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Drug interaction list


Query:
D00292  Dexamethasone (JP18/USP/INN); Decadron (TN); Maxidex (TN)

Interactions: 1456 hits    [ ATC classification | Therapeutic category ]

C01946  Oleandomycin; Amimycin; Landomycin; Matromycin; Romicil (P) unclassified
C04931  Argatroban; (2R,4R)-4-Methyl-1[Nalpha-[(3-methyl-1,2,3,4-tetrahydro-8-quinolinyl)sulfonyl]-L-arginyl]-2-piperadinecarboxylic acid (P) unclassified
C06174  Codeine; (5alpha,6alpha)-7,8-Didehydro-4,5-epoxy-3-methoxy-17-methylmorphinan-6-ol (P) unclassified
C07005  Flunisolide; Flunisolide anhydrous (P) unclassified
C07051  Indinavir (P) unclassified
D00066  Progesterone (JP18/USP/INN); Crinone (TN); Prometrium (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00067  Estrone (JAN/USP/INN); Estrone (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00085  Insulin (JAN/USP) (P) unclassified
D00105  Estradiol (JAN/USP/INN); Climara (TN); Divigel (TN); Estrace (TN); Estraderm (TN); Estrasorb (TN); Estring (TN); Estrogel (TN); Innofem (TN); Vagifem (TN); Vivelle (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00106  Epoprostenol (USAN/INN); Prostaglandin I2; Prostacyclin; Epoprostenol (TN) (P) unclassified
D00107  Tacrolimus (USP/INN); Tacrolimus hydrate (JP18); Prograf (TN); Protopic (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00109  Aspirin (JP18/USP); Aspalon (JAN); Acetylsalicylic acid; Easprin (TN); Durlaza (TN) (P) unclassified
D00123  Cyanamide (JP18); Cyanamide (TN) (CI) unclassified
D00124  Ephedrine (USP); Ephedrine (TN) (P) unclassified
D00127  Piroxicam (JP18/USP/INN); Feldene (TN) (P) unclassified
D00130  Diflunisal (JAN/USP/INN); Dolobid (TN) (P) unclassified
D00131  Disulfiram (JP18/USP/INN); Antabuse (TN) (CI) unclassified
D00136  Haloperidol (JP18/USP/INN); Haldol (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00140  Erythromycin (JP18/USP/INN); Akne-mycin (TN); Eryc (TN); Erygel (TN); Pce (TN); Staticin (TN); T-stat (TN) (P) unclassified
D00168  Cytarabine (JP18/USP/INN); ARA-C; Depocyt (TN) (P) unclassified
D00181  Argatroban (USP); Argatroban hydrate (JP18); Novastan (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00184  Cyclosporine (USP); Ciclosporin (JP18); Gengraf (TN); Neoral (TN); Restasis (TN); Sandimmune (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D00186  Ciprofloxacin (JP18/USP/INN); Cipro (TN); Otiprio (TN) (P) unclassified
D00195  Codeine (USP); Codeine hydrate (P) unclassified
D00197  Reserpine (JP18/USP/INN); Apoplon (TN); Serpalan (TN) (P) unclassified
D00198  Rescinnamine (JAN/INN); Tsuruselpi S (TN) (P) unclassified
D00203  Amphotericin B (JP18/USP/INN); Ambisome (TN); Amphotec (TN); Fungizone (TN) (P) unclassified
D00210  Norfloxacin (JP18/USP/INN); Noroxin (TN) (P) unclassified
D00211  Rifampin (USP); Rifampicin (JP18/INN); Rifadin (TN); Rimactane (TN) (P) CYP induction: CYP3A4
D00216  Acarbose (JAN/USAN/INN); Precose (TN) (P) unclassified
D00218  Acetazolamide (JP18/USP/INN); Diamox (TN) (P) unclassified
D00219  Acetohexamide (JP18/USP/INN); Dymelor (TN) (P) unclassified
D00246  Budesonide (JP18/USP/INN); Entocort EC (TN); Pulmicort (TN); Rhinocort (TN); Uceris (TN) (P) Enzyme: CYP3A4 / Target: NR3C1 / CYP induction: CYP3A4
D00247  Bumetanide (JP18/USP/INN); Bumex (TN) (P) unclassified
D00252  Carbamazepine (JP18/USP/INN); Equetro (TN); Tegretol (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00255  Carvedilol (JP18/USP/INN); Artist (TN); Coreg (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00271  Chlorpropamide (JP18/USP/INN); Diabinese (TN) (P) unclassified
D00272  Chlorthalidone (USP); Chlortalidone (JAN/INN); Hygroton (TN); Thalitone (TN) (P) unclassified
D00276  Clarithromycin (JP18/USP/INN); Biaxin (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D00281  Clonidine (JAN/USP/INN); Catarpres-TTS (TN) (P) unclassified
D00282  Clotrimazole (JP18/USP/INN); Lotrimin (TN); Mycelex (TN) (P) CYP inhibition: CYP3A4
D00283  Clozapine (JAN/USP/INN); Clozaril (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00287  Cyclophosphamide (USP); Cyclophosphamide hydrate (JP18); Cytoxan (TN); Neosar (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00292  Dexamethasone (JP18/USP/INN); Decadron (TN); Maxidex (TN) (P) Enzyme: CYP3A4 / Target: NR3C1 / CYP induction: CYP3A4
D00293  Diazepam (JP18/USP/INN); Diastat (TN); Valium (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00294  Diazoxide (JAN/USP/INN); Hyperstat (TN); Proglycem (TN) (P) unclassified
D00298  Digoxin (JP18/USP); Lanoxicaps (TN); Lanoxin (TN) (P) unclassified
D00302  Dipyridamole (JP18/USP/INN); Persantine (TN) (P) unclassified
D00303  Disopyramide (JP18/USAN/INN); Rythmodan P (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00312  Estrone sodium sulfate; Sodium estrone sulfate (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00313  Ethacrynic acid (USP); Etacrynic acid (JP18/INN) (P) unclassified
D00319  Felodipine (JP18/USP/INN); Plendil (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00320  Fentanyl (JAN/USP/INN); Duragesic (TN); Subsys (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00321  Finasteride (JAN/USP/INN); Propecia (TN); Proscar (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00322  Fluconazole (JP18/USP/INN); Diflucan (TN) (P) CYP inhibition: CYP3A4
D00324  Flunisolide (JAN/USP); Aerospan (TN); Nasalide (TN) (P) Enzyme: CYP3A4 / Target: NR3C1 / CYP induction: CYP3A4
D00330  Flurbiprofen (JP18/USP/INN); Ansaid (TN) (P) unclassified
D00331  Furosemide (JP18/USP/INN); Frusemide; Lasix (TN) (P) unclassified
D00335  Glipizide (USP/INN); Glucotrol (TN) (P) unclassified
D00336  Glyburide (USP); Glibenclamide (JP18/INN); Diabeta (TN); Glynase (TN); Micronase (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00340  Hydrochlorothiazide (JP18/USP/INN); Esidrix (TN); Microzide (TN) (P) unclassified
D00343  Ifosfamide (JAN/USP/INN); Ifex (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00345  Indapamide (JP18/USP); Lozol (TN); Natrix (TN) (P) unclassified
D00350  Itraconazole (JP18/USP); Itrizole (TN); Sporanox (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D00351  Ketoconazole (JP18/USP); Nizoral (TN); Xolegel (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D00355  Lansoprazole (JP18/USP/INN); Prevacid (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00358  Lidocaine (JP18/USP/INN); Dentipatch (TN); Xylocaine (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00359  Lovastatin (USP/INN); MK-803; ML-530B; Mevacor (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00364  Loratadine (JAN/USP/INN); Claritin (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00372  Thiabendazole (USP); Tiabendazole (JAN/INN); Mintezol (TN) (P) unclassified
D00377  Mesalamine (USP); Mesalazine (JP18/INN); Apriso (TN); Asacol (TN); Canasa (TN); Delzicol (TN); Lialda (TN); Mesalamine (TN); Pentasa (TN); Rowasa (TN); Sfrowasa (TN) (P) unclassified
D00379  Tolazamide (JAN/USP/INN); Tolinase (TN) (P) unclassified
D00380  Tolbutamide (JP18/USP/INN); Orinase (TN) (P) unclassified
D00382  Torsemide (USP); Torasemide (JAN/INN); Demadex (TN); Luprac (TN) (P) unclassified
D00386  Triamterene (JP18/USP/INN); Dyrenium (TN) (P) unclassified
D00387  Triazolam (JP18/USP/INN); Halcion (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00395  Troglitazone (JAN/USAN/INN); Rezulin (TN) (P) unclassified
D00405  Methyldopa (USP); Methyldopa hydrate (JP18); Aldomet (TN) (P) unclassified
D00407  Methylprednisolone (JP18/USP/INN); Medrol (TN) (P) Enzyme: CYP3A4 / Target: NR3C1 / CYP induction: CYP3A4
D00416  Miconazole (JP18/USP/INN); Monistat (TN); Oravig (TN) (P) unclassified
D00418  Minoxidil (JAN/USP/INN); Loniten (TN); Riup (TN); Rogaine (TN) (P) unclassified
D00420  Mitotane (JAN/USP/INN); Lysodren (TN) (P) unclassified
D00424  Rifabutin (JAN/USP/INN); Mycobutin (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00426  Risperidone (JP18/USP/INN); Risperdal (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00427  Ritonavir (JAN/USP/INN); Norvir (TN) (P) unclassified
D00428  Salsalate (USP/INN); Sasapyrine (JAN); Disalcid (TN) (P) unclassified
D00429  Saquinavir (JAN/USP/INN); Fortovase (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00431  Metolazone (JAN/USP/INN); Zaroxolyn (TN) (P) unclassified
D00434  Simvastatin (JP18/USP/INN); MK-733; Zocor (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00435  Nevirapine (JAN/USP/INN); Viramune (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00437  Nifedipine (JP18/USP/INN); Adalat (TN); Afeditab CR (TN); Procardia (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00438  Nimodipine (USP/INN); Nimotop (TN); Nymalize (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00443  Spironolactone (JP18/USP/INN); Aldactone (TN) (P) unclassified
D00448  Sulfasalazine (USP/INN); Salazosulfapyridine (JP18); Azulfidine (TN) (P) unclassified
D00453  Ofloxacin (JP18/USP/INN); Floxin (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00455  Omeprazole (JP18/USP/INN); Prilosec (TN) (P) unclassified
D00456  Ondansetron (JAN/USP/INN); Zofran ODT (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00457  Quazepam (JAN/USP/INN); Doral (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00458  Quetiapine fumarate (JP18/USP); Seroquel (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00461  Quinethazone (JAN/INN); Hydromox (TN) (P) unclassified
D00465  Oxybutynin (USAN/INN); Anturol (TN); Oxytrol (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00471  Praziquantel (JAN/USP/INN); Biltricide (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00483  Propranolol hydrochloride (JP18/USP); Inderal (TN); Innopran XL (TN) (P) unclassified
D00491  Paclitaxel (JAN/USP/INN); Abraxane (TN); Taxol (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00506  Phenobarbital (JP18/USP/INN); Luminal (TN) (P) unclassified
D00512  Phenytoin (JP18/USP/INN); Dilantin (TN) (P) unclassified
D00519  Chlorothiazide (JAN/USP/INN); Diuril (TN) (P) unclassified
D00528  Caffeine (USP); Anhydrous caffeine (JP18); Anhydrous caffeine (TN); Respia (TN) (P) unclassified
D00529  Montelukast sodium (JP18/USP); Singulair (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00530  Zaleplon (JAN/USP/INN); Sonata (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00537  Topiramate (JAN/USP/INN); Topamax (TN); Trokendi xr (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00539  Ethosuximide (JP18/USP/INN); Zarontin (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00542  Halothane (JP18/USP/INN); Fluothane (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00544  Methoxyflurane (USP/INN); Penthrane (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00550  Midazolam (JAN/USP/INN); Dormicum (TN); Buccolam (TN); Nayzilam (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00554  Ethinyl estradiol (USP); Ethinylestradiol (JP18/INN); Estinyl (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D00560  Pimozide (JP18/USP/INN); Orap (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00563  Mirtazapine (JAN/USP/INN); Remeron (TN); Reflex (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00564  Warfarin sodium (USP); Coumadin (TN); Jantoven (TN) (P) unclassified
D00566  Sodium salicylate (JP18/USP); Salsonin (TN) (P) unclassified
D00570  Colchicine (JP18/USP); Colchicine (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00578  Voriconazole (JP18/USP/INN); Vfend (TN) (P) unclassified
D00585  Mifepristone (JAN/USAN/INN); Korlym (TN); Mifeprex (TN) (P) Enzyme: CYP3A4 / Target: NR3C1 / CYP induction: CYP3A4
D00588  Levofloxacin (USP); Levofloxacin hydrate (JP18); Levofloxacin hemihydrate; Iquix (TN); Levaquin (TN); Quixin (TN) (P) unclassified
D00592  Dapsone (USP); Diaphenylsulfone (JAN); Aczone (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00593  Glimepiride (JP18/USP/INN); Amaryl (TN) (P) unclassified
D00594  Repaglinide (JAN/USP/INN); Prandin (TN); Surepost (TN) (P) unclassified
D00595  Buformin (USAN/INN) (P) unclassified
D00596  Rosiglitazone maleate (JAN/USP); Avandia (TN) (P) unclassified
D00604  Clonidine hydrochloride (JP18/USP); Nexiclon (TN); Kapvay (TN); Duraclon (TN); Catapres (TN) (P) unclassified
D00606  Guanfacine hydrochloride (JAN/USP); Intuniv (TN); Tenex (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00608  Doxazosin mesylate (USP); Doxazosin mesilate (JP18); Cardura (TN) (P) unclassified
D00609  Prazosin hydrochloride (JP18/USP); Minipress (TN) (P) unclassified
D00611  Mecamylamine hydrochloride (USP); Inversine (TN) (P) unclassified
D00612  Trimetaphan camsilate (JAN/INN); Trimetaphan camsylate; Arfonad (TN) (P) unclassified
D00614  Sodium nitroprusside (USP); Sodium nitroprusside hydrate (JAN); Nitropress (TN) (P) unclassified
D00615  Amlodipine besylate (USP); Amlodipine besilate (JP18); Norvasc (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00616  Diltiazem hydrochloride (JP18/USP); Cardizem (TN); Cartia XT (TN); Dilacor XR (TN); Dilt-CD (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00617  Nicardipine hydrochloride (JP18/USAN); Cardene (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00618  Nisoldipine (JAN/USAN/INN); Sular (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00619  Verapamil hydrochloride (JP18/USP); Calan (TN); Covera-hs (TN); Vasolan (TN); Verelan (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D00625  Miglitol (JP18/USAN/INN); Glyset (TN) (P) unclassified
D00629  Nitrendipine (JP18/USAN/INN); Baypress (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00631  Bepridil hydrochloride (USAN); Bepridil hydrochloride hydrate (JAN); Vascor (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00636  Amiodarone hydrochloride (JP18/USP); Ancaron (TN); Cordarone (TN); Nexterone (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00637  Disopyramide phosphate (JAN/USP); Norpace (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00640  Propafenone hydrochloride (JP18/USP); Rythmol (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00646  Tolterodine (USAN/INN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00649  Amiloride hydrochloride (USP); Midamor (TN) (P) unclassified
D00650  Bendroflumethiazide (JAN/USP/INN); Naturetin (TN) (P) unclassified
