrochloride (JAN); Prothiaden (TN) (P) unclassified
D01557  Glycol salicylate (JAN); Ethylene glycol salicylate; Norgesic (TN); Phlogont (TN) (P) unclassified
D01596  Oxytetracycline hydrochloride (JP19/USP); Terramycin (TN) (P) unclassified
D01599  Gliclazide (JP19/INN); Glimicron (TN) (P) unclassified
D01615  Dexamethasone palmitate (JAN); Dexamethasone 21-palmitate; Limethason (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D01619  Hydrocortisone butyrate (JP19/USP); Locoid (TN) (P) unclassified
D01632  Dexamethasone dipropionate (USAN); Dexamethasone propionate (JAN); Hifmeta (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D01637  Betamethasone dipropionate (JP19/USP); Diprolene (TN); Rinderon-DP (TN); Sernivo (TN) (P) unclassified
D01649  Propicillin potassium (JAN) (P) unclassified
D01665  Voglibose (JP19/USAN/INN); Basen (TN) (P) unclassified
D01668  Sultamicillin tosilate hydrate (JP19); Sultamicillin tosylate dihydrate; Unasyn (TN) (P) unclassified
D01689  Loteprednol etabonate (JAN/USAN); Lotemax (TN) (P) unclassified
D01696  Lenampicillin hydrochloride (JP19); Kbt 1585; Valacillin (TN) (P) unclassified
D01703  Ciclesonide (JAN/USAN/INN); Alvesco (TN); Omnaris (TN); Zetonna (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D01708  Fluticasone propionate (JAN/USP); Cutivate (TN); Flonase (TN); Flovent (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D01712  Theophylline sodium acetate (JAN) (P) unclassified
D01740  Barbital (JP19/INN) (P) unclassified
D01744  Brotizolam (JP19/USAN/INN); Lendormin (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D01745  Domperidone (JP19/USAN/INN); Motilium (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D01764  Diflucortolone valerate (JP19); Afusona (TN) (P) unclassified
D01799  Glyclopyramide (JAN/INN); Deamelin-S (TN) (P) unclassified
D01811  Salicylamide (JAN/USP/INN) (P) unclassified
D01820  Alclometasone dipropionate (JAN/USP); Aclovate (TN) (P) unclassified
D01825  Fluocinolone acetonide (JP19/USP/INN); Fluocet (TN); Retisert (TN); Synalar (TN) (P) unclassified
D01831  Buserelin acetate (JAN/USAN); Suprecur (TN) (P) unclassified
D01832  Modafinil (JAN/USP/INN); Provigil (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D01854  Mitiglinide calcium hydrate (JP19); Mitiglinide calcium dihydrate; Glufast (TN) (P) unclassified
D01886  Hydrocortisone probutate (USAN); Hydrocortisone butyrate propionate (JAN); Hydrocortisone buteprate; Pandel (TN) (P) unclassified
D01896  Cilostazol (JP19/USP/INN); Pletal (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D01898  Haloperidol decanoate (JAN/USP); Halomonth (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D01948  Dexamethasone valerate (JAN); Dexamethasone 17-valerate; DV-17; Voalla ointment (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D01977  Gefitinib (JP19/USAN/INN); Iressa (TN) (P) unclassified
D01998  Prednisolone farnesylate (JAN); PNF 21; Farnerate (TN) (P) unclassified
D02008  Tadalafil (JAN/USP/INN); Adcirca (TN); Cialis (TN); Zalutia (TN) (CI,P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D02032  Betamethasone butyrate propionate (JAN); Antebate (TN) (P) unclassified
D02096  Fosphenytoin sodium (USP); Cerebyx (TN); Sesquient (TN) (P) CYP induction: CYP3A4
D02103  Phenytoin sodium (USP); Phenytoin sodium for injection (JP19); Aleviatin (TN); Dilantin (TN) (P) unclassified
D02116  Histrelin acetate; Vantas (TN); Supprelin (TN) (P) unclassified
D02119  Ampicillin sodium (JP19/USP); Omnipen-N (TN); Viccillin (TN) (P) unclassified
D02122  Tetracycline hydrochloride (JP19/USP); Bristacycline (TN) (P) unclassified
D02129  Doxycycline hyclate (USP); Doxycycline hydrochloride hydrate (JP19); Doryx (TN); Lymepak (TN); Periostat (TN); Vibra-tabs (TN) (P) unclassified
D02137  Dicloxacillin sodium (USP); Dicloxacillin sodium hydrate (JP19); Dycill (TN) (P) unclassified
D02156  Prednisolone hemisuccinate (USP); Prednisolone succinate (JP19) (P) unclassified
D02157  Penicillin G benzathine (USP); Benzylpenicillin benzathine hydrate (JP19); Bicillin L-A (TN); Permapen (TN); Wycillin (TN); Stelues (TN) (P) unclassified
D02174  Dexamethasone acetate (JAN/USP); Decadronal (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D02190  Carbenicillin disodium (USP); Carbenicillin sodium (JAN); Geopen (TN) (P) unclassified
D02196  Methicillin sodium (USAN); Meticillin sodium (JAN); Methicillin sodium monohydrate; Staphcillin (TN) (P) unclassified
D02199  Carbenicillin phenyl sodium (USAN); Carfecillin sodium (JAN) (P) unclassified
D02201  Talampicillin hydrochloride (JP19/USAN); Aseocillin (TN) (P) unclassified
D02203  Hetacillin potassium (JAN/USAN); Hetacin-K (TN) (P) unclassified
D02206  Buformin hydrochloride (JP19); Dibetos-B (TN) (P) unclassified
D02219  Terbinafine hydrochloride (JP19/USP); Lamisil (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D02221  Mezlocillin sodium (JAN); Mezlocillin sodium monohydrate; Mezlin (TN) (P) unclassified
D02223  Sulbactam sodium (JP19/USP); SBT (P) unclassified
D02229  Sildenafil citrate (JAN/USP); Revatio (TN); Viagra (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D02231  Cloxacillin sodium (USP); Cloxacillin sodium hydrate (JP19); Cloxapen (TN); Tegopen (TN) (P) unclassified
D02241  Ticarcillin disodium (USP); Ticarcillin sodium (JAN); Ticar (TN) (P) unclassified
D02251  Piperacillin (USP); Piperacillin hydrate (JP19) (P) unclassified
D02252  Amobarbital sodium (JAN/USP); Amytal sodium (TN) (P) unclassified
D02253  Pentobarbital calcium (JP19); Ravona (TN) (P) unclassified
D02255  Chlortetracycline hydrochloride (JAN/USP); Aureomycin (TN) (P) unclassified
D02271  Morphine hydrochloride hydrate (JP19); Morphine hydrochloride trihydrate; Anpec (TN) (P) unclassified
D02282  Rolitetracycline (JAN/USAN/INN); Synterin (TN) (P) unclassified
D02286  Betamethasone benzoate (USP); Uticort (TN) (P) unclassified
D02287  Clocortolone pivalate (USP); Cloderm (TN) (P) unclassified
D02288  Hydrocortisone valerate (USP); Westcort (TN) (P) unclassified
D02289  Medrysone (USAN); HMS (TN) (P) unclassified
D02336  Benzylpenicillin (INN); Penicillin G (P) unclassified
D02339  Azlocillin (USAN/INN) (P) unclassified
D02348  Dicloxacillin (USAN/INN) (P) unclassified
D02369  Histrelin (USAN/INN); Vantas (TN) (P) unclassified
D02372  Perospirone hydrochloride hydrate (JP19); Lullan (TN) (P) unclassified
D02405  Penicillin V benzathine (USP) (P) unclassified
D02408  Trimipramine maleate (JAN/USP); Surmontil (TN) (P) unclassified
D02415  Apalcillin sodium (USAN) (P) unclassified
D02425  Carbutamide (INN); Invenol (TN) (P) unclassified
