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Drug interaction list


Query:
D05928  Stiripentol (JAN/USAN/INN); Diacomit (TN)

Interactions: 1280 hits    [ ATC classification | Therapeutic category ]

C01946  Oleandomycin; Amimycin; Landomycin; Matromycin; Romicil (P) unclassified
C06921  Clorazepate; Clorazepic acid (P) unclassified
C07051  Indinavir (P) unclassified
C07480  Theobromine; 3,7-Dimethylxanthine (P) unclassified
D00020  Tryptophan (USP/INN); L-Tryptophan (JP19) (P) unclassified
D00058  gamma-Aminobutyric acid (JAN); Gammalon (TN) (P) unclassified
D00066  Progesterone (JP19/USP/INN); Crinone (TN); Prometrium (TN) (P) Enzyme: CYP3A4 CYP2C19 / CYP inhibition: CYP3A4 CYP2C19
D00105  Estradiol (JAN/USP/INN); Climara (TN); Divigel (TN); Estrace (TN); Estraderm (TN); Estrasorb (TN); Estring (TN); Estrogel (TN); Innofem (TN); Vagifem (TN); Vivelle (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00107  Tacrolimus (USP/INN); Tacrolimus hydrate (JP19); Prograf (TN); Protopic (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00109  Aspirin (JP19/USP); Aspalon (JAN); Acetylsalicylic acid; Easprin (TN); Durlaza (TN) (P) unclassified
D00118  Naproxen (JP19/USP/INN); Naprosyn (TN) (P) unclassified
D00120  Sulindac (JP19/USP/INN); Clinoril (TN) (P) unclassified
D00126  Ibuprofen (JP19/USP/INN); Advil (TN); Motrin (TN) (P) CYP inhibition: CYP2C9
D00127  Piroxicam (JP19/USP/INN); Feldene (TN) (P) CYP inhibition: CYP2C9
D00130  Diflunisal (JAN/USP/INN); Dolobid (TN) (P) unclassified
D00132  Ketoprofen (JP19/USP/INN); Orudis (TN) (P) unclassified
D00136  Haloperidol (JP19/USP/INN); Haldol (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 CYP2D6
D00140  Erythromycin (JP19/USP/INN); Akne-mycin (TN); Eryc (TN); Erygel (TN); Pce (TN); Staticin (TN); T-stat (TN) (P) unclassified
D00141  Indomethacin (USP); Indometacin (JP19/INN); Aconip (TN); Indocin (TN) (P) unclassified
D00142  Methotrexate (JP19/USP/INN); Otrexup (TN); Xatmep (TN) (P) unclassified
D00151  Mefenamic acid (JP19/USP/INN); Ponstel (TN) (P) CYP inhibition: CYP2C9
D00158  Tolmetin sodium (JAN/USP); Tolmetin sodium dihydrate; Tolectin (TN) (P) unclassified
D00169  Meclofenamate sodium (USP); Meclofenamate sodium monohydrate; Meclomen (TN) (P) unclassified
D00184  Cyclosporine (USP); Ciclosporin (JP19); Gengraf (TN); Neoral (TN); Restasis (TN); Sandimmune (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00211  Rifampin (USP); Rifampicin (JP19/INN); Rifadin (TN); Rimactane (TN) (P) CYP induction: CYP3A4
D00225  Alprazolam (JP19/USP/INN); Xanax (TN) (P) unclassified
D00227  Aminophylline (USP/INN); Somophyllin (TN); Theophylline ethylenediamine (TN) (P) Enzyme: CYP1A2 / CYP inhibition: CYP1A2
D00228  Amoxapine (JP19/USP/INN); Asendin (TN) (P) CYP inhibition: CYP2D6
D00235  Atenolol (JP19/USP/INN); Tenormin (TN) (P) CYP inhibition: CYP2D6
D00238  Azathioprine (JP19/USP/INN); Azasan (TN); Imuran (TN); Jayempi (TN) (P) unclassified
D00246  Budesonide (JP19/USP/INN); Entocort EC (TN); Pulmicort (TN); Rhinocort (TN); Uceris (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00252  Carbamazepine (JP19/USP/INN); Equetro (TN); Tegretol (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D00255  Carvedilol (JP19/USP/INN); Artist (TN); Coreg (TN) (P) Enzyme: CYP3A4 CYP1A2 / CYP inhibition: CYP1A2 CYP3A4 CYP2D6 CYP2C9
D00267  Chlordiazepoxide (JP19/USP/INN); Libritabs (TN) (P) unclassified
D00276  Clarithromycin (JP19/USP/INN); Biaxin (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00280  Clonazepam (JP19/USP/INN); Klonopin (TN) (P) unclassified
D00282  Clotrimazole (JP19/USP/INN); Lotrimin (TN); Mycelex (TN) (P) CYP inhibition: CYP3A4
D00283  Clozapine (JAN/USP/INN); Clozaril (TN) (P) Enzyme: CYP1A2 CYP3A4 / CYP inhibition: CYP1A2 CYP3A4
D00292  Dexamethasone (JP19/USP/INN); Decadron (TN); Maxidex (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D00293  Diazepam (JP19/USP/INN); Diastat (TN); Valium (TN) (P) Enzyme: CYP2C19 CYP3A4 / CYP inhibition: CYP3A4 CYP2C19
D00295  Cimetidine (JP19/USP/INN); Tagamet (TN) (P) CYP inhibition: CYP3A4
D00304  Divalproex sodium (USP); Valproate semisodium (INN); Depakote (TN) (P) unclassified
D00311  Estazolam (JP19/USP/INN); ProSom (TN) (P) unclassified
D00315  Etodolac (JP19/USP/INN); Lodine (TN) (P) unclassified
D00319  Felodipine (JP19/USP/INN); Plendil (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00320  Fentanyl (JAN/USP/INN); Duragesic (TN); Subsys (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00322  Fluconazole (JP19/USP/INN); Diflucan (TN) (P) CYP inhibition: CYP2C19 CYP3A4
D00326  Fluoxetine (USAN/INN); Fluoxetine (TN) (P) CYP inhibition: CYP2C19 CYP2D6 CYP2C9
D00329  Flurazepam (JAN/INN); Insumin (TN) (P) unclassified
D00330  Flurbiprofen (JP19/USP/INN); Ansaid (TN) (P) CYP inhibition: CYP2C9
D00336  Glyburide (USP); Glibenclamide (JP19/INN); Diabeta (TN); Glynase (TN); Micronase (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 CYP2C9
D00338  Halazepam (USAN/INN); Paxipam (TN) (P) unclassified
D00346  Isoniazid (JP19/USP/INN); Laniazid (TN) (P) unclassified
D00349  Isradipine (USP/INN); Dynacirc (TN) (P) unclassified
D00350  Itraconazole (JP19/USP); Itrizole (TN); Sporanox (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00351  Ketoconazole (JP19/USP); Nizoral (TN); Xolegel (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00354  Lamotrigine (JAN/USP/INN); Lamictal (TN) (P) unclassified
D00355  Lansoprazole (JP19/USP/INN); Prevacid (TN) (P) Enzyme: CYP2C19 CYP3A4 / CYP inhibition: CYP2C19 CYP3A4
D00359  Lovastatin (USP/INN); Mevacor (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00365  Lorazepam (JP19/USP/INN); Ativan (TN) (P) unclassified
D00370  Temazepam (USP/INN); Restoril (TN) (P) unclassified
D00371  Theophylline (JP19); Elixophyllin (TN); Quibron-t (TN); Theo-24 (TN); Theodur G (TN); Theolair (TN); Uniphyl (TN) (P) Enzyme: CYP1A2 / CYP inhibition: CYP1A2
D00372  Thiabendazole (USP); Tiabendazole (JAN/INN); Mintezol (TN) (P) unclassified
D00375  Mephenytoin (USP/INN); Mesantoin (TN) (P) Enzyme: CYP2C19 / CYP inhibition: CYP2C19
D00377  Mesalamine (USP); Mesalazine (JP19/INN); Apriso (TN); Asacol (TN); Canasa (TN); Delzicol (TN); Lialda (TN); Mesalamine (TN); Pentasa (TN); Rowasa (TN); Sfrowasa (TN) (P) unclassified
D00378  Timolol (USAN); Timolol hemihydrate; Betimol (TN) (P) CYP inhibition: CYP2D6
D00387  Triazolam (JP19/USP/INN); Halcion (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00392  Trimethadione (JP19/INN); Tridione (TN) (P) unclassified
D00394  Trimipramine (USAN/INN) (P) unclassified
D00399  Valproic acid (USP); Depakene (TN) (P) unclassified
D00404  Methsuximide (USP); Mesuximide (INN); Celontin (TN) (P) unclassified
D00415  Zolmitriptan (JAN/USP/INN); Zomig (TN) (P) Enzyme: CYP1A2 / CYP inhibition: CYP1A2
D00416  Miconazole (JP19/USP/INN); Monistat (TN); Oravig (TN) (P) unclassified
D00420  Mitotane (JAN/USP/INN); Lysodren (TN) (P) unclassified
D00425  Nabumetone (JP19/USP/INN); Relafen (TN) (P) unclassified
D00426  Risperidone (JP19/USP/INN); Risperdal (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 CYP2D6
D00427  Ritonavir (JAN/USP/INN); Norvir (TN) (P) CYP inhibition: CYP2D6 / CYP induction: CYP1A2 CYP2C19
D00428  Salsalate (USP/INN); Sasapyrine (JAN); Disalcid (TN) (P) unclassified
D00429  Saquinavir (JAN/USP/INN); Fortovase (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00432  Nadolol (JP19/USP/INN); Corgard (TN) (P) unclassified
D00434  Simvastatin (JP19/USP/INN); MK-733; Zocor (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00435  Nevirapine (JAN/USP/INN); Viramune (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 CYP2D6
D00437  Nifedipine (JP19/USP/INN); Adalat (TN); Afeditab CR (TN); Procardia (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00438  Nimodipine (USP/INN); Nimotop (TN); Nymalize (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00448  Sulfasalazine (USP/INN); Salazosulfapyridine (JP19); Azulfidine (TN) (P) unclassified
D00452  Suprofen (JAN/USP/INN); Profenal (TN) (P) CYP inhibition: CYP2C9
D00455  Omeprazole (JP19/USP/INN); Prilosec (TN) (P) Enzyme: CYP2C19 / CYP inhibition: CYP2C19
D00457  Quazepam (JAN/USP/INN); Doral (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 CYP2C9
D00458  Quetiapine fumarate (JP19/USP); Seroquel (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00463  Oxaprozin (JP19/USP/INN); Daypro (TN) (P) unclassified
D00464  Oxazepam (JAN/USP/INN); Serax (TN) (P) unclassified
D00470  Prazepam (JP19/USAN/INN); Centrax (TN) (P) unclassified
D00472  Prednisolone (JP19/USP/INN); Delta-cortef (TN) (P) unclassified
D00474  Primidone (JP19/USP/INN); Mysoline (TN) (P) unclassified
D00483  Propranolol hydrochloride (JP19/USP); Inderal (TN); Innopran XL (TN) (P) Enzyme: CYP1A2 CYP2C19 / CYP inhibition: CYP1A2 CYP2D6 CYP2C19
D00484  Protriptyline hydrochloride (USP); Vivactil (TN) (P) unclassified
D00495  Paramethadione (INN); Paradione (TN) (P) unclassified
D00501  Pentoxifylline (JAN/USP/INN); Pentoxil (TN); Trental (TN) (P) unclassified
D00502  Pergolide mesylate (USP); Pergolide mesilate (JAN); Permax (TN) (P) unclassified
D00504  Phenacemide (JAN/INN); Phenurone (TN) (P) unclassified
D00505  Phenelzine sulfate (USP); Nardil (TN) (P) unclassified
D00506  Phenobarbital (JP19/USP/INN); Luminal (TN) (P) unclassified
D00508  Phensuximide (USP/INN); Milontin (TN) (P) unclassified
D00510  Phenylbutazone (JP19/USP/INN); Azolid (TN) (P) unclassified
D00512  Phenytoin (JP19/USP/INN); Dilantin (TN) (P) CYP inhibition: CYP2C9
D00513  Pindolol (JP19/USP/INN); Blocklin-L (TN); Carvisken (TN); Visken (TN) (P) CYP inhibition: CYP2D6
D00520  Dimenhydrinate (JP19/USP/INN); Dramamine (TN) (P) unclassified
D00528  Caffeine (USP); Anhydrous caffeine (JP19); Anhydrous caffeine (TN); Respia (TN) (P) Enzyme: CYP1A2 / CYP inhibition: CYP1A2
D00531  Nitrazepam (JP19/USAN/INN); Benzalin (TN); Nitrazepam (TN) (P) unclassified
D00533  Oxcarbazepine (JAN/USP/INN); Oxtellar (TN); Trileptal (TN) (P) CYP inhibition: CYP2C19
D00535  Vigabatrin (JAN/USP/INN); Sabril (TN) (P) unclassified
D00536  Felbamate (USPINN); Felbatol (TN) (P) unclassified
D00537  Topiramate (JAN/USP/INN); Topamax (TN); Trokendi xr (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00538  Zonisamide (JP19/USP/INN); Excegran (TN) (P) unclassified
D00539  Ethosuximide (JP19/USP/INN); Zarontin (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00542  Halothane (JP19/USP/INN); Fluothane (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00550  Midazolam (JAN/USP/INN); Dormicum (TN); Buccolam (TN); Nayzilam (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00553  Prilocaine (USP/INN); Propitocaine (JAN) (P) unclassified
D00556  Aminopyrine (JAN); Aminophenazone (INN) (P) unclassified
D00560  Pimozide (JP19/USP/INN); Orap (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00563  Mirtazapine (JAN/USP/INN); Remeron (TN); Reflex (TN) (P) Enzyme: CYP1A2 CYP3A4 / CYP inhibition: CYP1A2 CYP3A4 CYP2D6
D00564  Warfarin sodium (USP); Coumadin (TN); Jantoven (TN) (P) CYP inhibition: CYP2C9
D00566  Sodium salicylate (JP19/USP); Salsonin (TN) (P) unclassified
D00567  Celecoxib (JP19/USP/INN); Celebrex (TN); Onsenal (TN) (P) CYP inhibition: CYP2C9
D00568  Rofecoxib (JAN/USAN/INN); Vioxx (TN) (P) unclassified
D00570  Colchicine (JP19/USP) (CI,P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00578  Voriconazole (JP19/USP/INN); Vfend (TN) (P) unclassified
D00597  Acebutolol hydrochloride (JP19/USP); Sectral (TN) (P) unclassified
D00598  Betaxolol hydrochloride (JP19/USP); Betoptic (TN); Kerlone (TN) (P) unclassified
D00599  Carteolol hydrochloride (JP19/USP); Cartrol (TN); Ocupress (TN) (P) CYP inhibition: CYP2D6
D00601  Metoprolol tartrate (JP19/USP); Lopressor (TN) (P) CYP inhibition: CYP2D6
D00602  Penbutolol sulfate (JP19/USP); Levatol (TN) (P) unclassified
D00603  Timolol maleate (JP19/USP); Blocadren (TN); Istalol (TN); Timoptic (TN) (P) CYP inhibition: CYP2D6
D00606  Guanfacine hydrochloride (JAN/USP); Intuniv (TN); Tenex (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00615  Amlodipine besylate (USP); Amlodipine besilate (JP19); Norvasc (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00616  Diltiazem hydrochloride (JP19/USP); Cardizem (TN); Cartia XT (TN); Dilacor XR (TN); Dilt-CD (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00617  Nicardipine hydrochloride (JP19/USAN); Cardene (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00618  Nisoldipine (JAN/USAN/INN); Sular (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00619  Verapamil hydrochloride (JP19/USP); Calan (TN); Covera-hs (TN); Vasolan (TN); Verelan (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00629  Nitrendipine (JP19/USAN/INN); Baypress (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00631  Bepridil hydrochloride (USAN); Bepridil hydrochloride hydrate (JAN); Vascor (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 CYP2D6 CYP2C9
D00634  Bisoprolol fumarate (JP19/USP); Zebeta (TN) (P) unclassified
D00635  Metoprolol succinate (USP); Toprol XL (TN) (P) CYP inhibition: CYP2D6
