C01946 |
Oleandomycin; Amimycin; Landomycin; Matromycin; Romicil |
(P) unclassified |
C04931 |
Argatroban; (2R,4R)-4-Methyl-1[Nalpha-[(3-methyl-1,2,3,4-tetrahydro-8-quinolinyl)sulfonyl]-L-arginyl]-2-piperadinecarboxylic acid |
(P) unclassified |
C07051 |
Indinavir |
(P) unclassified |
C07521 |
Thiopental |
(P) unclassified |
D00085 |
Insulin (JAN/USP) |
(P) unclassified |
D00105 |
Estradiol (JAN/USP/INN); Climara (TN); Divigel (TN); Estrace (TN); Estraderm (TN); Estrasorb (TN); Estring (TN); Estrogel (TN); Innofem (TN); Vagifem (TN); Vivelle (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D00106 |
Epoprostenol (USAN/INN); Prostaglandin I2; Prostacyclin; Epoprostenol (TN) |
(P) unclassified |
D00107 |
Tacrolimus (USP/INN); Tacrolimus hydrate (JP18); Prograf (TN); Protopic (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D00109 |
Aspirin (JP18/USP); Aspalon (JAN); Acetylsalicylic acid; Easprin (TN); Durlaza (TN) |
(P) unclassified |
D00124 |
Ephedrine (USP); Ephedrine (TN) |
(P) unclassified |
D00127 |
Piroxicam (JP18/USP/INN); Feldene (TN) |
(P) unclassified |
D00130 |
Diflunisal (JAN/USP/INN); Dolobid (TN) |
(P) unclassified |
D00136 |
Haloperidol (JP18/USP/INN); Haldol (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D00140 |
Erythromycin (JP18/USP/INN); Akne-mycin (TN); Eryc (TN); Erygel (TN); Pce (TN); Staticin (TN); T-stat (TN) |
(P) unclassified |
D00168 |
Cytarabine (JP18/USP/INN); ARA-C; Depocyt (TN) |
(P) unclassified |
D00181 |
Argatroban (USP); Argatroban hydrate (JP18); Novastan (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D00184 |
Cyclosporine (USP); Ciclosporin (JP18); Gengraf (TN); Neoral (TN); Restasis (TN); Sandimmune (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4 |
D00186 |
Ciprofloxacin (JP18/USP/INN); Cipro (TN); Otiprio (TN) |
(P) unclassified |
D00197 |
Reserpine (JP18/USP/INN); Apoplon (TN); Serpalan (TN) |
(P) unclassified |
D00198 |
Rescinnamine (JAN/INN); Tsuruselpi S (TN) |
(P) unclassified |
D00203 |
Amphotericin B (JP18/USP/INN); Ambisome (TN); Amphotec (TN); Fungizone (TN) |
(P) unclassified |
D00210 |
Norfloxacin (JP18/USP/INN); Noroxin (TN) |
(P) unclassified |
D00211 |
Rifampin (USP); Rifampicin (JP18/INN); Rifadin (TN); Rimactane (TN) |
(P) CYP induction: CYP3A4 |
D00216 |
Acarbose (JAN/USAN/INN); Precose (TN) |
(P) unclassified |
D00218 |
Acetazolamide (JP18/USP/INN); Diamox (TN) |
(P) unclassified |
D00219 |
Acetohexamide (JP18/USP/INN); Dymelor (TN) |
(P) unclassified |
D00247 |
Bumetanide (JP18/USP/INN); Bumex (TN) |
(P) unclassified |
D00252 |
Carbamazepine (JP18/USP/INN); Equetro (TN); Tegretol (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D00271 |
Chlorpropamide (JP18/USP/INN); Diabinese (TN) |
(P) unclassified |
D00272 |
Chlorthalidone (USP); Chlortalidone (JAN/INN); Hygroton (TN); Thalitone (TN) |
(P) unclassified |
D00276 |
Clarithromycin (JP18/USP/INN); Biaxin (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4 |
D00281 |
Clonidine (JAN/USP/INN); Catarpres-TTS (TN) |
(P) unclassified |
D00282 |
Clotrimazole (JP18/USP/INN); Lotrimin (TN); Mycelex (TN) |
(P) CYP inhibition: CYP3A4 |
D00283 |
Clozapine (JAN/USP/INN); Clozaril (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D00287 |
Cyclophosphamide (USP); Cyclophosphamide hydrate (JP18); Cytoxan (TN); Neosar (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D00292 |
Dexamethasone (JP18/USP/INN); Decadron (TN); Maxidex (TN) |
(P) Enzyme: CYP3A4 / Target: NR3C1 / CYP induction: CYP3A4 |
D00293 |
Diazepam (JP18/USP/INN); Diastat (TN); Valium (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D00294 |
Diazoxide (JAN/USP/INN); Hyperstat (TN); Proglycem (TN) |
(P) unclassified |
D00298 |
Digoxin (JP18/USP); Lanoxicaps (TN); Lanoxin (TN) |
(P) unclassified |
D00302 |
Dipyridamole (JP18/USP/INN); Persantine (TN) |
(P) unclassified |
D00313 |
Ethacrynic acid (USP); Etacrynic acid (JP18/INN) |
(P) unclassified |
D00320 |
Fentanyl (JAN/USP/INN); Duragesic (TN); Subsys (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D00322 |
Fluconazole (JP18/USP/INN); Diflucan (TN) |
(P) CYP inhibition: CYP3A4 |
D00330 |
Flurbiprofen (JP18/USP/INN); Ansaid (TN) |
(P) unclassified |
D00331 |
Furosemide (JP18/USP/INN); Frusemide; Lasix (TN) |
(P) unclassified |
D00335 |
Glipizide (USP/INN); Glucotrol (TN) |
(P) unclassified |
D00336 |
Glyburide (USP); Glibenclamide (JP18/INN); Diabeta (TN); Glynase (TN); Micronase (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D00340 |
Hydrochlorothiazide (JP18/USP/INN); Esidrix (TN); Microzide (TN) |
(P) unclassified |
D00345 |
Indapamide (JP18/USP); Lozol (TN); Natrix (TN) |
(P) unclassified |
D00350 |
Itraconazole (JP18/USP); Itrizole (TN); Sporanox (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4 |
D00351 |
Ketoconazole (JP18/USP); Nizoral (TN); Xolegel (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4 |
D00372 |
Thiabendazole (USP); Tiabendazole (JAN/INN); Mintezol (TN) |
(P) unclassified |
D00377 |
Mesalamine (USP); Mesalazine (JP18/INN); Apriso (TN); Asacol (TN); Canasa (TN); Delzicol (TN); Lialda (TN); Mesalamine (TN); Pentasa (TN); Rowasa (TN); Sfrowasa (TN) |
(P) unclassified |
D00379 |
Tolazamide (JAN/USP/INN); Tolinase (TN) |
(P) unclassified |
D00380 |
Tolbutamide (JP18/USP/INN); Orinase (TN) |
(P) unclassified |
D00382 |
Torsemide (USP); Torasemide (JAN/INN); Demadex (TN); Luprac (TN) |
(P) unclassified |
D00386 |
Triamterene (JP18/USP/INN); Dyrenium (TN) |
(P) unclassified |
D00387 |
Triazolam (JP18/USP/INN); Halcion (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D00395 |
Troglitazone (JAN/USAN/INN); Rezulin (TN) |
(P) unclassified |
D00405 |
Methyldopa (USP); Methyldopa hydrate (JP18); Aldomet (TN) |
(P) unclassified |
D00416 |
Miconazole (JP18/USP/INN); Monistat (TN); Oravig (TN) |
(P) unclassified |
D00418 |
Minoxidil (JAN/USP/INN); Loniten (TN); Riup (TN); Rogaine (TN) |
(P) unclassified |
D00420 |
Mitotane (JAN/USP/INN); Lysodren (TN) |
(P) unclassified |
D00426 |
Risperidone (JP18/USP/INN); Risperdal (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D00427 |
Ritonavir (JAN/USP/INN); Norvir (TN) |
(P) unclassified |
D00428 |
Salsalate (USP/INN); Sasapyrine (JAN); Disalcid (TN) |
(P) unclassified |
D00429 |
Saquinavir (JAN/USP/INN); Fortovase (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D00430 |
Secobarbital (USP/INN); Seconal (TN) |
(P) unclassified |
D00431 |
Metolazone (JAN/USP/INN); Zaroxolyn (TN) |
(P) unclassified |
D00435 |
Nevirapine (JAN/USP/INN); Viramune (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D00443 |
Spironolactone (JP18/USP/INN); Aldactone (TN) |
(P) unclassified |
D00448 |
Sulfasalazine (USP/INN); Salazosulfapyridine (JP18); Azulfidine (TN) |
(P) unclassified |
D00453 |
Ofloxacin (JP18/USP/INN); Floxin (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D00458 |
Quetiapine fumarate (JP18/USP); Seroquel (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D00461 |
Quinethazone (JAN/INN); Hydromox (TN) |
(P) unclassified |
D00471 |
Praziquantel (JAN/USP/INN); Biltricide (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D00474 |
Primidone (JP18/USP/INN); Mysoline (TN) |
(P) unclassified |
D00483 |
Propranolol hydrochloride (JP18/USP); Inderal (TN); Innopran XL (TN) |
(P) unclassified |
D00491 |
Paclitaxel (JAN/USP/INN); Abraxane (TN); Taxol (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D00499 |
Pentobarbital (USP/INN); Nembutal (TN) |
(P) unclassified |
D00500 |
Pentobarbital sodium (JAN/USP); Nembutal sodium (TN) |
(P) unclassified |
D00506 |
Phenobarbital (JP18/USP/INN); Luminal (TN) |
(P) unclassified |
D00512 |
Phenytoin (JP18/USP/INN); Dilantin (TN) |
(P) unclassified |
D00519 |
Chlorothiazide (JAN/USP/INN); Diuril (TN) |
(P) unclassified |
D00528 |
Caffeine (USP); Anhydrous caffeine (JP18); Anhydrous caffeine (TN); Respia (TN) |
(P) unclassified |
D00537 |
Topiramate (JAN/USP/INN); Topamax (TN); Trokendi xr (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D00550 |
Midazolam (JAN/USP/INN); Dormicum (TN); Buccolam (TN); Nayzilam (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D00554 |
Ethinyl estradiol (USP); Ethinylestradiol (JP18/INN); Estinyl (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4 |
D00555 |
Amobarbital (JP18/INN); Isomytal (TN) |
(P) unclassified |
D00563 |
Mirtazapine (JAN/USP/INN); Remeron (TN); Reflex (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D00564 |
Warfarin sodium (USP); Coumadin (TN); Jantoven (TN) |
(P) unclassified |
D00566 |
Sodium salicylate (JP18/USP); Salsonin (TN) |
(P) unclassified |
D00578 |
Voriconazole (JP18/USP/INN); Vfend (TN) |
(P) unclassified |
D00588 |
Levofloxacin (USP); Levofloxacin hydrate (JP18); Levofloxacin hemihydrate; Iquix (TN); Levaquin (TN); Quixin (TN) |
(P) unclassified |
D00593 |
Glimepiride (JP18/USP/INN); Amaryl (TN) |
(P) unclassified |
D00594 |
Repaglinide (JAN/USP/INN); Prandin (TN); Surepost (TN) |
(P) unclassified |
D00595 |
Buformin (USAN/INN) |
(P) unclassified |
D00596 |
Rosiglitazone maleate (JAN/USP); Avandia (TN) |
(P) unclassified |
D00604 |
Clonidine hydrochloride (JP18/USP); Nexiclon (TN); Kapvay (TN); Duraclon (TN); Catapres (TN) |
(P) unclassified |
D00606 |
Guanfacine hydrochloride (JAN/USP); Intuniv (TN); Tenex (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D00608 |
Doxazosin mesylate (USP); Doxazosin mesilate (JP18); Cardura (TN) |
(P) unclassified |
D00609 |
Prazosin hydrochloride (JP18/USP); Minipress (TN) |
(P) unclassified |
D00611 |
Mecamylamine hydrochloride (USP); Inversine (TN) |
(P) unclassified |
D00612 |
Trimetaphan camsilate (JAN/INN); Trimetaphan camsylate; Arfonad (TN) |
(P) unclassified |
D00614 |
Sodium nitroprusside (USP); Sodium nitroprusside hydrate (JAN); Nitropress (TN) |
(P) unclassified |
D00615 |
Amlodipine besylate (USP); Amlodipine besilate (JP18); Norvasc (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D00625 |
Miglitol (JP18/USAN/INN); Glyset (TN) |
(P) unclassified |
D00636 |
Amiodarone hydrochloride (JP18/USP); Ancaron (TN); Cordarone (TN); Nexterone (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D00649 |
Amiloride hydrochloride (USP); Midamor (TN) |
(P) unclassified |
D00650 |
Bendroflumethiazide (JAN/USP/INN); Naturetin (TN) |