D02426  Glycyclamide (INN); Tolcyclamide (P) unclassified
D02427  Glibornuride (USAN/INN); Glutril (TN) (P) unclassified
D02428  Glisentide (INN); Glypentide; Staticum (TN) (P) unclassified
D02429  Glisolamide (INN); Glysolamide; Diabenor (TN) (P) unclassified
D02430  Gliquidone (INN); Glurenorm (TN) (P) unclassified
D02461  Penicillin G procaine (USP); Duracillin (TN) (P) unclassified
D02476  Meclocycline (USAN/INN) (P) unclassified
D02477  Meclocycline sulfosalicylate (USP); Meclan (TN) (P) unclassified
D02484  Artemether and lumefantrine; Coartem (TN) (P) unclassified
D02497  Fosamprenavir (INN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D02498  Lopinavir and ritonavir; Kaletra (TN) (P) unclassified
D02504  Aspoxicillin hydrate (JP19); ASPC; Doyle (TN) (P) unclassified
D02506  Phenoxymethylpenicillin benzathine (JAN); Penicillin V benzathine tetrahydrate (P) unclassified
D02508  Pivampicillin hydrochloride (USAN) (P) unclassified
D02554  Rifaximin (JAN/USAN/INN); Xifaxan (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D02565  Dimetacrine (INN) (P) unclassified
D02591  Dexamethasone acefurate (USAN/INN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D02592  Dexamethasone beloxil (USAN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D02618  Butobarbital (BAN); Butethal; Neonal (TN) (P) unclassified
D02624  Eszopiclone (JAN/USP/INN); Estorra (TN); Lunesta (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D02689  Ramelteon (JAN/USAN/INN); Rozerem (TN) (P) unclassified
D02691  Somatropin (USP/INN); Somatropin (genetical recombination) (JAN); Human growth hormone (JAN); Asellacrin (TN); Humatrope (TN); Nutropin (TN); Omnitrope (TN) (P) unclassified
D02704  Tampramine fumarate (USAN) (P) unclassified
D02715  Balsalazide disodium (USP); Colazide (TN) (P) unclassified
D02732  Pranlukast hydrate (JP19); Onon (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D02797  Albutoin (USAN/INN); Euprax (TN) (P) unclassified
D02817  Allobarbital (USAN/INN) (P) unclassified
D02861  Indinavir sulfate ethanolate (JAN); Crixivan (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D02867  Fosamprenavir calcium hydrate (JAN); Lexiva (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D02888  Amdinocillin (USAN); Mecillinam (INN); Coactin (TN) (P) unclassified
D02889  Pivmecillinam (INN); Amdinocillin pivoxil; Coactabs (TN) (P) unclassified
D02899  Amicycline (USAN/INN) (P) unclassified
D02925  Amoxicillin sodium (USAN) (P) unclassified
D02968  Aprepitant (JAN/USP/INN); Aponvie (TN); Emend (TN); Cinvanti (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D03001  Atevirdine mesylate (USAN) (P) unclassified
D03038  Azipramine hydrochloride (USAN) (P) unclassified
D03039  Azlocillin sodium; Azlin (TN) (P) unclassified
D03106  Bexarotene (JAN/USAN/INN); Targretin (TN) (P) unclassified
D03150  Bortezomib (JAN/USAN/INN); Velcade (TN) (P) unclassified
D03180  Butabarbital (USP); Secbutabarbital (BAN) (P) unclassified
D03182  Butalbital (USP/INN); Sandoptal (TN) (P) unclassified
D03199  Butriptyline hydrochloride (USAN) (P) unclassified
D03218  Axitinib (JAN/USAN); Inlyta (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D03230  Insulin human (USP/INN); Insulin human (genetical recombination) (JP19); Insulin human (biosynthesis) (JAN); Insulin human (synthesis) (JAN); Humulin (TN) (P) unclassified
D03250  Insulin glargine (USAN/INN); Insulin glargine (genetical recombination) (JP19); Insulin glargine (genetical recombination) [Insulin glargin biosimilar 1] (JAN); Insulin glargine (genetical recombination) [Insulin glargin biosimilar 2] (JAN); Insulin glargine-yfgn; Lantus (TN) (P) unclassified
D03253  Brecanavir (USAN) (P) unclassified
D03260  Vardenafil hydrochloride hydrate (JAN); Vardenafil monohydrochloride trihydrate; Levitra (TN); Staxyn (TN) (CI,P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D03267  Gonadorelin diacetate (JP19) (P) unclassified
D03301  Prednisolone valerate acetate (JAN); PDL; Spirazon (TN) (P) unclassified
D03325  Mometasone furoate hydrate (JAN); Mometasone furoate monohydrate; Nasonex (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D03371  Capravirine (USAN/INN) (P) unclassified
D03385  Carbaspirin calcium (USAN); Carbasalate calcium (INN) (P) unclassified
D03387  Carbenicillin potassium (USAN) (P) unclassified
D03451  Cetocycline hydrochloride (USAN) (P) unclassified
D03477  Chlortetracycline bisulfate (USP) (P) unclassified
D03491  Cidoxepin hydrochloride (USAN) (P) unclassified
D03541  Clocortolone acetate (USAN) (P) unclassified
D03561  Cloprednol (USAN/INN); Cloradryn (TN) (P) unclassified
D03571  Cloxacillin benzathine (USP) (P) unclassified
D03594  Cortivazol (USAN) (P) unclassified
D03656  Darunavir (USAN/INN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D03658  Dasatinib (JAN/INN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D03669  Deferasirox (JAN/USAN/INN); Exjade (TN); Jadenu (TN) (P) CYP induction: CYP3A4
D03671  Deflazacort (USAN/INN); Emflaza (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D03680  Demeclocycline (USP); Demethylchlortetracycline (JAN) (P) unclassified
D03681  Demecycline (USAN/INN) (P) unclassified
D03694  Deslorelin (USAN/INN) (P) unclassified
D03696  Desonide (USP/INN); Desowen (TN); Verdeso (TN) (P) unclassified
D03697  Desoximetasone (USP/INN); Topicort (TN) (P) unclassified
D03705  Sulbactam benzathine (USAN) (P) unclassified
D03706  Sulbactam pivoxil (USAN) (P) unclassified
D03707  Tazobactam sodium (JAN/USAN) (P) unclassified
D03799  Dienogest (JAN/USAN/INN); Endometrion (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D03812  Diflucortolone (USAN) (P) unclassified
D03813  Diflucortolone pivalate (USAN) (P) unclassified
D03820  Dutasteride (JAN/USP/INN); Avodart (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D03833  Indinavir (USAN); Indinavir hydrate (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D03835  Fosamprenavir calcium (USAN); Lexiva (TN); Telzir (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D03837  Fosamprenavir sodium (USAN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D03839  Droxinavir hydrochloride (USAN) (P) unclassified
D03840  Palinavir (USAN/INN) (P) unclassified
D03842  Telinavir (USAN/INN) (P) unclassified
D03843  Tipranavir disodium (USAN) (P) unclassified
D03903  Doxycycline calcium (USP) (P) unclassified
D03904  Doxycycline fosfatex (USAN) (P) unclassified
D04020  Epicillin (USAN/INN); Dexacillin (TN) (P) unclassified