D00636  Amiodarone hydrochloride (JP19/USP); Ancaron (TN); Cordarone (TN); Nexterone (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00644  Esmolol hydrochloride (JAN/USP); Brevibloc (TN) (P) unclassified
D00661  Cevimeline hydrochloride (USAN); Cevimeline hydrochloride hydrate (JAN); Evoxac (TN); Saligren (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 CYP2D6
D00665  Chlorpheniramine maleate (JP19/USP); Chlor-trimeton (TN); Teldrin (TN) (P) unclassified
D00670  Donepezil hydrochloride (JP19/USP); Aricept (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00679  Ergotamine tartrate (JP19/USP); Ergomar (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00680  Methylergonovine maleate (USP); Methylergometrine maleate (JP19); Methergine (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00681  Methysergide maleate (USP); Sansert (TN) (P) unclassified
D00687  Salmeterol xinafoate (JAN/USP); Serevent (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00691  Dyphylline (USP); Diprophylline (JAN/INN); Lufyllin (TN) (P) unclassified
D00693  Chlordiazepoxide hydrochloride (JAN/USP); Librium (TN) (P) unclassified
D00694  Clorazepate dipotassium (JP19/USP); Tranxene (TN) (P) unclassified
D00695  Flurazepam hydrochloride (USP); Flurazepam dihydrochloride; Dalmane (TN) (P) unclassified
D00696  Midazolam hydrochloride (USAN); Versed (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00700  Mephobarbital (JAN/USP); Methylphenobarbital (INN); Mebaral (TN) (P) Enzyme: CYP2C19 / CYP inhibition: CYP2C19
D00701  Phenobarbital sodium (JAN/USP/INN); Luminal sodium (TN) (P) unclassified
D00708  Ethotoin (JAN/USP/INN); Accenon (TN); Peganone (TN) (P) unclassified
D00709  Levetiracetam (JP19/USP/INN); Keppra (TN); E keppra (TN) (P) unclassified
D00710  Valproate sodium (USAN); Sodium valproate (JP19); Depakene (TN); Selenica (TN) (P) unclassified
D00722  Oxybutynin chloride (USP); Oxybutynin hydrochloride (JP19); Ditropan (TN); Gelnique (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00724  Rabeprazole sodium (JP19/USP); Aciphex (TN); Pariet (TN) (P) Enzyme: CYP2C19 CYP3A4 / CYP inhibition: CYP3A4 CYP2C19
D00727  Olsalazine sodium (USAN); Dipentum (TN) (P) unclassified
D00742  Etanercept (USAN/INN); Etanercept (genetical recombination) (JAN); Etanercept (genetical recombination) [Etanercept biosimilar 1] (JAN); Etanercept (genetical recombination) [Etanercept biosimilar 2] (JAN); Enbrel (TN) (P) unclassified
D00746  Interferon beta-1b (USAN/INN); Interferon beta-1b (genetical recombination) (JAN); Betaseron (TN); Extavia (TN) (P) unclassified
D00749  Leflunomide (JAN/USP/INN); Arava (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00752  Mycophenolate mofetil (JAN/USP); Cellcept (TN) (P) unclassified
D00753  Sirolimus (JAN/USAN/INN); Rapamune (TN); Rapamycin (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00754  Thalidomide (JAN/USP/INN); Thalomid (TN); Thaled (TN) (P) unclassified
D00765  Rocuronium bromide (JAN/USP/INN); Zemuron (TN) (P) unclassified
D00769  Clopidogrel bisulfate (USP); Clopidogrel sulfate (JP19); Clopidogrel sulfate tablets (JP19); Clopidogrel hydrogen sulphate; Isocover (TN); Plavix (TN) (P) Enzyme: CYP2C19 CYP1A2 / CYP inhibition: CYP1A2 CYP2C19
D00775  Riluzole (JAN/USP/INN); Rilutek (TN) (P) Enzyme: CYP1A2 / CYP inhibition: CYP1A2
D00780  Bromocriptine mesylate (USP); Bromocriptine mesilate (JP19); Parlodel (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00784  Ropinirole hydrochloride (JAN/USP); Requip (TN) (P) Enzyme: CYP1A2 / CYP inhibition: CYP1A2
D00789  Chlorpromazine hydrochloride (JP19/USP); Sonazine (TN) (P) CYP inhibition: CYP2D6
D00809  Amitriptyline hydrochloride (JP19/USP); Elavil (TN) (P) Enzyme: CYP3A4 CYP2C19 / CYP inhibition: CYP3A4 CYP2D6 CYP2C19
D00810  Choline salicylate (JAN/USAN/INN); Arthropan (TN) (P) unclassified
D00811  Clomipramine hydrochloride (JP19/USP); Anafranil (TN) (P) Enzyme: CYP3A4 CYP2C19 / CYP inhibition: CYP3A4 CYP2D6 CYP2C19
D00812  Desipramine hydrochloride (JAN/USP); Norpramin (TN) (P) unclassified
D00813  Ketorolac tromethamine (USP); Acular (TN); Toradol (TN) (P) unclassified
D00814  Doxepin hydrochloride (USP); Sinequan (TN); Zonalon (TN) (P) Enzyme: CYP2C19 / CYP inhibition: CYP2D6 CYP2C19 CYP2C9
D00815  Imipramine hydrochloride (JP19/USP); Tofranil (TN) (P) Enzyme: CYP3A4 CYP2C19 / CYP inhibition: CYP3A4 CYP2D6 CYP2C19
D00816  Nortriptyline hydrochloride (JP19/USP/INN); Pamelor (TN) (P) CYP inhibition: CYP2D6
D00817  Bupropion hydrochloride (JAN/USP); Wellbutrin (TN); Zyban (TN) (P) unclassified
D00818  Maprotiline hydrochloride (JP19/USP); Ludiomil (TN) (P) CYP inhibition: CYP2D6
D00819  Nefazodone hydrochloride (USP); Serzone (TN) (P) unclassified
D00820  Trazodone hydrochloride (JAN/USP); Desyrel (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 CYP2D6
D00821  Venlafaxine hydrochloride (JAN/USP); Effexor (TN) (P) CYP inhibition: CYP2D6
D00822  Citalopram hydrobromide (USP); Celexa (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP2C19 CYP3A4 CYP2D6
D00823  Fluoxetine hydrochloride (JAN/USP); Prozac (TN); Sarafem (TN) (P) CYP inhibition: CYP2C19 CYP2D6 CYP2C9
D00824  Fluvoxamine maleate (JP19/USP); Luvox (TN) (P) CYP inhibition: CYP1A2 CYP2C19 CYP3A4 CYP2D6
D00825  Sertraline hydrochloride (JAN/USP); Zoloft (TN) (P) Enzyme: CYP2C19 CYP3A4 / CYP inhibition: CYP3A4 CYP2C19 CYP2C9
D00826  Tranylcypromine sulfate (USP); Parnate (TN) (P) unclassified
D00827  Magnesium salicylate (USP); Magnesium salicylate tetrahydrate; Magan (TN) (P) unclassified
D00831  Mefloquine hydrochloride (JP19/USP); Lariam (TN) (P) unclassified
D00836  Buprenorphine hydrochloride (JP19/USP); Buprenex (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00848  Dextromethorphan hydrobromide (USP); Dextromethorphan hydrobromide hydrate (JP19); Benylin DM (TN) (P) CYP inhibition: CYP2D6
D00851  Erythromycin estolate (USP); Erythromycin estorate (JAN); Ilosone (TN) (P) unclassified
D00880  Butoconazole nitrate (USP); Femstat (TN); Gynazole-1 (TN) (P) unclassified
D00881  Econazole nitrate (JAN/USP); Ecoza (TN); Spectazole (TN) (P) unclassified
D00882  Miconazole nitrate (JP19/USP); Micatin (TN); Monistat (TN) (P) unclassified
D00885  Oxiconazole nitrate (JAN/USAN); Oxistat (TN) (P) unclassified
D00886  Sulconazole nitrate (JAN/USP); Exelderm (TN) (P) unclassified
D00887  Atorvastatin calcium anhydorous; Lipitor (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00888  Terconazole (USP/INN); Terazol 3 (TN) (P) unclassified
D00889  Cerivastatin sodium (JAN/USAN); Baycol (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00890  Tioconazole (JAN/USP/INN); Vagistat-1 (TN) (P) unclassified
D00892  Fluvastatin sodium (JAN/USP); Lescol (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 CYP2C9
D00893  Pravastatin sodium (JP19/USP); CS-514; Pravachol (TN) (P) unclassified
D00894  Amprenavir (JAN/USAN/INN); Agenerase (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00897  Indinavir sulfate (USP); Crixivan (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00899  Nelfinavir mesylate (USAN/INN); Nelfinavir mesilate (JAN); Viracept (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00903  Diclofenac potassium (USP); Cambia (TN); Cataflam (TN); Zipsor (TN) (P) CYP inhibition: CYP2C9
D00904  Diclofenac sodium (JP19/USP); Solaraze (TN); Voltaren (TN) (P) CYP inhibition: CYP2C9
D00950  Levonorgestrel (JAN/USP/INN); Mirena (TN); Norplant (TN); Skyla (TN) (P) unclassified
D00961  Bicalutamide (JP19/USP/INN); Casodex (TN) (P) CYP inhibition: CYP3A4
D00964  Letrozole (JAN/USP/INN); Femara (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D00968  Fenoprofen calcium (JAN/USP); Nalfon (TN) (P) unclassified
D00969  Meloxicam (JAN/USP/INN); Mobic (TN) (P) CYP inhibition: CYP2C9
D00970  Naproxen sodium (USP); Anaprox (TN) (P) unclassified
D00971  Sodium thiosalicylate; Thiosalicylic acid sodium salt; Rexolate (TN) (P) unclassified
D00987  Cabergoline (JP19/USP/INN); Cabaser (TN); Dostinex (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D01025  Levobunolol hydrochloride (JAN/USP); Betagan (TN) (P) unclassified
D01026  Sotalol hydrochloride (JAN/USP); Betapace (TN); Sorine (TN) (P) unclassified
D01037  1,4-Dimethyl-7-isopropylazulene (JAN); Guaiazulene; Azunol (TN) (P) unclassified
D01049  Nimesulide (JAN/INN) (P) unclassified
D01061  Irinotecan hydrochloride (USP); Irinotecan hydrochloride hydrate (JP19); Irinotecan hydrochloride trihydrate; CPT 11; CPT-11; Campto (TN); Camptosar (TN); Onivyde (TN) (P) unclassified
D01078  Telithromycin (JAN/USAN/INN); Ketek (TN) (P) CYP inhibition: CYP2D6
D01087  Methyl salicylate (JP19/NF) (P) unclassified
D01092  Lanoconazole (JP19/INN); Latoconazole; Astat (TN) (P) unclassified
D01104  Barnidipine hydrochloride (JAN); Hypoca (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D01107  Milnacipran hydrochloride (JAN/USAN); Savella (TN); Toledomin (TN) (P) unclassified
D01110  Melitracen hydrochloride (JAN/USAN) (P) unclassified
D01115  Eplerenone (JP19/USAN/INN); Inspra (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D01122  Ibuprofen piconol (JP19/USAN); Staderm (TN) (P) CYP inhibition: CYP2C9
D01145  Azelnidipine (JP19/INN); Calblock (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D01160  Saquinavir mesylate (USP); Saquinavir mesilate (JAN); Invirase (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D01163  Ergonovine maleate (USP); Ergometrine maleate (JP19); Ergometrine (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D01164  Aripiprazole (JP19/USP/INN); Abilify (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 CYP2D6
D01172  Diphenylpyraline hydrochloride (JAN); Hispril (TN); Vena (TN) (P) unclassified
D01173  Cilnidipine (JP19/INN); Atelec (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D01176  Blonanserin (JP19/INN); AD 5423 (CI,P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D01179  Duloxetine hydrochloride (JAN/USP); Cymbalta (TN); Yentreve (TN) (P) Enzyme: CYP1A2 / CYP inhibition: CYP1A2
D01182  Alprenolol hydrochloride (JP19/USAN); Regletin (TN) (P) CYP inhibition: CYP2D6
D01183  Tolfenamic acid (JAN/INN); Clotam (TN) (P) unclassified
D01185  Protizinic acid (JAN/INN) (P) unclassified
D01189  Metiazinic acid (JAN/INN) (P) unclassified
D01190  Ethylphenacemide (JAN); Pheneturide (INN) (P) unclassified
D01207  Omeprazole sodium (USAN); Losec sodium (TN) (P) Enzyme: CYP2C19 / CYP inhibition: CYP2C19
D01213  Tolvaptan (JP19/USAN/INN); Samsca (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D01230  Flunitrazepam (JP19/USAN/INN); Rohypnol (TN) (P) unclassified
D01235  Josamycin (JP19/USAN/INN); Leucomycin A3; JM (P) CYP inhibition: CYP3A4
D01239  Prednisolone sodium succinate (JP19/USP); Kohakusanin (TN) (P) unclassified
D01243  Prilocaine hydrochloride (USP); Propitocaine hydrochloride (JAN); Citanest (TN) (P) unclassified
D01245  Bromazepam (JP19/USAN/INN); Lectopam (TN) (P) unclassified
D01252  Alclofenac (JAN/USP/INN); Mervan (TN) (P) unclassified
D01253  Clobazam (JAN/USAN/INN); Mystan (TN); Onfi (TN) (P) Enzyme: CYP3A4 CYP2C19 / CYP inhibition: CYP3A4 CYP2C19
D01254  Tofisopam (JP19/INN); Emandaxin (TN) (P) unclassified
D01267  Floctafenine (JAN/USAN/INN); Idarac (TN) (P) unclassified
D01268  Cloxazolam (JP19/INN); Sepazon (TN) (P) unclassified
D01271  Bufexamac (JAN/INN); Anderm (TN) (P) unclassified
D01276  Atazanavir sulfate (JAN/USAN); Reyataz (TN) (P) CYP inhibition: CYP3A4
D01278  Oxazolam (JP19/INN); Serenal (TN) (P) unclassified
D01279  Flutoprazepam (JAN/INN); Restas (TN) (P) unclassified
D01280  Warfarin potassium (JP19); Athrombin-K (TN) (P) CYP inhibition: CYP2C9
D01285  Lofepramine hydrochloride (JAN/USAN); Amplit (TN) (P) unclassified
D01286  Flutazolam (JAN/INN); Coreminal (TN) (P) unclassified
D01287  Levobupivacaine hydrochloride (JAN/USAN); Chirocaine (TN) (P) Enzyme: CYP3A4 CYP1A2 / CYP inhibition: CYP1A2 CYP3A4
D01289  Suxibuzone (JAN/INN) (P) unclassified
D01290  Nicergoline (JP19/USAN/INN); Sermion (TN) (P) unclassified
D01292  Medazepam (JP19/INN); Pamnace (TN) (P) unclassified
D01293  Ethyl loflazepate (JP19/INN); Meilax (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D01296  Methylphenidate hydrochloride (JAN/USP); Concerta (TN); Metadate (TN); Quillivant xr (TN); Ritalin (TN) (P) unclassified
D01303  Flunarizine hydrochloride (JAN/USAN) (P) CYP inhibition: CYP2D6
D01305  Feprazone (JAN/INN) (P) unclassified
D01314  Dibenzepin hydrochloride (JAN/USAN) (P) unclassified
D01316  Mexazolam (JAN/INN); Melex (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D01322  Troleandomycin (USAN/INN); Triacetyloleandomycin (JAN); TAO; Tao (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D01325  Tiaprofenic acid (JAN/INN); Surgam (TN) (P) unclassified
D01328  Clotiazepam (JP19/INN); Rize (TN) (P) unclassified
D01330  Clidanac (JAN/INN) (P) unclassified
D01339  Midecamycin (JP19/INN); Medemycin (TN) (P) CYP inhibition: CYP3A4
D01341  Tiaramide hydrochloride (JP19/USAN); Solantal (TN) (P) unclassified
D01344  Fenbufen (JP19/USAN/INN) (P) unclassified
D01348  Terguride (JAN/INN); Teluron (TN) (P) unclassified
D01353  Emorfazone (JP19/INN); Pentoil (TN) (P) unclassified