D00651  Benzthiazide (JAN/INN); Exna (TN) (P) unclassified
D00653  Dorzolamide hydrochloride (JP18/USP); Trusopt (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00654  Hydroflumethiazide (JAN/USP/INN); Saluron (TN) (P) unclassified
D00656  Methyclothiazide (JAN/USP/INN); Enduron (TN) (P) unclassified
D00657  Polythiazide (JAN/USAN/INN); Renese (TN) (P) unclassified
D00658  Trichlormethiazide (JP18/USP/INN); Naqua (TN) (P) unclassified
D00661  Cevimeline hydrochloride (USAN); Cevimeline hydrochloride hydrate (JAN); Evoxac (TN); Saligren (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00670  Donepezil hydrochloride (JP18/USP); Aricept (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00674  Naratriptan hydrochloride (JAN/USP); Amerge (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00677  Granisetron hydrochloride (JAN/USP); Kytril (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00678  Ondansetron hydrochloride hydrate (JAN/USP); Ondansetron hydrochloride; Zofran (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00679  Ergotamine tartrate (JP18/USP); Ergomar (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00680  Methylergonovine maleate (USP); Methylergometrine maleate (JP18); Methergine (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00683  Albuterol sulfate (USP); Salbutamol sulfate (JP18); Accuneb (TN); Proventil (TN); Ventolin (TN) (P) unclassified
D00687  Salmeterol xinafoate (JAN/USP); Serevent (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00688  Terbutaline sulfate (JP18/USP); Brethine (TN) (P) unclassified
D00689  Beclomethasone dipropionate (USP); Beclometasone dipropionate (JP18); Beclovent (TN); Qnasl (TN); Vanceril (TN) (P) Enzyme: CYP3A4 / Target: NR3C1 / CYP induction: CYP3A4
D00690  Mometasone furoate (JAN/USP); Asmanex (TN); Elocon (TN) (P) Enzyme: CYP3A4 / Target: NR3C1 / CYP induction: CYP3A4
D00696  Midazolam hydrochloride (USAN); Versed (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00701  Phenobarbital sodium (JAN/USP/INN); Luminal sodium (TN) (P) unclassified
D00706  Zolpidem tartrate (JP18/USP); Ambien (TN); Intermezzo (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00722  Oxybutynin chloride (USP); Oxybutynin hydrochloride (JP18); Ditropan (TN); Gelnique (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00724  Rabeprazole sodium (JP18/USP); Aciphex (TN); Pariet (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00727  Olsalazine sodium (USAN); Dipentum (TN) (P) unclassified
D00729  Loperamide hydrochloride (JAN/USP); Imodium (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00749  Leflunomide (JAN/USP/INN); Arava (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00751  Methylprednisolone sodium succinate (JAN/USP); A-methapred (TN); Solu-medrol (TN) (P) Enzyme: CYP3A4 / Target: NR3C1 / CYP induction: CYP3A4
D00753  Sirolimus (JAN/USAN/INN); Rapamune (TN); Rapamycin (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D00754  Thalidomide (JAN/USP/INN); Thalomid (TN); Thaled (TN) (P) unclassified
D00762  Metyrosine (USP); Metirosine (JAN/INN); Demser (TN) (P) unclassified
D00765  Rocuronium bromide (JAN/USP/INN); Zemuron (TN) (P) unclassified
D00769  Clopidogrel bisulfate (USP); Clopidogrel sulfate (JP18); Clopidogrel sulfate tablets (JP18); Clopidogrel hydrogen sulphate; Isocover (TN); Plavix (TN) (P) unclassified
D00780  Bromocriptine mesylate (USP); Bromocriptine mesilate (JP18); Parlodel (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D00785  Selegiline hydrochloride (JAN/USP); Eldepryl (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00794  Loxapine succinate (USP); Loxitane (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00804  Ivermectin (JAN/USP/INN); Sklice (TN); Soolantra (TN); Stromectol (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00809  Amitriptyline hydrochloride (JP18/USP); Elavil (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00810  Choline salicylate (JAN/USAN/INN); Arthropan (TN) (P) unclassified
D00811  Clomipramine hydrochloride (JP18/USP); Anafranil (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00815  Imipramine hydrochloride (JP18/USP); Tofranil (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00820  Trazodone hydrochloride (JAN/USP); Desyrel (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00821  Venlafaxine hydrochloride (JAN/USP); Effexor (TN) (P) unclassified
D00822  Citalopram hydrobromide (USP); Celexa (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00825  Sertraline hydrochloride (JAN/USP); Zoloft (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00827  Magnesium salicylate (USP); Magnesium salicylate tetrahydrate; Magan (TN) (P) unclassified
D00831  Mefloquine hydrochloride (JP18/USP); Lariam (TN) (P) unclassified
D00836  Buprenorphine hydrochloride (JP18/USP); Buprenex (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00840  Levomethadyl acetate hydrochloride (USAN); Orlaam (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00847  Oxycodone hydrochloride (USP); Oxecta (TN); Oxycontin (TN); Roxicodone (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00851  Erythromycin estolate (USP); Erythromycin estorate (JAN); Ilosone (TN) (P) unclassified
D00873  Lomefloxacin hydrochloride (JAN/USAN); Maxaquin (TN) (P) unclassified
D00874  Moxifloxacin hydrochloride (JAN/USP); Avelox (TN); Vigamox (TN) (P) unclassified
D00879  Rifapentine (USAN/INN); Priftin (TN) (P) CYP induction: CYP3A4
D00880  Butoconazole nitrate (USP); Femstat (TN); Gynazole-1 (TN) (P) unclassified
D00881  Econazole nitrate (JAN/USP); Ecoza (TN); Spectazole (TN) (P) unclassified
D00882  Miconazole nitrate (JP18/USP); Micatin (TN); Monistat (TN) (P) unclassified
D00885  Oxiconazole nitrate (JAN/USAN); Oxistat (TN) (P) unclassified
D00886  Sulconazole nitrate (JAN/USP); Exelderm (TN) (P) unclassified
D00887  Atorvastatin calcium anhydorous; Lipitor (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00888  Terconazole (USP/INN); Terazol 3 (TN) (P) unclassified
D00889  Cerivastatin sodium (JAN/USAN); Baycol (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00890  Tioconazole (JAN/USP/INN); Vagistat-1 (TN) (P) unclassified
D00892  Fluvastatin sodium (JAN/USP); Lescol (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00894  Amprenavir (JAN/USAN/INN); Agenerase (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00896  Efavirenz (JAN/USP/INN); Sustiva (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00897  Indinavir sulfate (USP); Crixivan (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D00899  Nelfinavir mesylate (USAN/INN); Nelfinavir mesilate (JAN); Viracept (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D00904  Diclofenac sodium (JP18/USP); Solaraze (TN); Voltaren (TN) (P) unclassified
D00944  Metformin hydrochloride (JP18/USP); Glucophage (TN) (P) unclassified
D00945  Pioglitazone hydrochloride (JP18/USP); Actos (TN) (P) unclassified
D00948  Estropipate (USP); Piperazine estrone sulfate; Ogen (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00951  Medroxyprogesterone acetate (JP18/USP); Depo-provera (TN); Depo-subq provera 104 (TN); Provera (TN) (CI,P) unclassified
D00961  Bicalutamide (JP18/USP/INN); Casodex (TN) (P) CYP inhibition: CYP3A4
D00963  Exemestane (JAN/USP/INN); Aromasin (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00964  Letrozole (JAN/USP/INN); Femara (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00966  Tamoxifen citrate (JP18/USP); Nolvadex (TN); Soltamox (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00967  Toremifene citrate (JAN/USAN); Fareston (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D00969  Meloxicam (JAN/USP/INN); Mobic (TN) (P) unclassified
D00971  Sodium thiosalicylate; Thiosalicylic acid sodium salt; Rexolate (TN) (P) unclassified
D00975  Dexamethasone sodium phosphate (JAN/USP); Dalalone (TN); Maxidex (TN) (P) Enzyme: CYP3A4 / Target: NR3C1 / CYP induction: CYP3A4
D00979  Methylprednisolone acetate (JAN/USP); Depo-medrol (TN) (P) Enzyme: CYP3A4 / Target: NR3C1 / CYP induction: CYP3A4
D00987  Cabergoline (JP18/USP/INN); Cabaser (TN); Dostinex (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D01007  Propiverine hydrochloride (JP18); Bup-4 (TN); Mictonorm (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D01028  Ticlopidine hydrochloride (JP18/USP); Ticlid (TN) (P) unclassified
D01029  Tirofiban hydrochloride (USAN); Tirofiban hydrochloride hydrate; Aggrastat (TN) (P) unclassified
D01061  Irinotecan hydrochloride (USP); Irinotecan hydrochloride hydrate (JP18); Irinotecan hydrochloride trihydrate; CPT 11; CPT-11; Campto (TN); Camptosar (TN); Onivyde (TN) (P) unclassified
D01068  Vinblastine sulfate (JP18/USP); Exal (TN); Velban (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D01078  Telithromycin (JAN/USAN/INN); Ketek (TN) (P) unclassified
D01087  Methyl salicylate (JP18/NF); Methyl salicylate (TN) (P) unclassified
D01092  Lanoconazole (JP18/INN); Latoconazole; Astat (TN) (P) unclassified
D01098  Maxacalcitol (JAN/USAN/INN); Oxarol (TN); Prezios (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D01101  Bromperidol (JAN/USAN/INN); Impromen (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D01104  Barnidipine hydrochloride (JAN); Hypoca (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D01111  Nateglinide (JP18/USP/INN); Starsis (TN) (P) unclassified
D01115  Eplerenone (JP18/USAN/INN); Inspra (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D01121  Rebamipide (JP18/INN); Mucosta (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D01131  Lafutidine (JP18/INN); Protecadin (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D01144  Prulifloxacin (JAN/INN); Sword (TN) (P) unclassified
D01145  Azelnidipine (JP18/INN); Calblock (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D01148  Tolterodine tartrate (JAN/USP); Detrol (TN); Detrusitol (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D01160  Saquinavir mesylate (USP); Saquinavir mesilate (JAN); Invirase (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D01161  Fulvestrant (JAN/USP/INN); Faslodex (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D01163  Ergonovine maleate (USP); Ergometrine maleate (JP18); Ergometrine (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D01164  Aripiprazole (JAN/USP/INN); Abilify (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D01173  Cilnidipine (JP18/INN); Atelec (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D01176  Blonanserin (JAN/INN); AD 5423 (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D01196  Acetazolamide sodium (JAN); Diamox (TN) (P) unclassified
D01207  Omeprazole sodium (USAN); Losec sodium (TN) (P) unclassified
D01213  Tolvaptan (JAN/USAN/INN); Samsca (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D01217  Dydrogesterone (JP18/USP/INN); Duphaston (TN); Gynorest (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D01220  Trapidil (JP18/INN); Rocornal (TN) (P) unclassified
D01227  Bosentan (USAN); Bosentan hydrate (JAN); Tracleer (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D01235  Josamycin (JP18/USAN/INN); Leucomycin A3; JM; Josamycin (TN) (P) CYP inhibition: CYP3A4
D01236  Conivaptan hydrochloride (JAN/USAN); Vaprisol (TN) (P) unclassified
D01240  Deslanoside (JP18/USP/INN); Cedilanid-d (TN) (P) unclassified
D01241  Penflutizide (JAN/INN) (P) unclassified
D01246  Benzylhydrochlorothiazide (JAN); Behyd (TN) (P) unclassified
D01247  Ethiazide (JAN/INN) (P) unclassified
D01253  Clobazam (JAN/USAN/INN); Mystan (TN); Onfi (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D01256  Cyclothiazide (JAN/USAN/INN); Anhydron (TN) (P) unclassified
D01263  Ritodrine hydrochloride (JP18/USP); Yutopar (TN) (P) unclassified
D01269  Solifenacin succinate (JAN/USAN/INN); Vesicare (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D01276  Atazanavir sulfate (JAN/USAN); Reyataz (TN) (P) CYP inhibition: CYP3A4
D01280  Warfarin potassium (JP18); Athrombin-K (TN) (P) unclassified
D01287  Levobupivacaine hydrochloride (JAN/USAN); Chirocaine (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D01293  Ethyl loflazepate (JP18/INN); Meilax (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D01302  Hydralazine hydrochloride (JP18/USP); Apresoline (TN) (P) unclassified
D01316  Mexazolam (JAN/INN); Melex (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D01322  Troleandomycin (USAN/INN); Triacetyloleandomycin (JAN); TAO; Tao (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D01323  Azosemide (JP18/USAN/INN); Diart (TN) (P) unclassified
D01333  Urapidil (JP18/INN); Ebrantil (TN) (P) unclassified
D01337  Epoprostenol sodium (JAN/USAN); Flolan (TN); Veletri (TN) (P) unclassified
D01339  Midecamycin (JP18/INN); Medemycin (TN) (P) CYP inhibition: CYP3A4
D01355  Tramadol hydrochloride (JP18/USP); Ultram (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D01356  Glymidine sodium (JAN/USAN/INN) (P) unclassified
D01358  Mianserin hydrochloride (JAN/USAN); Tetramide (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D01360  Clenbuterol hydrochloride (JAN/USP); Spiropent (TN) (P) unclassified
D01361  Erythromycin ethylsuccinate (JP18/USP); E.E.S. (TN); Eryped (TN); Erythrocin W (TN) (P) unclassified
D01362  Tulobuterol hydrochloride (JP18); Hokunalin (TN); Respacal (TN) (P) unclassified
D01372  Zopiclone (JP18/INN); Amoban (TN); Zopiclone (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D01375  Methenolone acetate (USAN); Metenolone acetate (JP18); Primobolan (TN) (P) unclassified
D01386  Ephedrine hydrochloride (JP18/USP); Ephedrine hydrochloride (TN) (P) unclassified
D01390  Isoproterenol hydrochloride (USP); dl-Isoprenaline hydrochloride (JAN); Isuprel (TN); Proternol-S (TN) (P) unclassified
D01399  Fentanyl citrate (JP18/USP); Abstral (TN); Fentora (TN); Lazanda (TN); Oralet (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D01413  Estradiol valerate (JAN/USP/INN); Deladumone (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D01418  Tamibarotene (JAN/USAN/INN); Am 80; Amnoid (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D01425  Lopinavir (JAN/USP/INN) (P) unclassified
D01428  Fenoterol hydrobromide (JAN); Berotec (TN) (P) unclassified
D01429  Fosfluconazole (JAN/INN); Prodif (TN) (P) CYP inhibition: CYP3A4