D04023  Erlotinib hydrochloride (JAN/USAN); Tarceva (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D04024  Lapatinib ditosylate (USAN); Lapatinib tosilate hydrate (JAN); Lapatinib ditosylate monohydrate; Tykerb (TN); Tyverb (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D04030  Epitetracycline hydrochloride (USP) (P) unclassified
D04077  Eterobarb (USAN/INN); Antilon (TN) (P) unclassified
D04103  Etoformin hydrochloride (USAN) (P) unclassified
D04112  Etravirine (JAN/USAN/INN); Intelence (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D04121  Exenatide (JAN/USAN/INN); Byetta (TN) (P) unclassified
D04145  Fendosal (USAN/INN); Alnovin (TN) (P) unclassified
D04174  Fertirelin acetate (USAN) (P) unclassified
D04196  Floxacillin (USAN); Flucloxacillin (INN); Floxapen (TN) (P) unclassified
D04201  Flucloronide (USAN); Fluclorolone acetonide (INN) (P) unclassified
D04206  Flufenisal (USAN/INN) (P) unclassified
D04208  Flumethasone (USAN); Flumetasone (INN) (P) unclassified
D04214  Flunisolide acetate (USAN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D04217  Fluocortin butyl (USAN) (P) unclassified
D04218  Fluocortolone (USAN/INN) (P) unclassified
D04219  Fluocortolone caproate (USAN) (P) unclassified
D04221  Fluorometholone acetate (USP); Fluorometholone 17-acetate; Flarex (TN) (P) unclassified
D04225  Fluperolone acetate (USAN); Methral (TN) (P) unclassified
D04244  Formocortal (USAN/INN); Deflamene (TN) (P) unclassified
D04270  Fumoxicillin (USAN/INN) (P) unclassified
D04322  Gliamilide (USAN/INN) (P) unclassified
D04354  Glyhexamide (USAN/INN); Subose (TN) (P) unclassified
D04355  Glyoctamide (USAN/INN) (P) unclassified
D04356  Glyparamide (USAN) (P) unclassified
D04361  Gonadorelin acetate (USP); Luteinizing (TN) (P) unclassified
D04403  Guar gum (NF) (P) unclassified
D04405  Goserelin (USAN/INN) (P) unclassified
D04409  Halobetasol propionate (USP); Ulobetasol propionate; Ultravate (TN) (P) unclassified
D04467  Hydrocortisone hemisuccinate (USP) (P) unclassified
D04475  Insulin aspart (USP/INN); Insulin aspart (genetical recombination) (JP19); Insulin aspart (genetical recombination) [Insulin aspart biosimilar 1] (JAN); Insulin X 14; Insulin aspart-szjj; nsulin aspart-xjhz; Merilog (TN); NovoRapid (TN); Novolog (TN); Kirsty (TN) (P) unclassified
D04477  Insulin lispro (USP/INN); Insulin lispro (genetical recombination) (JAN); Insulin lispro (genetical recombination) [Insulin lispro Biosimilar 1] (JAN); Insulin lispro-aabc; Humalog (TN); Lyumjev (TN) (P) unclassified
D04539  Insulin detemir (USAN/INN); Insulin detemir (genetical recombination) (JAN); Levemir (TN) (P) unclassified
D04540  Insulin glulisine (USAN/INN); Insulin glulisine (genetical recombination) (JAN); Apidra (TN) (P) unclassified
D04541  Insulin human, isophane (USP) (P) unclassified
D04542  Insulin human zinc (USP) (P) unclassified
D04543  Insulin human zinc, extended (USP) (P) unclassified
D04547  Insulin, isophane (USP); Isophane insulin (aqueous suspension) (JAN); Humalog PEN (TN) (P) unclassified
D04550  Insulin zinc, prompt (USP); Semilente iletin (TN) (P) unclassified
D04551  Insulin zinc (USP); Lente iletin (TN) (P) unclassified
D04556  Intriptyline hydrochloride (USAN) (P) unclassified
D04605  Iprindole (USAN/INN) (P) unclassified
D04641  Istradefylline (JAN/USAN/INN); Nourianz (TN); Nouriast (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D04652  Ketipramine fumarate (USAN) (P) unclassified
D04666  Lanreotide acetate (JAN/USAN); Somatuline (TN) (P) unclassified
D04719  Levopropylcillin potassium (USAN) (P) unclassified
D04768  Lonafarnib (JAN/USAN/INN); Zokinvy (TN) (CI,P) unclassified
D04786  Loviride (USAN/INN) (P) unclassified
D04820  Lurasidone hydrochloride (JAN/USAN); SM 13496; Latuda (TN) (CI,P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D04823  Lutrelin acetate (USAN) (P) unclassified
D04966  Metformin (USAN/INN) (P) unclassified
D04972  Methacycline (USAN); Metacycline (INN) (P) unclassified
D04982  Methetoin (USAN/INN) (P) unclassified
D04985  Methohexital (USP/INN) (P) unclassified
D05000  Methylprednisolone hemisuccinate (USP); Methylprednisolone succinate (JP19) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D05001  Methylprednisolone sodium phosphate (USAN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D05002  Methylprednisolone suleptanate (USAN/INN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D05021  Mezlocillin (USAN/INN) (P) unclassified
D05022  Mezlocillin sodium (USP) (P) unclassified
D05045  Minocycline (USAN/INN) (P) unclassified
D05181  Aspirin aluminum (JP19) (P) unclassified
D05184  Nitrocycline (USAN/INN) (P) unclassified
D05231  Octriptyline phosphate (USAN) (P) unclassified
D05259  Omeprazole magnesium (USP); Prilosec OTC (TN) (P) unclassified
D05261  Omeprazole sodium injection (JAN); Omeprazole sodium hydrate; Omepral (TN) (P) unclassified
D05322  Oxytetracycline calcium (USP); Terramycin (TN) (P) unclassified
D05380  Pazopanib hydrochloride (JAN/USAN); Votrient (TN) (P) unclassified
D05406  Penamecillin (USAN/INN) (P) unclassified
D05408  Penicillin G sodium (USP); Benzylpenicillin sodium (P) unclassified
D05411  Penicillin V (USP); Phenoxymethylpenicillin (INN); V-Cillin (TN) (P) unclassified
D05413  Penicillin V hydrabamine (USP) (P) unclassified
D05462  Oxycodone hydrochloride hydrate (JP19) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D05494  Pirbenicillin sodium (USAN) (P) unclassified
D05496  Piridicillin sodium (USAN) (P) unclassified
D05520  Pivampicillin pamoate (USAN) (P) unclassified
D05521  Pivampicillin probenate (USAN) (P) unclassified
D05538  Mozenavir (INN) (P) unclassified
D05594  Pramlintide (USAN/INN) (P) unclassified
D05595  Pramlintide acetate (USAN); Symlin (TN) (P) unclassified
D05601  Prednicarbate (USP/INN); Dermatop (TN) (P) unclassified
D05622  Proinsulin human (USAN) (P) unclassified
D05719  Resocortol butyrate (USAN) (P) unclassified
D05729  Rimexolone (USP/INN); Vexol (TN) (P) unclassified
D05775  Rufinamide (JAN/USP/INN); Banzel (TN) (P) unclassified
D05788  Salcolex (USAN); Salcolex tetrahydrate (P) unclassified
D05789  Salethamide maleate (USAN) (P) unclassified
D05791  Salicylate meglumine (USAN) (P) unclassified
D05793  Salnacedin (USAN/INN) (P) unclassified
D05796  Sancycline (USAN/INN); Bonomycin (TN) (P) unclassified
D05805  Sarmoxicillin (USAN/INN) (P) unclassified
D05806  Sarpicillin (USAN) (P) unclassified
D05972  Sultamicillin (USAN/INN) (P) unclassified
D05974  Suncillin sodium (USAN) (P) unclassified
D05998  Talosalate (USAN/INN) (P) unclassified
D06064  Temocillin (USAN) (P) unclassified