D01354  Fludiazepam (JP19/INN); Erispan (TN) (P) unclassified
D01355  Tramadol hydrochloride (JP19/USP); Ultram (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 CYP2D6
D01358  Mianserin hydrochloride (JAN/USAN); Tetramide (TN) (P) Enzyme: CYP3A4 CYP1A2 / CYP inhibition: CYP1A2 CYP3A4 CYP2D6
D01361  Erythromycin ethylsuccinate (JP19/USP); E.E.S. (TN); Eryped (TN); Erythrocin W (TN) (P) unclassified
D01370  Cladribine (JAN/USP/INN); Leustatin (TN); Mavenclad (TN) (P) unclassified
D01372  Zopiclone (JP19/INN); Amoban (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D01380  Isopropylantipyrine (JP19); Propyphenazone (INN); Yoshipyrin (TN) (P) unclassified
D01382  Metharbital (JAN/INN); Gemonil (TN) (P) unclassified
D01394  Epirizole (JP19/USAN); Mebron (TN) (P) unclassified
D01397  Ampiroxicam (JP19/INN); Flucam (TN) (P) CYP inhibition: CYP2C9
D01399  Fentanyl citrate (JP19/USP); Abstral (TN); Fentora (TN); Lazanda (TN); Oralet (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D01408  Flurazepam hydrochloride (JP19); Flurazepam monohydrochloride; Dalmate (TN) (P) unclassified
D01410  Benzydamine hydrochloride (JAN/USAN); Tantum (TN) (P) unclassified
D01418  Tamibarotene (JAN/USAN/INN); Am 80; Amnoid (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D01425  Lopinavir (JAN/USP/INN) (P) unclassified
D01429  Fosfluconazole (JAN/INN); Prodif (TN) (P) CYP inhibition: CYP2C19 CYP3A4
D01437  Nifenazone (JAN/INN) (P) unclassified
D01453  Caffeine hydrate (JP19); Caffeine monohydrate (P) Enzyme: CYP1A2 / CYP inhibition: CYP1A2
D01454  Bupranolol hydrochloride (JP19) (P) unclassified
D01462  Lisuride maleate (JAN) (P) unclassified
D01466  Ethenzamide (JP19/INN) (P) unclassified
D01471  Esatenolol (JAN/INN); (S)-Atenolol (P) unclassified
D01475  Flurbiprofen axetil (JAN); FP 83; Ropion (TN) (P) CYP inhibition: CYP2C9
D01477  Opipramol hydrochloride (JAN/USAN); Insidon (TN) (P) unclassified
D01480  Isoconazole nitrate (JAN); Adestan-G (TN) (P) unclassified
D01492  Bucumolol hydrochloride (JP19) (P) unclassified
D01504  Bufetolol hydrochloride (JP19); Adobiol (TN) (P) unclassified
D01512  Befunolol hydrochloride (JAN); Bentos (TN) (P) unclassified
D01513  Alminoprofen (JP19/INN); Minalfen (TN) (P) unclassified
D01514  Etizolam (JP19/INN); Sedekopan (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 CYP2C9
D01545  Aceclofenac (JAN/INN) (P) unclassified
D01546  Dothiepin hydrochloride (USAN); Dosulepin hydrochloride (JAN); Prothiaden (TN) (P) CYP inhibition: CYP2D6
D01547  Zaltoprofen (JP19/INN); CN 100; Peon (TN) (P) unclassified
D01553  Manidipine hydrochloride (JP19); Manidipine dihydrochloride; Calslot (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D01557  Glycol salicylate (JAN); Ethylene glycol salicylate; Norgesic (TN); Phlogont (TN) (P) unclassified
D01562  Aranidipine (JAN/INN); Sapresta (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D01564  Rilmazafone hydrochloride hydrate (JP19); Rilmazafone hydrochloride dihydrate; Rilmazafone hydrochloride; Rhythmy (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D01565  Indometacin farnesil (JAN); Infree (TN) (P) unclassified
D01566  Gusperimus trihydrochloride (USAN); Gusperimus hydrochloride (JAN); Spanidin (TN) (P) unclassified
D01567  Ketophenylbutazone (JAN); Kebuzone (INN) (P) unclassified
D01578  Pranoprofen (JP19/INN); Elicapric (TN) (P) unclassified
D01581  Flufenamic acid (JAN/USAN/INN); Arlef (TN) (P) unclassified
D01582  Acemetacin (JP19/INN); Rantudil (TN) (P) unclassified
D01583  Pirfenidone (JAN/USAN/INN); Esbriet (TN) (P) Enzyme: CYP1A2 CYP2C19 / CYP inhibition: CYP1A2 CYP2D6 CYP2C19
D01593  Nimetazepam (JAN/INN); Erimin (TN) (P) unclassified
D01594  Bendazac (JAN/USAN/INN); Iwazac (TN) (P) unclassified
D01604  Efonidipine hydrochloride ethanolate (JAN); Efonidipine hydrochloride ethanol; Efonidipine hydrochloride; NZ 105 ethanolate; Landel (TN) (P) unclassified
D01614  Acetylkitasamycin (JP19); Neo-leucomycin H (TN) (P) unclassified
D01620  Neticonazole hydrochloride (JAN); Atolant (TN) (P) unclassified
D01627  Diphenylpyraline teoclate (JAN); Piprinhydrinate; Plokon (TN) (P) unclassified
D01630  Propentofylline (JAN/INN) (P) unclassified
D01636  Midecamycin acetate (JP19); Miocamycin; Miocamycin (TN) (P) CYP inhibition: CYP3A4
D01656  Brovincamine fumarate (JAN); Sabromin (TN) (P) unclassified
D01657  Lormetazepam (JAN/USAN/INN); Loramet (TN) (P) unclassified
D01661  Bucolome (JAN/INN); Paramidin (TN) (P) unclassified
D01664  Omoconazole nitrate (JAN/USAN) (P) unclassified
D01675  Felbinac (JP19/USAN/INN); Dolinac (TN) (P) unclassified
D01703  Ciclesonide (JAN/USAN/INN); Alvesco (TN); Omnaris (TN); Zetonna (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D01706  Migrenin (JP19) (P) unclassified
D01708  Fluticasone propionate (JAN/USP); Cutivate (TN); Flonase (TN); Flovent (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D01709  Loxoprofen sodium hydrate (JP19); Lorfenamin (TN); Loxonin (TN) (P) unclassified
D01710  Roxithromycin (JP19/USAN/INN); Rulide (TN) (P) unclassified
D01712  Theophylline sodium acetate (JAN) (P) Enzyme: CYP1A2 / CYP inhibition: CYP1A2
D01718  Mofezolac (JAN/INN) (P) CYP inhibition: CYP2C9
D01741  Celiprolol hydrochloride (JAN/USAN); Selectol (TN) (P) unclassified
D01744  Brotizolam (JP19/USAN/INN); Lendormin (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D01745  Domperidone (JP19/USAN/INN); Motilium (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D01758  Haloxazolam (JP19/INN); Somelin (TN) (P) unclassified
D01762  Dipyrone (USAN); Sulpyrine hydrate (JP19); Metamizole sodium salt monohydrate (P) unclassified
D01765  Proglumetacin maleate (JAN); Miridacin (TN) (P) unclassified
D01767  Tenoxicam (JAN/USAN/INN); Tilcotil (TN) (P) CYP inhibition: CYP2C9
D01771  Proxyphylline (JAN/INN); Monophyllin (TN) (P) unclassified
D01775  Bifonazole (JP19/USAN/INN); Mycospor (TN) (P) unclassified
D01776  Antipyrine (JP19/USP); Phenazone (INN) (P) unclassified
D01787  Sulthiame (USAN); Sultiame (JP19); Ospolot (TN) (P) unclassified
D01788  Amfenac sodium (USAN); Amfenac sodium hydrate (JAN); Fenazox (TN) (P) unclassified
D01793  Bifemelane hydrochloride (JAN) (P) unclassified
D01794  Bopindolol malonate (JAN); Sandonorm (TN) (P) CYP inhibition: CYP2D6
D01795  Tilisolol hydrochloride (JAN); Selecal (TN) (P) unclassified
D01806  Oxprenolol hydrochloride (JP19/USP); Okuspurecol (TN) (P) unclassified
D01811  Salicylamide (JAN/USP/INN) (P) unclassified
D01823  Ufenamate (JAN/INN); Flufenamic acid butyl ester; Combec (TN) (P) unclassified
D01832  Modafinil (JAN/USP/INN); Provigil (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP2C19 CYP3A4 / CYP induction: CYP1A2 CYP3A4
D01841  Felbinac ethyl (JAN); LM 001 (P) unclassified
D01847  Landiolol hydrochloride (JAN/USAN); ONO 1101 hydrochloride; Onoact (TN); Rapiblyk (TN) (P) unclassified
D01849  Lercanidipine hydrochloride (JAN/USAN); Cardiovasc (TN) (P) unclassified
D01851  Mepranoprofen arbamel (JAN); Y-23023 (P) unclassified
D01862  Pitavastatin calcium (JAN); NK 104; Livalo (TN) (P) CYP inhibition: CYP2C9
D01865  Pelubiprofen (JAN/INN) (P) unclassified
D01866  Lornoxicam (JP19/USAN/INN); Lorcam (TN) (P) CYP inhibition: CYP2C9
D01874  Vedaprofen (JAN/USAN/INN) (P) unclassified
D01896  Cilostazol (JP19/USP/INN); Pletal (TN) (P) Enzyme: CYP3A4 CYP2C19 / CYP inhibition: CYP3A4 CYP2C19
D01897  Rokitamycin (JAN/INN); Ricamycin (TN) (P) unclassified
D01898  Haloperidol decanoate (JAN/USP); Halomonth (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 CYP2D6
D01908  Nilvadipine (JP19/USAN/INN); Nivadil (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D01915  Rosuvastatin calcium (JP19/USP); ZD 4522; Crestor (TN) (P) unclassified
D01920  Tenatoprazole (JAN/INN); TU 199 (P) unclassified
D01933  Vatanidipine hydrochloride (JAN); AE 0047; Calbren (TN) (P) unclassified
D01958  Indenolol hydrochloride (JP19) (P) unclassified
D01963  Ibufenac (JAN/USAN/INN); Dytransin (TN) (P) unclassified
D01969  Gallopamil hydrochloride (JAN) (P) unclassified
D01973  Eletriptan hydrobromide (JAN/USAN); Relpax (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D01974  Tilmacoxib (JAN/USAN/INN) (P) unclassified
D01975  Fentiazac (JAN/USAN/INN) (P) unclassified
D01977  Gefitinib (JP19/USAN/INN); Iressa (TN) (P) unclassified
D01980  Luliconazole (JAN/USAN/INN); Lulicon (TN); Luzu (TN) (P) CYP inhibition: CYP2C19 CYP3A4
D01984  Esomeprazole magnesium (USP); Esomeprazole magnesium hydrate (JP19); Esomeprazole magnesium trihydrate; Nexium (TN) (P) Enzyme: CYP2C19 / CYP inhibition: CYP2C19
D02000  Kitasamycin tartrate (JP19); Leucomycin tartrate (TN) (P) unclassified
D02008  Tadalafil (JAN/USP/INN); Adcirca (TN); Cialis (TN); Zalutia (TN) (CI,P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D02009  Erythromycin lactobionate (JP19/USP); Erythrocin (TN) (P) unclassified
D02017  Oxtriphylline (USP); Choline theophyllinate (INN); Choline theophylline (JAN); Theophyline and choline; Theocolin (TN) (P) Enzyme: CYP1A2 / CYP inhibition: CYP1A2
D02045  Benidipine hydrochloride (JP19); KW 3049; Coniel (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D02075  Sodium gualenate (INN); Sodium guaiazulenesulfonate; Azunol ST (TN) (P) unclassified
D02081  Metipranolol hydrochloride; Optipranolol (TN) (P) unclassified
D02096  Fosphenytoin sodium (USP); Cerebyx (TN); Sesquient (TN) (P) CYP inhibition: CYP2C9 / CYP induction: CYP3A4
D02097  Tiagabine hydrochloride (USP); Gabitril (TN) (P) unclassified
D02101  Codeine phosphate (USP); Codeine phosphate hydrate (JP19) (P) CYP inhibition: CYP2D6
D02103  Phenytoin sodium (USP); Phenytoin sodium for injection (JP19); Aleviatin (TN); Dilantin (TN) (P) CYP inhibition: CYP2C9
D02110  Indomethacin sodium (USP); Indometacin sodium hydrate (JAN); Indomethacin sodium trihydrate; Indometacin sodium; Indocin I.V. (TN) (P) unclassified
D02114  Hydroxychloroquine sulfate (JAN/USP); Plaquenil (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D02115  Methotrexate sodium; Trexall (TN); Rasuvo (TN) (P) unclassified
D02134  Azithromycin hydrate (JP19); Azithromycin dihydrate; Zithromac (TN); Zmax (TN); Azimycin (TN) (P) unclassified
D02169  Croconazole hydrochloride (JP19); Pilzcin (TN) (P) unclassified
D02184  Erythromycin stearate (JP19/USP); Bristamycin (TN) (P) unclassified
D02186  Oleandomycin phosphate (JAN); Matromycin (TN) (P) unclassified
D02211  Dihydroergotamine mesylate (USP); Dihydroergotamine mesilate (JP19); Migranal (TN); Trudhesa (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D02229  Sildenafil citrate (JAN/USP); Revatio (TN); Viagra (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D02258  Atorvastatin calcium (USP); Atorvastatin calcium hydrate (JP19); Atorvastatin calcium trihydrate; Atorvaliq (TN); Lipitor (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D02260  Paroxetine hydrochloride hemihydrate (USP); Paroxetine hydrochloride hydrate (JP19); Paxil (TN) (P) CYP inhibition: CYP2D6
D02264  Dipotassium glycyrrhizinate (JAN); Glycyrrhizinate dipotassium; Neubormitin (TN) (P) unclassified
D02268  Ergoloid mesylates (USP); Dihydroergotoxine mesilate (JP19); Circanol (TN); Hydergine (TN); Inorter (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D02269  Kitasamycin (JP19/USAN); Leucomycin (TN) (P) unclassified
D02272  Quinidine sulfate (USP); Quinidine sulfate hydrate (JP19); Quinidex (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D02290  Flurbiprofen sodium (USP); Ocufen (TN) (P) CYP inhibition: CYP2C9
D02338  Acebutolol (USAN/INN) (P) unclassified
D02341  Meclofenamic acid (USAN/INN) (P) unclassified
D02342  Bisoprolol (JAN/USAN/INN) (P) unclassified
D02350  Fenoprofen (USAN/INN) (P) unclassified
D02355  Tolmetin (USAN/INN) (P) unclassified
D02356  Verapamil (USAN/INN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D02357  Methysergide (USAN/INN) (P) unclassified
D02358  Metoprolol (USAN/INN) (P) CYP inhibition: CYP2D6
D02360  Sertraline (INN) (P) Enzyme: CYP2C19 CYP3A4 / CYP inhibition: CYP3A4 CYP2C19 CYP2C9
D02362  Paroxetine (USP/INN) (P) CYP inhibition: CYP2D6
D02372  Perospirone hydrochloride hydrate (JP19); Lullan (TN) (P) unclassified
D02374  Metipranolol (USAN/INN) (P) unclassified
D02389  Primidolol (USAN/INN) (P) unclassified
D02408  Trimipramine maleate (JAN/USP); Surmontil (TN) (P) unclassified
D02420  Acetylspiramycin (JP19); Spiramycin II (P) unclassified
D02484  Artemether and lumefantrine; Coartem (TN) (P) unclassified
D02490  Tylosin (USP/INN); TS; Tylan (TN) (P) unclassified
D02492  Tilmicosin (USP/INN); TMS; Micotil (TN) (P) unclassified
D02493  Tilmicosin phosphate (USAN); TP (P) unclassified
D02497  Fosamprenavir (INN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D02498  Lopinavir and ritonavir; Kaletra (TN) (P) unclassified
D02523  Erythromycin acistrate (USAN); Erasis (TN) (P) unclassified
D02524  Erythromycin gluceptate (USP); Erythromycin glucoheptonate; Ilotycin gluceptate (TN) (P) unclassified
D02525  Erythromycin propionate (USAN) (P) unclassified
D02537  Dronedarone (INN) (P) unclassified
D02555  Posaconazole (JAN/USAN/INN); Noxafil (TN) (P) CYP inhibition: CYP3A4