D01436  Clorexolone (JAN/USAN/INN) (P) unclassified
D01441  Imatinib mesylate (USAN); Imatinib mesilate (JAN); Gleevec (TN); Glivec (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D01450  Bupivacaine hydrochloride (USP); Bupivacaine hydrochloride hydrate (JP18); Marcaine (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D01453  Caffeine hydrate (JP18); Caffeine monohydrate; Caffeine (TN) (P) unclassified
D01455  Cifenline succinate (USAN); Cibenzoline succinate (JP18); Cibenol (TN); Cipralan (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D01466  Ethenzamide (JP18/INN); Ethenzamide (TN) (P) unclassified
D01468  Nemonapride (JAN/INN); Emilace (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D01475  Flurbiprofen axetil (JAN); FP 83; Ropion (TN) (P) unclassified
D01478  Ebastine (JP18/USAN/INN); Kestine (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D01480  Isoconazole nitrate (JAN); Adestan-G (TN) (P) unclassified
D01481  Dihydrocodeine phosphate (JP18); Dihydro (TN) (P) unclassified
D01510  Dexamethasone metasulfobenzoate sodium (JAN); Dexamethazone metasulfobenzoate sodium; Dexapos; Santeson (TN) (P) Enzyme: CYP3A4 / Target: NR3C1 / CYP induction: CYP3A4
D01514  Etizolam (JP18/INN); Sedekopan (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D01551  Beraprost sodium (JP18/USAN); Procylin (TN) (P) unclassified
D01553  Manidipine hydrochloride (JP18); Manidipine dihydrochloride; Calslot (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D01557  Glycol salicylate (JAN); Ethylene glycol salicylate; Norgesic (TN); Phlogont (TN) (P) unclassified
D01562  Aranidipine (JAN/INN); Sapresta (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D01564  Rilmazafone hydrochloride hydrate (JP18); Rilmazafone hydrochloride dihydrate; Rilmazafone hydrochloride; Rhythmy (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D01599  Gliclazide (JP18/INN); Glimicron (TN) (P) unclassified
D01603  Bethanidine sulfate (JAN/USAN); Tenathan (TN) (P) unclassified
D01605  Meticrane (JP18/INN); Arresten (TN) (P) unclassified
D01614  Acetylkitasamycin (JP18); Neo-leucomycin H (TN) (P) unclassified
D01615  Dexamethasone palmitate (JAN); Dexamethasone 21-palmitate; Limethason (TN) (P) Enzyme: CYP3A4 / Target: NR3C1 / CYP induction: CYP3A4
D01617  Estradiol dipropionate (JAN); Ovahormon (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D01620  Neticonazole hydrochloride (JAN); Atolant (TN) (P) unclassified
D01624  Sarpogrelate hydrochloride (JP18); Anplag (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D01632  Dexamethasone dipropionate (USAN); Dexamethasone propionate (JAN); Hifmeta (TN) (P) Enzyme: CYP3A4 / Target: NR3C1 / CYP induction: CYP3A4
D01634  Piretanide (JAN/USAN/INN); Arelix (TN) (P) unclassified
D01636  Midecamycin acetate (JP18); Miocamycin; Miocamycin (TN) (P) CYP inhibition: CYP3A4
D01663  Quinine ethylcarbonate (JP18); Quinine ethylcarbonate (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D01664  Omoconazole nitrate (JAN/USAN) (P) unclassified
D01665  Voglibose (JP18/USAN/INN); Basen (TN) (P) unclassified
D01670  Nafamostat mesylate (USAN); Nafamostat mesilate (JP18); Ronastat (TN) (P) unclassified
D01672  Gabexate mesilate (JP18); Gabexate mesylate; Arodate (TN) (P) unclassified
D01683  Ozagrel hydrochloride hydrate (JAN); Ozagrel hydrochloride; Ozagrel (TN) (P) unclassified
D01684  Ozagrel sodium (JP18); Ozapen (TN) (P) unclassified
D01692  Alfuzosin hydrochloride (JAN/USAN); Uroxatral (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D01699  Darifenacin hydrobromide (JAN/USAN); Enablex (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D01703  Ciclesonide (JAN/USAN/INN); Alvesco (TN); Omnaris (TN); Zetonna (TN) (P) Enzyme: CYP3A4 / Target: NR3C1 / CYP induction: CYP3A4
D01708  Fluticasone propionate (JAN/USP); Cutivate (TN); Flonase (TN); Flovent (TN) (P) Enzyme: CYP3A4 / Target: NR3C1 / CYP induction: CYP3A4
D01710  Roxithromycin (JP18/USAN/INN); Rulide (TN) (P) unclassified
D01744  Brotizolam (JP18/USAN/INN); Lendormin (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D01745  Domperidone (JP18/USAN/INN); Motilium (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D01775  Bifonazole (JP18/USAN/INN); Mycospor (TN) (P) unclassified
D01799  Glyclopyramide (JAN/INN); Deamelin-S (TN) (P) unclassified
D01804  Cadralazine (JP18/INN); Cadral (TN) (P) unclassified
D01810  Nicorandil (JP18/USAN/INN); Sigmart (TN) (P) unclassified
D01811  Salicylamide (JAN/USP/INN); Salicylamide (TN) (P) unclassified
D01822  Clofenamide (JAN/INN) (P) unclassified
D01832  Modafinil (JAN/USP/INN); Provigil (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D01844  Fondaparinux sodium (JAN/USP/INN); Arixtra (TN) (P) unclassified
D01854  Mitiglinide calcium hydrate (JP18); Mitiglinide calcium dihydrate; Glufast (TN) (P) unclassified
D01855  Mozavaptane hydrochloride (JAN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D01872  Doxapram hydrochloride (USP); Doxapram hydrochloride hydrate (JP18); Dopram (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D01877  Mefruside (JP18/USAN/INN); Baycaron (TN) (P) unclassified
D01892  Icosapent ethyl (USAN); Ethyl icosapentate (JP18); Epadel S (TN); Vascepa (TN) (P) unclassified
D01895  Tripamide (JAN/USAN/INN); Normonal (TN) (P) unclassified
D01896  Cilostazol (JP18/USP/INN); Pletal (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D01897  Rokitamycin (JAN/INN); Ricamycin (TN) (P) unclassified
D01898  Haloperidol decanoate (JAN/USP); Halomonth (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D01908  Nilvadipine (JP18/USAN/INN); Nivadil (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D01935  Vinorelbine tartrate (USP); Vinorelbine ditartrate (JAN); KW 2307; Navelbine (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D01943  Canrenoate potassium (USAN); Potassium canrenoate (JP18); Soldactone (TN) (P) unclassified
D01948  Dexamethasone valerate (JAN); Dexamethasone 17-valerate; DV-17; Voalla ointment (TN) (P) Enzyme: CYP3A4 / Target: NR3C1 / CYP induction: CYP3A4
D01953  Estradiol benzoate (JP18/USP); Ovahormon (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D01965  Silodosin (JP18/INN); KMD 3213; Rapaflo (TN); Urief (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D01973  Eletriptan hydrobromide (JAN/USAN); Relpax (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D01977  Gefitinib (JP18/USAN/INN); Iressa (TN) (P) unclassified
D01980  Luliconazole (JAN/USAN/INN); Lulicon (TN); Luzu (TN) (P) CYP inhibition: CYP3A4
D01981  Ximelagatran (JAN/USAN/INN); Exanta (TN) (P) unclassified
D01984  Esomeprazole magnesium (USP); Esomeprazole magnesium hydrate (JAN); Esomeprazole magnesium trihydrate; Nexium (TN) (P) unclassified
D01994  Mosapride citrate hydrate (JP18); Mosapride citrate dihydrate; Gasmotin (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D01996  Tosufloxacin tosylate hydrate (JP18); Tosufloxacin tosilate; Ozex (TN); Tosuxacin (TN) (P) unclassified
D02000  Kitasamycin tartrate (JP18); Leucomycin tartrate (TN) (P) unclassified
D02008  Tadalafil (JAN/USP/INN); Adcirca (TN); Cialis (TN); Zalutia (TN) (CI,P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D02009  Erythromycin lactobionate (JP18/USP); Erythrocin (TN) (P) unclassified
D02045  Benidipine hydrochloride (JP18); KW 3049; Coniel (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D02061  Cyclopenthiazide (JAN/USAN/INN); Navidrex (TN) (P) unclassified
D02086  Lidocaine hydrochloride (JAN/USP); Dalcaine (TN); Xylocaine (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D02096  Fosphenytoin sodium (USP); Cerebyx (TN); Sesquient (TN) (P) CYP induction: CYP3A4
D02101  Codeine phosphate (USP); Codeine phosphate hydrate (JP18); Codeine (TN) (P) unclassified
D02102  Methadone hydrochloride (JAN/USP); Dolophine hydrochloride (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D02103  Phenytoin sodium (USP); Phenytoin sodium for injection (JP18); Aleviatin (TN); Dilantin (TN) (P) unclassified
D02109  dl-Methylephedrine hydrochloride (JP18); Methy-F (TN) (P) unclassified
D02112  Heparin sodium (JP18/USP/INN); Parnaparin sodium (INN); Liquemin sodium (TN) (P) unclassified
D02114  Hydroxychloroquine sulfate (JAN/USP); Plaquenil (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D02134  Azithromycin hydrate (JP18); Azithromycin dihydrate; Zithromac (TN); Zmax (TN); Azimycin (TN) (P) unclassified
D02150  l-Isoprenaline hydrochloride (JP18); Proternol-L (TN) (P) unclassified
D02151  Tulobuterol (JP18/INN); Atenos (TN); Hokunalin (TN) (P) unclassified
D02165  Docetaxel (USP); Docetaxel hydrate (JP18); Docetaxel trihydrate; Taxotere (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D02169  Croconazole hydrochloride (JP18); Pilzcin (TN) (P) unclassified
D02173  Galantamine hydrobromide (JAN/USP); Razadyne (TN); Reminyl (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D02174  Dexamethasone acetate (JAN/USP); Decadronal (TN) (P) Enzyme: CYP3A4 / Target: NR3C1 / CYP induction: CYP3A4
D02175  Compound oxycodone (JP18); Pavinal (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D02184  Erythromycin stearate (JP18/USP); Bristamycin (TN) (P) unclassified
D02186  Oleandomycin phosphate (JAN); Matromycin (TN) (P) unclassified
D02205  Ethylmorphine hydrochloride hydrate (JP18); Ethylmorphine hydrochloride dihydrate; Ethylmorphine hydrochloride (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D02206  Buformin hydrochloride (JP18); Dibetos-B (TN) (P) unclassified
D02211  Dihydroergotamine mesylate (USP); Dihydroergotamine mesilate (JP18); Migranal (TN); Trudhesa (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D02216  Ciprofloxacin hydrochloride (USP); Ciprofloxacin hydrochloride hydrate (JP18); Ciloxan (TN); Cipro (TN); Proquin XR (TN) (P) unclassified
D02219  Terbinafine hydrochloride (JP18/USP); Lamisil (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D02229  Sildenafil citrate (JAN/USP); Revatio (TN); Viagra (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D02235  Desmopressin acetate (USP); Desmopressin acetate hydrate (JAN); Desmopressin acetate trihydrate; DDAVP (TN); Minirinmelt (TN); Stimate (TN) (CI) unclassified
D02237  Guanethidine sulfate (USAN) (P) unclassified
D02258  Atorvastatin calcium (USP); Atorvastatin calcium hydrate (JP18); Atorvastatin calcium trihydrate; Atorvaliq (TN); Lipitor (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D02261  Quinine hydrochloride hydrate (JP18); Quinine hydrochloride dihydrate; Quinine hydrochloride (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D02262  Quinine sulfate (USP); Quinine sulfate hydrate (JP18); Quinine hydrogen sulfate; Coco-quinine (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D02268  Ergoloid mesylates (USP); Dihydroergotoxine mesilate (JP18); Circanol (TN); Hydergine (TN); Inorter (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D02269  Kitasamycin (JP18/USAN); Leucomycin (TN) (P) unclassified
D02323  Tolrestat (USAN/INN); Alredase (TN) (P) unclassified
D02340  Loxapine (USAN/INN); Adasuve (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D02356  Verapamil (USAN/INN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D02360  Sertraline (INN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D02363  Ketanserin (USAN/INN) (P) unclassified
D02372  Perospirone hydrochloride hydrate (JAN); Lullan (TN) (P) unclassified
D02375  Terbinafine (USAN/INN); Lamasil (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D02386  Ticrynafen (USAN); Tienilic acid (INN); Selacryn (TN) (P) unclassified
D02404  Procaterol hydrochloride (USAN); Pro-Air (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D02420  Acetylspiramycin (JP18); Spiramycin II; Acetylspiramycin (TN) (P) unclassified
D02425  Carbutamide (INN); Invenol (TN) (P) unclassified
D02426  Glycyclamide (INN); Tolcyclamide (P) unclassified
D02427  Glibornuride (USAN/INN); Glutril (TN) (P) unclassified
D02428  Glisentide (INN); Glypentide; Staticum (TN) (P) unclassified
D02429  Glisolamide (INN); Glysolamide; Diabenor (TN) (P) unclassified
D02430  Gliquidone (INN); Glurenorm (TN) (P) unclassified
D02453  Flumethiazide (INN); Ademol (TN) (P) unclassified
D02460  Clopamide (USAN/INN); Aquex (TN) (P) unclassified
D02475  Sitafloxacin (USAN); Sitafloxacin hydrate (JAN) (P) unclassified
D02478  Disulfamide (BAN) (P) unclassified
D02484  Artemether and lumefantrine; Coartem (TN) (P) unclassified
D02490  Tylosin (USP/INN); TS; Tylan (TN) (P) unclassified
D02492  Tilmicosin (USP/INN); TMS; Micotil (TN) (P) unclassified
D02493  Tilmicosin phosphate (USAN); TP (P) unclassified
D02497  Fosamprenavir (INN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D02498  Lopinavir and ritonavir; Kaletra (TN) (P) unclassified
D02501  Caspofungin acetate (JAN/USAN); Cancidas (TN) (P) unclassified
D02523  Erythromycin acistrate (USAN); Erasis (TN) (P) unclassified
D02524  Erythromycin gluceptate (USP); Erythromycin glucoheptonate; Ilotycin gluceptate (TN) (P) unclassified
D02525  Erythromycin propionate (USAN) (P) unclassified
D02540  Garenoxacin mesylate (USAN); Garenoxacin mesilate hydrate (JAN) (P) unclassified
D02554  Rifaximin (JAN/USAN/INN); Xifaxan (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D02555  Posaconazole (JAN/USAN/INN); Noxafil (TN) (P) CYP inhibition: CYP3A4
D02556  Ravuconazole (prop.INN) (P) unclassified
D02557  Chlormidazole (INN) (P) unclassified
D02564  Pargyline hydrochloride (USAN); Eutonyl (TN) (P) unclassified
D02567  Escitalopram oxalate (JAN/USP); Lexapro (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D02570  Desvenlafaxine succinate (USAN); Desvenlafaxine succinate hydrate (JAN); Desvenlafaxine succinate monohydrate; Pristiq (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D02577  Flibanserin (USAN/INN); Addyi (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D02582  Fenticonazole (INN) (P) unclassified
D02583  Fenticonazole nitrate (USAN); Lomexin (TN) (P) unclassified
D02584  Aliconazole (INN) (P) unclassified
D02585  Vibunazole; Bay N-7133 (P) unclassified
D02586  Alteconazole (INN) (P) unclassified
D02587  Metildigoxin (JP18); Lanirapid (TN) (P) unclassified
D02591  Dexamethasone acefurate (USAN/INN) (P) Enzyme: CYP3A4 / Target: NR3C1 / CYP induction: CYP3A4