(P) unclassified |
D00651 |
Benzthiazide (JAN/INN); Exna (TN) |
(P) unclassified |
D00654 |
Hydroflumethiazide (JAN/USP/INN); Saluron (TN) |
(P) unclassified |
D00656 |
Methyclothiazide (JAN/USP/INN); Enduron (TN) |
(P) unclassified |
D00657 |
Polythiazide (JAN/USAN/INN); Renese (TN) |
(P) unclassified |
D00658 |
Trichlormethiazide (JP18/USP/INN); Naqua (TN) |
(P) unclassified |
D00670 |
Donepezil hydrochloride (JP18/USP); Aricept (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D00678 |
Ondansetron hydrochloride hydrate (JAN/USP); Ondansetron hydrochloride; Zofran (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D00683 |
Albuterol sulfate (USP); Salbutamol sulfate (JP18); Accuneb (TN); Proventil (TN); Ventolin (TN) |
(P) unclassified |
D00687 |
Salmeterol xinafoate (JAN/USP); Serevent (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D00688 |
Terbutaline sulfate (JP18/USP); Brethine (TN) |
(P) unclassified |
D00698 |
Aprobarbital (INN); Alurate (TN) |
(P) unclassified |
D00699 |
Butabarbital sodium (USP); Secbutabarbital sodium (INN); Butabarb (TN); Butisol sodium (TN) |
(P) unclassified |
D00700 |
Mephobarbital (JAN/USP); Methylphenobarbital (INN); Mebaral (TN) |
(P) unclassified |
D00701 |
Phenobarbital sodium (JAN/USP/INN); Luminal sodium (TN) |
(P) unclassified |
D00712 |
Methohexital sodium (USP); Brevital sodium (TN) |
(P) unclassified |
D00713 |
Thiamylal sodium (JP18); Surital (TN) |
(P) unclassified |
D00714 |
Thiopental sodium (JP18/USP/INN); Pentothal (TN) |
(P) unclassified |
D00727 |
Olsalazine sodium (USAN); Dipentum (TN) |
(P) unclassified |
D00749 |
Leflunomide (JAN/USP/INN); Arava (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D00754 |
Thalidomide (JAN/USP/INN); Thalomid (TN); Thaled (TN) |
(P) unclassified |
D00762 |
Metyrosine (USP); Metirosine (JAN/INN); Demser (TN) |
(P) unclassified |
D00765 |
Rocuronium bromide (JAN/USP/INN); Zemuron (TN) |
(P) unclassified |
D00769 |
Clopidogrel bisulfate (USP); Clopidogrel sulfate (JP18); Clopidogrel sulfate tablets (JP18); Clopidogrel hydrogen sulphate; Isocover (TN); Plavix (TN) |
(P) unclassified |
D00809 |
Amitriptyline hydrochloride (JP18/USP); Elavil (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D00810 |
Choline salicylate (JAN/USAN/INN); Arthropan (TN) |
(P) unclassified |
D00827 |
Magnesium salicylate (USP); Magnesium salicylate tetrahydrate; Magan (TN) |
(P) unclassified |
D00831 |
Mefloquine hydrochloride (JP18/USP); Lariam (TN) |
(P) unclassified |
D00836 |
Buprenorphine hydrochloride (JP18/USP); Buprenex (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D00851 |
Erythromycin estolate (USP); Erythromycin estorate (JAN); Ilosone (TN) |
(P) unclassified |
D00873 |
Lomefloxacin hydrochloride (JAN/USAN); Maxaquin (TN) |
(P) unclassified |
D00874 |
Moxifloxacin hydrochloride (JAN/USP); Avelox (TN); Vigamox (TN) |
(P) unclassified |
D00880 |
Butoconazole nitrate (USP); Femstat (TN); Gynazole-1 (TN) |
(P) unclassified |
D00881 |
Econazole nitrate (JAN/USP); Ecoza (TN); Spectazole (TN) |
(P) unclassified |
D00882 |
Miconazole nitrate (JP18/USP); Micatin (TN); Monistat (TN) |
(P) unclassified |
D00885 |
Oxiconazole nitrate (JAN/USAN); Oxistat (TN) |
(P) unclassified |
D00886 |
Sulconazole nitrate (JAN/USP); Exelderm (TN) |
(P) unclassified |
D00888 |
Terconazole (USP/INN); Terazol 3 (TN) |
(P) unclassified |
D00890 |
Tioconazole (JAN/USP/INN); Vagistat-1 (TN) |
(P) unclassified |
D00894 |
Amprenavir (JAN/USAN/INN); Agenerase (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D00897 |
Indinavir sulfate (USP); Crixivan (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4 |
D00899 |
Nelfinavir mesylate (USAN/INN); Nelfinavir mesilate (JAN); Viracept (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4 |
D00904 |
Diclofenac sodium (JP18/USP); Solaraze (TN); Voltaren (TN) |
(P) unclassified |
D00944 |
Metformin hydrochloride (JP18/USP); Glucophage (TN) |
(P) unclassified |
D00945 |
Pioglitazone hydrochloride (JP18/USP); Actos (TN) |
(P) unclassified |
D00951 |
Medroxyprogesterone acetate (JP18/USP); Depo-provera (TN); Depo-subq provera 104 (TN); Provera (TN) |
(CI,P) unclassified |
D00961 |
Bicalutamide (JP18/USP/INN); Casodex (TN) |
(P) CYP inhibition: CYP3A4 |
D00964 |
Letrozole (JAN/USP/INN); Femara (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D00969 |
Meloxicam (JAN/USP/INN); Mobic (TN) |
(P) unclassified |
D00971 |
Sodium thiosalicylate; Thiosalicylic acid sodium salt; Rexolate (TN) |
(P) unclassified |
D01028 |
Ticlopidine hydrochloride (JP18/USP); Ticlid (TN) |
(P) unclassified |
D01029 |
Tirofiban hydrochloride (USAN); Tirofiban hydrochloride hydrate; Aggrastat (TN) |
(P) unclassified |
D01061 |
Irinotecan hydrochloride (USP); Irinotecan hydrochloride hydrate (JP18); Irinotecan hydrochloride trihydrate; CPT 11; CPT-11; Campto (TN); Camptosar (TN); Onivyde (TN) |
(P) unclassified |
D01071 |
Hexobarbital (JAN/INN) |
(P) unclassified |
D01078 |
Telithromycin (JAN/USAN/INN); Ketek (TN) |
(P) unclassified |
D01087 |
Methyl salicylate (JP18/NF); Methyl salicylate (TN) |
(P) unclassified |
D01092 |
Lanoconazole (JP18/INN); Latoconazole; Astat (TN) |
(P) unclassified |
D01111 |
Nateglinide (JP18/USP/INN); Starsis (TN) |
(P) unclassified |
D01115 |
Eplerenone (JP18/USAN/INN); Inspra (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D01144 |
Prulifloxacin (JAN/INN); Sword (TN) |
(P) unclassified |
D01160 |
Saquinavir mesylate (USP); Saquinavir mesilate (JAN); Invirase (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D01164 |
Aripiprazole (JAN/USP/INN); Abilify (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D01176 |
Blonanserin (JAN/INN); AD 5423 |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D01196 |
Acetazolamide sodium (JAN); Diamox (TN) |
(P) unclassified |
D01213 |
Tolvaptan (JAN/USAN/INN); Samsca (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D01220 |
Trapidil (JP18/INN); Rocornal (TN) |
(P) unclassified |
D01227 |
Bosentan (USAN); Bosentan hydrate (JAN); Tracleer (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D01235 |
Josamycin (JP18/USAN/INN); Leucomycin A3; JM; Josamycin (TN) |
(P) CYP inhibition: CYP3A4 |
D01236 |
Conivaptan hydrochloride (JAN/USAN); Vaprisol (TN) |
(P) unclassified |
D01240 |
Deslanoside (JP18/USP/INN); Cedilanid-d (TN) |
(P) unclassified |
D01241 |
Penflutizide (JAN/INN) |
(P) unclassified |
D01246 |
Benzylhydrochlorothiazide (JAN); Behyd (TN) |
(P) unclassified |
D01247 |
Ethiazide (JAN/INN) |
(P) unclassified |
D01253 |
Clobazam (JAN/USAN/INN); Mystan (TN); Onfi (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D01256 |
Cyclothiazide (JAN/USAN/INN); Anhydron (TN) |
(P) unclassified |
D01263 |
Ritodrine hydrochloride (JP18/USP); Yutopar (TN) |
(P) unclassified |
D01276 |
Atazanavir sulfate (JAN/USAN); Reyataz (TN) |
(P) CYP inhibition: CYP3A4 |
D01280 |
Warfarin potassium (JP18); Athrombin-K (TN) |
(P) unclassified |
D01302 |
Hydralazine hydrochloride (JP18/USP); Apresoline (TN) |
(P) unclassified |
D01310 |
Secobarbital sodium (JAN/USP); Seconal sodium (TN) |
(P) unclassified |
D01322 |
Troleandomycin (USAN/INN); Triacetyloleandomycin (JAN); TAO; Tao (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4 |
D01323 |
Azosemide (JP18/USAN/INN); Diart (TN) |
(P) unclassified |
D01333 |
Urapidil (JP18/INN); Ebrantil (TN) |
(P) unclassified |
D01337 |
Epoprostenol sodium (JAN/USAN); Flolan (TN); Veletri (TN) |
(P) unclassified |
D01339 |
Midecamycin (JP18/INN); Medemycin (TN) |
(P) CYP inhibition: CYP3A4 |
D01356 |
Glymidine sodium (JAN/USAN/INN) |
(P) unclassified |
D01358 |
Mianserin hydrochloride (JAN/USAN); Tetramide (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D01360 |
Clenbuterol hydrochloride (JAN/USP); Spiropent (TN) |
(P) unclassified |
D01361 |
Erythromycin ethylsuccinate (JP18/USP); E.E.S. (TN); Eryped (TN); Erythrocin W (TN) |
(P) unclassified |
D01362 |
Tulobuterol hydrochloride (JP18); Hokunalin (TN); Respacal (TN) |
(P) unclassified |
D01372 |
Zopiclone (JP18/INN); Amoban (TN); Zopiclone (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D01375 |
Methenolone acetate (USAN); Metenolone acetate (JP18); Primobolan (TN) |
(P) unclassified |
D01382 |
Metharbital (JAN/INN); Gemonil (TN) |
(P) unclassified |
D01386 |
Ephedrine hydrochloride (JP18/USP); Ephedrine hydrochloride (TN) |
(P) unclassified |
D01390 |
Isoproterenol hydrochloride (USP); dl-Isoprenaline hydrochloride (JAN); Isuprel (TN); Proternol-S (TN) |
(P) unclassified |
D01399 |
Fentanyl citrate (JP18/USP); Abstral (TN); Fentora (TN); Lazanda (TN); Oralet (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D01418 |
Tamibarotene (JAN/USAN/INN); Am 80; Amnoid (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D01425 |
Lopinavir (JAN/USP/INN) |
(P) unclassified |
D01428 |
Fenoterol hydrobromide (JAN); Berotec (TN) |
(P) unclassified |
D01429 |
Fosfluconazole (JAN/INN); Prodif (TN) |
(P) CYP inhibition: CYP3A4 |
D01436 |
Clorexolone (JAN/USAN/INN) |
(P) unclassified |
D01441 |
Imatinib mesylate (USAN); Imatinib mesilate (JAN); Gleevec (TN); Glivec (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D01453 |
Caffeine hydrate (JP18); Caffeine monohydrate; Caffeine (TN) |
(P) unclassified |
D01466 |
Ethenzamide (JP18/INN); Ethenzamide (TN) |
(P) unclassified |
D01475 |
Flurbiprofen axetil (JAN); FP 83; Ropion (TN) |
(P) unclassified |
D01480 |
Isoconazole nitrate (JAN); Adestan-G (TN) |
(P) unclassified |
D01551 |
Beraprost sodium (JP18/USAN); Procylin (TN) |
(P) unclassified |
D01557 |
Glycol salicylate (JAN); Ethylene glycol salicylate; Norgesic (TN); Phlogont (TN) |
(P) unclassified |
D01599 |
Gliclazide (JP18/INN); Glimicron (TN) |
(P) unclassified |
D01603 |
Bethanidine sulfate (JAN/USAN); Tenathan (TN) |
(P) unclassified |
D01605 |
Meticrane (JP18/INN); Arresten (TN) |
(P) unclassified |
D01614 |
Acetylkitasamycin (JP18); Neo-leucomycin H (TN) |
(P) unclassified |
D01620 |
Neticonazole hydrochloride (JAN); Atolant (TN) |
(P) unclassified |
D01624 |
Sarpogrelate hydrochloride (JP18); Anplag (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D01634 |
Piretanide (JAN/USAN/INN); Arelix (TN) |
(P) unclassified |
D01636 |
Midecamycin acetate (JP18); Miocamycin; Miocamycin (TN) |