D02556  Ravuconazole (prop.INN) (P) unclassified
D02557  Chlormidazole (INN) (P) unclassified
D02559  Toloxatone (INN); Humoryl (TN) (P) unclassified
D02561  Moclobemide (USAN/INN); Aurorix (TN) (P) Enzyme: CYP2C19 / CYP inhibition: CYP2C19
D02562  Rasagiline mesylate (USAN); Rasagiline mesilate (JAN); Azilect (TN) (P) Enzyme: CYP1A2 / CYP inhibition: CYP1A2
D02565  Dimetacrine (INN) (P) unclassified
D02566  Maprotiline (USAN) (P) CYP inhibition: CYP2D6
D02567  Escitalopram oxalate (JAN/USP); Lexapro (TN) (P) Enzyme: CYP3A4 CYP2C19 / CYP inhibition: CYP3A4 CYP2D6 CYP2C19
D02570  Desvenlafaxine succinate (USAN); Desvenlafaxine succinate hydrate (JAN); Desvenlafaxine succinate monohydrate; Pristiq (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D02572  Viloxazine hydrochloride (USAN); Qelbree (TN); Vivalan (TN) (P) CYP inhibition: CYP2D6
D02573  Reboxetine mesylate (USAN); Reboxetine mesilate; Vestra (TN) (P) unclassified
D02574  Atomoxetine hydrochloride (JAN/USP); Tomoxetine hydrochloride; Strattera (TN) (P) CYP inhibition: CYP2D6
D02575  Tianeptine (INN); Stablon (TN) (P) unclassified
D02578  Agomelatine (INN); Valdoxan (TN) (P) unclassified
D02579  Iproniazid (INN) (P) unclassified
D02580  Isocarboxazid (INN); Marplan (TN) (P) unclassified
D02582  Fenticonazole (INN) (P) unclassified
D02583  Fenticonazole nitrate (USAN); Lomexin (TN) (P) unclassified
D02584  Aliconazole (INN) (P) unclassified
D02585  Vibunazole; Bay N-7133 (P) unclassified
D02586  Alteconazole (INN) (P) unclassified
D02593  Pantoprazole sodium (USP); Pantoprazole sodium hydrate (JAN); Protonix (TN) (P) Enzyme: CYP2C19 / CYP inhibition: CYP2C19
D02596  Tocilizumab (USAN/INN); Tocilizumab (genetical recombination) (JAN); Tocilizumab (genetical recombination) [Tocilizumab biosimilar 1] (JAN); Tocilizumab (genetical recombination) [Tocilizumab biosimilar 2] (JAN); Tocilizumab-aazg; Tocilizumab-bavi; Tocilizumab-anoh; Actemra (TN); Avtozma (TN); Tofidence (TN); Tyenne (TN) (P) unclassified
D02597  Adalimumab (USAN/INN); Adalimumab (genetical recombination) (JAN); Adalimumab (genetical recombination) [Adalimumab biosimilar 1] (JAN); Adalimumab (genetical recombination) [Adalimumab biosimilar 2] (JAN); Adalimumab (genetical recombination) [Adalimumab biosimilar 3] (JAN); Adalimumab (genetical recombination) [Adalimumab biosimilar 4] (JAN); Adalimumab-adaz; Adalimumab-adbm; Adalimumab-afzb; Adalimumab-atto; Adalimumab-bwwd; Adalimumab-fkjp; Adalimumab-aaty; Adalimumab-aacf; Adalimumab-aqvh; Adalimumab-ryvk; Humira (TN); Abrilada (TN); Amjevita (TN); Cyltezo (TN); Hadlima (TN); Hyrimoz (TN) (P) unclassified
D02598  Infliximab (USAN/INN); Infliximab (genetical recombination) (JAN); Infliximab (genetical recombination) [Infliximab biosimilar 1] (JAN); Infliximab (genetical recombination) [Infliximab biosimilar 2] (JAN); Infliximab (genetical recombination) [Infliximab biosimilar 3] (JAN); Infliximab-dyyb; Infliximab-abda; Infliximab-axxq; Remicade (TN); Inflectra (TN); Renflexis (TN); Avsola (TN); Zymfentra (TN) (P) unclassified
D02600  Demoxepam (USAN/INN) (P) unclassified
D02624  Eszopiclone (JAN/USP/INN); Estorra (TN); Lunesta (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D02629  Fluspirilene (USAN/INN); Imap (TN) (P) unclassified
D02630  Penfluridol (USAN/INN); Semap (TN) (P) unclassified
D02633  Lomerizine hydrochloride (JAN); Terranas (TN) (P) unclassified
D02689  Ramelteon (JAN/USAN/INN); Rozerem (TN) (P) Enzyme: CYP1A2 / CYP inhibition: CYP1A2
D02691  Somatropin (USP/INN); Somatropin (genetical recombination) (JAN); Human growth hormone (JAN); Asellacrin (TN); Humatrope (TN); Nutropin (TN); Omnitrope (TN) (P) CYP inhibition: CYP2C19
D02706  Sodium gualenate hydrate (JAN); Azulene sulfonate sodium hydrate; Sodium guaiazulene sulfonate; Azunol (TN) (P) unclassified
D02709  Valdecoxib (USAN/INN); Bextra (TN) (P) unclassified
D02714  Everolimus (JAN/USAN/INN); Afinitor (TN); Votubia (TN); Zortress (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D02715  Balsalazide disodium (USP); Colazide (TN) (P) unclassified
D02732  Pranlukast hydrate (JP19); Onon (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D02765  Adaprolol maleate (USAN) (P) unclassified
D02766  Valpromide (INN); Depamide (TN) (P) unclassified
D02770  Adinazolam (USAN/INN) (P) unclassified
D02771  Adinazolam mesylate (USAN) (P) unclassified
D02787  Alaproclate (USAN/INN) (P) unclassified
D02800  Alefacept (USAN/INN); Amevive (TN) (P) unclassified
D02802  Alemtuzumab (USAN/INN); Alemtuzumab (genetical recombination) (JAN); Campath (TN); Lemtrada (TN) (P) unclassified
D02834  Alprenoxime hydrochloride (USAN) (P) unclassified
D02861  Indinavir sulfate ethanolate (JAN); Crixivan (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D02867  Fosamprenavir calcium hydrate (JAN); Lexiva (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D02884  Ambuphylline (USAN); Bufylline (BAN); Butaphyllamine (TN) (P) unclassified
D02893  Amesergide (USAN/INN) (P) unclassified
D02914  Amlodipine maleate (USAN); Amvaz (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D02934  Anakinra (USAN/INN); Anakinra (genetical recombination) (JAN); Kineret (TN) (P) unclassified
D02944  Anirolac (USAN/INN) (P) unclassified
D02968  Aprepitant (JAN/USP/INN); Aponvie (TN); Emend (TN); Cinvanti (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D02985  Arofylline (USAN/INN) (P) unclassified
D02995  Asenapine maleate (JAN/USAN); Saphris (TN) (P) Enzyme: CYP1A2 / CYP inhibition: CYP1A2
D03023  Azaconazole (USAN/INN) (P) unclassified
D03033  Azathioprine sodium (USP); Imuran (TN) (P) unclassified
D03051  Bamifylline hydrochloride (USAN) (P) unclassified
D03058  Basiliximab (USAN/INN); Basiliximab (genetical recombination) (JAN); Simulect (TN) (P) unclassified
D03067  Belfosdil (USAN/INN) (P) unclassified
D03068  Belimumab (USAN); Belimumab (genetical recombination) (JAN); Benlysta (TN); LymphoStat-B (TN) (P) unclassified
D03080  Benoxaprofen (USAN/INN); Oraflex (TN) (P) unclassified
D03083  Bentazepam (USAN/INN) (P) unclassified
D03098  Berythromycin (USAN/INN); Erythromycin B (P) unclassified
D03106  Bexarotene (JAN/USAN/INN); Targretin (TN) (P) unclassified
D03150  Bortezomib (JAN/USAN/INN); Velcade (TN) (P) unclassified
D03163  Bromfenac sodium (USAN); Bromfenac sodium hydrate (JP19); Bromfenac sodium sesquihydrate; Bromday (TN); Prolensa (TN); Xibrom (TN); Yellox (TN) (P) unclassified
D03164  Bromindione (USAN/INN) (P) unclassified
D03165  Bromocriptine (USAN/INN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D03170  Bucindolol hydrochloride (USAN) (P) unclassified
D03177  Bunolol hydrochloride (USAN) (P) unclassified
D03198  Butoxamine hydrochloride (USAN) (P) unclassified
D03199  Butriptyline hydrochloride (USAN) (P) unclassified
D03203  Abatacept (USAN/INN); Abatacept (genetical recombination) (JAN); Orencia (TN) (P) unclassified
D03204  Abetimus sodium (USAN) (P) unclassified
D03218  Axitinib (JAN/USAN); Inlyta (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D03222  Belatacept (USAN/INN); Nulojix (TN) (P) unclassified
D03253  Brecanavir (USAN) (P) unclassified
D03254  Flufenamate aluminum (JAN); Flufenamic acid aluminum; Opyrin (TN) (P) unclassified
D03260  Vardenafil hydrochloride hydrate (JAN); Vardenafil monohydrochloride trihydrate; Levitra (TN); Staxyn (TN) (CI,P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D03385  Carbaspirin calcium (USAN); Carbasalate calcium (INN) (P) unclassified
D03410  Carprofen (USP/INN); Rimadyl (TN) (P) unclassified
D03415  Carvedilol phosphate (USAN); Carvedilol phosphate hydrate (JAN); Coreg CR (TN) (P) Enzyme: CYP3A4 CYP1A2 / CYP inhibition: CYP1A2 CYP3A4 CYP2D6 CYP2C9
D03441  Certolizumab pegol (USAN/INN); Certolizumab pegol (genetical recombination) (JAN); Cimzia (TN) (P) unclassified
D03449  Cetamolol hydrochloride (USAN) (P) unclassified
D03489  Cicloprofen (USAN/INN) (P) unclassified
D03490  Cicloprolol hydrochloride (USAN) (P) unclassified
D03516  Cipamfylline (USAN/INN) (P) unclassified
D03526  Cisconazole (USAN/INN) (P) unclassified
D03536  Clentiazem maleate (JAN/USAN) (P) unclassified
D03540  Cliprofen (USAN/INN) (P) unclassified
D03560  Clopirac (USAN/INN) (P) unclassified
D03562  Clorazepate monopotassium (USAN) (P) unclassified
D03601  Crilvastatin (USAN/INN) (P) unclassified
D03631  Cyprazepam (USAN/INN) (P) unclassified
D03639  Daclizumab (USAN/INN); Zenapax (TN); Zinbryta (TN) (P) unclassified
D03643  Dalvastatin (USAN/INN) (P) unclassified
D03652  Darbufelone mesylate (USAN) (P) unclassified
D03655  Darodipine (USAN/INN) (P) unclassified
D03656  Darunavir (USAN/INN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D03658  Dasatinib (JAN/INN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D03669  Deferasirox (JAN/USAN/INN); Exjade (TN); Jadenu (TN) (P) CYP inhibition: CYP1A2 / CYP induction: CYP3A4
D03689  Deracoxib (USAN) (P) unclassified
D03710  Etoricoxib (USAN/INN) (P) unclassified
D03712  Firocoxib (USAN/INN); Equioxx (TN) [veterinary] (P) unclassified
D03714  Lumiracoxib (USAN/INN) (P) unclassified
D03715  Dexibuprofen (USAN/INN) (P) unclassified
D03716  Parecoxib (USAN/INN) (P) unclassified
D03717  Parecoxib sodium (USAN); Dynastat (TN) (P) unclassified
D03718  Dexibuprofen lysine (USAN); Dexibuprofen lysine monohydrate; Doctrin (TN) (P) unclassified
D03727  Dexpemedolac (USAN/INN) (P) unclassified
D03729  Dexpropranolol hydrochloride (USAN) (P) unclassified
D03737  Dextofisopam (USAN/INN) (P) unclassified
D03759  Diacetolol hydrochloride (USAN) (P) unclassified
D03798  Dicumarol (USAN); Dicoumarol (INN) (P) unclassified
D03799  Dienogest (JAN/USAN/INN); Endometrion (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D03816  Tenivastatin calcium (USAN) (P) unclassified
D03820  Dutasteride (JAN/USP/INN); Avodart (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D03830  Diltiazem malate (USAN); Tiamate (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D03833  Indinavir (USAN); Indinavir hydrate (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D03835  Fosamprenavir calcium (USAN); Lexiva (TN); Telzir (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D03837  Fosamprenavir sodium (USAN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D03839  Droxinavir hydrochloride (USAN) (P) unclassified
D03840  Palinavir (USAN/INN) (P) unclassified
D03842  Telinavir (USAN/INN) (P) unclassified
D03843  Tipranavir disodium (USAN) (P) unclassified
D03844  Phenytoin, phenobarbital and caffeine and sodium benzoate; Hydantol F (TN) (P) Enzyme: CYP2C19 / CYP inhibition: CYP2C19 CYP2C9
D03846  Dimethyl fumarate (JAN/USAN); Tecfidera (TN) (P) unclassified
D03865  Dirithromycin (USP/INN); Dynabac (TN) (P) unclassified
D03883  Doconazole (USAN/INN) (P) unclassified
D03898  Doxofylline (USAN/INN); Maxivent (TN) (P) unclassified
D03914  Dronedarone hydrochloride (USP); Multaq (TN) (P) unclassified
D03936  Econazole (USAN/INN) (P) unclassified
D03940  Eculizumab (USAN/INN); Eculizumab (genetical recombination) (JAN); Eculizumab-aagh; Eculizumab-aeeb; Soliris (TN); Bkemv (TN); Epysqli (TN) (P) unclassified
D03959  Efalizumab (USAN/INN); Raptiva (TN) (P) unclassified
D03997  Enilconazole (USAN/INN) (P) unclassified
D04003  Enolicam sodium (USAN); Enolicam sodium monohydrate (P) unclassified
D04006  Enprofylline (USAN/INN) (P) unclassified
D04023  Erlotinib hydrochloride (JAN/USAN); Tarceva (TN) (P) Enzyme: CYP3A4 CYP1A2 / CYP inhibition: CYP1A2 CYP3A4
D04024  Lapatinib ditosylate (USAN); Lapatinib tosilate hydrate (JAN); Lapatinib ditosylate monohydrate; Tykerb (TN); Tyverb (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D04048  Ropivacaine hydrochloride (USP); Ropivacaine hydrochloride hydrate (JAN); Anapeine (TN) (P) Enzyme: CYP1A2 CYP3A4 / CYP inhibition: CYP1A2 CYP3A4
D04054  Erythromycin salnacedin (USAN); Erythromycin salnacedin dihydrate (P) unclassified
D04056  Esomeprazole sodium (USAN); Nexium IV (TN) (P) Enzyme: CYP2C19 / CYP inhibition: CYP2C19
D04102  Etofenamate (USAN/INN) (P) unclassified
D04105  Etoperidone hydrochloride (USAN); Etonin (TN) (P) unclassified
D04142  Fenclofenac (USAN/INN) (P) unclassified
D04144  Fenclorac (USAN/INN) (P) unclassified
D04145  Fendosal (USAN/INN); Alnovin (TN) (P) unclassified
D04147  Fenethylline hydrochloride (USAN) (P) unclassified
D04148  Fenfluramine hydrochloride (JAN/USAN); Fintepla (TN); Pondimin (TN) (P) Enzyme: CYP1A2 CYP2C19 CYP3A4 / CYP inhibition: CYP1A2 CYP3A4 CYP2D6 CYP2C19
D04187  Fingolimod hydrochloride (JAN/USAN); Gilenya (TN) (P) unclassified
D04190  Flestolol sulfate (USAN) (P) unclassified
D04193  Flordipine (USAN/INN) (P) unclassified
D04206  Flufenisal (USAN/INN) (P) unclassified
D04248  Fosazepam (USAN/INN) (P) unclassified
D04260  Fostedil (USAN/INN) (P) unclassified
D04273  Furaprofen (USAN/INN) (P) unclassified
D04277  Furobufen (USAN/INN) (P) unclassified
D04300  Ganaxolone (USAN/INN); Ztalmy (TN) (P) Enzyme: CYP3A4 CYP2C19 / CYP inhibition: CYP3A4 CYP2D6 CYP2C19
D04314  Gepirone hydrochloride (USAN); Exxua (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D04340  Dextromethorphan hydrobromide and potassium cresolsulfonate; Medicon (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 CYP2D6