D02592  Dexamethasone beloxil (USAN) (P) Enzyme: CYP3A4 / Target: NR3C1 / CYP induction: CYP3A4
D02593  Pantoprazole sodium (USP); Pantoprazole sodium hydrate (JAN); Protonix (TN) (P) unclassified
D02624  Eszopiclone (JAN/USP/INN); Estorra (TN); Lunesta (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D02626  Bromperidol decanoate (USAN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D02666  Iloperidone (USAN/INN); Fanapt (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D02690  Cholestyramine resin (USP); Colestyramine (JAN/INN); Questran (TN) (P) unclassified
D02691  Somatropin (USP/INN); Somatropin (genetical recombination) (JAN); Human growth hormone (JAN); Asellacrin (TN); Humatrope (TN); Nutropin (TN); Omnitrope (TN) (P) unclassified
D02714  Everolimus (JAN/USAN/INN); Afinitor (TN); Votubia (TN); Zortress (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D02715  Balsalazide disodium (USP); Colazide (TN) (P) unclassified
D02720  Beraprost (USAN) (P) unclassified
D02721  Iloprost (USAN/INN); Ventavis (TN) (P) unclassified
D02722  Limaprost (INN) (P) unclassified
D02731  Vardenafil dihydrochoride (USAN); Levitra (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D02732  Pranlukast hydrate (JP18); Onon (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D02740  Lidocaine and prilocaine; Lidocaine and propitocaine; Emla (TN); Oraqix (TN); Lidocaine and prilocaine (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D02749  Teceleukin (USAN); Teceleukin (genetical recombination) (JP18); Imunace (TN) (P) unclassified
D02778  Abciximab (USAN/INN); Abciximab (genetical recombination) (JAN); Reopro (TN) (P) unclassified
D02824  Almotriptan (USAN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D02825  Almotriptan malate (USP); Axert (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D02829  Alosetron hydrochloride (USAN); Lotrpnex (TN) (P) unclassified
D02837  Alteplase (USP/INN); Alteplase (genetical recombination) (JAN); Activase (TN); Cathflo activase (TN) (P) unclassified
D02838  Althiazide (USAN); Altizide (INN) (P) unclassified
D02860  Limaprost alfadex (JP18); Opalmon (TN) (P) unclassified
D02861  Indinavir sulfate ethanolate (JAN); Crixivan (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D02867  Fosamprenavir calcium hydrate (JAN); Lexiva (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D02910  Amiodarone (USAN/INN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D02914  Amlodipine maleate (USAN); Amvaz (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D02938  Ancrod (USAN/INN); Viprinex (TN) (P) unclassified
D02947  Anistreplase (USAN/INN); Eminase (TN) (P) unclassified
D02968  Aprepitant (JAN/USP/INN); Aponvie (TN); Emend (TN); Cinvanti (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D02980  Adomiparin sodium (USAN); Ardeparin sodium (USAN/INN); Semuloparin sodium (USAN/INN); Normiflo (TN) (P) unclassified
D02994  Rituximab (USAN/INN); Rituximab (genetical recombination) (JAN); Rituximab (genetical recombination) [Rituximab biosimilar 1] (JAN); Rituximab (genetical recombination) [Rituximab biosimilar 2] (JAN); Rituximab-abbs; Rituximab-pvvr; Rituximab-arrx; Rituxan (TN); Riabni (TN); Truximab (TN) (P) unclassified
D03023  Azaconazole (USAN/INN) (P) unclassified
D03063  BCG vaccine (USP); Freeze-dried BCG vaccine (for percutaneous use) (JP18); BCG vaccine (TN) (CI) unclassified
D03098  Berythromycin (USAN/INN); Erythromycin B (P) unclassified
D03106  Bexarotene (JAN/USAN/INN); Targretin (TN) (P) unclassified
D03136  Bivalirudin (USAN/INN) (P) unclassified
D03150  Bortezomib (JAN/USAN/INN); Velcade (TN) (P) unclassified
D03157  Brinolase (USAN); Brinase (INN) (P) unclassified
D03164  Bromindione (USAN/INN) (P) unclassified
D03165  Bromocriptine (USAN/INN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D03189  Buthiazide (USAN); Butizide (INN) (P) unclassified
D03208  Aliskiren (USAN/INN); Rasilez (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D03213  Apixaban (JAN/USAN/INN); Eliquis (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D03215  Armodafinil (USAN/INN); Nuvigil (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D03217  Avanafil (USAN/INN); Stendra (TN); Spedra (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D03218  Axitinib (JAN/USAN); Inlyta (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D03230  Insulin human (USP/INN); Insulin human (genetical recombination) (JP18); Insulin human (biosynthesis) (JAN); Insulin human (synthesis) (JAN); Humulin (TN) (P) unclassified
D03250  Insulin glargine (USAN/INN); Insulin glargine (genetical recombination) (JP18); Insulin glargine (genetical recombination) [Insulin glargin biosimilar 1] (JAN); Insulin glargine (genetical recombination) [Insulin glargin biosimilar 2] (JAN); Lantus (TN) (P) unclassified
D03252  Bosutinib (USAN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D03253  Brecanavir (USAN) (P) unclassified
D03259  Gemtuzumab ozogamicin (USAN); Gemtuzumab ozogamicin (genetical recombination) (JAN); Gemtuzumab (INN); Mylotarg (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D03260  Vardenafil hydrochloride hydrate (JAN); Vardenafil monohydrochloride trihydrate; Levitra (TN); Staxyn (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D03278  Enviomycin sulfate (JP18); Tuberactin (TN) (P) unclassified
D03297  Mecasermin (USAN/INN); Mecasermin (genetical recombination) (JAN); Increlex (TN); Myotrophin (TN) (P) unclassified
D03324  Nasaruplase (cell culture) (JAN); Prourokinase (plasminogen activator prolyse) (P) unclassified
D03325  Mometasone furoate hydrate (JAN); Mometasone furoate monohydrate; Nasonex (TN) (P) Enzyme: CYP3A4 / Target: NR3C1 / CYP induction: CYP3A4
D03337  Reviparin sodium (JAN); Clivarine (TN) (P) unclassified
D03341  Urokinase (JP18/USAN/INN); Abbokinase (TN) (P) unclassified
D03342  Camiglibose (USAN) (P) unclassified
D03352  Batroxobin (JAN/INN); Defibrase (TN) (P) unclassified
D03353  Dalteparin sodium (JAN/USP/INN); Ardeparin sodium; Fragmin (TN) (P) unclassified
D03359  Cangrelor (USAN/INN) (P) unclassified
D03361  Cangrelor tetrasodium (USAN); Kengreal (TN) (P) unclassified
D03363  Canrenone (USAN) (P) unclassified
D03385  Carbaspirin calcium (USAN); Carbasalate calcium (INN) (P) unclassified
D03415  Carvedilol phosphate (USAN); Carvedilol phosphate hydrate (JAN); Coreg CR (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D03471  Chlorothiazide sodium (USP); Diuril (TN) (P) unclassified
D03492  Cifenline (USAN); Cibenzoline (INN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D03493  Ciglitazone (USAN/INN) (P) unclassified
D03504  Cinacalcet (USAN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D03505  Cinacalcet hydrochloride (JAN/USAN); Sensipar (TN); Mimpara (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D03526  Cisconazole (USAN/INN) (P) unclassified
D03579  Codeine polistirex (USAN) (P) unclassified
D03580  Codeine sulfate (USP); Codeine sulfate trihydrate; Codeine sulfate (TN) (P) unclassified
D03644  Danaparoid sodium (JAN/USAN); Orgaran (TN) (P) unclassified
D03653  Darglitazone sodium (USAN) (P) unclassified
D03654  Darifenacin (USAN/INN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D03656  Darunavir (USAN/INN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D03658  Dasatinib (JAN/INN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D03661  Dazmegrel (USAN/INN) (P) unclassified
D03663  Dazoxiben hydrochloride (USAN) (P) unclassified
D03664  Debrisoquin sulfate (USAN); Declinax (TN) (P) unclassified
D03669  Deferasirox (JAN/USAN/INN); Exjade (TN); Jadenu (TN) (P) CYP induction: CYP3A4
D03671  Deflazacort (USAN/INN); Emflaza (TN) (P) Enzyme: CYP3A4 / Target: NR3C1 / CYP induction: CYP3A4
D03673  Deligoparin sodium (USAN/INN) (P) unclassified
D03674  Enoxaparin sodium (JAN/USP/INN); Lovenox (TN) (P) unclassified
D03692  Desirudin (USAN/INN); Iprivask (TN) (P) unclassified
D03695  Desmoteplase (USAN/INN) (P) unclassified
D03722  Efegatran sulfate (USAN) (P) unclassified
D03725  Hydrocodone bitartrate (USP); Hydrocodone bitartrate hemipentahydrate; Dicodid (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D03728  Napsagatran (USAN) (P) unclassified
D03731  Selegiline (USAN/INN); Emsam (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D03783  Oxycodone terephthalate (USP) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D03798  Dicumarol (USAN); Dicoumarol (INN); Dicumarol (TN) (P) unclassified
D03799  Dienogest (JAN/USAN/INN); Endometrion (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D03820  Dutasteride (JAN/USP/INN); Avodart (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D03825  Dihydrocodeine bitartrate (USP) (P) unclassified
D03830  Diltiazem malate (USAN); Tiamate (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D03833  Indinavir (USAN); Indinavir hydrate (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D03835  Fosamprenavir calcium (USAN); Lexiva (TN); Telzir (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D03837  Fosamprenavir sodium (USAN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D03839  Droxinavir hydrochloride (USAN) (P) unclassified
D03840  Palinavir (USAN/INN) (P) unclassified
D03842  Telinavir (USAN/INN) (P) unclassified
D03843  Tipranavir disodium (USAN) (P) unclassified
D03852  Droperidol and fentanyl citrate; Innovar (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D03865  Dirithromycin (USP/INN); Dynabac (TN) (P) unclassified
D03883  Doconazole (USAN/INN) (P) unclassified
D03917  Drospirenone (JAN/USP/INN); Slynd (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D03918  Drotrecogin alfa (activated) (USAN); Drotrecogin alfa; Xigris (TN) (P) unclassified
D03936  Econazole (USAN/INN) (P) unclassified
D03941  Edaglitazone sodium (USAN) (P) unclassified
D03960  Aspirin and dialuminate; Aspirin, aluminum glycinate and magnesium carbonate; Bufferin (TN) (P) unclassified
D03994  Endralazine mesylate (USAN); Endralazine monomethanesulfonate; Migranal (TN) (P) unclassified
D03996  Englitazone sodium (USAN) (P) unclassified
D03997  Enilconazole (USAN/INN) (P) unclassified
D04018  Ephedrine sulfate (USP); Akovaz (TN); Corphedra (TN); Emerphed (TN) (P) unclassified
D04023  Erlotinib hydrochloride (JAN/USAN); Tarceva (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D04024  Lapatinib ditosylate (USAN); Lapatinib tosilate hydrate (JAN); Lapatinib ditosylate monohydrate; Tykerb (TN); Tyverb (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D04029  Razaxaban hydrochloride (USAN) (P) unclassified
D04033  Epithiazide (USAN); Epitizide (INN) (P) unclassified
D04048  Ropivacaine hydrochloride (USP); Ropivacaine hydrochloride hydrate (JAN); Anapeine (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D04052  Epinephrine and lidocaine hydrochloride; Adrenaline and lidocaine hydrochloride; Xylocaine (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D04054  Erythromycin salnacedin (USAN); Erythromycin salnacedin dihydrate (P) unclassified
D04056  Esomeprazole sodium (USAN); Nexium IV (TN) (P) unclassified
D04061  Estradiol acetate (USAN); Femring (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D04063  Estradiol cypionate (USP); Depo-estradiol (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D04064  Estradiol enanthate (USAN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D04065  Estradiol undecylate (USAN/INN); Delestrec (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D04070  Estrogens, conjugated (JAN/USP); Conjugated estrogens; Premarin (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D04079  Ethacrynate sodium (USP) (P) unclassified
D04103  Etoformin hydrochloride (USAN) (P) unclassified
D04111  Etozolin (USAN/INN) (P) unclassified
D04112  Etravirine (JAN/USAN/INN); Intelence (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D04121  Exenatide (JAN/USAN/INN); Byetta (TN) (P) unclassified
D04145  Fendosal (USAN/INN); Alnovin (TN) (P) unclassified
D04148  Fenfluramine hydrochloride (JAN/USAN); Fintepla (TN); Pondimin (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D04161  Fenquizone (USAN/INN) (P) unclassified
D04183  Fidexaban (USAN/INN) (P) unclassified
D04206  Flufenisal (USAN/INN) (P) unclassified
D04214  Flunisolide acetate (USAN) (P) Enzyme: CYP3A4 / Target: NR3C1 / CYP induction: CYP3A4
D04265  Reserpine, hydralazine hydrochloride and hydrochlorothiazide (P) unclassified
D04266  Benzylhydrochlorothiazide, Reserpine and Carbazochrome; Behyd RA (TN) (P) unclassified
D04276  Furegrelate sodium (USAN) (P) unclassified
D04292  Galantamine (USAN/INN); Reminyl (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D04300  Ganaxolone (USAN/INN); Ztalmy (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D04313  Dihydrocodeine phosphate, dl-methylephedrine hydrochloride and Chlorpheniramine maleate; Huscode (TN) (P) unclassified
D04314  Gepirone hydrochloride (USAN); Exxua (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D04318  Glatiramer acetate (JAN/USAN); Copaxone (TN) (P) unclassified
D04322  Gliamilide (USAN/INN) (P) unclassified
D04338  Dihydrocodeine phosphate, ephedrine hydrochloride and ammmonium chloride; Sekicode (TN) (P) unclassified
D04340  Dextromethorphan hydrobromide and potassium cresolsulfonate; Medicon (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D04354  Glyhexamide (USAN/INN); Subose (TN) (P) unclassified
D04355  Glyoctamide (USAN/INN) (P) unclassified
D04356  Glyparamide (USAN) (P) unclassified
D04370  Granisetron (JAN/USAN/INN); Sancuso (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D04382  Guanethidine monosulfate (USP); Guanethidine sulfate (JP18); Ismelin (TN) (P) unclassified
D04386  Guanoclor sulfate (USAN); Vatensol (TN) (P) unclassified
D04398  Guanoxabenz (USAN/INN) (P) unclassified
D04399  Guanoxan sulfate (USAN); Envacar (TN) (P) unclassified
D04403  Guar gum (NF) (P) unclassified
D04427  Heparin calcium (JP18); Nadroparin calcium (INN); Calciparin; Calciparine (TN) (P) unclassified
D04446  Betamethasone acetate and betamethasone sodium phosphate; Celestone soluspan (TN); Rinderon (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D04447  Betamethasone and d-chlorpheniramine maleate; Celestamine (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D04458  Hydralazine polistirex (USAN) (P) unclassified