(P) CYP inhibition: CYP3A4 |
D01664 |
Omoconazole nitrate (JAN/USAN) |
(P) unclassified |
D01665 |
Voglibose (JP18/USAN/INN); Basen (TN) |
(P) unclassified |
D01670 |
Nafamostat mesylate (USAN); Nafamostat mesilate (JP18); Ronastat (TN) |
(P) unclassified |
D01672 |
Gabexate mesilate (JP18); Gabexate mesylate; Arodate (TN) |
(P) unclassified |
D01683 |
Ozagrel hydrochloride hydrate (JAN); Ozagrel hydrochloride; Ozagrel (TN) |
(P) unclassified |
D01684 |
Ozagrel sodium (JP18); Ozapen (TN) |
(P) unclassified |
D01710 |
Roxithromycin (JP18/USAN/INN); Rulide (TN) |
(P) unclassified |
D01740 |
Barbital (JP18/INN); Barbital (TN) |
(P) unclassified |
D01744 |
Brotizolam (JP18/USAN/INN); Lendormin (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D01775 |
Bifonazole (JP18/USAN/INN); Mycospor (TN) |
(P) unclassified |
D01799 |
Glyclopyramide (JAN/INN); Deamelin-S (TN) |
(P) unclassified |
D01804 |
Cadralazine (JP18/INN); Cadral (TN) |
(P) unclassified |
D01810 |
Nicorandil (JP18/USAN/INN); Sigmart (TN) |
(P) unclassified |
D01811 |
Salicylamide (JAN/USP/INN); Salicylamide (TN) |
(P) unclassified |
D01822 |
Clofenamide (JAN/INN) |
(P) unclassified |
D01844 |
Fondaparinux sodium (JAN/USP/INN); Arixtra (TN) |
(P) unclassified |
D01854 |
Mitiglinide calcium hydrate (JP18); Mitiglinide calcium dihydrate; Glufast (TN) |
(P) unclassified |
D01855 |
Mozavaptane hydrochloride (JAN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D01877 |
Mefruside (JP18/USAN/INN); Baycaron (TN) |
(P) unclassified |
D01892 |
Icosapent ethyl (USAN); Ethyl icosapentate (JP18); Epadel S (TN); Vascepa (TN) |
(P) unclassified |
D01895 |
Tripamide (JAN/USAN/INN); Normonal (TN) |
(P) unclassified |
D01896 |
Cilostazol (JP18/USP/INN); Pletal (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D01897 |
Rokitamycin (JAN/INN); Ricamycin (TN) |
(P) unclassified |
D01898 |
Haloperidol decanoate (JAN/USP); Halomonth (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D01943 |
Canrenoate potassium (USAN); Potassium canrenoate (JP18); Soldactone (TN) |
(P) unclassified |
D01973 |
Eletriptan hydrobromide (JAN/USAN); Relpax (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D01977 |
Gefitinib (JP18/USAN/INN); Iressa (TN) |
(P) unclassified |
D01980 |
Luliconazole (JAN/USAN/INN); Lulicon (TN); Luzu (TN) |
(P) CYP inhibition: CYP3A4 |
D01981 |
Ximelagatran (JAN/USAN/INN); Exanta (TN) |
(P) unclassified |
D01996 |
Tosufloxacin tosylate hydrate (JP18); Tosufloxacin tosilate; Ozex (TN); Tosuxacin (TN) |
(P) unclassified |
D02000 |
Kitasamycin tartrate (JP18); Leucomycin tartrate (TN) |
(P) unclassified |
D02008 |
Tadalafil (JAN/USP/INN); Adcirca (TN); Cialis (TN); Zalutia (TN) |
(CI,P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D02009 |
Erythromycin lactobionate (JP18/USP); Erythrocin (TN) |
(P) unclassified |
D02061 |
Cyclopenthiazide (JAN/USAN/INN); Navidrex (TN) |
(P) unclassified |
D02102 |
Methadone hydrochloride (JAN/USP); Dolophine hydrochloride (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D02103 |
Phenytoin sodium (USP); Phenytoin sodium for injection (JP18); Aleviatin (TN); Dilantin (TN) |
(P) unclassified |
D02109 |
dl-Methylephedrine hydrochloride (JP18); Methy-F (TN) |
(P) unclassified |
D02112 |
Heparin sodium (JP18/USP/INN); Parnaparin sodium (INN); Liquemin sodium (TN) |
(P) unclassified |
D02134 |
Azithromycin hydrate (JP18); Azithromycin dihydrate; Zithromac (TN); Zmax (TN); Azimycin (TN) |
(P) unclassified |
D02150 |
l-Isoprenaline hydrochloride (JP18); Proternol-L (TN) |
(P) unclassified |
D02151 |
Tulobuterol (JP18/INN); Atenos (TN); Hokunalin (TN) |
(P) unclassified |
D02169 |
Croconazole hydrochloride (JP18); Pilzcin (TN) |
(P) unclassified |
D02184 |
Erythromycin stearate (JP18/USP); Bristamycin (TN) |
(P) unclassified |
D02186 |
Oleandomycin phosphate (JAN); Matromycin (TN) |
(P) unclassified |
D02206 |
Buformin hydrochloride (JP18); Dibetos-B (TN) |
(P) unclassified |
D02216 |
Ciprofloxacin hydrochloride (USP); Ciprofloxacin hydrochloride hydrate (JP18); Ciloxan (TN); Cipro (TN); Proquin XR (TN) |
(P) unclassified |
D02229 |
Sildenafil citrate (JAN/USP); Revatio (TN); Viagra (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D02235 |
Desmopressin acetate (USP); Desmopressin acetate hydrate (JAN); Desmopressin acetate trihydrate; DDAVP (TN); Minirinmelt (TN); Stimate (TN) |
(CI) unclassified |
D02237 |
Guanethidine sulfate (USAN) |
(P) unclassified |
D02252 |
Amobarbital sodium (JAN/USP); Amytal sodium (TN) |
(P) unclassified |
D02253 |
Pentobarbital calcium (JP18); Ravona (TN) |
(P) unclassified |
D02269 |
Kitasamycin (JP18/USAN); Leucomycin (TN) |
(P) unclassified |
D02323 |
Tolrestat (USAN/INN); Alredase (TN) |
(P) unclassified |
D02363 |
Ketanserin (USAN/INN) |
(P) unclassified |
D02372 |
Perospirone hydrochloride hydrate (JAN); Lullan (TN) |
(P) unclassified |
D02386 |
Ticrynafen (USAN); Tienilic acid (INN); Selacryn (TN) |
(P) unclassified |
D02420 |
Acetylspiramycin (JP18); Spiramycin II; Acetylspiramycin (TN) |
(P) unclassified |
D02425 |
Carbutamide (INN); Invenol (TN) |
(P) unclassified |
D02426 |
Glycyclamide (INN); Tolcyclamide |
(P) unclassified |
D02427 |
Glibornuride (USAN/INN); Glutril (TN) |
(P) unclassified |
D02428 |
Glisentide (INN); Glypentide; Staticum (TN) |
(P) unclassified |
D02429 |
Glisolamide (INN); Glysolamide; Diabenor (TN) |
(P) unclassified |
D02430 |
Gliquidone (INN); Glurenorm (TN) |
(P) unclassified |
D02453 |
Flumethiazide (INN); Ademol (TN) |
(P) unclassified |
D02460 |
Clopamide (USAN/INN); Aquex (TN) |
(P) unclassified |
D02475 |
Sitafloxacin (USAN); Sitafloxacin hydrate (JAN) |
(P) unclassified |
D02478 |
Disulfamide (BAN) |
(P) unclassified |
D02484 |
Artemether and lumefantrine; Coartem (TN) |
(P) unclassified |
D02490 |
Tylosin (USP/INN); TS; Tylan (TN) |
(P) unclassified |
D02492 |
Tilmicosin (USP/INN); TMS; Micotil (TN) |
(P) unclassified |
D02493 |
Tilmicosin phosphate (USAN); TP |
(P) unclassified |
D02497 |
Fosamprenavir (INN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4 |
D02498 |
Lopinavir and ritonavir; Kaletra (TN) |
(P) unclassified |
D02501 |
Caspofungin acetate (JAN/USAN); Cancidas (TN) |
(P) unclassified |
D02523 |
Erythromycin acistrate (USAN); Erasis (TN) |
(P) unclassified |
D02524 |
Erythromycin gluceptate (USP); Erythromycin glucoheptonate; Ilotycin gluceptate (TN) |
(P) unclassified |
D02525 |
Erythromycin propionate (USAN) |
(P) unclassified |
D02540 |
Garenoxacin mesylate (USAN); Garenoxacin mesilate hydrate (JAN) |
(P) unclassified |
D02555 |
Posaconazole (JAN/USAN/INN); Noxafil (TN) |
(P) CYP inhibition: CYP3A4 |
D02556 |
Ravuconazole (prop.INN) |
(P) unclassified |
D02557 |
Chlormidazole (INN) |
(P) unclassified |
D02564 |
Pargyline hydrochloride (USAN); Eutonyl (TN) |
(P) unclassified |
D02582 |
Fenticonazole (INN) |
(P) unclassified |
D02583 |
Fenticonazole nitrate (USAN); Lomexin (TN) |
(P) unclassified |
D02584 |
Aliconazole (INN) |
(P) unclassified |
D02585 |
Vibunazole; Bay N-7133 |
(P) unclassified |
D02586 |
Alteconazole (INN) |
(P) unclassified |
D02587 |
Metildigoxin (JP18); Lanirapid (TN) |
(P) unclassified |
D02618 |
Butobarbital (BAN); Butethal; Neonal (TN) |
(P) unclassified |
D02624 |
Eszopiclone (JAN/USP/INN); Estorra (TN); Lunesta (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D02690 |
Cholestyramine resin (USP); Colestyramine (JAN/INN); Questran (TN) |
(P) unclassified |
D02691 |
Somatropin (USP/INN); Somatropin (genetical recombination) (JAN); Human growth hormone (JAN); Asellacrin (TN); Humatrope (TN); Nutropin (TN); Omnitrope (TN) |
(P) unclassified |
D02714 |
Everolimus (JAN/USAN/INN); Afinitor (TN); Votubia (TN); Zortress (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D02715 |
Balsalazide disodium (USP); Colazide (TN) |
(P) unclassified |
D02720 |
Beraprost (USAN) |
(P) unclassified |
D02721 |
Iloprost (USAN/INN); Ventavis (TN) |
(P) unclassified |
D02722 |
Limaprost (INN) |
(P) unclassified |
D02732 |
Pranlukast hydrate (JP18); Onon (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D02749 |
Teceleukin (USAN); Teceleukin (genetical recombination) (JP18); Imunace (TN) |
(P) unclassified |
D02778 |
Abciximab (USAN/INN); Abciximab (genetical recombination) (JAN); Reopro (TN) |
(P) unclassified |
D02817 |
Allobarbital (USAN/INN) |
(P) unclassified |
D02837 |
Alteplase (USP/INN); Alteplase (genetical recombination) (JAN); Activase (TN); Cathflo activase (TN) |
(P) unclassified |
D02838 |
Althiazide (USAN); Altizide (INN) |
(P) unclassified |
D02860 |
Limaprost alfadex (JP18); Opalmon (TN) |
(P) unclassified |
D02861 |
Indinavir sulfate ethanolate (JAN); Crixivan (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4 |
D02867 |
Fosamprenavir calcium hydrate (JAN); Lexiva (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4 |
D02938 |
Ancrod (USAN/INN); Viprinex (TN) |
(P) unclassified |
D02947 |
Anistreplase (USAN/INN); Eminase (TN) |
(P) unclassified |
D02968 |
Aprepitant (JAN/USP/INN); Aponvie (TN); Emend (TN); Cinvanti (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4 |
D02980 |
Adomiparin sodium (USAN); Ardeparin sodium (USAN/INN); Semuloparin sodium (USAN/INN); Normiflo (TN) |
(P) unclassified |
D02994 |
Rituximab (USAN/INN); Rituximab (genetical recombination) (JAN); Rituximab (genetical recombination) [Rituximab biosimilar 1] (JAN); Rituximab (genetical recombination) [Rituximab biosimilar 2] (JAN); Rituximab-abbs; Rituximab-pvvr; Rituximab-arrx; Rituxan (TN); Riabni (TN); Truximab (TN) |
(P) unclassified |
D03023 |
Azaconazole (USAN/INN) |
(P) unclassified |
D03063 |
BCG vaccine (USP); Freeze-dried BCG vaccine (for percutaneous use) (JP18); BCG vaccine (TN) |
(CI) unclassified |
D03098 |
Berythromycin (USAN/INN); Erythromycin B |
(P) unclassified |
D03106 |
Bexarotene (JAN/USAN/INN); Targretin (TN) |
(P) unclassified |
D03136 |
Bivalirudin (USAN/INN) |
(P) unclassified |
D03150 |
Bortezomib (JAN/USAN/INN); Velcade (TN) |
(P) unclassified |
D03157 |
Brinolase (USAN); Brinase (INN) |
(P) unclassified |
D03164 |
Bromindione (USAN/INN) |
(P) unclassified |
D03180 |
Butabarbital (USP); Secbutabarbital (BAN) |
(P) unclassified |
D03182 |
Butalbital (USP/INN); Sandoptal (TN) |
(P) unclassified |
D03189 |
Buthiazide (USAN); Butizide (INN) |