D04358  Golimumab (USAN/INN); Golimumab (genetical recombination) (JAN); Golimumab (genetical recombination) [Golimumab biosimilar 1] (JAN); Simponi (TN) (P) unclassified
D04483  Ethinylestradiol and norethisterone; Norethindrone and ethinyl estradiol; Synphase T28 (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D04490  Ibuprofen aluminum (USAN) (P) CYP inhibition: CYP2C9
D04530  Indoprofen (USAN/INN) (P) unclassified
D04554  Interferon beta-1a (USAN); Interferon beta-1a (genetical recombination) (JAN); Avonex (TN); Rebif (TN) (P) unclassified
D04605  Iprindole (USAN/INN) (P) unclassified
D04624  Isoconazole (USAN/INN) (P) unclassified
D04638  Isoxepac (USAN/INN); Artil (TN) (P) unclassified
D04639  Isoxicam (USAN/INN); Maxicam (TN) (P) unclassified
D04641  Istradefylline (JAN/USAN/INN); Nourianz (TN); Nouriast (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D04650  Ketazolam (USAN/INN) (P) unclassified
D04657  Lacidipine (USAN/INN); Motens (TN) (P) unclassified
D04666  Lanreotide acetate (JAN/USAN); Somatuline (TN) (P) unclassified
D04687  Lenalidomide (JAN/USAN/INN); Revlimid (TN) (P) unclassified
D04693  Lergotrile (USAN/INN) (P) unclassified
D04694  Lergotrile mesylate (USAN) (P) unclassified
D04710  Levobetaxolol hydrochloride (USAN); Betaxon (TN) (P) unclassified
D04721  Levotofisopam (USAN/INN) (P) unclassified
D04725  Lexithromycin (USAN/INN) (P) unclassified
D04733  Lidoflazine (USAN/INN); Angex (TN) (P) unclassified
D04748  Lisofylline (USAN/INN); ProTec (TN) (P) unclassified
D04768  Lonafarnib (JAN/USAN/INN); Zokinvy (TN) (CI,P) CYP inhibition: CYP2C19
D04820  Lurasidone hydrochloride (JAN/USAN); SM 13496; Latuda (TN) (CI,P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D04863  Mavacoxib (USAN) (P) unclassified
D04882  Medazepam hydrochloride (USAN); Nobrium (TN) (P) unclassified
D04888  Medroxalol (USAN/INN) (P) unclassified
D04889  Medroxalol hydrochloride (USAN) (P) unclassified
D04896  Megalomicin potassium phosphate (USAN) (P) unclassified
D05011  Metoprolol fumarate (USP); Lopressor (TN) (P) CYP inhibition: CYP2D6
D05024  Mibefradil dihydrochloride (USAN); Posicor (TN) (P) CYP inhibition: CYP1A2
D05028  Midazolam maleate (USAN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D05039  Minaprine (USAN/INN); Cantor (TN) (P) CYP inhibition: CYP2D6
D05040  Minaprine hydrochloride (USAN) (P) CYP inhibition: CYP2D6
D05092  Muromonab-CD3 (JAN/USAN/INN); Orthoclone okt3 (TN) (P) unclassified
D05094  Mycophenolate mofetil hydrochloride (USAN); Cellcept (TN) (P) unclassified
D05095  Mycophenolate sodium (USP); Myfortic (TN) (P) unclassified
D05096  Mycophenolic acid (USAN/INN) (P) unclassified
D05121  Naproxol (USAN/INN) (P) unclassified
D05125  Naxifylline (USAN/INN) (P) unclassified
D05127  Nebivolol (USAN/INN) (P) CYP inhibition: CYP2D6
D05143  Nepafenac (JAN/USAN/INN); Nevanac (TN) (P) unclassified
D05153  Neutramycin (USAN) (P) unclassified
D05181  Aspirin aluminum (JP19) (P) unclassified
D05200  Nomifensine maleate (USAN); Merital (TN) (P) unclassified
D05218  Ocrelizumab (USAN); Ocrelizumab (genetical recombination) (JAN); Ocrevus (TN) (P) unclassified
D05259  Omeprazole magnesium (USP); Prilosec OTC (TN) (P) Enzyme: CYP2C19 / CYP inhibition: CYP2C19
D05261  Omeprazole sodium injection (JAN); Omeprazole sodium hydrate; Omepral (TN) (P) Enzyme: CYP2C19 / CYP inhibition: CYP2C19
D05268  Orconazole nitrate (USAN) (P) unclassified
D05319  Oxyphenbutazone hydrate; Tandearil (TN) (P) unclassified
D05345  Pamatolol sulfate (USAN) (P) unclassified
D05351  Josamycin propionate (JP19); Josamy (TN) (P) CYP inhibition: CYP3A4
D05353  Pantoprazole (USAN/INN) (P) Enzyme: CYP2C19 / CYP inhibition: CYP2C19
D05367  Parconazole hydrochloride (USAN) (P) unclassified
D05374  Paroxetine hydrochloride (USP); Paxil (TN) (P) CYP inhibition: CYP2D6
D05375  Paroxetine mesylate (USAN); Brisdelle (TN); Pexeva (TN) (P) CYP inhibition: CYP2D6
D05380  Pazopanib hydrochloride (JAN/USAN); Votrient (TN) (P) unclassified
D05404  Pemedolac (USAN/INN) (P) unclassified
D05429  Aminophylline hydrate (JP19) (P) Enzyme: CYP1A2 / CYP inhibition: CYP1A2
D05442  Perhexiline maleate (USAN) (P) CYP inhibition: CYP2D6
D05451  Phenbutazone sodium glycerate (USAN) (P) unclassified
D05457  Phenprocoumon (USAN/INN); Liquamar (TN) (P) unclassified
D05462  Oxycodone hydrochloride hydrate (JP19) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D05511  Piroxicam betadex (USAN) (P) CYP inhibition: CYP2C9
D05512  Piroxicam cinnamate (USAN) (P) CYP inhibition: CYP2C9
D05513  Piroxicam olamine (USAN) (P) CYP inhibition: CYP2C9
D05515  Pirprofen (USAN/INN) (P) unclassified
D05538  Mozenavir (INN) (P) unclassified
D05587  Practolol (USAN) (P) unclassified
D05598  Pravadoline maleate (USAN) (P) unclassified
D05619  Prodolic acid (USAN/INN) (P) unclassified
D05621  Progabide (USAN/INN); Gabren (TN) (P) unclassified
D05710  Reclazepam (USAN/INN) (P) unclassified
D05713  Relomycin (USAN/INN) (P) unclassified
D05717  Repromicin (USAN/INN) (P) unclassified
D05722  Revaprazan hydrochloride (USAN) (P) unclassified
D05757  Rosaramicin (USAN/INN) (P) unclassified
D05758  Rosaramicin butyrate (USAN) (P) unclassified
D05759  Rosaramicin propionate (USAN) (P) unclassified
D05760  Rosaramicin sodium phosphate (USAN) (P) unclassified
D05761  Rosaramicin stearate (USAN) (P) unclassified
D05775  Rufinamide (JAN/USP/INN); Banzel (TN) (P) unclassified
D05788  Salcolex (USAN); Salcolex tetrahydrate (P) unclassified
D05789  Salethamide maleate (USAN) (P) unclassified
D05791  Salicylate meglumine (USAN) (P) unclassified
D05793  Salnacedin (USAN/INN) (P) unclassified
D05800  Saperconazole (USAN/INN) (P) unclassified
D05811  Sedecamycin (USAN/INN) (P) unclassified
D05829  Sergolexole maleate (USAN) (P) unclassified
D05830  Sermetacin (USAN/INN) (P) unclassified
D05900  Timoprazole (INN) (P) unclassified
D05901  Picoprazole (INN) (P) unclassified
D05906  Leminoprazole (INN) (P) unclassified
D05908  Spiramycin (JAN/USAN/INN); Rovamycin (TN) (P) unclassified
D05928  Stiripentol (JAN/USAN/INN); Diacomit (TN) (P) Enzyme: CYP1A2 CYP2C19 CYP3A4 / CYP inhibition: CYP1A2 CYP3A4 CYP2C19
D05937  Sudoxicam (USAN/INN) (P) unclassified
D05942  Sulazepam (USAN/INN) (P) unclassified
D05995  Talmetacin (USAN/INN) (P) unclassified
D05998  Talosalate (USAN/INN) (P) unclassified
D06012  Tazifylline hydrochloride (USAN) (P) unclassified
D06060  Teludipine hydrochloride (USAN) (P) unclassified
D06068  Temsirolimus (JAN/USAN/INN); Torisel (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D06082  Tesicam (USAN) (P) unclassified
D06103  Theophylline (USP); Theophylline monohydrate; Accurbron (TN) (P) Enzyme: CYP1A2 / CYP inhibition: CYP1A2
D06104  Theophylline sodium glycinate (USP); Asbron (TN) (P) Enzyme: CYP1A2 / CYP inhibition: CYP1A2
D06143  Tifurac sodium (USAN) (P) unclassified
D06156  Tiopinac (USAN/INN) (P) unclassified
D06199  Trabectedin (JAN/USAN/INN); Yondelis (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D06231  Triflubazam (USAN/INN) (P) unclassified
D06258  Tulathromycin (JAN/USAN/INN) (P) unclassified
D06273  Imidafenacin (JAN/INN); Uritos (TN); Staybla (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D06291  Verofylline (USAN/INN) (P) unclassified
D06315  Fluticasone furoate (JAN/USAN/INN); Veramyst (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D06334  Xanthinol niacinate (USAN); Xantinol nicotinate; Complamin (TN) (P) unclassified
D06363  Ziconotide (USAN/INN); Prialt (TN) (P) unclassified
D06364  Zidometacin (USAN/INN) (P) unclassified
D06367  Zimeldine hydrochloride (USAN); Zimeldine hydrochloride hydrate (P) unclassified
D06373  Zinoconazole hydrochloride (USAN) (P) unclassified
D06382  Zomepirac sodium (USAN); Zomepirac sodium dihydrate (P) unclassified
D06390  Azithromycin (USP); Zmax (TN) (P) unclassified
D06402  Sunitinib malate (JAN/USAN); Sutent (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D06405  Nalfurafine hydrochloride (JAN/USAN); Remitch (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D06413  Nilotinib hydrochloride hydrate (JAN); Nilotinib monohydrochloride monohydrate; Tasigna (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D06414  Dasatinib (USAN); Dasatinib hydrate (JAN); Sprycel (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D06478  Darunavir ethanolate (JAN); Prezista (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D06573  Carisbamate (USAN) (P) unclassified
D06597  Fosaprepitant dimeglumine (USAN); Fosaprepitant meglumine (JAN); Proemend (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D06598  Gamithromycin (USAN/INN) (P) unclassified
D06606  Ibuprofen lysine (USAN); Ibuprofen L-lysine (JAN); Solufenum; Neoprofen (TN) (P) CYP inhibition: CYP2C9
D06622  Nebivolol hydrochloride (USAN); Bystolic (TN) (P) CYP inhibition: CYP2D6
D06630  Pramiconazole (USAN/INN) (P) unclassified
D06635  Rilonacept (USAN/INN); Arcalyst (TN) (P) unclassified
D06637  Romidepsin (JAN/USAN/INN); Istodax (TN) (P) unclassified
D06646  Epanolol (USAN/INN) (P) unclassified
D06883  Sertaconazole (INN) (P) unclassified
D06886  Natalizumab (USAN/INN); Natalizumab (genetical recombination) (JAN); Natalizumab-sztn; Tysabri (TN); Tyruko (TN) (P) unclassified
D07062  Acefylline piperazine (INN); Epicophylline (TN) (P) unclassified
D07064  Acenocoumarol (INN); Acenocoumarin; Mini-sintrom (TN) (P) unclassified
D07131  Ethyl biscoumacetate (INN) (P) unclassified
D07135  Clorindione (INN); G-25766 (P) unclassified
D07136  Diphenadione (INN) (P) unclassified
D07137  Tioclomarol (INN) (P) unclassified
D07139  Cloricromen (INN) (P) unclassified
D07141  Indobufen (INN) (P) unclassified
D07151  Cafedrine (BAN) (P) unclassified
D07155  Theodrenaline (INN) (P) unclassified
D07156  Alprenolol (INN) (P) CYP inhibition: CYP2D6
D07174  Pentifylline (INN) (P) unclassified
D07181  Mepindolol (INN) (P) unclassified
D07182  Tertatolol (INN) (P) unclassified
D07183  Cloranolol (INN) (P) unclassified
D07184  Talinolol (INN) (P) unclassified
D07185  Fendiline (INN) (P) unclassified
D07193  Flutrimazole (INN) (P) unclassified
D07217  Quinagolide (INN/BAN) (P) unclassified
D07218  Metergoline (INN) (P) unclassified
D07219  Flunoxaprofen (INN) (P) unclassified
D07242  Flurithromycin (INN) (P) unclassified
D07262  Mofebutazone (INN); Monazone (TN) (P) unclassified
D07263  Clofezone (JAN/INN); Clofezone dihydrate (P) unclassified
D07264  Bumadizone (INN) (P) unclassified
D07265  Lonazolac (INN) (P) unclassified
D07266  Oxametacin (INN) (P) unclassified
D07267  Droxicam (INN) (P) unclassified
D07268  Ibuproxam (INN); Ibudros (TN) (P) unclassified
D07269  Dexketoprofen (INN) (P) unclassified
D07283  Esketamine (USAN/INN) (P) Enzyme: CYP2C19 CYP3A4 / CYP inhibition: CYP3A4 CYP2C19
D07290  Dipyrocetyl (INN) (P) unclassified
D07291  Benorilate (INN); Benorylate (P) unclassified
D07292  Guacetisal (INN); Prontomucil (TN) (P) unclassified
D07293  Imidazole salicylate (INN); Selezen (TN) (P) unclassified
D07298  Barbexaclone (INN); Maliasin (TN) (P) unclassified
D07299  Lacosamide (JAN/USAN/INN); Erlosamide; Vimpat (TN) (P) Enzyme: CYP2C19 CYP3A4 / CYP inhibition: CYP3A4 CYP2C19 CYP2C9
D07300  Beclamide (INN) (P) unclassified
D07314  Pinazepam (INN); Domar (TN) (P) unclassified
D07315  Camazepam (INN) (P) unclassified
D07326  Loprazolam (INN); Dormonoct (TN) (P) unclassified
D07327  Doxefazepam (INN) (P) unclassified
D07328  Cinolazepam (INN); Gerodorm (TN) (P) unclassified
D07335  Amineptine (INN); Survector (TN) (P) unclassified
D07336  Quinupramine (INN) (P) unclassified
D07337  Nialamide (INN); Niamid (TN) (P) unclassified
D07338  Iproclozide (INN) (P) unclassified
D07339  Oxitriptan (INN); Levothym (TN) (P) unclassified
D07340  Oxaflozane (INN) (P) unclassified
D07341  Medifoxamine (INN) (P) unclassified
D07342  Pivagabine (INN) (P) unclassified
D07378  Etamiphylline (INN) (P) unclassified
D07421  Aloxiprin (INN); Superpyrin (TN) (P) unclassified
D07436  Afelimomab (INN) (P) unclassified
D07443  Amfenac (INN) (P) unclassified
D07448  Amitriptyline (INN); Laroxyl (TN) (P) Enzyme: CYP2C19 CYP3A4 / CYP inhibition: CYP3A4 CYP2D6 CYP2C19
D07450  Amlodipine (USP/INN); Norvasc (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D07453  Amtolmetin guacil (INN); Artromed (TN) (P) unclassified
D07457  Anisindione (INN); Miradon (TN) (P) unclassified
D07471  Atazanavir (INN); Reyataz (TN) (P) CYP inhibition: CYP3A4
D07474  Atorvastatin (INN); Lipitor (TN); Sortis (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D07486  Azithromycin (INN); Azasite (TN) (P) unclassified
D07488  Balsalazide (INN) (P) unclassified
D07491  Bamifylline (INN) (P) unclassified
D07494  Barnidipine (INN); Vasexten (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D07496  Befunolol (INN) (P) unclassified
D07503  Bendazac lysine (BAN); Bendalina (TN) (P) unclassified
D07505  Latanoprost and timolol maleate; Xalacom (TN) (P) unclassified
D07509  Benidipine (INN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D07516  Benzydamine (INN) (P) unclassified
D07517  Benzydamine salicylate; Fulgium (TN) (P) unclassified