D06068  Temsirolimus (JAN/USAN/INN); Torisel (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D06098  Tetracycline metaphosphate (JAN); Tetracycline phosphate complex; Tetrax (TN) (P) unclassified
D06103  Theophylline (USP); Theophylline monohydrate; Accurbron (TN) (P) unclassified
D06104  Theophylline sodium glycinate (USP); Asbron (TN) (P) unclassified
D06106  Thiamylal (P) unclassified
D06113  Thiphencillin potassium (USAN) (P) unclassified
D06137  Ticarcillin cresyl sodium (USAN) (P) unclassified
D06138  Ticarcillin monosodium (USP); Ticarcillin monosodium hydrate (P) unclassified
D06171  Tixocortol pivalate (USAN) (P) unclassified
D06177  Tolbutamide sodium, sterile (P) unclassified
D06186  Tolpyrramide (USAN/INN) (P) unclassified
D06199  Trabectedin (JAN/USAN/INN); Yondelis (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D06216  Triamcinolone acetonide sodium phosphate (USAN) (P) unclassified
D06247  Triptorelin (USAN/INN) (P) unclassified
D06248  Triptorelin pamoate (USAN); Trelstar (TN); Triptodur (TN) (P) unclassified
D06273  Imidafenacin (JAN/INN); Uritos (TN); Staybla (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D06315  Fluticasone furoate (JAN/USAN/INN); Veramyst (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D06402  Sunitinib malate (JAN/USAN); Sutent (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D06404  Liraglutide (USAN/INN); Liraglutide (genetical recombination) (JAN); Victoza (TN) (P) unclassified
D06405  Nalfurafine hydrochloride (JAN/USAN); Remitch (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D06413  Nilotinib hydrochloride hydrate (JAN); Nilotinib monohydrochloride monohydrate; Tasigna (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D06414  Dasatinib (USAN); Dasatinib hydrate (JAN); Sprycel (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D06478  Darunavir ethanolate (JAN); Prezista (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D06553  Alogliptin benzoate (JAN/USAN); Vipidia (TN); Nesina (TN) (P) unclassified
D06597  Fosaprepitant dimeglumine (USAN); Fosaprepitant meglumine (JAN); Proemend (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D06637  Romidepsin (JAN/USAN/INN); Istodax (TN) (P) unclassified
D06645  Sitagliptin phosphate (USAN); Sitagliptin phosphate hydrate (JP19); Sitagliptin phosphate monohydrate; Januvia (TN) (P) unclassified
D06673  Meprednisone (USP/INN) (P) unclassified
D06876  Hydrocortisone aceponate (INN); Efficort (TN) (P) unclassified
D06884  Lymecycline (INN) (P) unclassified
D06885  Clomocycline (INN) (P) unclassified
D06887  Talbutal (INN); Lotusate (TN) (P) unclassified
D07073  Dexamethasone cipecilate (JAN/INN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D07080  Vildagliptin (JAN/USAN/INN); Equa (TN); Galvus (TN) (P) unclassified
D07116  Alclometasone (INN) (P) unclassified
D07117  Metahexamide (INN) (P) unclassified
D07118  Glisoxepide (INN) (P) unclassified
D07192  Benfluorex (INN/BAN); Mediaxal (TN) (P) unclassified
D07201  Fluprednidene (INN) (P) unclassified
D07202  Halometasone (INN) (P) unclassified
D07203  Methylprednisolone aceponate (INN); Advantan (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D07230  Prednylidene (INN) (P) unclassified
D07234  Metampicillin (INN) (P) unclassified
D07235  Azidocillin (INN) (P) unclassified
D07236  Clometocillin (INN) (P) unclassified
D07259  Buserelin (INN); Tiloryth (TN) (P) unclassified
D07290  Dipyrocetyl (INN) (P) unclassified
D07291  Benorilate (INN); Benorylate (P) unclassified
D07292  Guacetisal (INN); Prontomucil (TN) (P) unclassified
D07293  Imidazole salicylate (INN); Selezen (TN) (P) unclassified
D07298  Barbexaclone (INN); Maliasin (TN) (P) unclassified
D07321  Vinylbital (INN); Vinylbitone (P) unclassified
D07322  Vinbarbital (INN) (P) unclassified
D07323  Cyclobarbital (INN) (P) unclassified
D07324  Proxibarbal (INN); Centralgol (TN) (P) unclassified
D07334  Imipraminoxide (INN) (P) unclassified
D07335  Amineptine (INN); Survector (TN) (P) unclassified
D07336  Quinupramine (INN) (P) unclassified
D07421  Aloxiprin (INN); Superpyrin (TN) (P) unclassified
D07448  Amitriptyline (INN); Laroxyl (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D07452  Amoxicillin (INN); AMPC (P) unclassified
D07464  Paramethasone (INN); Dillar (TN) (P) unclassified
D07469  Aspoxicillin (JAN/INN); ASPC; Doyle (TN) (P) unclassified
D07471  Atazanavir (INN); Reyataz (TN) (P) CYP inhibition: CYP3A4
D07484  Azidocillin sodium salt; InfectoBicillin H-Tabletten (TN); Longatren (TN) (P) unclassified
D07487  Bacampicillin (INN); Penglobe (TN) (P) unclassified
D07488  Balsalazide (INN) (P) unclassified
D07495  Beclometasone (INN) (P) unclassified
D07508  Benfluorex hydrochloride; Mediator (TN) (P) unclassified
D07538  Bosentan (INN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D07569  Candesartan cilexetil and anmlodipine besylate (JP19); Unisia (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D07570  Ampicillin benzathine; Durapen (TN) (P) unclassified
D07579  Aspirin calcium salt; Notras (TN) (P) unclassified
D07580  Aspirin DL-lysine (JAN); Aspirin lysine salt; Aspegic (TN) (P) unclassified
D07581  Aspirin magnesium salt; Mobidin (TN) (P) unclassified
D07582  Aspirin sodium; Sodium acetylsalicylate; Catalgine (TN) (P) unclassified
D07583  Phenytoin and phenobarbital; Aleviatin with phenobarbital (TN) (P) unclassified
D07595  Fosphenytoin sodium hydrate (JAN); Fostoin (TN) (P) CYP induction: CYP3A4
D07601  Butriptyline (INN); Evadyne (TN) (P) unclassified
D07612  Sodium salamidacetate; o-Carbamoylphenoxyacetic acid sodium salt; Clinit-n (TN) (P) unclassified
D07614  Carbenicillin (INN) (P) unclassified
D07621  Carindacillin (INN); Carbenicillin indanyl (P) unclassified
D07689  Chlortetracycline (INN); Aureomycin (TN) (P) unclassified
D07712  Clemizole penicillin (INN) (P) unclassified
D07715  Clobetasol (INN); Clobecort Amex (TN) (P) unclassified
D07717  Clobetasone (INN) (P) unclassified
D07719  Clocortolone (INN) (P) unclassified
D07727  Clomipramine (INN); Anafranil (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D07733  Cloxacillin (INN); Orbenin (TN) (P) unclassified
D07735  Clometocillin potassium; Rixapen (TN) (P) unclassified
D07749  Cortisone (INN) (P) unclassified
D07757  Cyclobarbital calcium (BAN); Phanodorn calcium (TN) (P) unclassified
D07782  Delavirdine (INN) (P) unclassified
D07791  Desipramine (INN) (P) unclassified