(P) unclassified |
D03213 |
Apixaban (JAN/USAN/INN); Eliquis (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D03218 |
Axitinib (JAN/USAN); Inlyta (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D03230 |
Insulin human (USP/INN); Insulin human (genetical recombination) (JP18); Insulin human (biosynthesis) (JAN); Insulin human (synthesis) (JAN); Humulin (TN) |
(P) unclassified |
D03250 |
Insulin glargine (USAN/INN); Insulin glargine (genetical recombination) (JP18); Insulin glargine (genetical recombination) [Insulin glargin biosimilar 1] (JAN); Insulin glargine (genetical recombination) [Insulin glargin biosimilar 2] (JAN); Lantus (TN) |
(P) unclassified |
D03253 |
Brecanavir (USAN) |
(P) unclassified |
D03259 |
Gemtuzumab ozogamicin (USAN); Gemtuzumab ozogamicin (genetical recombination) (JAN); Gemtuzumab (INN); Mylotarg (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D03260 |
Vardenafil hydrochloride hydrate (JAN); Vardenafil monohydrochloride trihydrate; Levitra (TN); Staxyn (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D03278 |
Enviomycin sulfate (JP18); Tuberactin (TN) |
(P) unclassified |
D03297 |
Mecasermin (USAN/INN); Mecasermin (genetical recombination) (JAN); Increlex (TN); Myotrophin (TN) |
(P) unclassified |
D03324 |
Nasaruplase (cell culture) (JAN); Prourokinase (plasminogen activator prolyse) |
(P) unclassified |
D03337 |
Reviparin sodium (JAN); Clivarine (TN) |
(P) unclassified |
D03341 |
Urokinase (JP18/USAN/INN); Abbokinase (TN) |
(P) unclassified |
D03342 |
Camiglibose (USAN) |
(P) unclassified |
D03352 |
Batroxobin (JAN/INN); Defibrase (TN) |
(P) unclassified |
D03353 |
Dalteparin sodium (JAN/USP/INN); Ardeparin sodium; Fragmin (TN) |
(P) unclassified |
D03359 |
Cangrelor (USAN/INN) |
(P) unclassified |
D03361 |
Cangrelor tetrasodium (USAN); Kengreal (TN) |
(P) unclassified |
D03363 |
Canrenone (USAN) |
(P) unclassified |
D03385 |
Carbaspirin calcium (USAN); Carbasalate calcium (INN) |
(P) unclassified |
D03471 |
Chlorothiazide sodium (USP); Diuril (TN) |
(P) unclassified |
D03493 |
Ciglitazone (USAN/INN) |
(P) unclassified |
D03505 |
Cinacalcet hydrochloride (JAN/USAN); Sensipar (TN); Mimpara (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D03526 |
Cisconazole (USAN/INN) |
(P) unclassified |
D03644 |
Danaparoid sodium (JAN/USAN); Orgaran (TN) |
(P) unclassified |
D03653 |
Darglitazone sodium (USAN) |
(P) unclassified |
D03656 |
Darunavir (USAN/INN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4 |
D03658 |
Dasatinib (JAN/INN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D03661 |
Dazmegrel (USAN/INN) |
(P) unclassified |
D03663 |
Dazoxiben hydrochloride (USAN) |
(P) unclassified |
D03664 |
Debrisoquin sulfate (USAN); Declinax (TN) |
(P) unclassified |
D03669 |
Deferasirox (JAN/USAN/INN); Exjade (TN); Jadenu (TN) |
(P) CYP induction: CYP3A4 |
D03673 |
Deligoparin sodium (USAN/INN) |
(P) unclassified |
D03674 |
Enoxaparin sodium (JAN/USP/INN); Lovenox (TN) |
(P) unclassified |
D03692 |
Desirudin (USAN/INN); Iprivask (TN) |
(P) unclassified |
D03695 |
Desmoteplase (USAN/INN) |
(P) unclassified |
D03722 |
Efegatran sulfate (USAN) |
(P) unclassified |
D03728 |
Napsagatran (USAN) |
(P) unclassified |
D03798 |
Dicumarol (USAN); Dicoumarol (INN); Dicumarol (TN) |
(P) unclassified |
D03799 |
Dienogest (JAN/USAN/INN); Endometrion (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D03833 |
Indinavir (USAN); Indinavir hydrate |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4 |
D03835 |
Fosamprenavir calcium (USAN); Lexiva (TN); Telzir (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4 |
D03837 |
Fosamprenavir sodium (USAN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4 |
D03839 |
Droxinavir hydrochloride (USAN) |
(P) unclassified |
D03840 |
Palinavir (USAN/INN) |
(P) unclassified |
D03842 |
Telinavir (USAN/INN) |
(P) unclassified |
D03843 |
Tipranavir disodium (USAN) |
(P) unclassified |
D03865 |
Dirithromycin (USP/INN); Dynabac (TN) |
(P) unclassified |
D03883 |
Doconazole (USAN/INN) |
(P) unclassified |
D03918 |
Drotrecogin alfa (activated) (USAN); Drotrecogin alfa; Xigris (TN) |
(P) unclassified |
D03936 |
Econazole (USAN/INN) |
(P) unclassified |
D03941 |
Edaglitazone sodium (USAN) |
(P) unclassified |
D03960 |
Aspirin and dialuminate; Aspirin, aluminum glycinate and magnesium carbonate; Bufferin (TN) |
(P) unclassified |
D03994 |
Endralazine mesylate (USAN); Endralazine monomethanesulfonate; Migranal (TN) |
(P) unclassified |
D03996 |
Englitazone sodium (USAN) |
(P) unclassified |
D03997 |
Enilconazole (USAN/INN) |
(P) unclassified |
D04018 |
Ephedrine sulfate (USP); Akovaz (TN); Corphedra (TN); Emerphed (TN) |
(P) unclassified |
D04023 |
Erlotinib hydrochloride (JAN/USAN); Tarceva (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D04024 |
Lapatinib ditosylate (USAN); Lapatinib tosilate hydrate (JAN); Lapatinib ditosylate monohydrate; Tykerb (TN); Tyverb (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D04029 |
Razaxaban hydrochloride (USAN) |
(P) unclassified |
D04033 |
Epithiazide (USAN); Epitizide (INN) |
(P) unclassified |
D04054 |
Erythromycin salnacedin (USAN); Erythromycin salnacedin dihydrate |
(P) unclassified |
D04070 |
Estrogens, conjugated (JAN/USP); Conjugated estrogens; Premarin (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D04077 |
Eterobarb (USAN/INN); Antilon (TN) |
(P) unclassified |
D04079 |
Ethacrynate sodium (USP) |
(P) unclassified |
D04103 |
Etoformin hydrochloride (USAN) |
(P) unclassified |
D04111 |
Etozolin (USAN/INN) |
(P) unclassified |
D04121 |
Exenatide (JAN/USAN/INN); Byetta (TN) |
(P) unclassified |
D04145 |
Fendosal (USAN/INN); Alnovin (TN) |
(P) unclassified |
D04161 |
Fenquizone (USAN/INN) |
(P) unclassified |
D04183 |
Fidexaban (USAN/INN) |
(P) unclassified |
D04206 |
Flufenisal (USAN/INN) |
(P) unclassified |
D04265 |
Reserpine, hydralazine hydrochloride and hydrochlorothiazide |
(P) unclassified |
D04266 |
Benzylhydrochlorothiazide, Reserpine and Carbazochrome; Behyd RA (TN) |
(P) unclassified |
D04276 |
Furegrelate sodium (USAN) |
(P) unclassified |
D04318 |
Glatiramer acetate (JAN/USAN); Copaxone (TN) |
(P) unclassified |
D04322 |
Gliamilide (USAN/INN) |
(P) unclassified |
D04338 |
Dihydrocodeine phosphate, ephedrine hydrochloride and ammmonium chloride; Sekicode (TN) |
(P) unclassified |
D04354 |
Glyhexamide (USAN/INN); Subose (TN) |
(P) unclassified |
D04355 |
Glyoctamide (USAN/INN) |
(P) unclassified |
D04356 |
Glyparamide (USAN) |
(P) unclassified |
D04382 |
Guanethidine monosulfate (USP); Guanethidine sulfate (JP18); Ismelin (TN) |
(P) unclassified |
D04386 |
Guanoclor sulfate (USAN); Vatensol (TN) |
(P) unclassified |
D04398 |
Guanoxabenz (USAN/INN) |
(P) unclassified |
D04399 |
Guanoxan sulfate (USAN); Envacar (TN) |
(P) unclassified |
D04403 |
Guar gum (NF) |
(P) unclassified |
D04427 |
Heparin calcium (JP18); Nadroparin calcium (INN); Calciparin; Calciparine (TN) |
(P) unclassified |
D04458 |
Hydralazine polistirex (USAN) |
(P) unclassified |
D04463 |
Norgestrel and ethinylestradiol tablets (JP18); Low-ogestrel (TN); Planovar (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D04475 |
Insulin aspart (USP/INN); Insulin aspart (genetical recombination) (JP18); Insulin aspart (genetical recombination) [Insulin aspart biosimilar 1] (JAN); Insulin X 14; NovoRapid (TN); Novolog (TN) |
(P) unclassified |
D04477 |
Insulin lispro (USP/INN); Insulin lispro (genetical recombination) (JAN); Insulin lispro (genetical recombination) [Insulin lispro Biosimilar 1] (JAN); Insulin lispro-aabc; Humalog (TN); Lyumjev (TN) |
(P) unclassified |
D04482 |
Ethinylestradiol and levonorgestrel; Ange (TN); Levora (TN); Lo/ovral (TN); Seasonique (TN); Triphasil-21 (TN); Trivora (TN) |
(P) unclassified |
D04483 |
Ethinylestradiol and norethisterone; Norethindrone and ethinyl estradiol; Synphase T28 (TN) |
(P) unclassified |
D04484 |
Desogestrel and ethinylestradiol; Marvelon21 (TN); Ortho-cept (TN) |
(P) unclassified |
D04520 |
Indacrinone (USAN/INN) |
(P) unclassified |
D04531 |
Indoramin (USAN/INN) |
(P) unclassified |
D04532 |
Indoramin hydrochloride (USAN) |
(P) unclassified |
D04539 |
Insulin detemir (USAN/INN); Insulin detemir (genetical recombination) (JAN); Levemir (TN) |
(P) unclassified |
D04540 |
Insulin glulisine (USAN/INN); Insulin glulisine (genetical recombination) (JAN); Apidra (TN) |
(P) unclassified |
D04541 |
Insulin human, isophane (USP) |
(P) unclassified |
D04542 |
Insulin human zinc (USP) |
(P) unclassified |
D04543 |
Insulin human zinc, extended (USP) |
(P) unclassified |
D04547 |
Insulin, isophane (USP); Isophane insulin human (genetical recombination) injectable aqueous suspension (JP18); Isophane insulin (aqueous suspension) (JAN); Humalog PEN (TN) |
(P) unclassified |
D04548 |
Insulin, neutral (USAN); Neutral insulin injection (INN) |
(P) unclassified |
D04550 |
Insulin zinc, prompt (USP); Semilente iletin (TN) |
(P) unclassified |
D04551 |
Insulin zinc (USP); Lente iletin (TN) |
(P) unclassified |
D04624 |
Isoconazole (USAN/INN) |
(P) unclassified |
D04641 |
Istradefylline (JAN/USAN/INN); Nourianz (TN); Nouriast (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4 |
D04665 |
Lanoteplase (USAN/INN); Lanoteplase (genetical recombination) (JAN) |
(P) unclassified |
D04666 |
Lanreotide acetate (JAN/USAN); Somatuline (TN) |
(P) unclassified |
D04725 |
Lexithromycin (USAN/INN) |
(P) unclassified |
D04752 |
Lixivaptan (USAN/INN) |
(P) unclassified |
D04768 |
Lonafarnib (JAN/USAN/INN); Zokinvy (TN) |
(P) unclassified |
D04799 |
Heparinoid (JAN); Hirudoid (TN) |
(P) unclassified |
D04820 |
Lurasidone hydrochloride (JAN/USAN); SM 13496; Latuda (TN) |
(CI,P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D04866 |
Freeze-dried live attenuated measles vaccine (JP18) |
(CI) unclassified |
D04896 |
Megalomicin potassium phosphate (USAN) |
(P) unclassified |
D04966 |
Metformin (USAN/INN) |
(P) unclassified |
D04970 |
Methacholine chloride (JAN/USP/INN); Provocholine (TN) |
(P) unclassified |
D04976 |
Methalthiazide (USAN) |
(P) unclassified |
D04977 |
Parnaparin sodium (JP18); Lowhepa (TN) |
(P) unclassified |
D04985 |
Methohexital (USP/INN) |
(P) unclassified |
D05037 |