D07520  Bepridil (INN); Bepadin (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 CYP2D6 CYP2C9
D07523  Betaine (JAN); Cystadane (TN) (P) unclassified
D07526  Betaxolol (INN) (P) unclassified
D07528  Bifemelane (INN) (P) unclassified
D07537  Bopindolol (INN); Sandonorm (TN) (P) CYP inhibition: CYP2D6
D07541  Bromfenac (INN) (P) unclassified
D07545  Brovincamine (INN); Sarbromin (TN) (P) unclassified
D07549  Bumadizone calcium salt hemihydrate; Desflam (TN); Eumotol (TN) (P) unclassified
D07569  Candesartan cilexetil and anmlodipine besylate (JP19); Unisia (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D07579  Aspirin calcium salt; Notras (TN) (P) unclassified
D07580  Aspirin DL-lysine (JAN); Aspirin lysine salt; Aspegic (TN) (P) unclassified
D07581  Aspirin magnesium salt; Mobidin (TN) (P) unclassified
D07582  Aspirin sodium; Sodium acetylsalicylate; Catalgine (TN) (P) unclassified
D07583  Phenytoin and phenobarbital; Aleviatin with phenobarbital (TN) (P) CYP inhibition: CYP2C9
D07585  Isopropylantipyrine, ergotamine tartrate and anhydrous caffeine; Cleamine A (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D07590  Bupranolol (INN) (P) unclassified
D07591  Bupropion (INN) (P) unclassified
D07595  Fosphenytoin sodium hydrate (JAN); Fostoin (TN) (P) CYP inhibition: CYP2C9 / CYP induction: CYP3A4
D07598  Butoconazole (INN); Gynofort (TN) (P) unclassified
D07601  Butriptyline (INN); Evadyne (TN) (P) unclassified
D07603  Caffeine citrate (USP); Cafcit (TN) (P) Enzyme: CYP1A2 / CYP inhibition: CYP1A2
D07608  Carazolol (INN); Conducton (TN); Suacron [veterinary] (TN) (P) unclassified
D07612  Sodium salamidacetate; o-Carbamoylphenoxyacetic acid sodium salt; Clinit-n (TN) (P) unclassified
D07624  Carteolol (INN) (P) CYP inhibition: CYP2D6
D07660  Celiprolol (INN) (P) unclassified
D07661  Cerivastatin (INN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D07676  Chlormidazole hydrochloride; Unfungicid (TN) (P) unclassified
D07704  Citalopram (USP/INN); Citadur (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 CYP2D6 CYP2C19
D07705  Citalopram hydrochloride; Seropram (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 CYP2D6 CYP2C19
D07710  Clarithromycin lactobionate; Klacid (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D07714  Climazolam (INN); Climasol [veterinary] (TN) (P) unclassified
D07727  Clomipramine (INN); Anafranil (TN) (P) Enzyme: CYP2C19 CYP3A4 / CYP inhibition: CYP3A4 CYP2D6 CYP2C19
D07736  Cloricromen hydrohloride; Proendotel (TN) (P) unclassified
D07752  Croconazole (INN) (P) unclassified
D07784  Delorazepam (INN); Dadumir (TN) (P) unclassified
D07791  Desipramine (INN) (P) unclassified
D07793  Desvenlafaxine (INN); Khedezla (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D07812  Dibenzepin (INN) (P) unclassified
D07816  Diclofenac (USAN/INN); Solaraze (TN); Zorvolex (TN) (P) CYP inhibition: CYP2C9
D07817  Diclofenac diethylamine; Voltaren Emulgel (TN) (P) CYP inhibition: CYP2C9
D07818  Diclofenac epolamine; Diclofenac hydroxyethylpyrrolidine; Flector (TN) (P) CYP inhibition: CYP2C9
D07819  Diclofenac calcium; Voltaren Actingo Extra (TN) (P) CYP inhibition: CYP2C9
D07824  Diethylamine salicylate; Algesal (TN) (P) unclassified
D07833  Dihydroergocristine mesilate (BAN); Diertine (TN) (P) unclassified
D07834  Dihydroergocristine (BAN) (P) unclassified
D07835  Dihydroergocryptine (P) unclassified
D07836  Dihydroergocryptine mesilate; Almirid (TN) (P) unclassified
D07837  Dihydroergotamine (INN); Neomigran (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D07838  Dihydroergotamine tartrate; Divegal (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D07839  Dihydroergotoxine; Co-Dergocrin (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D07845  Diltiazem (INN); Surazem (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D07862  Diphenylpyraline (INN) (P) unclassified
D07869  Donepezil (JAN/INN); Donaz (TN); Allydone (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D07872  Dosulepin (INN); Dothiepin; Dothep (TN) (P) CYP inhibition: CYP2D6
D07875  Doxepin (INN); Sinequan (TN) (P) Enzyme: CYP2C19 / CYP inhibition: CYP2D6 CYP2C19 CYP2C9
D07880  Duloxetine (INN); Yentreve (TN) (P) Enzyme: CYP1A2 / CYP inhibition: CYP1A2
D07882  Eberconazole (INN) (P) unclassified
D07884  Eberconazole nitrate; Ebernet (TN) (P) unclassified
D07886  Efonidipine (INN) (P) unclassified
D07888  Eltenac (INN); Telzenac (TN) (P) unclassified
D07905  Ergometrine (INN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D07906  Ergotamine (INN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D07909  Erythromycin thiocyanate; Erythrocin (TN) (P) unclassified
D07910  Erythromycin stinoprate (INN); Erysec (TN) (P) unclassified
D07913  Escitalopram (INN); Esertia (TN) (P) Enzyme: CYP2C19 CYP3A4 / CYP inhibition: CYP3A4 CYP2D6 CYP2C19
D07916  Esmolol (INN) (P) unclassified
D07917  Esomeprazole (INN); Inexium paranova (TN) (P) Enzyme: CYP2C19 / CYP inhibition: CYP2C19
D07923  Etamiphylline hydrochloride; Solufilina (TN) (P) unclassified
D07933  Etofylline (INN); Oxyphyllin (TN) (P) unclassified
D07938  Bupropion hydrobromide (USAN); Aplenzin (TN) (P) unclassified
D07943  Fendiline hydrochloride; Sensit (TN) (P) unclassified
D07944  Fenetylline (INN); Fenethylline; Fitton (TN) (P) unclassified
D07945  Fenfluramine (INN); Ponderax (TN) (P) Enzyme: CYP1A2 CYP2C19 CYP3A4 / CYP inhibition: CYP1A2 CYP3A4 CYP2D6 CYP2C19
D07969  Fluindione (INN); Previsccan (TN) (P) unclassified
D07971  Flunarizine (INN); Sibelium (TN) (P) CYP inhibition: CYP2D6
D07983  Fluvastatin (INN); Fluvas (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 CYP2C9
D07984  Fluvoxamine (INN) (P) CYP inhibition: CYP2D6 CYP1A2 CYP2C19 CYP3A4
D07991  Fosfosal (INN); Aydolid (TN) (P) unclassified
D07993  Fosphenytoin (INN) (P) CYP inhibition: CYP2C9 / CYP induction: CYP3A4
D08009  Gallopamil (INN) (P) unclassified
D08021  Glucametacin (INN); Glucametan (TN) (P) unclassified
D08032  Gusperimus (INN); 15-Deoxyspergualin (P) unclassified
D08035  Haloperidol lactate; Haldol (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 CYP2D6
D08058  Ibuprofen arginine salt; Zafen (TN) (P) CYP inhibition: CYP2C9
D08059  Ibuprofen sodium; Ibuprofen sodium anhydrous; Esprenit (TN) (P) CYP inhibition: CYP2C9
D08070  Imipramine (INN); Tofranil (TN) (P) Enzyme: CYP2C19 CYP3A4 / CYP inhibition: CYP3A4 CYP2D6 CYP2C19
D08071  Imipramine pamoate (USP); Imipramine embonate; Tofranil-pm (TN) (P) Enzyme: CYP2C19 CYP3A4 / CYP inhibition: CYP3A4 CYP2D6 CYP2C19
D08074  Penbutolol (INN) (P) unclassified
D08078  Indenolol (INN) (P) unclassified
D08083  Vedolizumab (USAN); Vedolizumab (genetical recombination) (JAN); Entyvio (TN) (P) unclassified
D08085  Iproniazid phosphate; Marsilid (TN) (P) unclassified
D08095  Ivabradine hydrochloride (JAN/USAN); Ivabrandine hydrochloride; Corlanor (TN); Corlentor (TN); Coralan (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D08102  Ketoprofen lysine; Artrosilene (TN) (P) unclassified
D08103  Ketoprofen sodium; Orudis (TN) (P) unclassified
D08104  Ketorolac (INN); Toradol (TN) (P) unclassified
D08111  Lercanidipine (INN); Lercanil (TN) (P) unclassified
D08115  Levobunolol (INN) (P) unclassified
D08132  Lisuride (INN) (P) unclassified
D08140  Lofepramine (INN) (P) unclassified
D08142  Lonazolac calcium salt; Argun (TN) (P) unclassified
D08145  Loprazolam mesilate; Loprazolam mesylate; Loprazolam methanesulfonate; Havlane (TN) (P) unclassified
D08149  Loxoprofen (INN) (P) unclassified
D08153  Mabuprofen (INN); Aldospray analgesico (TN) (P) unclassified
D08155  Manidipine (INN); Manidipine 6300; Artedil (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D08162  Meclofenamate sodium; Meclomen (TN) (P) unclassified
D08170  Melatonin (JAN); Melatonina (TN); Melatobel (TN) (P) Enzyme: CYP1A2 / CYP inhibition: CYP1A2
D08171  Melitracen (INN); Adelax (TN) (P) unclassified
D08190  Dipyrone (BAN); Metamizole sodium; Vetalgin (TN) (P) unclassified
D08207  Methylergometrine (INN); Ergotyl (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D08216  Mianserin (INN); Tolvon (TN) (P) Enzyme: CYP1A2 CYP3A4 / CYP inhibition: CYP1A2 CYP3A4 CYP2D6
D08217  Mibefradil (INN) (P) CYP inhibition: CYP1A2
D08222  Milnacipran (INN) (P) unclassified
D08257  Nefazodone (INN) (P) unclassified
D08259  Nelfinavir (INN); Viracept (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D08270  Nicardipine (INN); Cardene (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D08271  Nicergoline tartrate; Sermion (TN) (P) unclassified
D08275  Niflumic acid (INN); Niflugel (TN) (P) unclassified
D08283  Nordazepam (INN); Calmday (TN) (P) Enzyme: CYP2C19 CYP3A4 / CYP inhibition: CYP3A4 CYP2C19
D08288  Nortriptyline (INN); Nortrilen (TN) (P) CYP inhibition: CYP2D6
D08295  Olsalazine (INN) (P) unclassified
D08296  Omoconazole (INN) (P) unclassified
D08297  Opipramol (INN) (P) unclassified
D08313  Oxiconazole (INN) (P) unclassified
D08318  Oxprenolol (INN) (P) unclassified
D08324  Oxyphenbutazone (INN); Reozon (TN) (P) unclassified
D08339  Pergolide (INN); Permax (TN) (P) unclassified
D08340  Perhexiline (INN) (P) CYP inhibition: CYP2D6
D08349  Phenelzine (BAN) (P) unclassified
D08354  Phenindione (INN); Hedulin (TN) (P) unclassified
D08356  Phenobarbital diethylamine; Gratusminal (TN) (P) unclassified
D08363  Phenylbutazone calcium; Peralgin (TN) (P) unclassified
D08364  Phenylbutazone sodium; Ambene (TN) (P) unclassified
D08374  Piketoprofen (INN); Calmatel (TN) (P) unclassified
D08375  Piketoprofen hydrochloride; Triparsean (TN) (P) unclassified
D08410  Pravastatin (INN); Pravator (TN) (P) unclassified
D08427  Proglumetacin (INN); Bruxel (TN) (P) unclassified
D08443  Propranolol (INN) (P) Enzyme: CYP1A2 CYP2C19 / CYP inhibition: CYP1A2 CYP2D6 CYP2C19
D08447  Protriptyline (INN) (P) unclassified
D08457  Quinagolide hydrochloride (BAN); Norprolac (TN) (P) unclassified
D08463  Rabeprazole (INN); Eraloc (TN) (P) Enzyme: CYP2C19 CYP3A4 / CYP inhibition: CYP3A4 CYP2C19
D08472  Reboxetine (INN); Edronax (TN) (P) unclassified
D08481  Rilmazafone (INN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D08488  Amlodipine besilate and atorvastatin calcium; Caduet (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D08492  Rosuvastatin (INN); Creston (TN) (P) unclassified
D08493  Dorzolamide hydrochloride and timolol maleate (JP19); Cosopt (TN) (P) Enzyme: CYP2C19 CYP3A4 / CYP inhibition: CYP3A4 CYP2D6 CYP2C19 CYP2C9
D08497  Rupatadine fumarate (JAN/USAN); Rinialer (TN); Rupafin (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D08501  Trolamine salicylate (USP); Salicylic acid trolamine; Salicylic acid triethanolamine; Arthricream (TN) (P) unclassified
D08510  Sertaconazole nitrate; Ertaczo (TN); Zalain (TN) (P) unclassified
D08525  Sotalol (INN); Darob mite (TN) (P) unclassified
D08527  Spiramycin adipate; Rovamycina (TN); Spiramaicina (TN) (P) unclassified
D08528  Spiramycin embonate; Cofamix STS (TN) (P) unclassified
D08535  Sulconazole (INN) (P) unclassified
D08556  Tacrolimus (INN); Prograf (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D08572  Tertatolol hydrochloride; Artex (TN) (P) unclassified
D08575  Tetrabenazine (JAN/INN); Nitoman (TN); Xenazine (TN) (P) Enzyme: CYP1A2 / CYP inhibition: CYP1A2 CYP2D6
D08586  Thiosalicylic acid; Pirosal (TN); Thiocyl (TN) (P) unclassified
D08588  Tiagabine (INN); Gabitril (TN) (P) unclassified
D08589  Tianeptine sodium; Stablon (TN) (P) unclassified
D08592  Tiaramide (INN) (P) unclassified
D08598  Tilisolol (INN) (P) unclassified
D08600  Timolol (INN); Betimol (TN) (P) CYP inhibition: CYP2D6
D08605  Tipranavir (INN); Aptivus (TN) (P) unclassified
D08625  Tranylcypromine (INN); Parnate (TN) (P) unclassified
D08626  Trazodone (INN); Trittico (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 CYP2D6
D08630  Tribuzone (prop.INN); Benetazon (TN) (P) unclassified
D08657  Apricoxib (USAN/INN) (P) unclassified
D08667  Calcium valproate; Valproic acid calcium salt; Convulsofin (TN) (P) unclassified
D08670  Venlafaxine (INN); Efectin (TN) (P) CYP inhibition: CYP2D6
D08673  Viloxazine (INN) (P) CYP inhibition: CYP2D6
D08682  Warfarin (INN); Warfarine; Choice (TN) (P) CYP inhibition: CYP2C9
D08686  Ziconotide acetate; Prialt (TN) (P) unclassified
D08699  Salmeterol xinafoate and fluticasone propionate; Adoair diskus (TN); Aerivio Spiromax (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D08856  Anamorelin hydrochloride (JAN/USAN); Adlumiz (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D08860  Apremilast (JAN/USAN); Otezla (TN) (P) unclassified
D08879  Brivaracetam (JAN/USAN/INN); Briviact (TN) (P) Enzyme: CYP2C19 / CYP inhibition: CYP2C19
D08892  Clevidipine (USAN/INN); Clevidipine butyrate; Cleviprex (TN) (P) unclassified
D08903  Dexlansoprazole (INN/USAN); Dexilant (TN) (P) Enzyme: CYP2C19 CYP3A4 / CYP inhibition: CYP3A4 CYP2C19
D08923  Fesoterodine fumarate (JAN/USAN); Toviaz (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 CYP2D6
D08962  Pamabrom (USP) (P) unclassified
D08964  Perampanel (JAN/USAN); Fycompa (TN) (P) unclassified