D07796  Dexamethasone 21-acetate; Dexamethasone acetate anhydrous; Decaject-L.A. (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D07797  Dexamethasone isonicotinate; Dexamethasone 21-isonicotinate; Voren [veterinary] (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D07798  Dexamethasone sodium hemisulfate; Dexamethasone 21-sodium sulfate (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D07799  Dexamethasone 21-tebutate; Dexamethasone tertiary butyl acetate; Dexamedium [veterinary] (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D07800  Dexamethasone 21-valerate; Voalla (TN); Zalucs (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D07801  Dexamethasone phenylpropionate; Dexafort [veterinary] (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D07802  Dexamethasone phosphate; Decadron-phosphate (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D07812  Dibenzepin (INN) (P) unclassified
D07824  Diethylamine salicylate; Algesal (TN) (P) unclassified
D07827  Diflorasone (INN); Murode (TN) (P) unclassified
D07869  Donepezil (JAN/INN); Donaz (TN); Allydone (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D07872  Dosulepin (INN); Dothiepin; Dothep (TN) (P) unclassified
D07875  Doxepin (INN); Sinequan (TN) (P) unclassified
D07876  Doxycycline (INN); Doxychel (TN) (P) unclassified
D07877  Doxycycline hydrochloride; Vibramycin (TN) (P) unclassified
D07957  Fertirelin (INN) (P) unclassified
D07965  Flucloxacillin sodium salt; Floxapen (TN) (P) unclassified
D07967  Fludrocortisone (INN); Astonin-H (TN) (P) unclassified
D07972  Fluocortin (INN) (P) unclassified
D07973  Fluocortolone 21-pivalate; Fluocortolone pivalate; Ultradil (TN) (P) unclassified
D07980  Fluprednidene acetate; Fluprednidene 21-acetate; Decoderm (TN) (P) unclassified
D07981  Fluticasone (INN); Fluticaps (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D07991  Fosfosal (INN); Aydolid (TN) (P) unclassified
D07993  Fosphenytoin (INN) (P) CYP induction: CYP3A4
D08017  Flucloxacillin magnesium; Floxapen (TN) (P) unclassified
D08027  Gonadorelin (INN); Fertagyl (TN) (P) unclassified
D08070  Imipramine (INN); Tofranil (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D08071  Imipramine pamoate (USP); Imipramine embonate; Tofranil-pm (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D08072  Imipraminoxide hydrochloride; Elepsin (TN) (P) unclassified
D08080  Insulin injection, biphasic isophane (BAN); Biphasic isophane insuline human (genetical recombination) injectable aqueous suspension (JP19); Insulin Humacart (TN) (P) unclassified
D08095  Ivabradine hydrochloride (JAN/USAN); Ivabrandine hydrochloride; Corlanor (TN); Corlentor (TN); Coralan (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D08110  Lenampicillin (INN) (P) unclassified
D08113  Leuprolide (USAN); Leuprorelin (INN); Enantone (TN) (P) unclassified
D08140  Lofepramine (INN) (P) unclassified
D08147  Loteprednol (INN) (P) unclassified
D08171  Melitracen (INN); Adelax (TN) (P) unclassified
D08191  Metampicillin sodium; Serfabiotic (TN) (P) unclassified
D08227  Mometasone (INN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D08233  Morphine (BAN); Substitol (TN) (P) unclassified
D08234  Morphine tartrate (P) unclassified
D08241  Nafarelin (INN) (P) unclassified
D08242  Nafcillin (INN) (P) unclassified
D08259  Nelfinavir (INN); Viracept (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D08288  Nortriptyline (INN); Nortrilen (TN) (P) unclassified
D08295  Olsalazine (INN) (P) unclassified
D08297  Opipramol (INN) (P) unclassified
D08307  Oxacillin (INN) (P) unclassified
D08329  Penethamate hydriodide (BAN); Mamyzin [veterinary] (TN) (P) unclassified
D08350  Pheneticillin (INN); Phenethicillin (P) unclassified
D08351  Phenformin (BAN) (P) unclassified
D08352  Phenformin hydrochloride; Debei (TN) (P) unclassified
D08356  Phenobarbital diethylamine; Gratusminal (TN) (P) unclassified
D08360  Phenoxymethylpenicillin calcium; Calcipen (TN) (P) unclassified
D08378  Pioglitazone (INN); Actos (TN) (P) unclassified
D08380  Piperacillin (INN); Peracin (TN) (P) unclassified
D08396  Pivampicillin (INN); Pondocillin (TN) (P) unclassified
D08412  Prednisolone pivalate; Prednisolone 21-pivalate; Ultracortenol (TN) (P) unclassified
D08413  Prednisolone sodium metazoate (USAN); Prednisolone metasulfobenzoate sodium; Prednisolone 21-(sodium 3-sulfobenzoate); Predenema (TN) (P) unclassified
D08414  Prednisolone 21-(sodium tetrahydrophthalate); Prednisolone sodium tetrahydrophthalate; Fenicort (TN) (P) unclassified
D08415  Prednisolone steaglate (BAN); Prednisolone 21-steaglate; Sintisone (TN) (P) unclassified
D08416  Prednisone acetate; Prednisone 21-acetate (P) unclassified
D08438  Propicillin (BAN) (P) unclassified
D08447  Protriptyline (INN) (P) unclassified
D08476  Resocortol (INN) (P) unclassified
D08479  Rifampicin sodium; Rifadine (TN) (P) CYP induction: CYP3A4
D08488  Amlodipine besilate and atorvastatin calcium; Caduet (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D08491  Rosiglitazone (INN); Gaudil (TN) (P) unclassified
D08497  Rupatadine fumarate (JAN/USAN); Rinialer (TN); Rupafin (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D08501  Trolamine salicylate (USP); Salicylic acid trolamine; Salicylic acid triethanolamine; Arthricream (TN) (P) unclassified
D08516  Sitagliptin (USAN/INN) (P) unclassified
D08533  Sulbactam (INN) (P) unclassified
D08534  Sulbenicillin (INN) (P) unclassified
D08557  Talampicillin (INN) (P) unclassified
D08567  Temocillin disodium salt; Negaban (TN) (P) unclassified
D08586  Thiosalicylic acid; Pirosal (TN); Thiocyl (TN) (P) unclassified
D08593  Ticarcillin (INN); Ticillin [veterinary] (TN) (P) unclassified
D08605  Tipranavir (INN); Aptivus (TN) (P) unclassified
D08610  Tixocortol (INN) (P) unclassified
D08616  Teneligliptin (INN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D08649  Triptorelin acetate; Decapeptyl (TN) (P) unclassified
D08660  Ulobetasol (INN); Halobetasol (P) unclassified
D08699  Salmeterol xinafoate and fluticasone propionate; Adoair diskus (TN); Aerivio Spiromax (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D08843  Albiglutide (USAN); Albiglutide (genetical recombination) (JAN); Tanzeum (TN) (P) unclassified
D08856  Anamorelin hydrochloride (JAN/USAN); Adlumiz (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D08897  Dapagliflozin (JAN/USAN/INN); Forxiga (TN) (P) unclassified
D08923  Fesoterodine fumarate (JAN/USAN); Toviaz (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D08964  Perampanel (JAN/USAN); Fycompa (TN) (P) unclassified
D08976  Pomalidomide (JAN/USAN/INN); Pomalyst (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D08996  Saxagliptin (USAN/INN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D09017  Ticagrelor (JAN/USAN/INN); Brilinta (TN) (CI,P) unclassified