Trimetoquinol hydrochloride hydrate (JP18); Tretoquinol hydrate; Caluyon (TN) |
(P) unclassified |
D05087 |
Moxonidine (USAN/INN); Cynt (TN) |
(P) unclassified |
D05089 |
Freeze-dried live attenuated mumps vaccine (JP18); Freeze-dried live attenuated mumps vaccine (TN) |
(CI) unclassified |
D05093 |
Muzolimine (USAN/INN) |
(P) unclassified |
D05123 |
Nasaruplase beta (USAN/INN); Prolyse (TN) |
(P) unclassified |
D05150 |
Netoglitazone (USAN/INN) |
(P) unclassified |
D05153 |
Neutramycin (USAN) |
(P) unclassified |
D05181 |
Aspirin aluminum (JP18) |
(P) unclassified |
D05248 |
Freeze-dried inactivated tissue culture ravies vaccine (JP18) |
(P) unclassified |
D05268 |
Orconazole nitrate (USAN) |
(P) unclassified |
D05277 |
Formoterol fumarate hydrate (JP18); Formoterol fumarate dihydrate; Atock (TN); Foradil (TN) |
(P) unclassified |
D05323 |
Ozolinone (USAN) |
(P) unclassified |
D05351 |
Josamycin propionate (JP18); Josamy (TN) |
(P) CYP inhibition: CYP3A4 |
D05366 |
Procaterol hydrochloride hydrate (JP18); Meptin (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D05367 |
Parconazole hydrochloride (USAN) |
(P) unclassified |
D05380 |
Pazopanib hydrochloride (JAN/USAN); Votrient (TN) |
(P) unclassified |
D05382 |
Pazufloxacin mesilate (JP18); Pazufloxacin methanesulfonate; Pasil (TN) |
(P) unclassified |
D05387 |
Pegaspargase (JAN/USAN/INN); Oncaspar (TN) |
(P) unclassified |
D05410 |
Pamiteplase (INN); Pamiteplase (genetical recombination) (JAN); Solinase (TN) |
(P) unclassified |
D05412 |
Monteplase (INN); Monteplase (genetical recombination) (JAN); Cleactor (TN) |
(P) unclassified |
D05457 |
Phenprocoumon (USAN/INN); Liquamar (TN) |
(P) unclassified |
D05462 |
Oxycodone hydrochloride hydrate (JP18) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D05482 |
Pinacidil (USAN); Pinacidil hydrate; Pindac (TN) |
(P) unclassified |
D05502 |
Pirmagrel (USAN/INN); CGS 13080 |
(P) unclassified |
D05538 |
Mozenavir (INN) |
(P) unclassified |
D05594 |
Pramlintide (USAN/INN) |
(P) unclassified |
D05595 |
Pramlintide acetate (USAN); Symlin (TN) |
(P) unclassified |
D05597 |
Prasugrel hydrochloride (JAN/USAN); Effient (TN) |
(P) unclassified |
D05622 |
Proinsulin human (USAN) |
(P) unclassified |
D05640 |
Prorenoate potassium (USAN/INN) |
(P) unclassified |
D05705 |
Rauwolfia serpentina (USP); Rauwolfia extract; Himolfia (TN) |
(P) unclassified |
D05713 |
Relomycin (USAN/INN) |
(P) unclassified |
D05717 |
Repromicin (USAN/INN) |
(P) unclassified |
D05721 |
Reteplase (USAN/INN); Retevase (TN) |
(P) unclassified |
D05727 |
Ridogrel (USAN/INN) |
(P) unclassified |
D05739 |
Rivoglitazone (USAN/INN) |
(P) unclassified |
D05757 |
Rosaramicin (USAN/INN) |
(P) unclassified |
D05758 |
Rosaramicin butyrate (USAN) |
(P) unclassified |
D05759 |
Rosaramicin propionate (USAN) |
(P) unclassified |
D05760 |
Rosaramicin sodium phosphate (USAN) |
(P) unclassified |
D05761 |
Rosaramicin stearate (USAN) |
(P) unclassified |
D05775 |
Rufinamide (JAN/USP/INN); Banzel (TN) |
(P) unclassified |
D05788 |
Salcolex (USAN); Salcolex tetrahydrate |
(P) unclassified |
D05789 |
Salethamide maleate (USAN) |
(P) unclassified |
D05791 |
Salicylate meglumine (USAN) |
(P) unclassified |
D05793 |
Salnacedin (USAN/INN) |
(P) unclassified |
D05800 |
Saperconazole (USAN/INN) |
(P) unclassified |
D05811 |
Sedecamycin (USAN/INN) |
(P) unclassified |
D05908 |
Spiramycin (JAN/USAN/INN); Rovamycin (TN) |
(P) unclassified |
D05912 |
Spiroxasone (USAN/INN) |
(P) unclassified |
D05932 |
Streptozocin (JAN/USAN/INN); Streptozotocin; Zanosar (TN) |
(P) unclassified |
D05998 |
Talosalate (USAN/INN) |
(P) unclassified |
D06068 |
Temsirolimus (JAN/USAN/INN); Torisel (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D06070 |
Tenecteplase (USAN/INN); Tnkase (TN) |
(P) unclassified |
D06106 |
Thiamylal |
(P) unclassified |
D06142 |
Tifacogin (USAN/INN) |
(P) unclassified |
D06177 |
Tolbutamide sodium, sterile; Orinase diagnostic (TN) |
(P) unclassified |
D06186 |
Tolpyrramide (USAN/INN) |
(P) unclassified |
D06199 |
Trabectedin (JAN/USAN/INN); Yondelis (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D06213 |
Treprostinil (JAN/USAN/INN); Remodulin (TN) |
(P) unclassified |
D06234 |
Trimazosin hydrochloride (USAN); Trimazosin hydrochloride monohydrate |
(P) unclassified |
D06256 |
Tuberculin (USP); Purified tuberculin; Aplisol (TN) |
(P) unclassified |
D06258 |
Tulathromycin (JAN/USAN/INN) |
(P) unclassified |
D06270 |
Urokinase alfa (USAN/INN); r-UK (TN) |
(P) unclassified |
D06272 |
Sorafenib tosylate (USAN); Sorafenib tosilate (JAN); Nexavar (TN) |
(P) unclassified |
D06341 |
Xipamide (USAN) |
(P) unclassified |
D06347 |
Yellow fever vaccine (USP); YF-Vax (TN) |
(CI) unclassified |
D06373 |
Zinoconazole hydrochloride (USAN) |
(P) unclassified |
D06390 |
Azithromycin (USP); Zmax (TN) |
(P) unclassified |
D06398 |
Tinzaparin sodium (USAN); Innohep (TN) |
(P) unclassified |
D06401 |
Indapamide hydrate; Tenaxil (TN) |
(P) unclassified |
D06402 |
Sunitinib malate (JAN/USAN); Sutent (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D06404 |
Liraglutide (USAN/INN); Liraglutide (genetical recombination) (JAN); Victoza (TN) |
(P) unclassified |
D06407 |
Vandetanib (JAN/USAN/INN); Caprelsa (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D06410 |
Thrombomodulin alfa (USAN/INN); Thrombomodulin alfa (genetical recombination) (JAN) |
(P) unclassified |
D06413 |
Nilotinib hydrochloride hydrate (JAN); Nilotinib monohydrochloride monohydrate; Tasigna (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D06414 |
Dasatinib (USAN); Dasatinib hydrate (JAN); Sprycel (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D06466 |
Freeze-dried BCG for intravesical use; Immunobladder (TN); Tice BCG (TN) |
(CI) unclassified |
D06478 |
Darunavir ethanolate (JAN); Prezista (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4 |
D06511 |
Freeze-dried smallpox vaccine prepared in cell culture (JP18) |
(CI) unclassified |
D06512 |
Freeze-dried live attenuated rubella vaccine (JP18) |
(CI) unclassified |
D06553 |
Alogliptin benzoate (JAN/USAN); Vipidia (TN); Nesina (TN) |
(P) unclassified |
D06571 |
Antithrombin III human (USP); Antithrombin III (INN); Kybernin (TN) |
(P) unclassified |
D06578 |
Denagliptin tosylate (USAN) |
(P) unclassified |
D06597 |
Fosaprepitant dimeglumine (USAN); Fosaprepitant meglumine (JAN); Proemend (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4 |
D06598 |
Gamithromycin (USAN/INN) |
(P) unclassified |
D06606 |
Ibuprofen lysine (USAN); Ibuprofen L-lysine (JAN); Solufenum; Neoprofen (TN) |
(P) unclassified |
D06630 |
Pramiconazole (USAN/INN) |
(P) unclassified |
D06641 |
Sergliflozin etabonate (USAN) |
(P) unclassified |
D06645 |
Sitagliptin phosphate (USAN); Sitagliptin phosphate hydrate (JP18); Sitagliptin phosphate monohydrate; Januvia (TN) |
(P) unclassified |
D06879 |
Streptokinase (INN); Streptase (TN) |
(P) unclassified |
D06880 |
Lepirudin (INN); Refludan (TN) |
(P) unclassified |
D06883 |
Sertaconazole (INN) |
(P) unclassified |
D06887 |
Talbutal (INN); Lotusate (TN) |
(P) unclassified |
D06888 |
Eptifibatide (INN); Integrilin (TN) |
(P) unclassified |
D07064 |
Acenocoumarol (INN); Acenocoumarin; Mini-sintrom (TN) |
(P) unclassified |
D07077 |
Ambrisentan (JAN/INN); Letairis (TN); Volibris (TN) |
(P) unclassified |
D07080 |
Vildagliptin (JAN/USAN/INN); Equa (TN); Galvus (TN) |
(P) unclassified |
D07082 |
Dabigatran etexilate mesylate (USAN); Dabigatran etexilate methanesulfonate (JAN); Dabigatran etexilate mesilate; Pradaxa (TN) |
(P) unclassified |
D07086 |
Rivaroxaban (JAN/USAN/INN); Xarelto (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D07117 |
Metahexamide (INN) |
(P) unclassified |
D07118 |
Glisoxepide (INN) |
(P) unclassified |
D07131 |
Ethyl biscoumacetate (INN) |
(P) unclassified |
D07132 |
Buprenorphine (JAN/INN); Temgesic (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D07135 |
Clorindione (INN); G-25766 |
(P) unclassified |
D07136 |
Diphenadione (INN) |
(P) unclassified |
D07137 |
Tioclomarol (INN) |
(P) unclassified |
D07138 |
Ditazole (INN) |
(P) unclassified |
D07139 |
Cloricromen (INN) |
(P) unclassified |
D07140 |
Picotamide (BAN); Plactidil (TN) |
(P) unclassified |
D07141 |
Indobufen (INN) |
(P) unclassified |
D07142 |
Triflusal (INN) |
(P) unclassified |
D07143 |
Melagatran (INN) |
(P) unclassified |
D07144 |
Dabigatran etexilate (USAN/INN); Pradaxa (TN) |
(P) unclassified |
D07166 |
Methoserpidine (INN) |
(P) unclassified |
D07167 |
Bietaserpine (prop.INN) |
(P) unclassified |
D07168 |
Tolonidine (INN) |
(P) unclassified |
D07169 |
Guanazodine (INN) |
(P) unclassified |
D07170 |
Dihydralazine (INN) |
(P) unclassified |
D07171 |
Sitaxentan (USAN/INN) |
(P) unclassified |
D07172 |
Mebutizide (INN) |
(P) unclassified |
D07192 |
Benfluorex (INN/BAN); Mediaxal (TN) |
(P) unclassified |
D07193 |
Flutrimazole (INN) |
(P) unclassified |
D07242 |
Flurithromycin (INN) |
(P) unclassified |
D07290 |
Dipyrocetyl (INN) |
(P) unclassified |
D07291 |
Benorilate (INN); Benorylate |
(P) unclassified |
D07292 |
Guacetisal (INN); Prontomucil (TN) |
(P) unclassified |
D07293 |
Imidazole salicylate (INN); Selezen (TN) |
(P) unclassified |
D07298 |
Barbexaclone (INN); Maliasin (TN) |
(P) unclassified |
D07321 |
Vinylbital (INN); Vinylbitone |
(P) unclassified |
D07322 |
Vinbarbital (INN) |
(P) unclassified |
D07323 |
Cyclobarbital (INN); Ciclobarbital (TN) |
(P) unclassified |
D07324 |
Proxibarbal (INN); Centralgol (TN) |
(P) unclassified |
D07421 |
Aloxiprin (INN); Superpyrin (TN) |
(P) unclassified |
D07422 |
Fibrinolysin (human) (INN); Fibrinolysin, human; Fibrogammin (TN) |
(P) unclassified |
D07447 |
Amiloride (INN); Amiclaran (TN) |
(P) unclassified |
D07457 |
Anisindione (INN); Miradon (TN) |
(P) unclassified |
D07471 |
Atazanavir (INN); Reyataz (TN) |
(P) CYP inhibition: CYP3A4 |
D07486 |
Azithromycin (INN); Azasite (TN); Azithromycin (TN) |
(P) unclassified |
D07488 |
Balsalazide (INN) |
(P) unclassified |
D07508 |
Benfluorex hydrochloride; Mediator (TN) |
(P) unclassified |
D07510 |
Adomiparin (USAN); Semuloparin (USAN); Heparin (BAN); Enoxaparin; Bemiparin; Parnaparin; Nadroparin; Heparin (TN) |
(P) unclassified |
D07538 |
Bosentan (INN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D07569 |