D04461  Hydrocodone polistirex (USAN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D04463  Norgestrel and ethinylestradiol tablets (JP18); Low-ogestrel (TN); Planovar (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D04475  Insulin aspart (USP/INN); Insulin aspart (genetical recombination) (JP18); Insulin aspart (genetical recombination) [Insulin aspart biosimilar 1] (JAN); Insulin X 14; NovoRapid (TN); Novolog (TN) (P) unclassified
D04477  Insulin lispro (USP/INN); Insulin lispro (genetical recombination) (JAN); Insulin lispro (genetical recombination) [Insulin lispro Biosimilar 1] (JAN); Insulin lispro-aabc; Humalog (TN); Lyumjev (TN) (P) unclassified
D04482  Ethinylestradiol and levonorgestrel; Ange (TN); Levora (TN); Lo/ovral (TN); Seasonique (TN); Triphasil-21 (TN); Trivora (TN) (P) unclassified
D04483  Ethinylestradiol and norethisterone; Norethindrone and ethinyl estradiol; Synphase T28 (TN) (P) unclassified
D04484  Desogestrel and ethinylestradiol; Marvelon21 (TN); Ortho-cept (TN) (P) unclassified
D04520  Indacrinone (USAN/INN) (P) unclassified
D04531  Indoramin (USAN/INN) (P) unclassified
D04532  Indoramin hydrochloride (USAN) (P) unclassified
D04539  Insulin detemir (USAN/INN); Insulin detemir (genetical recombination) (JAN); Levemir (TN) (P) unclassified
D04540  Insulin glulisine (USAN/INN); Insulin glulisine (genetical recombination) (JAN); Apidra (TN) (P) unclassified
D04541  Insulin human, isophane (USP) (P) unclassified
D04542  Insulin human zinc (USP) (P) unclassified
D04543  Insulin human zinc, extended (USP) (P) unclassified
D04547  Insulin, isophane (USP); Isophane insulin human (genetical recombination) injectable aqueous suspension (JP18); Isophane insulin (aqueous suspension) (JAN); Humalog PEN (TN) (P) unclassified
D04548  Insulin, neutral (USAN); Neutral insulin injection (INN) (P) unclassified
D04550  Insulin zinc, prompt (USP); Semilente iletin (TN) (P) unclassified
D04551  Insulin zinc (USP); Lente iletin (TN) (P) unclassified
D04624  Isoconazole (USAN/INN) (P) unclassified
D04641  Istradefylline (JAN/USAN/INN); Nourianz (TN); Nouriast (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D04645  Ixabepilone (JAN/USAN/INN); Ixempra (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D04665  Lanoteplase (USAN/INN); Lanoteplase (genetical recombination) (JAN) (P) unclassified
D04666  Lanreotide acetate (JAN/USAN); Somatuline (TN) (P) unclassified
D04716  Levomethadyl acetate (USAN); Levacetylmethadol (INN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D04725  Lexithromycin (USAN/INN) (P) unclassified
D04752  Lixivaptan (USAN/INN) (P) unclassified
D04768  Lonafarnib (JAN/USAN/INN); Zokinvy (TN) (P) unclassified
D04799  Heparinoid (JAN); Hirudoid (TN) (P) unclassified
D04813  Lidocaine hydrochloride and epinephrine bitartrate; Lidocaine hydrochloride and adrenaline bitartrate; Ora (TN); Lidosite (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D04820  Lurasidone hydrochloride (JAN/USAN); SM 13496; Latuda (TN) (CI,P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D04859  Maribavir (JAN/USAN/INN); Camvia (TN); Livtencity (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D04866  Freeze-dried live attenuated measles vaccine (JP18) (CI) unclassified
D04895  Mefloquine (USAN/INN) (P) unclassified
D04896  Megalomicin potassium phosphate (USAN) (P) unclassified
D04966  Metformin (USAN/INN) (P) unclassified
D04970  Methacholine chloride (JAN/USP/INN); Provocholine (TN) (P) unclassified
D04976  Methalthiazide (USAN) (P) unclassified
D04977  Parnaparin sodium (JP18); Lowhepa (TN) (P) unclassified
D05000  Methylprednisolone hemisuccinate (USP); Methylprednisolone succinate (JP18) (P) Enzyme: CYP3A4 / Target: NR3C1 / CYP induction: CYP3A4
D05001  Methylprednisolone sodium phosphate (USAN) (P) Enzyme: CYP3A4 / Target: NR3C1 / CYP induction: CYP3A4
D05002  Methylprednisolone suleptanate (USAN/INN) (P) Enzyme: CYP3A4 / Target: NR3C1 / CYP induction: CYP3A4
D05028  Midazolam maleate (USAN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D05029  Midostaurin (JAN/USAN/INN); Rydapt (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D05037  Trimetoquinol hydrochloride hydrate (JP18); Tretoquinol hydrate; Caluyon (TN) (P) unclassified
D05087  Moxonidine (USAN/INN); Cynt (TN) (P) unclassified
D05089  Freeze-dried live attenuated mumps vaccine (JP18); Freeze-dried live attenuated mumps vaccine (TN) (CI) unclassified
D05093  Muzolimine (USAN/INN) (P) unclassified
D05123  Nasaruplase beta (USAN/INN); Prolyse (TN) (P) unclassified
D05150  Netoglitazone (USAN/INN) (P) unclassified
D05153  Neutramycin (USAN) (P) unclassified
D05181  Aspirin aluminum (JP18) (P) unclassified
D05248  Freeze-dried inactivated tissue culture ravies vaccine (JP18) (P) unclassified
D05259  Omeprazole magnesium (USP); Prilosec OTC (TN) (P) unclassified
D05261  Omeprazole sodium injection (JAN); Omeprazole sodium hydrate; Omepral (TN) (P) unclassified
D05268  Orconazole nitrate (USAN) (P) unclassified
D05277  Formoterol fumarate hydrate (JP18); Formoterol fumarate dihydrate; Atock (TN); Foradil (TN) (P) unclassified
D05312  Oxycodone (USAN/INN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D05323  Ozolinone (USAN) (P) unclassified
D05333  Paclitaxel poliglumex (USAN/INN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D05343  Palonosetron hydrochloride (JAN/USP); Aloxi (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D05351  Josamycin propionate (JP18); Josamy (TN) (P) CYP inhibition: CYP3A4
D05353  Pantoprazole (USAN/INN) (P) unclassified
D05366  Procaterol hydrochloride hydrate (JP18); Meptin (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D05367  Parconazole hydrochloride (USAN) (P) unclassified
D05380  Pazopanib hydrochloride (JAN/USAN); Votrient (TN) (P) unclassified
D05382  Pazufloxacin mesilate (JP18); Pazufloxacin methanesulfonate; Pasil (TN) (P) unclassified
D05387  Pegaspargase (JAN/USAN/INN); Oncaspar (TN) (P) unclassified
D05410  Pamiteplase (INN); Pamiteplase (genetical recombination) (JAN); Solinase (TN) (P) unclassified
D05412  Monteplase (INN); Monteplase (genetical recombination) (JAN); Cleactor (TN) (P) unclassified
D05457  Phenprocoumon (USAN/INN); Liquamar (TN) (P) unclassified
D05462  Oxycodone hydrochloride hydrate (JP18) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D05482  Pinacidil (USAN); Pinacidil hydrate; Pindac (TN) (P) unclassified
D05502  Pirmagrel (USAN/INN); CGS 13080 (P) unclassified
D05538  Mozenavir (INN) (P) unclassified
D05594  Pramlintide (USAN/INN) (P) unclassified
D05595  Pramlintide acetate (USAN); Symlin (TN) (P) unclassified
D05597  Prasugrel hydrochloride (JAN/USAN); Effient (TN) (P) unclassified
D05622  Proinsulin human (USAN) (P) unclassified
D05640  Prorenoate potassium (USAN/INN) (P) unclassified
D05681  Quinine ascorbate (USAN); Quinine biascorbate (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D05705  Rauwolfia serpentina (USP); Rauwolfia extract; Himolfia (TN) (P) unclassified
D05713  Relomycin (USAN/INN) (P) unclassified
D05717  Repromicin (USAN/INN) (P) unclassified
D05721  Reteplase (USAN/INN); Retevase (TN) (P) unclassified
D05727  Ridogrel (USAN/INN) (P) unclassified
D05739  Rivoglitazone (USAN/INN) (P) unclassified
D05744  Roflumilast (JAN/USAN/INN); Daliresp (TN); Zoryve (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D05757  Rosaramicin (USAN/INN) (P) unclassified
D05758  Rosaramicin butyrate (USAN) (P) unclassified
D05759  Rosaramicin propionate (USAN) (P) unclassified
D05760  Rosaramicin sodium phosphate (USAN) (P) unclassified
D05761  Rosaramicin stearate (USAN) (P) unclassified
D05775  Rufinamide (JAN/USP/INN); Banzel (TN) (P) unclassified
D05788  Salcolex (USAN); Salcolex tetrahydrate (P) unclassified
D05789  Salethamide maleate (USAN) (P) unclassified
D05791  Salicylate meglumine (USAN) (P) unclassified
D05792  Salmeterol (USAN/INN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D05793  Salnacedin (USAN/INN) (P) unclassified
D05800  Saperconazole (USAN/INN) (P) unclassified
D05811  Sedecamycin (USAN/INN) (P) unclassified
D05908  Spiramycin (JAN/USAN/INN); Rovamycin (TN) (P) unclassified
D05912  Spiroxasone (USAN/INN) (P) unclassified
D05928  Stiripentol (JAN/USAN/INN); Diacomit (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D05932  Streptozocin (JAN/USAN/INN); Streptozotocin; Zanosar (TN) (P) unclassified
D05987  Synthetic conjugated estrogens, B (USAN); Enjuvia (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D05998  Talosalate (USAN/INN) (P) unclassified
D06068  Temsirolimus (JAN/USAN/INN); Torisel (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D06070  Tenecteplase (USAN/INN); Tnkase (TN) (P) unclassified
D06142  Tifacogin (USAN/INN) (P) unclassified
D06177  Tolbutamide sodium, sterile; Orinase diagnostic (TN) (P) unclassified
D06186  Tolpyrramide (USAN/INN) (P) unclassified
D06199  Trabectedin (JAN/USAN/INN); Yondelis (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D06213  Treprostinil (JAN/USAN/INN); Remodulin (TN) (P) unclassified
D06234  Trimazosin hydrochloride (USAN); Trimazosin hydrochloride monohydrate (P) unclassified
D06256  Tuberculin (USP); Purified tuberculin; Aplisol (TN) (P) unclassified
D06258  Tulathromycin (JAN/USAN/INN) (P) unclassified
D06270  Urokinase alfa (USAN/INN); r-UK (TN) (P) unclassified
D06272  Sorafenib tosylate (USAN); Sorafenib tosilate (JAN); Nexavar (TN) (P) unclassified
D06273  Imidafenacin (JAN/INN); Uritos (TN); Staybla (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D06315  Fluticasone furoate (JAN/USAN/INN); Veramyst (TN) (P) Enzyme: CYP3A4 / Target: NR3C1 / CYP induction: CYP3A4
D06341  Xipamide (USAN) (P) unclassified
D06347  Yellow fever vaccine (USP); YF-Vax (TN) (CI) unclassified
D06373  Zinoconazole hydrochloride (USAN) (P) unclassified
D06390  Azithromycin (USP); Zmax (TN) (P) unclassified
D06398  Tinzaparin sodium (USAN); Innohep (TN) (P) unclassified
D06401  Indapamide hydrate; Tenaxil (TN) (P) unclassified
D06402  Sunitinib malate (JAN/USAN); Sutent (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D06404  Liraglutide (USAN/INN); Liraglutide (genetical recombination) (JAN); Victoza (TN) (P) unclassified
D06405  Nalfurafine hydrochloride (JAN/USAN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D06407  Vandetanib (JAN/USAN/INN); Caprelsa (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D06410  Thrombomodulin alfa (USAN/INN); Thrombomodulin alfa (genetical recombination) (JAN) (P) unclassified
D06412  Aliskiren fumarate (JAN/USAN); Aliskiren hemifumarate; Tekturna (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D06413  Nilotinib hydrochloride hydrate (JAN); Nilotinib monohydrochloride monohydrate; Tasigna (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D06414  Dasatinib (USAN); Dasatinib hydrate (JAN); Sprycel (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D06466  Freeze-dried BCG for intravesical use; Immunobladder (TN); Tice BCG (TN) (CI) unclassified
D06478  Darunavir ethanolate (JAN); Prezista (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D06511  Freeze-dried smallpox vaccine prepared in cell culture (JP18) (CI) unclassified
D06512  Freeze-dried live attenuated rubella vaccine (JP18) (CI) unclassified
D06553  Alogliptin benzoate (JAN/USAN); Vipidia (TN); Nesina (TN) (P) unclassified
D06571  Antithrombin III human (USP); Antithrombin III (INN); Kybernin (TN) (P) unclassified
D06578  Denagliptin tosylate (USAN) (P) unclassified
D06597  Fosaprepitant dimeglumine (USAN); Fosaprepitant meglumine (JAN); Proemend (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D06598  Gamithromycin (USAN/INN) (P) unclassified
D06606  Ibuprofen lysine (USAN); Ibuprofen L-lysine (JAN); Solufenum; Neoprofen (TN) (P) unclassified
D06630  Pramiconazole (USAN/INN) (P) unclassified
D06641  Sergliflozin etabonate (USAN) (P) unclassified
D06645  Sitagliptin phosphate (USAN); Sitagliptin phosphate hydrate (JP18); Sitagliptin phosphate monohydrate; Januvia (TN) (P) unclassified
D06670  Maraviroc (JAN/INN); Selzentry (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D06879  Streptokinase (INN); Streptase (TN) (P) unclassified
D06880  Lepirudin (INN); Refludan (TN) (P) unclassified
D06883  Sertaconazole (INN) (P) unclassified
D06888  Eptifibatide (INN); Integrilin (TN) (P) unclassified
D07064  Acenocoumarol (INN); Acenocoumarin; Mini-sintrom (TN) (P) unclassified
D07073  Dexamethasone cipecilate (JAN/INN) (P) Enzyme: CYP3A4 / Target: NR3C1 / CYP induction: CYP3A4
D07077  Ambrisentan (JAN/INN); Letairis (TN); Volibris (TN) (P) unclassified
D07080  Vildagliptin (JAN/USAN/INN); Equa (TN); Galvus (TN) (P) unclassified
D07082  Dabigatran etexilate mesylate (USAN); Dabigatran etexilate methanesulfonate (JAN); Dabigatran etexilate mesilate; Pradaxa (TN) (P) unclassified
D07086  Rivaroxaban (JAN/USAN/INN); Xarelto (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D07113  Loperamide oxide (INN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D07117  Metahexamide (INN) (P) unclassified
D07118  Glisoxepide (INN) (P) unclassified
D07124  Alfuzosin (INN); Xatral (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D07129  Alosetron (INN) (P) unclassified
D07131  Ethyl biscoumacetate (INN) (P) unclassified
D07132  Buprenorphine (JAN/INN); Temgesic (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D07135  Clorindione (INN); G-25766 (P) unclassified
D07136  Diphenadione (INN) (P) unclassified
D07137  Tioclomarol (INN) (P) unclassified
D07138  Ditazole (INN) (P) unclassified
D07139  Cloricromen (INN) (P) unclassified
D07140  Picotamide (BAN); Plactidil (TN) (P) unclassified
D07141  Indobufen (INN) (P) unclassified
D07142  Triflusal (INN) (P) unclassified
D07143  Melagatran (INN) (P) unclassified
D07144  Dabigatran etexilate (USAN/INN); Pradaxa (TN) (P) unclassified
D07165  Ivabradine (USAN/INN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D07166  Methoserpidine (INN) (P) unclassified
D07167  Bietaserpine (prop.INN) (P) unclassified
D07168  Tolonidine (INN) (P) unclassified
D07169  Guanazodine (INN) (P) unclassified
D07170  Dihydralazine (INN) (P) unclassified
D07171  Sitaxentan (USAN/INN) (P) unclassified
D07172  Mebutizide (INN) (P) unclassified