D09033  Voclosporin (JAN/USAN/INN); Lupkynis (TN) (CI,P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D09319  Indacaterol maleate (JAN/USAN); Arcapta (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D09348  Fostamatinib disodium (USAN); Fostamatinib sodium hydrate (JAN); Fostamatinib disodium hexahydrate; Tavalisse (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D09365  Palovarotene (JAN/USAN/INN); Sohonos (TN) (CI,P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D09566  Linagliptin (JAN/USAN/INN); Tradjenta (TN) (P) unclassified
D09572  Riociguat (JAN/USAN/INN); Adempas (TN) (P) unclassified
D09587  Brentuximab vedotin (USAN/INN); Brentuximab vedotin (genetical recombination) (JAN); Adcetris (TN) (P) unclassified
D09592  Canagliflozin (USAN/INN); Canagliflozin hydrate (JAN); Invokana (TN) (P) unclassified
D09595  Budesonide and formoterol fumarate dihydrate; Symbicort (TN); Budeforu (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D09634  Lersivirine (USAN/INN) (P) unclassified
D09638  Lomitapide mesylate (USAN); Lomitapide mesilate (JAN); Juxtapid (TN); Lojuxta (TN) (CI,P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D09647  Omadacycline (USAN) (P) unclassified
D09720  Rilpivirine (JAN/USAN/INN); Rekambys (TN) (P) unclassified
D09727  Insulin degludec (USAN/INN); Insulin degludec (genetical recombination) (JAN); Tresiba (TN) (P) unclassified
D09728  Bosutinib hydrate (JAN); Bosutinib monohydrate; Bosulif (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D09729  Lixisenatide (JAN/USAN/INN); Adlyxin (TN); Lyxumia (TN) (P) unclassified
D09730  Olaparib (JAN/USAN/INN); Lynparza (TN) (P) unclassified
D09731  Crizotinib (JAN/USAN/INN); Xalkori (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D09743  Telmisartan and amlodipine besilate (JP19); Telmisartan and amlodipine besylate; Micamlo (TN); Twynsta (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D09744  Pioglitazone hydrochloride and metformin hydrochloride (JP19); Pioglitazone and metformin; Metact (TN) (P) unclassified
D09745  Valsartan and amlodipine besilate; Exforge (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D09753  Saxagliptin hydrate (JAN); Onglyza (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D09756  Teneligliptin hydrobromide hydrate (JAN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D09763  Dapagliflozin propanediol (USAN); Dapagliflozin propylene glycolate hydrate (JP19); Dapagliflozin propandiol monohydrate; Forxiga (TN); Farxiga (TN) (P) unclassified
D09783  Tofacitinib citrate (JAN/USAN); Tasocitinib citrate; Xeljanz (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D09796  Hydrocortisone caproate (JAN) (P) unclassified
D09799  Carotegrast methyl (JAN); Carogra (TN) (P) CYP inhibition: CYP3A4
D09848  Pioglitazone hydrochloride and glimepiride tablets (JP19); Pioglitazone and glimepiride; Duetact (TN); Sonias (TN) (P) unclassified
D09889  Dulaglutide (USAN/INN); Dulaglutide (genetical recombination) (JAN); Trulicity (TN) (P) unclassified
D09894  Eliglustat tartrate (JAN/USAN); Eliglustat hemitartrate; Cerdelga (TN) (CI,P) unclassified
D09906  Fosdevirine (USAN/INN) (P) unclassified
D09940  Omadacycline tosylate (USAN); Nuzyra (TN) (P) unclassified
D09951  Ponatinib hydrochloride (JAN/USAN); Iclusig (TN) (P) unclassified
D09956  Quizartinib dihydrochloride (USAN); Quizartinib hydrochloride (JAN); Vanflyta (TN) (P) unclassified
D09958  Rilpivirine hydrochloride (JAN/USAN); Edurant (TN) (P) unclassified
D09960  Ruxolitinib phosphate (JAN/USAN); Jakafi (TN); Jakavi (TN); Opzelura (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D09996  Vemurafenib (JAN/USAN/INN); Zelboraf (TN) (P) CYP induction: CYP3A4
D09999  Tramadol hydrochloride and acetaminophen; Tramcet (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D10003  Hemin (JAN); Normosang (TN); Panhematin (TN) (P) CYP induction: CYP3A4
D10024  Selumetinib sulfate (JAN/USAN); Koselugo (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D10025  Semaglutide (USAN/INN); Semaglutide (genetical recombination) (JAN); Ozempic (TN) (P) unclassified
D10082  Suvorexant (JAN/USAN); MK-4305; Belsomra (TN) (P) unclassified
D10095  Cabozantinib s-malate (USAN); Cabozantinib malate (JAN); Cometriq (TN); Cabometyx (TN) (P) unclassified
D10104  Dabrafenib mesylate (USAN); Dabrafenib mesilate (JAN); Tafinlar (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D10127  Glycerol phenylbutyrate (JAN/USAN); Ravicti (TN) (P) unclassified
D10135  Macitentan (JAN/USAN); Opsumit (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D10137  Regorafenib hydrate (JAN); Stivarga (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D10159  Alogliptin benzoate and pioglitazone hydrochloride; Liovel (TN); Oseni (TN); Incresync (TN) (P) unclassified
D10160  Mitiglinide calcium hydrate and voglibose; Glubes (TN) (P) unclassified
D10161  Sarilumab (USAN); Sarilumab (genetical receombination) (JAN); Kevzara (TN) (P) unclassified
D10195  Luseogliflozin hydrate (JAN); Lusefi (TN) (P) unclassified
D10196  Ipragliflozin (INN) (P) unclassified
D10200  Ipragliflozin L-proline (JAN); Suglat (TN) (P) unclassified
D10218  Enzalutamide (JAN/USAN); Xtandi (TN) (P) unclassified
D10223  Ibrutinib (JAN/USAN); Imbruvica (TN) (P) unclassified
D10243  Irbesartan and amlodipine besilate (JP19); Aimix (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D10244  Metformin hydrochloride and rosiglitazone maleate; Avandamet (TN) (P) unclassified
D10251  Glimepiride and rosiglitazone maleate; Avandaryl (TN) (P) unclassified
D10253  Alogliptin benzoate and metformin hydrochloride; Kazano (TN); Vipdomet (TN) (P) unclassified
D10258  Simvastatin and sitagliptin phosphate; Juvisync (TN) (P) unclassified
D10261  Metformin hydrochloride and sitagliptin phosphate; Janumet (TN) (P) unclassified
D10262  Saxagliptin hydrochloride; Onglyza (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D10263  Metformin hydrochloride and saxagliptin hydrochloride; Kombiglyze (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D10264  Linagliptin and metformin hydrochloride; Jentaduet (TN) (P) unclassified
D10265  Glipizide and metformin hydrochloride; Metaglip (TN) (P) unclassified
D10266  Glyburide and metformin hydrochloride; Glibenclamide and metformin hydrochloride; Glucovance (TN) (P) unclassified
D10307  Avatrombopag maleate (JAN/USAN); Doptelet (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D10309  Brexpiprazole (JAN/USAN/INN); Rexulti (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D10313  Ertugliflozin (USAN/INN) (P) unclassified