Candesartan cilexetil and anmlodipine besylate (JP18); Unisia (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D07579 |
Aspirin calcium salt; Notras (TN) |
(P) unclassified |
D07580 |
Aspirin DL-lysine (JAN); Aspirin lysine salt; Aspegic (TN) |
(P) unclassified |
D07581 |
Aspirin magnesium salt; Mobidin (TN) |
(P) unclassified |
D07582 |
Aspirin sodium; Sodium acetylsalicylate; Catalgine (TN) |
(P) unclassified |
D07583 |
Phenytoin and phenobarbital; Aleviatin with phenobarbital (TN) |
(P) unclassified |
D07595 |
Fosphenytoin sodium hydrate (JAN); Fostoin (TN) |
(P) CYP induction: CYP3A4 |
D07598 |
Butoconazole (INN); Gynofort (TN) |
(P) unclassified |
D07603 |
Caffeine citrate (USP); Cafcit (TN) |
(P) unclassified |
D07612 |
Sodium salamidacetate; o-Carbamoylphenoxyacetic acid sodium salt; Clinit-n (TN) |
(P) unclassified |
D07676 |
Chlormidazole hydrochloride; Unfungicid (TN) |
(P) unclassified |
D07710 |
Clarithromycin lactobionate; Klacid (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4 |
D07729 |
Clopidogrel (USP/INN); Clopidogrel (TN); Plavix (TN) |
(P) unclassified |
D07736 |
Cloricromen hydrohloride; Proendotel (TN) |
(P) unclassified |
D07748 |
Conivaptan (INN) |
(P) unclassified |
D07752 |
Croconazole (INN) |
(P) unclassified |
D07757 |
Cyclobarbital calcium (BAN); Phanodorn calcium (TN) |
(P) unclassified |
D07824 |
Diethylamine salicylate; Algesal (TN) |
(P) unclassified |
D07830 |
Dihydralazine sulfate; Dihydralazine hydrogen sulfate; Nepresol (TN) |
(P) unclassified |
D07869 |
Donepezil (JAN/INN); Donaz (TN); Allydone (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D07874 |
Doxazosin (INN); Cardura XL (TN) |
(P) unclassified |
D07882 |
Eberconazole (INN) |
(P) unclassified |
D07884 |
Eberconazole nitrate; Ebernet (TN) |
(P) unclassified |
D07895 |
Losartan potassium and hydrochlorothiazide (JP18); Hydrochlorothiazide and losartan potassium; Hyzaar (TN); Losarhyd (TN) |
(P) unclassified |
D07909 |
Erythromycin thiocyanate; Erythrocin (TN) |
(P) unclassified |
D07910 |
Erythromycin stinoprate (INN); Erysec (TN) |
(P) unclassified |
D07955 |
Fenquizone potassium salt; Idrolone (TN) |
(P) unclassified |
D07969 |
Fluindione (INN); Previsccan (TN) |
(P) unclassified |
D07991 |
Fosfosal (INN); Aydolid (TN) |
(P) unclassified |
D07999 |
Sodium furosemide; Frosemide sodium; Lasix (TN) |
(P) unclassified |
D08001 |
Furosemide diolamine; Furosemide diethanolamine salt; Nuriban (TN) |
(P) unclassified |
D08004 |
Gabexate (INN) |
(P) unclassified |
D08030 |
Guanethidine (INN) |
(P) unclassified |
D08031 |
Guanfacine (INN); Estulic (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D08044 |
Hydralazine (INN); Hidral (TN) |
(P) unclassified |
D08065 |
Iloprost tromethamine; Iloprost trometamol; Ventavis (TN) |
(P) unclassified |
D08080 |
Insulin injection, biphasic isophane (BAN); Biphasic isophane insuline human (genetical recombination) injectable aqueous suspension (JP18); Insulin Humacart (TN) |
(P) unclassified |
D08095 |
Ivabradine hydrochloride (JAN/USAN); Ivabrandine hydrochloride; Corlanor (TN); Corlentor (TN); Coralan (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D08099 |
Ketanserin tartrate; Sufrexal (TN) |
(P) unclassified |
D08194 |
Deserpidine (INN); Halmonyl (TN) |
(P) unclassified |
D08205 |
Methyldopa (INN); Aldomet (TN) |
(P) unclassified |
D08212 |
Trimazosin (INN) |
(P) unclassified |
D08240 |
Nafamostat (INN) |
(P) unclassified |
D08254 |
Endralazine (INN) |
(P) unclassified |
D08256 |
Nateplase (INN); Milyzer (TN); Tepase (TN) |
(P) unclassified |
D08259 |
Nelfinavir (INN); Viracept (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4 |
D08295 |
Olsalazine (INN) |
(P) unclassified |
D08296 |
Omoconazole (INN) |
(P) unclassified |
D08313 |
Oxiconazole (INN) |
(P) unclassified |
D08327 |
Ozagrel (INN); Cataclot (TN) |
(P) unclassified |
D08351 |
Phenformin (BAN) |
(P) unclassified |
D08352 |
Phenformin hydrochloride; Debei (TN) |
(P) unclassified |
D08354 |
Phenindione (INN); Hedulin (TN) |
(P) unclassified |
D08356 |
Phenobarbital diethylamine; Gratusminal (TN) |
(P) unclassified |
D08378 |
Pioglitazone (INN); Actos (TN) |
(P) unclassified |
D08411 |
Prazosin (INN); Minipress (TN) |
(P) unclassified |
D08453 |
Pargyline (INN) |
(P) unclassified |
D08479 |
Rifampicin sodium; Rifadine (TN) |
(P) CYP induction: CYP3A4 |
D08482 |
Rilmenidine (INN); Hyperium (TN) |
(P) unclassified |
D08488 |
Amlodipine besilate and atorvastatin calcium; Caduet (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D08491 |
Rosiglitazone (INN); Gaudil (TN) |
(P) unclassified |
D08501 |
Trolamine salicylate (USP); Salicylic acid trolamine; Salicylic acid triethanolamine; Arthricream (TN) |
(P) unclassified |
D08508 |
Sarpogrelate (INN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D08510 |
Sertaconazole nitrate; Ertaczo (TN); Zalain (TN) |
(P) unclassified |
D08516 |
Sitagliptin (USAN/INN) |
(P) unclassified |
D08517 |
Sitaxentan sodium (USAN); Thelin (TN) |
(P) unclassified |
D08527 |
Spiramycin adipate; Rovamycina (TN); Spiramaicina (TN) |
(P) unclassified |
D08528 |
Spiramycin embonate; Cofamix STS (TN) |
(P) unclassified |
D08535 |
Sulconazole (INN) |
(P) unclassified |
D08536 |
Suleparoid; Heparitin sulfate; Aremin (TN) |
(P) unclassified |
D08547 |
Sulodexide (INN); Vessel (TN) |
(P) unclassified |
D08586 |
Thiosalicylic acid; Pirosal (TN); Thiocyl (TN) |
(P) unclassified |
D08594 |
Ticlopidine (INN); Ticlopidin-Puren (TN) |
(P) unclassified |
D08605 |
Tipranavir (INN); Aptivus (TN) |
(P) unclassified |
D08607 |
Tirofiban (INN); Agrastat (TN) |
(P) unclassified |
D08609 |
Tisokinase (JAN) |
(P) unclassified |
D08616 |
Teneligliptin (INN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4 |
D08619 |
Torasemide sodium; Torem (TN) |
(P) unclassified |
D08628 |
Treprostinil monosodium salt; Treprostinil sodium; Trepulmix (TN) |
(P) unclassified |
D08631 |
Carmegliptin (USAN/INN) |
(P) unclassified |
D08662 |
Urapidil hydrochloride; Ebrantil (TN) |
(P) unclassified |
D08682 |
Warfarin (INN); Warfarine; Choice (TN) |
(P) unclassified |
D08699 |
Salmeterol xinafoate and fluticasone propionate; Adoair diskus (TN); Aerivio Spiromax (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D08777 |
Freeze-dried live attenuated varicella vaccine |
(CI) unclassified |
D08795 |
Human antithrombin III, freeze-dried concentrated; Neuart (TN) |
(P) unclassified |
D08804 |
Freeze-dried live attenuated measles-rubella combined vaccine; Mearubik (TN) |
(CI) unclassified |
D08843 |
Albiglutide (USAN); Albiglutide (genetical recombination) (JAN); Tanzeum (TN) |
(P) unclassified |
D08856 |
Anamorelin hydrochloride (JAN/USAN); Adlumiz (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D08858 |
Antithrombin alfa (INN/USAN); Atryn (TN) |
(P) unclassified |
D08860 |
Apremilast (JAN/USAN); Otezla (TN) |
(P) unclassified |
D08873 |
Betrixaban (USAN); Bevyxxa (TN) |
(P) unclassified |
D08897 |
Dapagliflozin (JAN/USAN/INN); Forxiga (TN) |
(P) unclassified |
D08913 |
Eribaxaban (USAN) |
(P) unclassified |
D08923 |
Fesoterodine fumarate (JAN/USAN); Toviaz (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D08962 |
Pamabrom (USP) |
(P) unclassified |
D08996 |
Saxagliptin (USAN/INN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D09013 |
Teplizumab (USAN/INN); Teplizumab-mzwv; Tzield (TN) |
(P) unclassified |
D09017 |
Ticagrelor (JAN/USAN/INN); Brilinta (TN) |
(CI,P) unclassified |
D09196 |
Candesartan cilexetil and hydrochlorothiazide (JP18); Ecard HD (TN); Ecard LD (TN) |
(P) unclassified |
D09197 |
Valsartan and hydrochlorothiazide (JP18); Co-dio (TN) |
(P) unclassified |
D09206 |
Saruplase (INN); Prourokinase (enzyme activating) (human clone pUK4/pUK18), nonglycosylated |
(P) unclassified |
D09219 |
Telmisartan and hydrochlorothiazide (JP18); Micombi (TN); Micardis hct (TN) |
(P) unclassified |
D09319 |
Indacaterol maleate (JAN/USAN); Arcapta neohaler (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D09326 |
Carmegliptin dihydrochloride (USAN) |
(P) unclassified |
D09333 |
Dutogliptin (USAN) |
(P) unclassified |
D09334 |
Dutogliptin tartrate (USAN) |
(P) unclassified |
D09348 |
Fostamatinib disodium (USAN); Fostamatinib sodium hydrate (JAN); Fostamatinib disodium hexahydrate; Tavalisse (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D09394 |
Fidaxomicin (JAN/USAN); Dificid (TN); Dificlir (TN) |
(P) CYP inhibition: CYP3A4 |
D09546 |
Edoxaban tosilate hydrate (JAN); Edoxaban tosylate monohydrate; Lixiana (TN); Savaysa (TN) |
(P) unclassified |
D09566 |
Linagliptin (JAN/USAN/INN); Tradjenta (TN) |
(P) unclassified |
D09572 |
Riociguat (JAN/USAN/INN); Adempas (TN) |
(P) unclassified |
D09592 |
Canagliflozin (USAN/INN); Canagliflozin hydrate (JAN); Invokana (TN) |
(P) unclassified |
D09595 |
Budesonide and formoterol fumarate dihydrate; Symbicort (TN); Budeforu (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D09605 |
Duvoglustat (USAN/INN); 1-Deoxynojirimycin |
(P) unclassified |
D09606 |
Duvoglustat hydrochloride (USAN) |
(P) unclassified |
D09625 |
Gosogliptin (USAN/INN) |
(P) unclassified |
D09638 |
Lomitapide mesylate (USAN); Lomitapide mesilate (JAN); Juxtapid (TN); Lojuxta (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D09642 |
Modithromycin (USAN/INN) |
(P) unclassified |
D09676 |
Tecarfarin (USAN/INN) |
(P) unclassified |
D09677 |
Tecarfarin sodium (USAN) |
(P) unclassified |
D09701 |
Abiraterone acetate (JAN/USP); Zytiga (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D09702 |
Albaconazole (USAN/INN) |
(P) unclassified |
D09707 |
Dabigatran (USAN/INN) |
(P) unclassified |
D09710 |
Edoxaban (USAN/INN) |
(P) unclassified |
D09720 |
Rilpivirine (JAN/USAN/INN); Rekambys (TN) |
(CI) unclassified |
D09723 |
Taspoglutide (USAN/INN) |
(P) unclassified |
D09727 |
Insulin degludec (USAN/INN); Insulin degludec (genetical recombination) (JAN); Tresiba (TN) |
(P) unclassified |
D09728 |
Bosutinib hydrate (JAN); Bosutinib monohydrate; Bosulif (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D09729 |
Lixisenatide (JAN/USAN/INN); Adlyxin (TN); Lyxumia (TN) |
(P) unclassified |
D09730 |
Olaparib (JAN/USAN/INN); Lynparza (TN) |
(P) unclassified |
D09731 |