D07175  Palonosetron (INN); Aloxi (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D07192  Benfluorex (INN/BAN); Mediaxal (TN) (P) unclassified
D07193  Flutrimazole (INN) (P) unclassified
D07203  Methylprednisolone aceponate (INN); Advantan (TN) (P) Enzyme: CYP3A4 / Target: NR3C1 / CYP induction: CYP3A4
D07226  Fesoterodine (INN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D07242  Flurithromycin (INN) (P) unclassified
D07283  Esketamine (USAN/INN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D07290  Dipyrocetyl (INN) (P) unclassified
D07291  Benorilate (INN); Benorylate (P) unclassified
D07292  Guacetisal (INN); Prontomucil (TN) (P) unclassified
D07293  Imidazole salicylate (INN); Selezen (TN) (P) unclassified
D07299  Lacosamide (JAN/USAN/INN); Erlosamide; Vimpat (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D07402  Levocetirizine (USAN/INN); Xazal (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D07407  Rupatadine (INN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D07421  Aloxiprin (INN); Superpyrin (TN) (P) unclassified
D07422  Fibrinolysin (human) (INN); Fibrinolysin, human; Fibrogammin (TN) (P) unclassified
D07447  Amiloride (INN); Amiclaran (TN) (P) unclassified
D07448  Amitriptyline (INN); Laroxyl (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D07450  Amlodipine (USP/INN); Norvasc (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D07457  Anisindione (INN); Miradon (TN) (P) unclassified
D07471  Atazanavir (INN); Reyataz (TN) (P) CYP inhibition: CYP3A4
D07474  Atorvastatin (INN); Lipitor (TN); Sortis (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D07486  Azithromycin (INN); Azasite (TN); Azithromycin (TN) (P) unclassified
D07488  Balsalazide (INN) (P) unclassified
D07494  Barnidipine (INN); Vasexten (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D07508  Benfluorex hydrochloride; Mediator (TN) (P) unclassified
D07509  Benidipine (INN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D07510  Adomiparin (USAN); Semuloparin (USAN); Heparin (BAN); Enoxaparin; Bemiparin; Parnaparin; Nadroparin; Heparin (TN) (P) unclassified
D07520  Bepridil (INN); Bepadin (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D07538  Bosentan (INN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D07552  Bupivacaine (USAN/INN); Bucaine (TN); Exparel (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D07569  Candesartan cilexetil and anmlodipine besylate (JP18); Unisia (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D07579  Aspirin calcium salt; Notras (TN) (P) unclassified
D07580  Aspirin DL-lysine (JAN); Aspirin lysine salt; Aspegic (TN) (P) unclassified
D07581  Aspirin magnesium salt; Mobidin (TN) (P) unclassified
D07582  Aspirin sodium; Sodium acetylsalicylate; Catalgine (TN) (P) unclassified
D07583  Phenytoin and phenobarbital; Aleviatin with phenobarbital (TN) (P) unclassified
D07585  Isopropylantipyrine, ergotamine tartrate and anhydrous caffeine; Cleamine A (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D07595  Fosphenytoin sodium hydrate (JAN); Fostoin (TN) (P) CYP induction: CYP3A4
D07598  Butoconazole (INN); Gynofort (TN) (P) unclassified
D07603  Caffeine citrate (USP); Cafcit (TN) (P) unclassified
D07612  Sodium salamidacetate; o-Carbamoylphenoxyacetic acid sodium salt; Clinit-n (TN) (P) unclassified
D07626  Caspofungin (INN); Cancidas (TN) (P) unclassified
D07661  Cerivastatin (INN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D07667  Cevimeline (INN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D07676  Chlormidazole hydrochloride; Unfungicid (TN) (P) unclassified
D07704  Citalopram (USP/INN); Citadur (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D07705  Citalopram hydrochloride; Seropram (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D07710  Clarithromycin lactobionate; Klacid (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D07727  Clomipramine (INN); Anafranil (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D07729  Clopidogrel (USP/INN); Clopidogrel (TN); Plavix (TN) (P) unclassified
D07736  Cloricromen hydrohloride; Proendotel (TN) (P) unclassified
D07740  Codeine hydrochloride; Bisoltus (TN) (P) unclassified
D07748  Conivaptan (INN) (P) unclassified
D07752  Croconazole (INN) (P) unclassified
D07760  Cyclophosphamide (INN); Cyclophosphamide (TN); Cytoxan (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D07793  Desvenlafaxine (INN); Khedezla (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D07796  Dexamethasone 21-acetate; Dexamethasone acetate anhydrous; Decaject-L.A. (TN) (P) Enzyme: CYP3A4 / Target: NR3C1 / CYP induction: CYP3A4
D07797  Dexamethasone isonicotinate; Dexamethasone 21-isonicotinate; Voren [veterinary] (TN) (P) Enzyme: CYP3A4 / Target: NR3C1 / CYP induction: CYP3A4
D07798  Dexamethasone sodium hemisulfate; Dexamethasone 21-sodium sulfate; Colircusi Dexametasona (TN) (P) Enzyme: CYP3A4 / Target: NR3C1 / CYP induction: CYP3A4
D07799  Dexamethasone 21-tebutate; Dexamethasone tertiary butyl acetate; Dexamedium [veterinary] (TN) (P) Enzyme: CYP3A4 / Target: NR3C1 / CYP induction: CYP3A4
D07800  Dexamethasone 21-valerate; Voalla (TN); Zalucs (TN) (P) Enzyme: CYP3A4 / Target: NR3C1 / CYP induction: CYP3A4
D07801  Dexamethasone phenylpropionate; Dexafort [veterinary] (TN) (P) Enzyme: CYP3A4 / Target: NR3C1 / CYP induction: CYP3A4
D07802  Dexamethasone phosphate; Decadron-phosphate (TN) (P) Enzyme: CYP3A4 / Target: NR3C1 / CYP induction: CYP3A4
D07824  Diethylamine salicylate; Algesal (TN) (P) unclassified
D07830  Dihydralazine sulfate; Dihydralazine hydrogen sulfate; Nepresol (TN) (P) unclassified
D07831  Dihydrocodeine (INN); Remedacen (TN) (P) unclassified
D07832  Dihydrocodeine thiocyanate; Paracodin (TN) (P) unclassified
D07837  Dihydroergotamine (INN); Neomigran (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D07838  Dihydroergotamine tartrate; Divegal (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D07839  Dihydroergotoxine; Co-Dergocrin (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D07845  Diltiazem (INN); Surazem (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D07866  Docetaxel (JAN/INN); Docetaxel (TN); Taxotere (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D07868  Domperidone maleate; Domperidone (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D07869  Donepezil (JAN/INN); Donaz (TN); Allydone (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D07871  Dorzolamide (INN); Trusopt (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D07873  Doxapram (INN); Docatone (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D07874  Doxazosin (INN); Cardura XL (TN) (P) unclassified
D07882  Eberconazole (INN) (P) unclassified
D07884  Eberconazole nitrate; Ebernet (TN) (P) unclassified
D07887  Eletriptan (INN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D07895  Losartan potassium and hydrochlorothiazide (JP18); Hydrochlorothiazide and losartan potassium; Hyzaar (TN); Losarhyd (TN) (P) unclassified
D07905  Ergometrine (INN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D07906  Ergotamine (INN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D07907  Erlotinib (INN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D07909  Erythromycin thiocyanate; Erythrocin (TN) (P) unclassified
D07910  Erythromycin stinoprate (INN); Erysec (TN) (P) unclassified
D07913  Escitalopram (INN); Esertia (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D07917  Esomeprazole (INN); Inexium paranova (TN) (P) unclassified
D07918  Estradiol hemihydrate; Estrasorb (TN); Vagifem (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D07919  Estradiol 17 beta-hemisuccinate; 17beta-Estradiol hemisuccinate; Eutocol (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D07928  Ethinylestradiol propanesulfonate; Turisteron (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D07929  Ethylmorphine (BAN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D07945  Fenfluramine (INN); Ponderax (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D07955  Fenquizone potassium salt; Idrolone (TN) (P) unclassified
D07969  Fluindione (INN); Previsccan (TN) (P) unclassified
D07981  Fluticasone (INN); Fluticaps (TN) (P) Enzyme: CYP3A4 / Target: NR3C1 / CYP induction: CYP3A4
D07983  Fluvastatin (INN); Fluvas (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D07991  Fosfosal (INN); Aydolid (TN) (P) unclassified
D07993  Fosphenytoin (INN) (P) CYP induction: CYP3A4
D07999  Sodium furosemide; Frosemide sodium; Lasix (TN) (P) unclassified
D08001  Furosemide diolamine; Furosemide diethanolamine salt; Nuriban (TN) (P) unclassified
D08004  Gabexate (INN) (P) unclassified
D08030  Guanethidine (INN) (P) unclassified
D08031  Guanfacine (INN); Estulic (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D08035  Haloperidol lactate; Haldol (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D08044  Hydralazine (INN); Hidral (TN) (P) unclassified
D08045  Hydrocodone (INN); Dihydrocodeinone (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D08046  Hydrocodone hydrochloride; Dihydrocodeinone hydrochloride; Dicodid (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D08050  Hydroxychloroquine (INN); Polirreumin (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D08065  Iloprost tromethamine; Iloprost trometamol; Ventavis (TN) (P) unclassified
D08066  Imatinib (INN); Glamox (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D08070  Imipramine (INN); Tofranil (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D08071  Imipramine pamoate (USP); Imipramine embonate; Tofranil-pm (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D08080  Insulin injection, biphasic isophane (BAN); Biphasic isophane insuline human (genetical recombination) injectable aqueous suspension (JP18); Insulin Humacart (TN) (P) unclassified
D08086  Irinotecan (INN); Biotecan (TN) (P) unclassified
D08095  Ivabradine hydrochloride (JAN/USAN); Ivabrandine hydrochloride; Corlanor (TN); Corlentor (TN); Coralan (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D08099  Ketanserin tartrate; Sufrexal (TN) (P) unclassified
D08108  Lapatinib (INN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D08116  Levobupivacaine (INN); Novabupi (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D08118  Levocetirizine dihydrochloride (USP); Levocetirizine hydrochloride (JAN); Xyzal (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D08127  Lidocaine hydrochloride monohydrate; Lidocaine (TN); Zingo (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D08144  Loperamide (INN); Diamide (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D08148  Loxapine hydrochloride; Desconex (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D08155  Manidipine (INN); Manidipine 6300; Artedil (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D08194  Deserpidine (INN); Halmonyl (TN) (P) unclassified
D08195  Methadone (BAN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D08205  Methyldopa (INN); Aldomet (TN) (P) unclassified
D08207  Methylergometrine (INN); Ergotyl (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D08212  Trimazosin (INN) (P) unclassified
D08216  Mianserin (INN); Tolvon (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D08227  Mometasone (INN) (P) Enzyme: CYP3A4 / Target: NR3C1 / CYP induction: CYP3A4
D08229  Montelukast (INN); Brondilat (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D08236  Mosapride (INN); Mosart (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D08240  Nafamostat (INN) (P) unclassified
D08254  Endralazine (INN) (P) unclassified
D08255  Naratriptan (INN); Naramig (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D08256  Nateplase (INN); Milyzer (TN); Tepase (TN) (P) unclassified
D08259  Nelfinavir (INN); Viracept (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D08270  Nicardipine (INN); Cardene (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D08283  Nordazepam (INN); Calmday (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D08291  Ofloxacin hydrochloride; Tarivid (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D08295  Olsalazine (INN) (P) unclassified
D08296  Omoconazole (INN) (P) unclassified
D08313  Oxiconazole (INN) (P) unclassified
D08327  Ozagrel (INN); Cataclot (TN) (P) unclassified
D08351  Phenformin (BAN) (P) unclassified
D08352  Phenformin hydrochloride; Debei (TN) (P) unclassified
D08354  Phenindione (INN); Hedulin (TN) (P) unclassified
D08356  Phenobarbital diethylamine; Gratusminal (TN) (P) unclassified
D08378  Pioglitazone (INN); Actos (TN) (P) unclassified
D08408  Pranlukast (INN); Azlaire (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D08411  Prazosin (INN); Minipress (TN) (P) unclassified
D08424  Procaterol (INN); Meptin (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D08435  Propafenone (INN); Propafenon hexal (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D08441  Propiverine (INN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D08453  Pargyline (INN) (P) unclassified
D08456  Quetiapine (INN); Norsic (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D08460  Quinine (BAN); Kinder Quinina (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D08461  Quinine dihydrochloride; Quinine (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D08463  Rabeprazole (INN); Eraloc (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D08479  Rifampicin sodium; Rifadine (TN) (P) CYP induction: CYP3A4
D08481  Rilmazafone (INN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D08482  Rilmenidine (INN); Hyperium (TN) (P) unclassified
D08488  Amlodipine besilate and atorvastatin calcium; Caduet (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D08490  Ropivacaine (INN); Naropin (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D08491  Rosiglitazone (INN); Gaudil (TN) (P) unclassified
D08493  Dorzolamide hydrochloride and timolol maleate (JP18); Cosopt (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D08497  Rupatadine fumarate (JAN); Rinialer (TN); Rupafin (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D08501  Trolamine salicylate (USP); Salicylic acid trolamine; Salicylic acid triethanolamine; Arthricream (TN) (P) unclassified
D08508  Sarpogrelate (INN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D08510  Sertaconazole nitrate; Ertaczo (TN); Zalain (TN) (P) unclassified