D10369  Eravacycline (USAN/INN) (P) unclassified
D10372  Palbociclib (JAN/USAN); Ibrance (TN) (P) unclassified
D10421  Eravacycline dihydrochloride (USAN); Xerava (TN) (P) unclassified
D10450  Alectinib hydrochloride (JAN); Alecensa (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D10452  Cabazitaxel acetonate (JAN); Cabazitaxel acetone; Jevtana (TN) (P) unclassified
D10459  Empagliflozin (JAN/USAN/INN); Jardiance (TN) (P) unclassified
D10466  Vonoprazan fumarate (JAN/USAN); Takecab (TN); Voquezna (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D10473  Insulin peglispro (USAN/INN) (P) unclassified
D10478  Naldemedine tosylate (JAN/USAN); Naldemedine tosilate; Symproic (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D10500  Metformin hydrochloride and repaglinide; Prandimet (TN) (P) unclassified
D10501  Fluticasone furoate and vilanterol trifenatate; Breo ellipta (TN); Relvar ellipita (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D10502  Gemigliptin (INN) (P) unclassified
D10505  Glycopyrronium bromide and indacaterol maleate; Ultibro (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D10506  Fluticasone propionate and formoterol fumarate hydrate; Flutiform (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D10516  Aripiprazole hydrate (JAN); Aripiprazole monohydrate; Abilify maintena (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D10524  Azilsartan and amlodipine besilate; Zacras (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D10528  Aldosterone (INN) (P) unclassified
D10533  Umeclidinium bromide and vilanterol; Anoro (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D10551  Ceritinib (JAN/USAN/INN); Zykadia (TN) (P) unclassified
D10564  Amenamevir (JAN/INN); Amenalief (TN) (P) unclassified
D10566  Pasireotide pamoate (JAN); Signifor lar (TN) (P) unclassified
D10570  Insulin degludec (genetical recombination) and insulin aspart (genetical recombination); Ryzodeg (TN) (P) unclassified
D10586  Dapagliflozin and metformin; Xigduo xr (TN) (P) unclassified
D10587  Canagliflozin and metformin; Invokamet (TN) (P) unclassified
D10588  Empagliflozin and linagliptin; Glyxambi (TN) (P) unclassified
D10624  Doravirine (JAN/USAN/INN); Pifeltro (TN) (P) unclassified
D10633  Finerenone (JAN/USAN/INN); Kerendia (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D10643  Isavuconazonium sulfate (JAN/USAN); Cresemba (TN) (P) unclassified
D10663  Rimegepant sulfate (USAN); Rimegepant sulfate hydrate (JAN); Nurtec odt (TN); Vydura (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D10666  Sarecycline (USAN/INN) (P) unclassified
D10667  Sarecycline hydrochloride (USAN); Seysara (TN) (P) unclassified
D10669  Sotagliflozin (USAN/INN); Inpefa (TN) (P) unclassified
D10679  Venetoclax (JAN/USAN/INN); Venclexta (TN) (CI,P) unclassified
D10688  Abemaciclib (JAN/USAN/INN); Verzenio (TN) (P) unclassified
D10743  Vildagliptin and metformin hydrochloride (P) unclassified
D10752  Empagliflozin and metformin; Synjardy (TN) (P) unclassified
D10755  Elvitegravir, cobicistat, emtricitabine and tenofovir alafenamide; Genvoya (TN) (P) unclassified
D10761  Polatuzumab vedotin (USAN); Polatuzumab vedotin (genetical recombination) (JAN); Polatuzumab vedotin-piiq; Polivy (TN) (P) unclassified
D10762  Fosravuconazole L-lysine ethanolate (JAN) (P) unclassified
D10774  Vonoprazan, amoxicillin and metronidazole; Vonopion (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D10775  Vonoprazan, amoxicillin and clarithromycin; Vonosap (TN); Voquenza (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D10780  Perampanel hydrate (JAN); Fycompa (TN) (P) unclassified
D10800  Gilteritinib fumarate (JAN/USAN); Xospata (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D10801  Letermovir (JAN/USAN/INN); Prevymis (TN) (P) unclassified
D10805  Telmisartan, amlodipine and hydrochlorothiazide; Micatrio (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D10826  Saxagliptin and dapagliflozin; Qtern (TN) (P) unclassified
D10832  Darunavir and cobicistat; Prezcobix (TN); Rezolsta (TN) (P) unclassified
D10865  Bexagliflozin (USAN); Brenzavvy (TN) (P) unclassified
D10866  Brigatinib (JAN/USAN); Alunbrig (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D10891  Capmatinib hydrochloride (USAN); Capmatinib hydrochloride hydrate (JAN); Tabrecta (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D10892  Esaxerenone (JAN/INN) (P) unclassified
D10893  Acalabrutinib (JAN/USAN/INN); Calquence (TN) (P) unclassified
D10926  Entrectinib (JAN/USAN/INN); Rozlytrek (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D10927  Erdafitinib (JAN/USAN/INN); Balversa (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D10931  Etrasimod arginine (USAN); Etrasimod L-arginine (JAN); Velsipity (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D10990  Somatrogon (USAN/INN); Somatrogon (genetical recombination) (JAN); Somatrogon-ghla; Ngenla (TN) (P) unclassified
D10993  Tucidinostat (JAN/USAN/INN); Hiyasta (TN) (P) unclassified
D10999  Valbenazine tosylate (USAN); Valbenazine tosilate (JAN); Valbenazine ditosylate; Ingrezza (TN); Dysval (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D11000  Vamorolone (USAN/INN); Agamree (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D11012  Lorlatinib (JAN/USAN/INN); Lorbrena (TN) (P) unclassified
D11014  Glecaprevir and pibrentasvir; Mavyret (TN) (P) unclassified
D11022  Lemborexant (JAN/USAN/INN); Dayvigo (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D11023  Evogliptin (INN) (P) unclassified
D11034  Insulin glargine and lixisenatide; Insulin glargine (genetical recombination) and lixisenatide; Soliqua (TN) (P) unclassified
D11035  Fluticasone furoate, umeclidinium bromide and vilanterol; Trelegy ellipta (TN) (P) unclassified
D11040  Apalutamide (JAN/INN); Erleada (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D11043  Ertugliflozin pidolate; Ertugliflozin L-pyroglutamic acid; Steglatro (TN) (P) unclassified
D11048  Upadacitinib hydrate (JAN); Upadacitinib hemihydrate; Rinvoq (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D11053  Encorafenib (JAN/USAN/INN); Braftovi (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D11066  Ertugliflozin and sitagliptin; Steglujan (TN) (P) unclassified
D11067  Ertugliflozin and metformin; Segluromet (TN) (P) unclassified
D11070  Tirabrutinib hydrochloride (JAN/USAN); Velexbru (TN) (P) unclassified
D11090  Ivosidenib (JAN/USAN/INN); Tibsovo (TN) (P) unclassified
D11093  Avacopan (JAN/USAN/INN); Tavneos (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D11109  Anagliptin and Metformin hydrochloride (P) unclassified