Crizotinib (JAN/USAN/INN); Xalkori (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D09736 |
Iron (III) hexacyanoferrate (II); Radiogardase (TN) |
(P) unclassified |
D09741 |
Drospirenone and ethinylestradiol; Drospirenone and ethinylestradiol betadex; Angeliq (TN); Yaz (TN); Flexyess (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D09743 |
Telmisartan and amlodipine besilate (JP18); Telmisartan and amlodipine besylate; Micamlo (TN); Twynsta (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D09744 |
Pioglitazone hydrochloride and metformin hydrochloride (JP18); Pioglitazone and metformin; Metact (TN) |
(P) unclassified |
D09745 |
Valsartan and amlodipine besilate; Exforge (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D09753 |
Saxagliptin hydrate (JAN); Onglyza (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D09756 |
Teneligliptin hydrobromide hydrate (JAN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4 |
D09763 |
Dapagliflozin propanediol (USAN); Dapagliflozin propylene glycolate hydrate (JAN); Dapagliflozin propandiol monohydrate; Forxiga (TN); Farxiga (TN) |
(P) unclassified |
D09765 |
Vorapaxar (USAN/INN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D09766 |
Vorapaxar sulfate (JAN/USAN); Zontivity (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D09772 |
Alilusem potassium (JAN); M17055 |
(P) unclassified |
D09779 |
Emiglitate (JAN/INN) |
(P) unclassified |
D09780 |
Anagliptin (JAN/INN) |
(P) unclassified |
D09783 |
Tofacitinib citrate (JAN/USAN); Tasocitinib citrate; Xeljanz (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D09799 |
Carotegrast methyl (JAN); Carogra (TN) |
(P) CYP inhibition: CYP3A4 |
D09807 |
Difethiarol (JAN); Difethialone |
(P) unclassified |
D09809 |
Tylosin acetate isovalerte (JAN) |
(P) unclassified |
D09814 |
Silteplase (INN); Silteplase (genetical recombination) (JAN) |
(P) unclassified |
D09817 |
Darexaban maleate (JAN); YM150 |
(P) unclassified |
D09823 |
Duteplase (INN); Duteplase (genetical recombination) (JAN) |
(P) unclassified |
D09848 |
Pioglitazone hydrochloride and glimepiride tablets (JP18); Pioglitazone and glimepiride; Duetact; Sonias (TN) |
(P) unclassified |
D09873 |
Bedaquiline fumarate (JAN/USAN); Sirturo (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D09889 |
Dulaglutide (USAN/INN); Dulaglutide (genetical recombination) (JAN); Trulicity (TN) |
(P) unclassified |
D09894 |
Eliglustat tartrate (JAN/USAN); Eliglustat hemitartrate; Cerdelga (TN) |
(P) unclassified |
D09920 |
Lenvatinib mesylate (USAN); Lenvatinib mesilate (JAN); Lenvima (TN) |
(P) unclassified |
D09923 |
Letaxaban (USAN/INN) |
(P) unclassified |
D09951 |
Ponatinib hydrochloride (JAN/USAN); Iclusig (TN) |
(P) unclassified |
D09956 |
Quizartinib dihydrochloride (USAN); Quizartinib hydrochloride (JAN); Vanflyta (TN) |
(P) unclassified |
D09958 |
Rilpivirine hydrochloride (JAN/USAN); Edurant (TN) |
(CI) unclassified |
D09960 |
Ruxolitinib phosphate (JAN/USAN); Jakafi (TN); Jakavi (TN); Opzelura (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D09978 |
Tofogliflozin (USAN); Tofogliflozin hydrate (JAN); Apleway (TN); Deberza (TN) |
(P) unclassified |
D09994 |
Selexipag (JAN/USAN/INN); Uptravi (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D09996 |
Vemurafenib (JAN/USAN/INN); Zelboraf (TN) |
(P) CYP induction: CYP3A4 |
D10003 |
Hemin (JAN); Normosang (TN); Panhematin (TN) |
(P) CYP induction: CYP3A4 |
D10021 |
Efinaconazole (JAN/USAN/INN); Clenafin (TN); Jublia (TN) |
(P) unclassified |
D10024 |
Selumetinib sulfate (JAN/USAN); Koselugo (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D10025 |
Semaglutide (USAN/INN); Semaglutide (genetical recombination) (JAN); Ozempic (TN) |
(P) unclassified |
D10032 |
Tylvalosin (USAN/INN) |
(P) unclassified |
D10033 |
Tylosin tartrate (USP) |
(P) unclassified |
D10034 |
Tylvalosin tartrate (USAN); Aiviosin [veterinary] (TN) |
(P) unclassified |
D10055 |
Remogliflozin etabonate (USAN/INN) |
(P) unclassified |
D10082 |
Suvorexant (JAN/USAN); MK-4305; Belsomra (TN) |
(P) unclassified |
D10093 |
Asunaprevir (JAN/USAN); Sunvepra (TN) |
(CI) CYP induction: CYP3A4 |
D10095 |
Cabozantinib s-malate (USAN); Cabozantinib malate (JAN); Cometriq (TN); Cabometyx (TN) |
(P) unclassified |
D10104 |
Dabrafenib mesylate (USAN); Dabrafenib mesilate (JAN); Tafinlar (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D10105 |
Daclatasvir dihydrochloride (USAN); Daclatasvir hydrochloride (JAN); Daklinza (TN) |
(CI) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D10131 |
Ixazomib citrate (JAN/USAN); Ninlaro (TN) |
(P) unclassified |
D10135 |
Macitentan (JAN/USAN); Opsumit (TN) |
(CI,P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D10137 |
Regorafenib hydrate (JAN); Stivarga (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D10159 |
Alogliptin benzoate and pioglitazone hydrochloride; Liovel (TN); Oseni (TN); Incresync (TN) |
(P) unclassified |
D10160 |
Mitiglinide calcium hydrate and voglibose; Glubes (TN) |
(P) unclassified |
D10161 |
Sarilumab (USAN); Sarilumab (genetical receombination) (JAN); Kevzara (TN) |
(P) unclassified |
D10178 |
Trelagliptin (USAN) |
(P) unclassified |
D10179 |
Trelagliptin succinate (JAN/USAN); Zafatek (TN) |
(P) unclassified |
D10185 |
Vortioxetine hydrobromide (JAN/USAN); Brintellix (TN); Trintellix (TN) |
(P) unclassified |
D10192 |
Recombinant adsorbed quadrivalent human papillomavirus virus-like particle vaccine (yeast origin); Gardasil (TN); Silgard (TN) |
(P) unclassified |
D10195 |
Luseogliflozin hydrate (JAN); Lusefi (TN) |
(P) unclassified |
D10196 |
Ipragliflozin (INN) |
(P) unclassified |
D10200 |
Ipragliflozin L-proline (JAN); Suglat (TN) |
(P) unclassified |
D10218 |
Enzalutamide (JAN/USAN); Xtandi (TN) |
(P) unclassified |
D10223 |
Ibrutinib (JAN/USAN); Imbruvica (TN) |
(P) unclassified |
D10243 |
Irbesartan and amlodipine besilate (JP18); Aimix (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D10244 |
Metformin hydrochloride and rosiglitazone maleate; Avandamet (TN) |
(P) unclassified |
D10251 |
Glimepiride and rosiglitazone maleate; Avandaryl (TN) |
(P) unclassified |
D10253 |
Alogliptin benzoate and metformin hydrochloride; Kazano (TN); Vipdomet (TN) |
(P) unclassified |
D10258 |
Simvastatin and sitagliptin phosphate; Juvisync (TN) |
(P) unclassified |
D10261 |
Metformin hydrochloride and sitagliptin phosphate; Janumet (TN) |
(P) unclassified |
D10262 |
Saxagliptin hydrochloride; Onglyza (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D10263 |
Metformin hydrochloride and saxagliptin hydrochloride; Kombiglyze (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D10264 |
Linagliptin and metformin hydrochloride; Jentaduet (TN) |
(P) unclassified |
D10265 |
Glipizide and metformin hydrochloride; Metaglip (TN) |
(P) unclassified |
D10266 |
Glyburide and metformin hydrochloride; Glibenclamide and metformin hydrochloride; Glucovance (TN) |
(P) unclassified |
D10267 |
Methyldopa and hydrochlorothiazide; Methyldopa and hydrochlorothiazide (TN) |
(P) unclassified |
D10309 |
Brexpiprazole (JAN/USAN/INN); Rexulti (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D10313 |
Ertugliflozin (USAN/INN) |
(P) unclassified |
D10317 |
Omarigliptin (JAN/USAN/INN) |
(P) unclassified |
D10372 |
Palbociclib (JAN/USAN); Ibrance (TN) |
(P) unclassified |
D10430 |
Treprostinil diolamine (USAN); Orenitram (TN) |
(P) unclassified |
D10450 |
Alectinib hydrochloride (JAN); Alecensa (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D10452 |
Cabazitaxel acetonate (JAN); Cabazitaxel acetone; Jevtana (TN) |
(P) unclassified |
D10459 |
Empagliflozin (JAN/USAN/INN); Jardiance (TN) |
(P) unclassified |
D10466 |
Vonoprazan fumarate (JAN/USAN); Takecab (TN); Voquezna (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D10471 |
Idraparinux sodium (USAN) |
(P) unclassified |
D10473 |
Insulin peglispro (USAN/INN) |
(P) unclassified |
D10478 |
Naldemedine tosylate (JAN/USAN); Naldemedine tosilate; Symproic (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D10480 |
Irbesartan and trichlormethiazide; Irtra (TN) |
(P) unclassified |
D10492 |
Tildipirosin (USAN/INN); Zuprevo [veterinary] (TN) |
(P) unclassified |
D10500 |
Metformin hydrochloride and repaglinide; Prandimet (TN) |
(P) unclassified |
D10502 |
Gemigliptin (INN) |
(P) unclassified |
D10505 |
Glycopyrronium bromide and indacaterol maleate; Ultibro (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D10506 |
Fluticasone propionate and formoterol fumarate hydrate; Flutiform (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D10513 |
Clopidogrel sulfate and aspirin; Clopidogrel and acetylsalicyclic acid; Complavin (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D10516 |
Aripiprazole hydrate (JAN); Aripiprazole monohydrate; Abilify maintena (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D10524 |
Azilsartan and amlodipine besilate; Zacras (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D10527 |
Acetylsalicylic acid and lansoprazole; Acetylsalicylic acid and lansoprazole; Takelda (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D10551 |
Ceritinib (JAN/USAN/INN); Zykadia (TN) |
(P) unclassified |
D10564 |
Amenamevir (JAN/INN); Amenalief (TN) |
(P) unclassified |
D10566 |
Pasireotide pamoate (JAN); Signifor lar (TN) |
(P) unclassified |
D10570 |
Insulin degludec (genetical recombination) and insulin aspart (genetical recombination); Ryzodeg (TN) |
(P) unclassified |
D10586 |
Dapagliflozin and metformin; Xigduo xr (TN) |
(P) unclassified |
D10587 |
Canagliflozin and metformin; Invokamet (TN) |
(P) unclassified |
D10588 |
Empagliflozin and linagliptin; Glyxambi (TN) |
(P) unclassified |
D10591 |
Clonidine and chlorthalidone; Clorpres (TN) |
(P) unclassified |
D10633 |
Finerenone (JAN/USAN/INN); Kerendia (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D10643 |
Isavuconazonium sulfate (JAN/USAN); Cresemba (TN) |
(P) unclassified |
D10669 |
Sotagliflozin (USAN/INN); Inpefa (TN) |
(P) unclassified |
D10677 |
Etelcalcetide hydrochloride (JAN/USAN); Velcalcetide hydrochloride (USAN); Parsabiv (TN) |
(P) unclassified |
D10679 |
Venetoclax (JAN/USAN/INN); Venclexta (TN) |
(P) unclassified |
D10684 |
Antithrombin gamma (INN); Antithrombin gamma (genetical recombination) (JAN); Acoalan (TN) |