D08514  Sildenafil (INN); Aphrodil (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D08516  Sitagliptin (USAN/INN) (P) unclassified
D08517  Sitaxentan sodium (USAN); Thelin (TN) (P) unclassified
D08522  Solifenacin (INN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D08527  Spiramycin adipate; Rovamycina (TN); Spiramaicina (TN) (P) unclassified
D08528  Spiramycin embonate; Cofamix STS (TN) (P) unclassified
D08535  Sulconazole (INN) (P) unclassified
D08536  Suleparoid; Heparitin sulfate; Aremin (TN) (P) unclassified
D08547  Sulodexide (INN); Vessel (TN) (P) unclassified
D08552  Sunitinib (INN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D08556  Tacrolimus (INN); Prograf (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D08559  Tamoxifen (INN); Tamoxifen (TN); Tamoplex (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D08575  Tetrabenazine (JAN/INN); Nitoman (TN); Xenazine (TN) (P) unclassified
D08586  Thiosalicylic acid; Pirosal (TN); Thiocyl (TN) (P) unclassified
D08594  Ticlopidine (INN); Ticlopidin-Puren (TN) (P) unclassified
D08605  Tipranavir (INN); Aptivus (TN) (P) unclassified
D08607  Tirofiban (INN); Agrastat (TN) (P) unclassified
D08609  Tisokinase (JAN) (P) unclassified
D08616  Teneligliptin (INN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D08619  Torasemide sodium; Torem (TN) (P) unclassified
D08620  Toremifene (INN); Fareston (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D08623  Tramadol (INN); Amanda (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D08626  Trazodone (INN); Trittico (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D08628  Treprostinil monosodium salt; Treprostinil sodium; Trepulmix (TN) (P) unclassified
D08631  Carmegliptin (USAN/INN) (P) unclassified
D08662  Urapidil hydrochloride; Ebrantil (TN) (P) unclassified
D08668  Vardenafil (USAN/INN); Levitra (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D08670  Venlafaxine (INN); Efectin (TN) (P) unclassified
D08675  Vinblastine (INN); Vinblastina (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D08680  Vinorelbine (INN); Navelbine (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D08682  Warfarin (INN); Warfarine; Choice (TN) (P) unclassified
D08690  Zolpidem (INN); Sanval (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D08695  dl-Methylephedrine hydrochloride, dihydrocodeine phosphate, diprophylline, diphenhydramine salicylate, acetaminophen and bromovalerylurea; Coughcode N (TN) (P) unclassified
D08697  Platycodon fluidextract, glycyrrhiza extract, plantago herb extract, peony root extract and dihydrocodeine phosphate; Opisezol codeine (TN) (P) unclassified
D08699  Salmeterol xinafoate and fluticasone propionate; Adoair diskus (TN); Aerivio Spiromax (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D08774  Amoxicillin hydrate, clarithromycin and lansoprazole; Lansap (TN); Prevpac (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D08777  Freeze-dried live attenuated varicella vaccine (CI) unclassified
D08795  Human antithrombin III, freeze-dried concentrated; Neuart (TN) (P) unclassified
D08804  Freeze-dried live attenuated measles-rubella combined vaccine; Mearubik (TN) (CI) unclassified
D08843  Albiglutide (USAN); Albiglutide (genetical recombination) (JAN); Tanzeum (TN) (P) unclassified
D08856  Anamorelin hydrochloride (JAN/USAN); Adlumiz (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D08858  Antithrombin alfa (INN/USAN); Atryn (TN) (P) unclassified
D08860  Apremilast (JAN/USAN); Otezla (TN) (P) unclassified
D08870  Belinostat (USAN/INN); Beleodaq (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D08873  Betrixaban (USAN); Bevyxxa (TN) (P) unclassified
D08897  Dapagliflozin (JAN/USAN/INN); Forxiga (TN) (P) unclassified
D08903  Dexlansoprazole (INN/USAN); Dexilant (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D08913  Eribaxaban (USAN) (P) unclassified
D08914  Eribulin mesylate (USAN); Eribulin mesilate (JAN); Halaven (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D08923  Fesoterodine fumarate (JAN/USAN); Toviaz (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D08950  Neratinib (USAN/INN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D08953  Nilotinib (USAN/INN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D08962  Pamabrom (USP) (P) unclassified
D08969  Pimavanserin tartrate (USAN); Nuplazide (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D08976  Pomalidomide (JAN/USAN/INN); Pomalyst (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D08988  Rolapitant hydrochloride (USAN); Varubi (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D08996  Saxagliptin (USAN/INN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D09012  Telaprevir (JAN/USAN/INN); Incivek (TN); Incivo (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D09013  Teplizumab (USAN/INN); Teplizumab-mzwv; Tzield (TN) (P) unclassified
D09017  Ticagrelor (JAN/USAN/INN); Brilinta (TN) (CI,P) unclassified
D09033  Voclosporin (JAN/USAN/INN); Lupkynis (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D09187  Estradiol and levonorgestrel; Wellnara (TN); Climara pro (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D09188  Estradiol and norethindrone; Menoaid (TN); Activella (TN); Combipatch (TN); Estradiol and norethindrone acetate (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D09196  Candesartan cilexetil and hydrochlorothiazide (JP18); Ecard HD (TN); Ecard LD (TN) (P) unclassified
D09197  Valsartan and hydrochlorothiazide (JP18); Co-dio (TN) (P) unclassified
D09206  Saruplase (INN); Prourokinase (enzyme activating) (human clone pUK4/pUK18), nonglycosylated (P) unclassified
D09215  Eslicarbazepine (USAN/INN) (P) CYP induction: CYP3A4
D09219  Telmisartan and hydrochlorothiazide (JP18); Micombi (TN); Micardis hct (TN) (P) unclassified
D09318  Indacaterol (USAN/INN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D09319  Indacaterol maleate (JAN/USAN); Arcapta neohaler (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D09326  Carmegliptin dihydrochloride (USAN) (P) unclassified
D09333  Dutogliptin (USAN) (P) unclassified
D09334  Dutogliptin tartrate (USAN) (P) unclassified
D09339  Esomeprazole potassium (USAN) (P) unclassified
D09347  Fostamatinib (USAN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D09348  Fostamatinib disodium (USAN); Fostamatinib sodium hydrate (JAN); Fostamatinib disodium hexahydrate; Tavalisse (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D09365  Palovarotene (JAN/USAN/INN); Sohonos (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D09388  Tasimelteon (USAN/INN); Hetlioz (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D09394  Fidaxomicin (JAN/USAN); Dificid (TN); Dificlir (TN) (P) CYP inhibition: CYP3A4
D09535  Mirabegron (JAN/USAN/INN); Myrbetriq (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D09544  Ozenoxacin (JAN/USAN/INN); Xepi (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D09546  Edoxaban tosilate hydrate (JAN); Edoxaban tosylate monohydrate; Lixiana (TN); Savaysa (TN) (P) unclassified
D09566  Linagliptin (JAN/USAN/INN); Tradjenta (TN) (P) unclassified
D09572  Riociguat (JAN/USAN/INN); Adempas (TN) (P) unclassified
D09592  Canagliflozin (USAN/INN); Canagliflozin hydrate (JAN); Invokana (TN) (P) unclassified
D09594  Olmesartan medoxomil and azelnidipine; Rezaltas (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D09595  Budesonide and formoterol fumarate dihydrate; Symbicort (TN); Budeforu (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D09605  Duvoglustat (USAN/INN); 1-Deoxynojirimycin (P) unclassified
D09606  Duvoglustat hydrochloride (USAN) (P) unclassified
D09612  Eslicarbazepine acetate (USAN); Zebinix (TN); Aptiom (TN) (P) CYP induction: CYP3A4
D09625  Gosogliptin (USAN/INN) (P) unclassified
D09637  Lomitapide (USAN/INN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D09638  Lomitapide mesylate (USAN); Lomitapide mesilate (JAN); Juxtapid (TN); Lojuxta (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D09642  Modithromycin (USAN/INN) (P) unclassified
D09666  Selumetinib (USAN/INN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D09676  Tecarfarin (USAN/INN) (P) unclassified
D09677  Tecarfarin sodium (USAN) (P) unclassified
D09683  Tivozanib (USAN/INN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D09698  Vilazodone (USAN/INN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D09699  Vilazodone hydrochloride (USAN); Viibryd (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D09701  Abiraterone acetate (JAN/USP); Zytiga (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D09702  Albaconazole (USAN/INN) (P) unclassified
D09707  Dabigatran (USAN/INN) (P) unclassified
D09710  Edoxaban (USAN/INN) (P) unclassified
D09720  Rilpivirine (JAN/USAN/INN); Rekambys (TN) (CI) unclassified
D09723  Taspoglutide (USAN/INN) (P) unclassified
D09727  Insulin degludec (USAN/INN); Insulin degludec (genetical recombination) (JAN); Tresiba (TN) (P) unclassified
D09728  Bosutinib hydrate (JAN); Bosutinib monohydrate; Bosulif (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D09729  Lixisenatide (JAN/USAN/INN); Adlyxin (TN); Lyxumia (TN) (P) unclassified
D09730  Olaparib (JAN/USAN/INN); Lynparza (TN) (P) unclassified
D09731  Crizotinib (JAN/USAN/INN); Xalkori (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D09736  Iron (III) hexacyanoferrate (II); Radiogardase (TN) (P) unclassified
D09741  Drospirenone and ethinylestradiol; Drospirenone and ethinylestradiol betadex; Angeliq (TN); Yaz (TN); Flexyess (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D09742  Lansoprazole, amoxicillin hydrate and metronidazole; Lampion (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D09743  Telmisartan and amlodipine besilate (JP18); Telmisartan and amlodipine besylate; Micamlo (TN); Twynsta (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D09744  Pioglitazone hydrochloride and metformin hydrochloride (JP18); Pioglitazone and metformin; Metact (TN) (P) unclassified
D09745  Valsartan and amlodipine besilate; Exforge (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D09753  Saxagliptin hydrate (JAN); Onglyza (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D09756  Teneligliptin hydrobromide hydrate (JAN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D09763  Dapagliflozin propanediol (USAN); Dapagliflozin propylene glycolate hydrate (JAN); Dapagliflozin propandiol monohydrate; Forxiga (TN); Farxiga (TN) (P) unclassified
D09765  Vorapaxar (USAN/INN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D09766  Vorapaxar sulfate (JAN/USAN); Zontivity (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D09772  Alilusem potassium (JAN); M17055 (P) unclassified
D09779  Emiglitate (JAN/INN) (P) unclassified
D09780  Anagliptin (JAN/INN) (P) unclassified
D09783  Tofacitinib citrate (JAN/USAN); Tasocitinib citrate; Xeljanz (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D09785  Delamanid (JAN/USAN); Deltyba (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D09799  Carotegrast methyl (JAN); Carogra (TN) (P) CYP inhibition: CYP3A4
D09807  Difethiarol (JAN); Difethialone (P) unclassified
D09809  Tylosin acetate isovalerte (JAN) (P) unclassified
D09814  Silteplase (INN); Silteplase (genetical recombination) (JAN) (P) unclassified
D09817  Darexaban maleate (JAN); YM150 (P) unclassified
D09823  Duteplase (INN); Duteplase (genetical recombination) (JAN) (P) unclassified
D09848  Pioglitazone hydrochloride and glimepiride tablets (JP18); Pioglitazone and glimepiride; Duetact; Sonias (TN) (P) unclassified
D09872  Bedaquiline (USAN/INN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D09873  Bedaquiline fumarate (JAN/USAN); Sirturo (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D09876  Cariprazine hydrochloride (JAN/USAN); Vraylar (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D09889  Dulaglutide (USAN/INN); Dulaglutide (genetical recombination) (JAN); Trulicity (TN) (P) unclassified
D09893  Eliglustat (USAN/INN) (P) unclassified
D09894  Eliglustat tartrate (JAN/USAN); Eliglustat hemitartrate; Cerdelga (TN) (P) unclassified
D09920  Lenvatinib mesylate (USAN); Lenvatinib mesilate (JAN); Lenvima (TN) (P) unclassified
D09923  Letaxaban (USAN/INN) (P) unclassified
D09951  Ponatinib hydrochloride (JAN/USAN); Iclusig (TN) (P) unclassified
D09956  Quizartinib dihydrochloride (USAN); Quizartinib hydrochloride (JAN); Vanflyta (TN) (P) unclassified
D09958  Rilpivirine hydrochloride (JAN/USAN); Edurant (TN) (CI) unclassified
D09959  Ruxolitinib (USAN/INN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D09960  Ruxolitinib phosphate (JAN/USAN); Jakafi (TN); Jakavi (TN); Opzelura (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D09970  Tofacitinib (USAN); Tasocitinib (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D09978  Tofogliflozin (USAN); Tofogliflozin hydrate (JAN); Apleway (TN); Deberza (TN) (P) unclassified
D09989  Vardenafil hydrochloride (USP) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D09994  Selexipag (JAN/USAN/INN); Uptravi (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D09996  Vemurafenib (JAN/USAN/INN); Zelboraf (TN) (P) CYP induction: CYP3A4
D09997  Cariprazine (USAN/INN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D09999  Tramadol hydrochloride and acetaminophen; Tramcet (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D10003  Hemin (JAN); Normosang (TN); Panhematin (TN) (P) CYP induction: CYP3A4
D10019  Panobinostat lactate (JAN); Farydak (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D10021  Efinaconazole (JAN/USAN/INN); Clenafin (TN); Jublia (TN) (P) unclassified
D10024  Selumetinib sulfate (JAN/USAN); Koselugo (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D10025  Semaglutide (USAN/INN); Semaglutide (genetical recombination) (JAN); Ozempic (TN) (P) unclassified
D10032  Tylvalosin (USAN/INN) (P) unclassified
D10033  Tylosin tartrate (USP) (P) unclassified
D10034  Tylvalosin tartrate (USAN); Aiviosin [veterinary] (TN) (P) unclassified
D10055  Remogliflozin etabonate (USAN/INN) (P) unclassified
D10064  Dabrafenib (USAN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D10065  Daclatasvir (USAN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D10066  Dolutegravir (USAN); Tivicay (TN) (P) unclassified