D11138  Larotrectinib sulfate (JAN/USAN); Vitrakvi (TN) (P) unclassified
D11159  Leniolisib phosphate (JAN/USAN); Joenja (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D11194  Somapacitan (USAN/INN); Somapacitan (genetical recombination) (JAN); Somapacitan-beco; Sogroya (TN) (P) unclassified
D11246  Dapivirine (USAN/INN) (P) unclassified
D11296  Fedratinib hydrochloride (USAN); Fedratinib hydrochloride hydrate (JAN); Fedratinib dihydrochloride monohydrate; Inrebic (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D11342  Dorzagliatin (USAN) (P) unclassified
D11360  Tirzepatide (JAN/USAN); Mounjaro (TN); Zepbound (TN) (P) unclassified
D11370  Fosnetupitant chloride hydrochloride (JAN/USAN); Arokaris (TN) (P) unclassified
D11371  Capivasertib (JAN/USAN); Truqap (TN) (P) unclassified
D11382  Darunavir, cobicistat, emtricitabine and tenofovir alafenamide; Symtuza (TN) (P) unclassified
D11417  Pemigatinib (JAN/USAN/INN); Pemazyre (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D11422  Zanubrutinib (JAN/USAN/INN); Brukinsa (TN) (P) unclassified
D11454  Repotrectinib (JAN/USAN); Augtyro (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D11485  Tazemetostat hydrobromide (JAN/USAN); Tazverik (TN) (P) unclassified
D11525  Enfortumab vedotin (USAN); Enfortumab vedotin (genetical recombination) (JAN); Enfortumab vedotin-ejfv; Padcev (TN) (P) unclassified
D11557  Tecovirimat hydrate (JAN); Tecovirimat monohydrate; Tpoxx (TN); Tepoxx (TN) (P) unclassified
D11567  Insulin degludec and liraglutide; Xultophy (TN) (P) unclassified
D11572  Beclomethasone dipropionate monohydrate; Beconase aq (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D11584  Budesonide, glycopyrronium bromide and formoterol fumarate; Budesonide, glycopyrrolate and formoterol fumarate; Breztri (TN) (P) unclassified
D11659  Tolvaptan sodium phosphate (JAN); Samtasu (TN) (P) unclassified
D11662  Valemetostat tosilate (JAN); Valemetostat tosylate; Ezharmia (TN) (P) unclassified
D11674  Berotralstat hydrochloride (JAN/USAN); Orladeyo (TN) (P) CYP inhibition: CYP3A4
D11711  Dapagliflozin, metformin and saxagliptin; Qternmet xr (TN) (P) unclassified
D11713  Selpercatinib (JAN/USAN/INN); Retevmo (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D11725  Futibatinib (JAN/USAN/INN); Lytgobi (TN) (P) unclassified
D11793  Zuranolone (JAN/USAN/INN); Zurzuvae (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D11804  Aspirin and vonoprazan; Cabpirin (TN) (P) unclassified
D11807  Imeglimin hydrochloride (JAN); Twymeeg (TN) (P) unclassified
D11814  Tisotumab vedotin (USAN/INN); Tisotumab vedotin (genetical recombination) (JAN); Tisotumab vedotin-tftv; Tivdak (TN) (P) unclassified
D11816  Belumosudil mesylate (USAN); Belumosudil mesilate (JAN); Rezurock (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D11835  Vorasidenib citrate (USAN); Vorasidenib citric acid hydrate (JAN); Voranigo (TN) (P) unclassified
D11856  Empagliflozin, linagliptin and metformin hydrochloride; Trijardy xr (TN) (P) unclassified
D11861  Indacaterol acetate, glycopyrronium bromide and mometasone furoate; Enerzair (TN) (P) unclassified
D11862  Indacaterol and mometasone furoate; Atectura (TN) (P) unclassified
D11887  Daridorexant hydrochloride (JAN/USAN); Quviviq (TN) (P) unclassified
D11920  Pimitespib (JAN); Jeselhy (TN) (P) unclassified
D11923  Lobeglitazone (INN) (P) unclassified
D11924  Beinaglutide (INN) (P) unclassified
D11954  Belzutifan (JAN/USAN/INN); Welireg (TN) (P) unclassified
D11968  Teneligliptin hydrobromide (JAN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D11970  Ritlecitinib tosylate (USAN); Ritlecitinib tosilate (JAN); Litfulo (TN) (P) unclassified
D12015  St. John's wort; SJW (P) unclassified
D12050  Pirtobrutinib (JAN/USAN); Jaypirca (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D12055  Sotorasib (JAN/USAN); Lumakras (TN) (P) unclassified
D12217  Imlunestrant tosylate (USAN); Imlunestrant tosilate (JAN); Inluriyo (TN) (P) Enzyme: CYP3A4 / Target: ESR1 / CYP inhibition: CYP3A4
D12245  Lazertinib mesylate (USAN); Lazertinib mesilate hydrate (JAN); Lazcluze (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D12252  Iptacopan hydrochloride (USAN); Iptacopan hydrochloride hydrate (JAN); Iptacopan hydrochloride monohydrate; Fabhalta (TN) (P) CYP induction: CYP3A4
D12265  Mavacamten (JAN/USAN/INN); Camzyos (TN) (P) unclassified
D12269  Nirmatrelvir and ritonavir; Paxlovid (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D12294  Sitagliptin phosphate (JAN) (P) unclassified
D12311  Bortezomib hydrate (JAN) (P) unclassified
D12337  Leuprolide mesylate (USAN); Leuprorelin mesylate; Leuprorelin mesilate; Camcevi (TN) (P) unclassified
D12358  Insulin icodec (USAN/INN); Insulin icodec (genetical recombination) (JAN); Insulin icodec-abae; Awiqli (TN) (P) unclassified
D12364  Taletrectinib adipate (JAN/USAN); Ibtrozi (TN) (P) unclassified
D12396  Sebetralstat (JAN/USAN/INN); Ekterly (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D12442  Tucatinib ethanolate (JAN); Tucatinib hemiethanolate; Tukysa (TN) (P) unclassified
D12444  Nilotinib hydrochloride dihydrate (JAN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D12484  Carfloglitazar (INN) (P) unclassified
D12586  Mifepristone and misoprostol; Mefeego (TN) (P) unclassified
D12595  Aspirin trelamine (USAN) (P) unclassified
D12596  Aspirin trelamine hydrochloride (USAN) (P) unclassified
D12611  Vornorexant hydrate (JAN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D12637  Darunavir hydrate (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D12703  Linagliptin hydrate (JAN); Linagliptin hemihydrate (P) unclassified
D12704  Acalabrutinib maleate hydrate (JAN); Acalabrutinib maleate monohydrate; Calquence (TN) (P) unclassified
D12752  Darunavir propylene glycolate (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D12837  Risovalisib mesilate hydrate (JAN); Risovalisib mesylate dihydrate; Haizexin (TN) (P) unclassified
D12963  Macitentan and tadalafil; Opsynvi (TN); Yuvanci (TN) (CI,P) unclassified
D13015  Enavogliflozin (INN) (P) unclassified
D13018  Elsulfavirine (INN) (P) unclassified
D13026  Atogepant hydrate (JAN); Aquipta (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D13028  Insulin efsitora alfa (INN); Insulin efsitora alfa (genetical recombination) (JAN) (P) unclassified
D13055  Sitagliptin hydrochloride; Sitagliptin monohydrochloride monohydrate; Brynovin (TN) (P) unclassified
D13245  Insulin icodec (genetical recombination) and semaglutide (genetical recombination); Kyinsu (TN) (P) unclassified