(P) unclassified |
D10688 |
Abemaciclib (JAN/USAN/INN); Verzenio (TN) |
(P) unclassified |
D10711 |
Pemafibrate (JAN); Parmodia (TN) |
(P) unclassified |
D10743 |
Vildagliptin and metformin hydrochloride |
(P) unclassified |
D10744 |
Tiotropium and olodaterol; Spiolto (TN); Stiolto respimat (TN) |
(P) unclassified |
D10746 |
Esflurbiprofen and mentha oil; Loqoa (TN) |
(P) unclassified |
D10750 |
Isavuconazole (INN); Cresemba (TN) |
(P) unclassified |
D10752 |
Empagliflozin and metformin; Synjardy (TN) |
(P) unclassified |
D10755 |
Elvitegravir, cobicistat, emtricitabine and tenofovir alafenamide; Genvoya (TN) |
(P) unclassified |
D10762 |
Fosravuconazole L-lysine ethanolate (JAN) |
(P) unclassified |
D10766 |
Osimertinib mesylate (USAN); Osimertinib mesilate (JAN); Tagrisso (TN) |
(P) unclassified |
D10772 |
Lascufloxacin hydrochloride (JAN); Lasvic (TN) |
(P) unclassified |
D10774 |
Vonoprazan, amoxicillin and metronidazole; Vonopion (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D10775 |
Vonoprazan, amoxicillin and clarithromycin; Vonosap (TN); Voquenza (TN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4 |
D10780 |
Perampanel hydrate (JAN); Fycompa (TN) |
(P) unclassified |
D10793 |
Sodium picosulfate hydrate, magnesium oxide and citric acid, anhydrous; Picoprep (TN); Prepopik (TN); Clenpiq (TN) |
(P) unclassified |
D10800 |
Gilteritinib fumarate (JAN/USAN); Xospata (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D10801 |
Letermovir (JAN/USAN/INN); Prevymis (TN) |
(P) unclassified |
D10805 |
Telmisartan, amlodipine and hydrochlorothiazide; Micatrio (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D10823 |
Clopidogrel hydrochloride; Clopidogrel (TN) |
(P) unclassified |
D10824 |
Clopidogrel besilate; Clopidogrel besylate; Clopidogrel (TN) |
(P) unclassified |
D10826 |
Saxagliptin and dapagliflozin; Qtern (TN) |
(P) unclassified |
D10832 |
Darunavir and cobicistat; Prezcobix (TN); Rezolsta (TN) |
(P) unclassified |
D10836 |
Emtricitabine, rilpivirine and tenofovir alafenamide; Odefsey (TN) |
(CI) unclassified |
D10865 |
Bexagliflozin (USAN); Brenzavvy (TN) |
(P) unclassified |
D10866 |
Brigatinib (JAN/USAN); Alunbrig (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D10891 |
Capmatinib hydrochloride (USAN); Capmatinib hydrochloride hydrate (JAN); Tabrecta (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D10892 |
Esaxerenone (JAN/INN) |
(P) unclassified |
D10893 |
Acalabrutinib (JAN/USAN/INN); Calquence (TN) |
(P) unclassified |
D10897 |
Teneligliptin and canagliflozin; Teneligliptin and canagliflozin; Canalia (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D10926 |
Entrectinib (JAN/USAN/INN); Rozlytrek (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D10970 |
Pegapamodutide (USAN/INN) |
(P) unclassified |
D10990 |
Somatrogon (USAN/INN); Somatrogon (genetical recombination) (JAN); Somatrogon-ghla; Ngenla (TN) |
(P) unclassified |
D10999 |
Valbenazine tosylate (USAN); Valbenazine tosilate (JAN); Valbenazine ditosylate; Ingrezza (TN); Dysval (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D11012 |
Lorlatinib (JAN/USAN/INN); Lorbrena (TN) |
(P) unclassified |
D11022 |
Lemborexant (JAN/USAN/INN); Dayvigo (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D11023 |
Evogliptin (INN) |
(P) unclassified |
D11029 |
Andexanet alfa (USAN/INN); Andexanet alfa (genetical recombination) (JAN); Andexxa (TN); Ondexxya (TN) |
(P) unclassified |
D11034 |
Insulin glargine and lixisenatide; Insulin glargine (genetical recombination) and lixisenatide; Soliqua (TN) |
(P) unclassified |
D11036 |
Glycopyrrolate and formoterol; Bevespi (TN) |
(P) unclassified |
D11040 |
Apalutamide (JAN/INN); Erleada (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D11043 |
Ertugliflozin pidolate; Ertugliflozin L-pyroglutamic acid; Steglatro (TN) |
(P) unclassified |
D11045 |
Darolutamide (JAN/USAN/INN); Nebeqa (TN) |
(P) unclassified |
D11048 |
Upadacitinib hydrate (JAN); Upadacitinib hemihydrate; Rinvoq (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D11063 |
Evocalcet (JAN/INN); Orkedia (TN) |
(P) unclassified |
D11064 |
Sitagliptin and ipragliflozin; Sujanu (TN) |
(P) unclassified |
D11066 |
Ertugliflozin and sitagliptin; Steglujan (TN) |
(P) unclassified |
D11067 |
Ertugliflozin and metformin; Segluromet (TN) |
(P) unclassified |
D11070 |
Tirabrutinib hydrochloride (JAN/USAN); Velexbru (TN) |
(P) unclassified |
D11072 |
Siponimod fumarate (USAN); Siponimod fumaric acid (JAN); Mayzent (TN) |
(P) unclassified |
D11093 |
Avacopan (JAN/USAN/INN); Tavneos (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D11109 |
Anagliptin and Metformin hydrochloride |
(P) unclassified |
D11138 |
Larotrectinib sulfate (JAN/USAN); Vitrakvi (TN) |
(P) unclassified |
D11160 |
Caplacizumab (USAN/INN); Caplacizumab (genetical recombination) (JAN); Caplacizumab-yhdp; Cablivi (TN) |
(P) unclassified |
D11194 |
Somapacitan (USAN/INN); Somapacitan (genetical recombination) (JAN); Somapacitan-beco; Sogroya (TN) |
(P) unclassified |
D11280 |
Bivalirudin trifluoroacetate (USAN); Angiomax (TN) |
(P) unclassified |
D11282 |
Dolutegravir sodium and rilpivirine hydrochloride; Juluca (TN) |
(CI) unclassified |
D11342 |
Dorzagliatin (USAN) |
(P) unclassified |
D11360 |
Tirzepatide (JAN/USAN); Mounjaro (TN) |
(P) unclassified |
D11370 |
Fosnetupitant chloride hydrochloride (JAN/USAN); Arokaris (TN) |
(P) unclassified |
D11371 |
Capivasertib (JAN/USAN); Truqap (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D11382 |
Darunavir, cobicistat, emtricitabine and tenofovir alafenamide; Symtuza (TN) |
(P) unclassified |
D11417 |
Pemigatinib (JAN/USAN/INN); Pemazyre (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D11441 |
Aprocitentan (USAN/INN); Tryvio (TN) |
(P) unclassified |
D11485 |
Tazemetostat hydrobromide (JAN/USAN); Tazverik (TN) |
(P) unclassified |
D11564 |
Upacicalcet sodium hydrate (JAN); Upasita (TN) |
(P) unclassified |
D11567 |
Insulin degludec and liraglutide; Xultophy (TN) |
(P) unclassified |
D11568 |
Edoxaban tosylate (USAN) |
(P) unclassified |
D11584 |
Budesonide, glycopyrronium bromide and formoterol fumarate; Budesonide, glycopyrrolate and formoterol fumarate; Breztri (TN) |
(P) unclassified |
D11603 |
Leriglitazone (USAN/INN); 1-Hydroxypioglitazone |
(P) unclassified |
D11604 |
Leriglitazone hydrochloride (USAN) |
(P) unclassified |
D11659 |
Tolvaptan sodium phosphate (JAN); Samtasu (TN) |
(P) unclassified |
D11662 |
Valemetostat tosilate (JAN); Valemetostat tosylate; Ezharmia (TN) |
(P) unclassified |
D11674 |
Berotralstat hydrochloride (JAN/USAN); Orladeyo (TN) |
(P) CYP inhibition: CYP3A4 |
D11711 |
Dapagliflozin, metformin and saxagliptin; Qternmet xr (TN) |
(P) unclassified |
D11713 |
Selpercatinib (JAN/USAN/INN); Retevmo (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D11725 |
Futibatinib (JAN/USAN/INN); Lytgobi (TN) |
(P) unclassified |
D11757 |
Inebilizumab (USAN/INN); Inebilizumab (genetical recombination) (JAN); Inebilizumab-cdon; Uplizna (TN) |
(P) unclassified |
D11785 |
Oteseconazole (USAN/INN); Vivijoa (TN) |
(P) unclassified |
D11804 |
Aspirin and vonoprazan; Cabpirin (TN) |
(P) unclassified |
D11807 |
Imeglimin hydrochloride (JAN); Twymeeg (TN) |
(P) unclassified |
D11816 |
Belumosudil mesylate (USAN); Belumosudil mesilate (JAN); Rezurock (TN) |
(P) unclassified |
D11856 |
Empagliflozin, linagliptin and metformin hydrochloride; Trijardy xr (TN) |
(P) unclassified |
D11861 |
Indacaterol acetate, glycopyrronium bromide and mometasone furoate; Enerzair (TN) |
(P) unclassified |
D11862 |
Indacaterol and mometasone furoate; Atectura (TN) |
(P) unclassified |
D11863 |
Human papillomavirus 9-valent vaccine, recombinant; Recombinant adsorbed 9-valent human papillomavirus virus-like particle vaccine (yeast origin); Gardasil 9 (TN); Silgard 9 (TN) |
(P) unclassified |
D11910 |
Danuglipron (USAN) |
(P) unclassified |
D11911 |
Danuglipron tromethamine (USAN) |
(P) unclassified |
D11920 |
Pimitespib (JAN); Jeselhy (TN) |
(P) unclassified |
D11923 |
Lobeglitazone (INN) |
(P) unclassified |
D11924 |
Beinaglutide (INN) |
(P) unclassified |
D11968 |
Teneligliptin hydrobromide (JAN) |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4 |
D11970 |
Ritlecitinib tosylate (USAN); Ritlecitinib tosilate (JAN); Litfulo (TN) |
(P) unclassified |
D12005 |
Treprostinil palmitil (USAN/INN) |
(P) unclassified |
D12055 |
Sotorasib (JAN/USAN); Lumakras (TN) |
(P) unclassified |
D12162 |
Lenacapavir sodium (JAN/USAN); Sunlenca (TN) |
(P) unclassified |
D12205 |
Pneumococcal 15-valent conjugate vaccine; Vaxneuvance (TN) |
(P) unclassified |
D12225 |
Mazdutide (USAN) |
(P) unclassified |
D12269 |
Nirmatrelvir and ritonavir; Paxlovid (TN) |
(P) Enzyme: CYP3A4 / CYP induction: CYP3A4 |
D12294 |
Sitagliptin phosphate (JAN) |
(P) unclassified |
D12311 |
Bortezomib hydrate (JAN) |
(P) unclassified |
D12326 |
Opelconazole (USAN/INN) |
(P) unclassified |
D12341 |
Vurolenatide (USAN/INN) |
(P) unclassified |
D12353 |
Ensitrelvir fumarate (USAN); Ensitrelvir fumaric acid (JAN); Xocova (TN) |
(P) unclassified |
D12358 |
Insulin icodec (USAN/INN); Insulin icodec (genetical recombination) (JAN) |
(P) unclassified |
D12446 |
Anpocogin (USAN) |
(P) unclassified |
D12484 |
Carfloglitazar (INN) |
(P) unclassified |
D12529 |
Orforglipron calcium (USAN) |
(P) unclassified |
D12536 |
Orforglipron (USAN) |
(P) unclassified |
D12555 |
Lotiglipron (USAN) |
(P) unclassified |
D12586 |
Mifepristone and misoprostol; Mefeego (TN) |
(CI,P) unclassified |
D12595 |
Aspirin trelamine (USAN) |
(P) unclassified |
D12596 |
Aspirin trelamine hydrochloride (USAN) |
(P) unclassified |
D12629 |
Treprostinil phosphate (USAN); Treprostinil biphosphate |
(P) unclassified |
D12637 |
Darunavir hydrate |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4 |
D12703 |
Linagliptin hydrate (JAN); Linagliptin hemihydrate |
(P) unclassified |
D12735 |
Lotiglipron tromethamine (USAN) |
(P) unclassified |
D12752 |
Darunavir propylene glycolate |
(P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4 |
D12861 |
Pemvidutide (USAN/INN) |
(P) unclassified |
D12874 |
Live attenuated influenza virus vaccine, intranasal; Flumist (TN) |
(CI) unclassified |