D08976  Pomalidomide (JAN/USAN/INN); Pomalyst (TN) (P) Enzyme: CYP1A2 CYP3A4 / CYP inhibition: CYP1A2 CYP3A4
D08989  Rolofylline (USAN) (P) unclassified
D09017  Ticagrelor (JAN/USAN/INN); Brilinta (TN) (CI,P) unclassified
D09033  Voclosporin (JAN/USAN/INN); Lupkynis (TN) (CI,P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D09188  Estradiol and norethindrone; Menoaid (TN); Activella (TN); Combipatch (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D09190  Anti-human thymocyte immunoglobulin, rabbit (JAN); Thymoglobuline (TN) (P) unclassified
D09214  Ustekinumab (USAN/INN); Ustekinumab (genetical recombination) (JAN); Ustekinumab (genetical recombination) [Ustekinumab biosimilar 1] (JAN); Ustekinumab (genetical recombination) [Ustekinumab biosimilar 2] (JAN); Ustekinumab (genetical recombination) [Ustekinumab biosimilar 3] (JAN); Ustekinumab (genetical recombination) [Ustekinumab biosimilar 4] (JAN); Ustekinumab-aauz; Ustekinumab-auub; Ustekinumab-ttwe; Ustekinumab-aekn; Ustekinumab-srlf; Ustekinumab-hmny; Stelara (TN); Otulfi (TN); Pyzchiva (TN); Wezlana (TN) (P) unclassified
D09215  Eslicarbazepine (USAN/INN) (P) CYP inhibition: CYP2C19 / CYP induction: CYP3A4
D09314  Ofatumumab (USAN/INN); Ofatumumab (genetical recombination) (JAN); Arzerra (TN); Kesimpta (TN) (P) unclassified
D09315  Canakinumab (USAN/INN); Canakinumab (genetical recombination) (JAN); Ilaris (TN) (P) unclassified
D09319  Indacaterol maleate (JAN/USAN); Arcapta (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D09339  Esomeprazole potassium (USAN) (P) Enzyme: CYP2C19 / CYP inhibition: CYP2C19
D09348  Fostamatinib disodium (USAN); Fostamatinib sodium hydrate (JAN); Fostamatinib disodium hexahydrate; Tavalisse (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D09365  Palovarotene (JAN/USAN/INN); Sohonos (TN) (CI,P) Enzyme: CYP2C19 CYP3A4 / CYP inhibition: CYP3A4 CYP2C19
D09394  Fidaxomicin (JAN/USAN); Dificid (TN); Dificlir (TN) (P) CYP inhibition: CYP2C19 CYP3A4
D09568  Naproxcinod (USAN/INN) (P) unclassified
D09569  Ezogabine (USAN); Retigabine (INN); Potiga (TN) (P) unclassified
D09572  Riociguat (JAN/USAN/INN); Adempas (TN) (P) unclassified
D09587  Brentuximab vedotin (USAN/INN); Brentuximab vedotin (genetical recombination) (JAN); Adcetris (TN) (P) unclassified
D09588  Briakinumab (USAN/INN) (P) unclassified
D09595  Budesonide and formoterol fumarate dihydrate; Symbicort (TN); Budeforu (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D09612  Eslicarbazepine acetate (USAN); Zebinix (TN); Aptiom (TN) (P) CYP inhibition: CYP2C19 / CYP induction: CYP3A4
D09638  Lomitapide mesylate (USAN); Lomitapide mesilate (JAN); Juxtapid (TN); Lojuxta (TN) (CI,P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D09642  Modithromycin (USAN/INN) (P) unclassified
D09669  Siltuximab (USAN/INN); Sylvant (TN) (P) unclassified
D09676  Tecarfarin (USAN/INN) (P) unclassified
D09677  Tecarfarin sodium (USAN) (P) unclassified
D09680  Teprotumumab (USAN/INN); Teprotumumab (genetical recombination) (JAN); Teprotumumab-trbw; Tepezza (TN) (P) unclassified
D09684  Tonapofylline (USAN/INN) (P) unclassified
D09698  Vilazodone (USAN/INN) (P) Enzyme: CYP2C19 CYP3A4 / CYP inhibition: CYP3A4 CYP2C19
D09699  Vilazodone hydrochloride (USAN); Viibryd (TN) (P) Enzyme: CYP2C19 CYP3A4 / CYP inhibition: CYP3A4 CYP2C19
D09702  Albaconazole (USAN/INN) (P) unclassified
D09728  Bosutinib hydrate (JAN); Bosutinib monohydrate; Bosulif (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D09730  Olaparib (JAN/USAN/INN); Lynparza (TN) (P) unclassified
D09731  Crizotinib (JAN/USAN/INN); Xalkori (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D09743  Telmisartan and amlodipine besilate (JP19); Telmisartan and amlodipine besylate; Micamlo (TN); Twynsta (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D09745  Valsartan and amlodipine besilate; Exforge (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D09753  Saxagliptin hydrate (JAN); Onglyza (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D09760  Ibuprofen sodium (USAN); Ibuprofen sodium hydrate (P) CYP inhibition: CYP2C9
D09783  Tofacitinib citrate (JAN/USAN); Tasocitinib citrate; Xeljanz (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D09789  Kirenidipine hydrochloride (JAN) (P) unclassified
D09799  Carotegrast methyl (JAN); Carogra (TN) (P) CYP inhibition: CYP3A4
D09807  Difethiarol (JAN); Difethialone (P) unclassified
D09809  Tylosin acetate isovalerte (JAN) (P) unclassified
D09813  Lenalidomide hydrate (JAN); Revlimid (TN) (P) unclassified
D09815  Travoprost and timolol maleate; Duotrav (TN) (P) unclassified
D09837  Penaprazole sodium hydrate (JAN) (P) unclassified
D09843  Beradilol monoethyl maleate (JAN); TZC-5665 (P) unclassified
D09894  Eliglustat tartrate (JAN/USAN); Eliglustat hemitartrate; Cerdelga (TN) (CI,P) CYP inhibition: CYP2D6
D09951  Ponatinib hydrochloride (JAN/USAN); Iclusig (TN) (P) unclassified
D09956  Quizartinib dihydrochloride (USAN); Quizartinib hydrochloride (JAN); Vanflyta (TN) (P) unclassified
D09960  Ruxolitinib phosphate (JAN/USAN); Jakafi (TN); Jakavi (TN); Opzelura (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D09967  Secukinumab (USAN/INN); Secukinumab (genetical recombination) (JAN); Cosentyx (TN) (P) unclassified
D09970  Tofacitinib (USAN); Tasocitinib (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D09996  Vemurafenib (JAN/USAN/INN); Zelboraf (TN) (P) CYP inhibition: CYP1A2 / CYP induction: CYP3A4
D10001  Fingolimod (INN); Gilenya (TN) (P) unclassified
D10003  Hemin (JAN); Normosang (TN); Panhematin (TN) (P) CYP induction: CYP3A4
D10017  Naproxen etemesil (USAN) (P) unclassified
D10021  Efinaconazole (JAN/USAN/INN); Clenafin (TN); Jublia (TN) (P) unclassified
D10024  Selumetinib sulfate (JAN/USAN); Koselugo (TN) (P) Enzyme: CYP1A2 CYP3A4 / CYP inhibition: CYP1A2 CYP3A4 CYP2C9
D10032  Tylvalosin (USAN/INN) (P) unclassified
D10033  Tylosin tartrate (USP) (P) unclassified
D10034  Tylvalosin tartrate (USAN); Aiviosin [veterinary] (TN) (P) unclassified
D10061  Brodalumab (USAN); Brodalumab (genetical recombination) (JAN); Siliq (TN) (P) unclassified
D10071  Ixekizumab (USAN); Ixekizumab (genetical recombination) (JAN); Taltz (TN) (P) unclassified
D10072  Levomilnacipran (USAN/INN) (P) unclassified
D10080  Sirukumab (USAN); Sirukumab (genetical recombination) (JAN) (P) unclassified
D10082  Suvorexant (JAN/USAN); MK-4305; Belsomra (TN) (P) unclassified
D10095  Cabozantinib s-malate (USAN); Cabozantinib malate (JAN); Cometriq (TN); Cabometyx (TN) (P) unclassified
D10104  Dabrafenib mesylate (USAN); Dabrafenib mesilate (JAN); Tafinlar (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D10120  Esomeprazole strontium (USAN); Esomeprazole strontium tetrahydrate (P) Enzyme: CYP2C19 / CYP inhibition: CYP2C19
D10127  Glycerol phenylbutyrate (JAN/USAN); Ravicti (TN) (P) unclassified
D10133  Levomilnacipran hydrochloride (USAN); Fetzima (TN) (P) unclassified
D10135  Macitentan (JAN/USAN); Opsumit (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D10137  Regorafenib hydrate (JAN); Stivarga (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D10161  Sarilumab (USAN); Sarilumab (genetical receombination) (JAN); Kevzara (TN) (P) unclassified
D10172  Teriflunomide (USAN); Aubagio (TN) (P) unclassified
D10184  Vortioxetine (USAN); Brintellix (TN) (P) Enzyme: CYP2C19 / CYP inhibition: CYP2D6 CYP2C19 CYP2C9
D10185  Vortioxetine hydrobromide (JAN/USAN); Brintellix (TN); Trintellix (TN) (P) Enzyme: CYP2C19 / CYP inhibition: CYP2D6 CYP2C19 CYP2C9
D10218  Enzalutamide (JAN/USAN); Xtandi (TN) (P) unclassified
D10223  Ibrutinib (JAN/USAN); Imbruvica (TN) (P) unclassified
D10243  Irbesartan and amlodipine besilate (JP19); Aimix (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D10254  Esflurbiprofen (JAN/USAN) (P) CYP inhibition: CYP2C9
D10298  Brimonidine tartrate and timolol maleate; Combigan (TN); Aibeta (TN) (P) unclassified
D10307  Avatrombopag maleate (JAN/USAN); Doptelet (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 CYP2C9
D10308  Baricitinib (JAN/USAN/INN); Olumiant (TN) (P) unclassified
D10309  Brexpiprazole (JAN/USAN/INN); Rexulti (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 CYP2D6
D10372  Palbociclib (JAN/USAN); Ibrance (TN) (P) unclassified
D10400  Tildrakizumab (USAN); Tildrakizumab (genetical recombination) (JAN); Tildrakizumab-asmn; Ilumya (TN) (P) unclassified
D10438  Guselkumab (USAN/INN); Guselkumab (genetical recombination) (JAN); Tremfya (TN) (P) unclassified
D10450  Alectinib hydrochloride (JAN); Alecensa (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D10452  Cabazitaxel acetonate (JAN); Cabazitaxel acetone; Jevtana (TN) (P) unclassified
D10466  Vonoprazan fumarate (JAN/USAN); Takecab (TN); Voquezna (TN) (P) Enzyme: CYP2C19 CYP3A4 / CYP inhibition: CYP3A4 CYP2D6 CYP2C19
D10478  Naldemedine tosylate (JAN/USAN); Naldemedine tosilate; Symproic (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D10492  Tildipirosin (USAN/INN); Zuprevo [veterinary] (TN) (P) unclassified
D10501  Fluticasone furoate and vilanterol trifenatate; Breo ellipta (TN); Relvar ellipita (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D10505  Glycopyrronium bromide and indacaterol maleate; Ultibro (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D10506  Fluticasone propionate and formoterol fumarate hydrate; Flutiform (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D10512  Brinzolamide and timolol maleate; Azorga (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 CYP2D6 CYP2C9
D10513  Clopidogrel sulfate and aspirin; Clopidogrel and acetylsalicyclic acid; Complavin (TN) (P) Enzyme: CYP2C19 CYP3A4 / CYP inhibition: CYP3A4 CYP2C19
D10516  Aripiprazole hydrate (JAN); Aripiprazole monohydrate; Abilify maintena (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 CYP2D6
D10524  Azilsartan and amlodipine besilate; Zacras (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D10533  Umeclidinium bromide and vilanterol; Anoro (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 CYP2D6
D10551  Ceritinib (JAN/USAN/INN); Zykadia (TN) (P) unclassified
D10564  Amenamevir (JAN/INN); Amenalief (TN) (P) unclassified
D10566  Pasireotide pamoate (JAN); Signifor lar (TN) (P) unclassified
D10568  Pitavastatin calcium hydrate (JP19); Pitabastatin calcium pentahydrate; Livalo (TN) (P) CYP inhibition: CYP2C9
D10569  Tafluprost and timolol maleate; Tapcom (TN) (P) unclassified
D10627  Esketamine hydrochloride (JAN/USAN); Spravato (TN) (P) Enzyme: CYP2C19 CYP3A4 / CYP inhibition: CYP3A4 CYP2C19
D10633  Finerenone (JAN/USAN/INN); Kerendia (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D10643  Isavuconazonium sulfate (JAN/USAN); Cresemba (TN) (P) unclassified
D10653  Peficitinib (USAN/INN) (P) unclassified
D10656  Polmacoxib (USAN/INN) (P) unclassified
D10663  Rimegepant sulfate (USAN); Rimegepant sulfate hydrate (JAN); Nurtec odt (TN); Vydura (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D10679  Venetoclax (JAN/USAN/INN); Venclexta (TN) (CI,P) unclassified
D10688  Abemaciclib (JAN/USAN/INN); Verzenio (TN) (P) unclassified
D10721  Peficitinib hydrobromide (JAN/USAN); Smyraf (TN) (P) unclassified
D10746  Esflurbiprofen and mentha oil; Loqoa (TN) (P) CYP inhibition: CYP2C9
D10750  Isavuconazole (INN); Cresemba (TN) (P) unclassified
D10761  Polatuzumab vedotin (USAN); Polatuzumab vedotin (genetical recombination) (JAN); Polatuzumab vedotin-piiq; Polivy (TN) (P) unclassified
D10762  Fosravuconazole L-lysine ethanolate (JAN) (P) unclassified
D10774  Vonoprazan, amoxicillin and metronidazole; Vonopion (TN) (P) Enzyme: CYP2C19 CYP3A4 / CYP inhibition: CYP3A4 CYP2D6 CYP2C19
D10775  Vonoprazan, amoxicillin and clarithromycin; Vonosap (TN); Voquenza (TN) (P) Enzyme: CYP2C19 CYP3A4 / CYP inhibition: CYP3A4 CYP2D6 CYP2C19
D10780  Perampanel hydrate (JAN); Fycompa (TN) (P) unclassified
D10800  Gilteritinib fumarate (JAN/USAN); Xospata (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D10801  Letermovir (JAN/USAN/INN); Prevymis (TN) (P) CYP induction: CYP2C19
D10805  Telmisartan, amlodipine and hydrochlorothiazide; Micatrio (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D10866  Brigatinib (JAN/USAN); Alunbrig (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D10871  Filgotinib (USAN/INN) (P) unclassified
D10872  Filgotinib hydrochloride (USAN) (P) unclassified
D10891  Capmatinib hydrochloride (USAN); Capmatinib hydrochloride hydrate (JAN); Tabrecta (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D10892  Esaxerenone (JAN/INN) (P) unclassified
D10893  Acalabrutinib (JAN/USAN/INN); Calquence (TN) (P) unclassified
D10915  Cannabidiol (JAN/USAN/INN); CBD; Epidiolex (TN) (P) Enzyme: CYP2C19 CYP3A4 / CYP inhibition: CYP3A4 CYP2C19
D10926  Entrectinib (JAN/USAN/INN); Rozlytrek (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D10927  Erdafitinib (JAN/USAN/INN); Balversa (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 CYP2C9
D10930  Etrasimod (USAN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 CYP2C9
D10931  Etrasimod arginine (USAN); Etrasimod L-arginine (JAN); Velsipity (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 CYP2C9
D10932  Etripamil (USAN/INN); Cardamyst (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D10944  Itacitinib (USAN/INN) (P) unclassified
D10945  Itacitinib adipate (JAN/USAN) (P) unclassified
D10967  Ozanimod hydrochloride (JAN/USAN); Zeposia (TN) (P) unclassified
D10968  Ozanimod (USAN/INN) (P) unclassified
D10990  Somatrogon (USAN/INN); Somatrogon (genetical recombination) (JAN); Somatrogon-ghla; Ngenla (TN) (P) unclassified
D10993  Tucidinostat (JAN/USAN/INN); Hiyasta (TN) (P) unclassified
D10994  Upadacitinib (USAN/INN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D10995  Upadacitinib tartrate (USAN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D10999  Valbenazine tosylate (USAN); Valbenazine tosilate (JAN); Valbenazine ditosylate; Ingrezza (TN); Dysval (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D11012  Lorlatinib (JAN/USAN/INN); Lorbrena (TN) (P) unclassified
D11022  Lemborexant (JAN/USAN/INN); Dayvigo (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D11027  Ropeginterferon alfa-2b (INN); Ropeginterferon alfa-2b (genetical recombination) (JAN); Ropeginterferon alfa-2b-njft; Besremi (TN) (P) unclassified
D11035  Fluticasone furoate, umeclidinium bromide and vilanterol; Trelegy ellipta (TN) (P) unclassified
D11040  Apalutamide (JAN/INN); Erleada (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4 CYP2C19
D11048  Upadacitinib hydrate (JAN); Upadacitinib hemihydrate; Rinvoq (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D11052  Risankizumab (USAN/INN); Risankizumab (genetical recombination) (JAN); Risankizumab-rzaa; Skyrizi (TN) (P) unclassified
D11053  Encorafenib (JAN/USAN/INN); Braftovi (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D11054  Ravulizumab (USAN/INN); Ravulizumab (genetical recombination) (JAN); Ultomiris (TN) (P) unclassified
D11056  Mirtazapine hydrate (JAN) (P) Enzyme: CYP1A2 CYP3A4 / CYP inhibition: CYP1A2 CYP3A4 CYP2D6
D11062  Osilodrostat phosphate (JAN/USAN); Isturisa (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 CYP2D6
D11070  Tirabrutinib hydrochloride (JAN/USAN); Velexbru (TN) (P) unclassified
D11072  Siponimod fumarate (USAN); Siponimod fumaric acid (JAN); Mayzent (TN) (P) CYP inhibition: CYP2C9
D11079  Satralizumab (USAN/INN); Satralizumab (genetical recombination) (JAN); satralizumab-mwge; Enspryng (TN) (P) unclassified
D11082  Anifrolumab (USAN); Anifrolumab (genetical recombination) (JAN); Anifrolumab-fnia; Saphnelo (TN) (P) unclassified
D11090  Ivosidenib (JAN/USAN/INN); Tibsovo (TN) (P) unclassified
D11092  Pitavastatin magnesium; Zypitamag (TN) (P) CYP inhibition: CYP2C9
D11093  Avacopan (JAN/USAN/INN); Tavneos (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D11095  Atorvastatin calcium propylene glycol solvate (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D11106  Filgotinib maleate (JAN/USAN); Jyseleca (TN) (P) unclassified
D11114  Esomeprazole magnesium dihydrate (P) Enzyme: CYP2C19 / CYP inhibition: CYP2C19
D11120  Emapalumab (USAN/INN); Emapalumab (genetical recombination) (JAN); Emapalumab-lzsg; Gamifant (TN) (P) unclassified
D11123  Mirikizumab (USAN/INN); Mirikizumab (genetical recombination) (JAN); Mirikizumab-mrkz; Omvoh (TN) (P) unclassified
D11138  Larotrectinib sulfate (JAN/USAN); Vitrakvi (TN) (P) unclassified
D11149  Brexanolone (USAN/INN); Zulresso (TN) (P) unclassified
D11150  Cenobamate (JAN/USAN/INN); Xcopri (TN) (P) Enzyme: CYP2C19 CYP3A4 / CYP inhibition: CYP3A4 CYP2C19
D11154  Diroximel fumarate (JAN/USAN/INN); Vumerity (TN) (P) unclassified
D11159  Leniolisib phosphate (JAN/USAN); Joenja (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D11194  Somapacitan (USAN/INN); Somapacitan (genetical recombination) (JAN); Somapacitan-beco; Sogroya (TN) (P) unclassified
D11215  Ponesimod (USAN/INN); Ponvory (TN) (P) unclassified
D11243  Ublituximab (USAN/INN); Briumvi (TN) (P) unclassified
D11296  Fedratinib hydrochloride (USAN); Fedratinib hydrochloride hydrate (JAN); Fedratinib dihydrochloride monohydrate; Inrebic (TN) (P) Enzyme: CYP2C19 CYP3A4 / CYP inhibition: CYP3A4 CYP2C19
D11370  Fosnetupitant chloride hydrochloride (JAN/USAN); Arokaris (TN) (P) unclassified
D11371  Capivasertib (JAN/USAN); Truqap (TN) (P) unclassified
D11397  Darvadstrocel (INN); Alofisel (TN) (P) unclassified
D11400  Abrocitinib (JAN/USAN); Cibinqo (TN) (P) Enzyme: CYP2C19 / CYP inhibition: CYP2C19 CYP2C9
D11417  Pemigatinib (JAN/USAN/INN); Pemazyre (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D11422  Zanubrutinib (JAN/USAN/INN); Brukinsa (TN) (P) unclassified
D11454  Repotrectinib (JAN/USAN); Augtyro (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D11460  Siponimod (USAN/INN) (P) CYP inhibition: CYP2C9
D11470  Imlifidase (USAN/INN); Idefirix (TN) (P) unclassified
D11477  Pozelimab (USAN); Pozelimab-bbfg; Veopoz (TN) (P) unclassified
D11485  Tazemetostat hydrobromide (JAN/USAN); Tazverik (TN) (P) unclassified
D11492  Monomethyl fumarate (USAN); Bafiertam (TN) (P) unclassified
D11525  Enfortumab vedotin (USAN); Enfortumab vedotin (genetical recombination) (JAN); Enfortumab vedotin-ejfv; Padcev (TN) (P) unclassified
D11530  Sutimlimab (USAN/INN); Sutimlimab (genetical recombination) (JAN); Sutimlimab-jome; Enjaymo (TN) (P) unclassified
D11550  Bimekizumab (USAN/INN); Bimekizumab (genetical recombination) (JAN); Bimzelx (TN) (P) unclassified
D11557  Tecovirimat hydrate (JAN); Tecovirimat monohydrate; Tpoxx (TN); Tepoxx (TN) (P) unclassified
D11584  Budesonide, glycopyrronium bromide and formoterol fumarate; Budesonide, glycopyrrolate and formoterol fumarate; Breztri (TN) (P) unclassified
D11613  Pegcetacoplan (JAN/USAN/INN); Empaveli (TN) (P) unclassified
D11619  Desvenlafaxine succinate anhydrous (P) unclassified
D11630  Aminophylline dihydrate (P) Enzyme: CYP1A2 / CYP inhibition: CYP1A2
D11641  Danicopan (JAN/USAN/INN); Voydeya (TN) (P) unclassified
D11659  Tolvaptan sodium phosphate (JAN); Samtasu (TN) (P) unclassified
D11662  Valemetostat tosilate (JAN); Valemetostat tosylate; Ezharmia (TN) (P) unclassified
D11666  Nipocalimab (USAN); Nipocalimab (genetical recombination) (JAN); Nipocalimab-aahu; Imaavy (TN) (P) unclassified
D11674  Berotralstat hydrochloride (JAN/USAN); Orladeyo (TN) (P) CYP inhibition: CYP3A4
D11696  Crovalimab (USAN/INN); Crovalimab (genetical recombination) (JAN); Crovalimab-akkz; Piasky (TN) (P) unclassified
D11703  Opinercept (INN) (P) unclassified
D11708  Givosiran sodium (JAN); Givlaari (TN) (P) unclassified
D11713  Selpercatinib (JAN/USAN/INN); Retevmo (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D11725  Futibatinib (JAN/USAN/INN); Lytgobi (TN) (P) unclassified
D11757  Inebilizumab (USAN/INN); Inebilizumab (genetical recombination) (JAN); Inebilizumab-cdon; Uplizna (TN) (P) unclassified
D11784  Vonoprazan (USAN/INN) (P) Enzyme: CYP2C19 CYP3A4 / CYP inhibition: CYP3A4 CYP2D6 CYP2C19
D11785  Oteseconazole (USAN/INN); Vivijoa (TN) (P) unclassified
D11793  Zuranolone (JAN/USAN/INN); Zurzuvae (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D11804  Aspirin and vonoprazan; Cabpirin (TN) (P) unclassified
D11814  Tisotumab vedotin (USAN/INN); Tisotumab vedotin (genetical recombination) (JAN); Tisotumab vedotin-tftv; Tivdak (TN) (P) unclassified
D11815  Belumosudil (USAN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D11816  Belumosudil mesylate (USAN); Belumosudil mesilate (JAN); Rezurock (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D11817  Deucravacitinib (JAN/USAN); Sotyktu (TN) (P) Enzyme: CYP1A2 / CYP inhibition: CYP1A2 CYP2D6
D11835  Vorasidenib citrate (USAN); Vorasidenib citric acid hydrate (JAN); Voranigo (TN) (P) Enzyme: CYP1A2 CYP2C19 / CYP inhibition: CYP1A2 CYP2D6 CYP2C19 CYP2C9
D11838  Vilobelimab (USAN); Gohibic (TN) (P) unclassified
D11843  Cendakimab (USAN/INN); Cendakimab (genetical recombination) (JAN) (P) unclassified
D11861  Indacaterol acetate, glycopyrronium bromide and mometasone furoate; Enerzair (TN) (P) unclassified
D11862  Indacaterol and mometasone furoate; Atectura (TN) (P) unclassified
D11866  Deuruxolitinib (USAN) (P) Enzyme: CYP1A2 / CYP inhibition: CYP1A2 CYP2C9
D11867  Deuruxolitinib phosphate (USAN); Leqselvi (TN) (P) Enzyme: CYP1A2 / CYP inhibition: CYP1A2 CYP2C9
D11876  Efgartigimod alfa (USAN/INN); Efgartigimod alfa (genetical recombination) (JAN); Efgartigimod alfa-fcab; Vyvgart (TN) (P) unclassified
D11881  Amlodipine benzoate; Katerzia (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D11887  Daridorexant hydrochloride (JAN/USAN); Quviviq (TN) (P) unclassified
D11920  Pimitespib (JAN); Jeselhy (TN) (P) unclassified
D11952  Axatilimab (USAN/INN); Axatilimab (genetical recombination) (JAN); Axatilimab-csfr; Niktimvo (TN) (P) unclassified
D11954  Belzutifan (JAN/USAN/INN); Welireg (TN) (P) Enzyme: CYP2C19 / CYP inhibition: CYP2C19
D11970  Ritlecitinib tosylate (USAN); Ritlecitinib tosilate (JAN); Litfulo (TN) (P) CYP inhibition: CYP1A2
D12015  St. John's wort; SJW (P) unclassified
D12050  Pirtobrutinib (JAN/USAN); Jaypirca (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 CYP2C19
D12055  Sotorasib (JAN/USAN); Lumakras (TN) (P) unclassified
D12066  Spesolimab (USAN/INN); Spesolimab (genetical recombination) (JAN); Spesolimab-sbzo; Spevigo (TN) (P) unclassified
D12182  Rozanolixizumab (USAN/INN); Rozanolixizumab (genetical recombination) (JAN); rozanolixizumab-noli; Rystiggo (TN) (P) unclassified
D12213  Tolebrutinib (JAN/USAN/INN) (P) unclassified
D12217  Imlunestrant tosylate (USAN); Imlunestrant tosilate (JAN); Inluriyo (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D12245  Lazertinib mesylate (USAN); Lazertinib mesilate hydrate (JAN); Lazcluze (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D12246  Tegoprazan (INN) (P) unclassified
D12251  Iptacopan (USAN/INN) (P) CYP induction: CYP3A4
D12252  Iptacopan hydrochloride (USAN); Iptacopan hydrochloride hydrate (JAN); Iptacopan hydrochloride monohydrate; Fabhalta (TN) (P) CYP induction: CYP3A4
D12265  Mavacamten (JAN/USAN/INN); Camzyos (TN) (P) Enzyme: CYP2C19 / CYP inhibition: CYP2C19 CYP2C9
D12285  Remibrutinib (JAN/USAN/INN); Rhapsido (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D12311  Bortezomib hydrate (JAN) (P) unclassified
D12326  Opelconazole (USAN/INN) (P) unclassified
D12356  Zilucoplan sodium (JAN); Zilbrysq (TN) (P) unclassified
D12357  Zilucoplan (USAN/INN) (P) unclassified
D12364  Taletrectinib adipate (JAN/USAN); Ibtrozi (TN) (P) CYP inhibition: CYP2C9
D12374  Sibeprenlimab (USAN/INN); Sibeprenlimab (genetical recombination) (JAN); Sibeprenlimab-szsi; Voyxact (TN) (P) unclassified
D12396  Sebetralstat (JAN/USAN/INN); Ekterly (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D12403  Venlafaxine besylate monohydrate; Venlafaxine besylate (TN) (P) CYP inhibition: CYP2D6
D12410  Landiolol (USAN/INN) (P) unclassified
D12442  Tucatinib ethanolate (JAN); Tucatinib hemiethanolate; Tukysa (TN) (P) unclassified
D12444  Nilotinib hydrochloride dihydrate (JAN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D12487  Olokizumab (INN) (P) unclassified
D12493  Dextromethorphan hydrobromide and bupropion hydrochloride; Auvelity (TN) (P) CYP inhibition: CYP2D6
D12544  Vortioxetine hemihydrobromide (USAN) (P) Enzyme: CYP2C19 / CYP inhibition: CYP2D6 CYP2C19 CYP2C9
D12586  Mifepristone and misoprostol; Mefeego (TN) (P) unclassified
D12595  Aspirin trelamine (USAN) (P) unclassified
D12596  Aspirin trelamine hydrochloride (USAN) (P) unclassified
D12597  Ibuprofen trelamine (USAN); Ibuprofen diethylaminoethyl ester (P) CYP inhibition: CYP2C9
D12598  Ibuprofen trelamine hydrochloride (USAN) (P) CYP inhibition: CYP2C9
D12611  Vornorexant hydrate (JAN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D12637  Darunavir hydrate (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D12684  Efgartigimod alfa and hyaluronidase; Efgartigimod alfa (genetical recombination) and vorhyaluronidase alfa (genetical recombination); Efgartigimod alfa and hyaluronidase-qvfc; Vyvgard hytrulo (TN); Vyvdura (TN) (P) unclassified
D12704  Acalabrutinib maleate hydrate (JAN); Acalabrutinib maleate monohydrate; Calquence (TN) (P) unclassified
D12747  Divozilimab (INN) (P) unclassified
D12748  Levilimab (INN) (P) unclassified
D12752  Darunavir propylene glycolate (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D12816  Dexlansoprazole sesquihydrate (P) Enzyme: CYP2C19 CYP3A4 / CYP inhibition: CYP3A4 CYP2C19
D12837  Risovalisib mesilate hydrate (JAN); Risovalisib mesylate dihydrate; Haizexin (TN) (P) CYP induction: CYP2C19
D12963  Macitentan and tadalafil; Opsynvi (TN); Yuvanci (TN) (CI,P) Enzyme: CYP2C19 / CYP inhibition: CYP2C19 CYP2C9
D12975  Nerandomilast (JAN/USAN/INN); Jascayd (TN) (P) unclassified
D13012  Fexuprazan (INN); Abeprazan (P) unclassified
D13013  Ilaprazole (INN) (P) unclassified
D13026  Atogepant hydrate (JAN); Aquipta (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4
D13167  Tegomil fumarate (INN); Riulvy (TN) (P) unclassified
D13197  Linaprazan glurate (USAN/INN) (P) unclassified
D13198  Linaprazan glurate hydrochloride (USAN) (P) unclassified
D13231  Dimdazenil (INN) (P) unclassified
D13240  Zastaprazan (INN) (P) unclassified
D13243  Nafithromycin (INN) (P) unclassified