D10082  Suvorexant (JAN/USAN); MK-4305; Belsomra (TN) (P) unclassified
D10093  Asunaprevir (JAN/USAN); Sunvepra (TN) (P) CYP induction: CYP3A4
D10095  Cabozantinib s-malate (USAN); Cabozantinib malate (JAN); Cometriq (TN); Cabometyx (TN) (P) unclassified
D10104  Dabrafenib mesylate (USAN); Dabrafenib mesilate (JAN); Tafinlar (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D10105  Daclatasvir dihydrochloride (USAN); Daclatasvir hydrochloride (JAN); Daklinza (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D10113  Dolutegravir sodium (JAN/USAN); Tivicay (TN) (P) unclassified
D10120  Esomeprazole strontium (USAN); Esomeprazole strontium tetrahydrate; Esomeprazole strontium (TN) (P) unclassified
D10131  Ixazomib citrate (JAN/USAN); Ninlaro (TN) (P) unclassified
D10135  Macitentan (JAN/USAN); Opsumit (TN) (CI,P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D10137  Regorafenib hydrate (JAN); Stivarga (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D10138  Regorafenib (USAN/INN); Stivarga (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D10158  Safinamide (USAN/INN) (P) unclassified
D10159  Alogliptin benzoate and pioglitazone hydrochloride; Liovel (TN); Oseni (TN); Incresync (TN) (P) unclassified
D10160  Mitiglinide calcium hydrate and voglibose; Glubes (TN) (P) unclassified
D10161  Sarilumab (USAN); Sarilumab (genetical receombination) (JAN); Kevzara (TN) (P) unclassified
D10178  Trelagliptin (USAN) (P) unclassified
D10179  Trelagliptin succinate (JAN/USAN); Zafatek (TN) (P) unclassified
D10184  Vortioxetine (USAN); Brintellix (TN) (P) unclassified
D10185  Vortioxetine hydrobromide (JAN/USAN); Brintellix (TN); Trintellix (TN) (P) unclassified
D10188  Naldemedine (USAN/INN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D10190  Tivozanib hydrochloride (USAN); Tivozanib hydrochloride monohydrate; Fotivda (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D10191  Safinamide mesylate (USAN); Safinamide mesilate (JAN); Safinamide methanesulfonate; Xadago (TN); Equfina (TN) (P) unclassified
D10192  Recombinant adsorbed quadrivalent human papillomavirus virus-like particle vaccine (yeast origin); Gardasil (TN); Silgard (TN) (P) unclassified
D10195  Luseogliflozin hydrate (JAN); Lusefi (TN) (P) unclassified
D10196  Ipragliflozin (INN) (P) unclassified
D10200  Ipragliflozin L-proline (JAN); Suglat (TN) (P) unclassified
D10218  Enzalutamide (JAN/USAN); Xtandi (TN) (P) unclassified
D10223  Ibrutinib (JAN/USAN); Imbruvica (TN) (P) unclassified
D10243  Irbesartan and amlodipine besilate (JP18); Aimix (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D10244  Metformin hydrochloride and rosiglitazone maleate; Avandamet (TN) (P) unclassified
D10246  Omeprazole, clarithromycin and amoxicillin; Omeclamox-pak (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D10251  Glimepiride and rosiglitazone maleate; Avandaryl (TN) (P) unclassified
D10253  Alogliptin benzoate and metformin hydrochloride; Kazano (TN); Vipdomet (TN) (P) unclassified
D10258  Simvastatin and sitagliptin phosphate; Juvisync (TN) (P) unclassified
D10261  Metformin hydrochloride and sitagliptin phosphate; Janumet (TN) (P) unclassified
D10262  Saxagliptin hydrochloride; Onglyza (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D10263  Metformin hydrochloride and saxagliptin hydrochloride; Kombiglyze (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D10264  Linagliptin and metformin hydrochloride; Jentaduet (TN) (P) unclassified
D10265  Glipizide and metformin hydrochloride; Metaglip (TN) (P) unclassified
D10266  Glyburide and metformin hydrochloride; Glibenclamide and metformin hydrochloride; Glucovance (TN) (P) unclassified
D10267  Methyldopa and hydrochlorothiazide; Methyldopa and hydrochlorothiazide (TN) (P) unclassified
D10306  Avatrombopag (USAN/INN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D10307  Avatrombopag maleate (JAN/USAN); Doptelet (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D10309  Brexpiprazole (JAN/USAN/INN); Rexulti (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D10313  Ertugliflozin (USAN/INN) (P) unclassified
D10315  Momelotinib (USAN/INN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D10317  Omarigliptin (JAN/USAN/INN) (P) unclassified
D10319  Panobinostat (USAN/INN); Farydak (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D10355  Aripiprazole cavoxil (USAN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D10358  Momelotinib dihydrochloride (USAN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D10364  Aripiprazole lauroxil (USAN); Aristada (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D10372  Palbociclib (JAN/USAN); Ibrance (TN) (P) unclassified
D10385  Ezetimibe and atorvastatin; Atozet (TN); Liptruzet (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D10430  Treprostinil diolamine (USAN); Orenitram (TN) (P) unclassified
D10433  Vibegron (JAN/USAN/INN); Beova (TN); Gemtesa (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D10450  Alectinib hydrochloride (JAN); Alecensa (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D10452  Cabazitaxel acetonate (JAN); Cabazitaxel acetone; Jevtana (TN) (P) unclassified
D10459  Empagliflozin (JAN/USAN/INN); Jardiance (TN) (P) unclassified
D10466  Vonoprazan fumarate (JAN/USAN); Takecab (TN); Voquezna (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D10471  Idraparinux sodium (USAN) (P) unclassified
D10473  Insulin peglispro (USAN/INN) (P) unclassified
D10478  Naldemedine tosylate (JAN/USAN); Naldemedine tosilate; Symproic (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D10480  Irbesartan and trichlormethiazide; Irtra (TN) (P) unclassified
D10492  Tildipirosin (USAN/INN); Zuprevo [veterinary] (TN) (P) unclassified
D10500  Metformin hydrochloride and repaglinide; Prandimet (TN) (P) unclassified
D10501  Fluticasone furoate and vilanterol trifenatate; Breo ellipta (TN); Relvar ellipita (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D10502  Gemigliptin (INN) (P) unclassified
D10505  Glycopyrronium bromide and indacaterol maleate; Ultibro (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D10506  Fluticasone propionate and formoterol fumarate hydrate; Flutiform (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D10512  Brinzolamide and timolol maleate; Azorga (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D10513  Clopidogrel sulfate and aspirin; Clopidogrel and acetylsalicyclic acid; Complavin (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D10516  Aripiprazole hydrate (JAN); Aripiprazole monohydrate; Abilify maintena (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D10519  Rabeprazole, amoxicillin and clarithromycin; Rabecure (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D10520  Rabeprazole, amoxicillin and metronidazole; Rabefine (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D10524  Azilsartan and amlodipine besilate; Zacras (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D10525  Valsartan and cilnidipine; Atedio (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D10527  Acetylsalicylic acid and lansoprazole; Acetylsalicylic acid and lansoprazole; Takelda (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D10533  Umeclidinium bromide and vilanterol; Anoro (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D10542  Alectinib (USAN/INN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D10551  Ceritinib (JAN/USAN/INN); Zykadia (TN) (P) unclassified
D10564  Amenamevir (JAN/INN); Amenalief (TN) (P) unclassified
D10566  Pasireotide pamoate (JAN); Signifor lar (TN) (P) unclassified
D10570  Insulin degludec (genetical recombination) and insulin aspart (genetical recombination); Ryzodeg (TN) (P) unclassified
D10572  Fosnetupitant and palonosetron hydrochloride; Netupitant and palonosetron hydrochloride; Akynzeo (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D10586  Dapagliflozin and metformin; Xigduo xr (TN) (P) unclassified
D10587  Canagliflozin and metformin; Invokamet (TN) (P) unclassified
D10588  Empagliflozin and linagliptin; Glyxambi (TN) (P) unclassified
D10591  Clonidine and chlorthalidone; Clorpres (TN) (P) unclassified
D10600  Dolutegravir, abacavir and lamivudine; Triumeq (TN) (P) unclassified
D10612  Benzhydrocodone (USAN/INN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D10627  Esketamine hydrochloride (JAN/USAN); Spravato (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D10630  Fedratinib (USAN/INN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D10633  Finerenone (JAN/USAN/INN); Kerendia (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D10642  Irinotecan sucrosofate (USAN) (P) unclassified
D10643  Isavuconazonium sulfate (JAN/USAN); Cresemba (TN) (P) unclassified
D10662  Rimegepant (USAN/INN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D10663  Rimegepant sulfate (USAN); Nurtec odt (TN); Vydura (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D10669  Sotagliflozin (USAN/INN); Inpefa (TN) (P) unclassified
D10673  Ubrogepant (USAN/INN); Ubrelvy (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D10675  Valbenazine (USAN/INN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D10676  Etelcalcetide (USAN/INN); Velcalcetide (P) unclassified
D10677  Etelcalcetide hydrochloride (JAN/USAN); Velcalcetide hydrochloride (USAN); Parsabiv (TN) (P) unclassified
D10679  Venetoclax (JAN/USAN/INN); Venclexta (TN) (P) unclassified
D10684  Antithrombin gamma (INN); Antithrombin gamma (genetical recombination) (JAN); Acoalan (TN) (P) unclassified
D10688  Abemaciclib (JAN/USAN/INN); Verzenio (TN) (P) unclassified
D10692  Benzhydrocodone hydrochloride (USAN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D10696  Capmatinib (USAN/INN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D10709  Gilteritinib (USAN/INN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D10711  Pemafibrate (JAN); Parmodia (TN) (P) unclassified
D10742  Rolapitant (USAN/INN); Varubi (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D10743  Vildagliptin and metformin hydrochloride (P) unclassified
D10744  Tiotropium and olodaterol; Spiolto (TN); Stiolto respimat (TN) (P) unclassified
D10745  Ombitasvir, paritaprevir and ritonavir; Technivie (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D10746  Esflurbiprofen and mentha oil; Loqoa (TN) (P) unclassified
D10749  Pitolisant (USAN/INN); Wakix (TN); Ozawade (TN) (P) unclassified
D10750  Isavuconazole (INN); Cresemba (TN) (P) unclassified
D10752  Empagliflozin and metformin; Synjardy (TN) (P) unclassified
D10753  Atazanavir and cobicistat; Evotaz (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D10755  Elvitegravir, cobicistat, emtricitabine and tenofovir alafenamide; Genvoya (TN) (P) unclassified
D10762  Fosravuconazole L-lysine ethanolate (JAN) (P) unclassified
D10766  Osimertinib mesylate (USAN); Osimertinib mesilate (JAN); Tagrisso (TN) (P) unclassified
D10772  Lascufloxacin hydrochloride (JAN); Lasvic (TN) (P) unclassified
D10774  Vonoprazan, amoxicillin and metronidazole; Vonopion (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D10775  Vonoprazan, amoxicillin and clarithromycin; Vonosap (TN); Voquenza (TN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D10780  Perampanel hydrate (JAN); Fycompa (TN) (P) unclassified
D10793  Sodium picosulfate hydrate, magnesium oxide and citric acid, anhydrous; Picoprep (TN); Prepopik (TN); Clenpiq (TN) (P) unclassified
D10800  Gilteritinib fumarate (JAN/USAN); Xospata (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D10801  Letermovir (JAN/USAN/INN); Prevymis (TN) (P) unclassified
D10805  Telmisartan, amlodipine and hydrochlorothiazide; Micatrio (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D10811  Fentanyl hydrochloride (JAN); Ionsys (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D10823  Clopidogrel hydrochloride; Clopidogrel (TN) (P) unclassified
D10824  Clopidogrel besilate; Clopidogrel besylate; Clopidogrel (TN) (P) unclassified
D10826  Saxagliptin and dapagliflozin; Qtern (TN) (P) unclassified
D10827  Sofosbuvir and velpatasvir; Epclusa (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D10832  Darunavir and cobicistat; Prezcobix (TN); Rezolsta (TN) (P) unclassified
D10836  Emtricitabine, rilpivirine and tenofovir alafenamide; Odefsey (TN) (CI) unclassified
D10865  Bexagliflozin (USAN); Brenzavvy (TN) (P) unclassified
D10866  Brigatinib (JAN/USAN); Alunbrig (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D10882  Daclatasvir, asunaprevir and beclabuvir; Ximency (TN) (P) CYP induction: CYP3A4
D10883  Ribociclib (USAN/INN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D10889  Momelotinib hydrochloride hydrate (JAN); Momelotinib dihydrochloride monohydrate; Ojjaara (TN); Omjjara (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D10891  Capmatinib hydrochloride (USAN); Capmatinib hydrochloride hydrate (JAN); Tabrecta (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D10892  Esaxerenone (JAN/INN) (P) unclassified
D10893  Acalabrutinib (JAN/USAN/INN); Calquence (TN) (P) unclassified
D10895  Fosaprepitant (INN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D10897  Teneligliptin and canagliflozin; Teneligliptin and canagliflozin; Canalia (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D10898  Neratinib maleate; Nerlynx (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D10915  Cannabidiol (USAN/INN); CBD; Epidiolex (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D10926  Entrectinib (JAN/USAN/INN); Rozlytrek (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D10927  Erdafitinib (JAN/USAN/INN); Balversa (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D10930  Etrasimod (USAN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D10931  Etrasimod arginine (USAN); Etrasimod L-arginine (JAN); Velsipity (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D10954  Mirvetuximab soravtansine (USAN/INN); Mirvetuximab soravtansine-gynx; Elahere (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D10960  Nirogacestat (USAN/INN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D10970  Pegapamodutide (USAN/INN) (P) unclassified
D10979  Ribociclib succinate (USAN); Kisqali (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D10990  Somatrogon (USAN/INN); Somatrogon (genetical recombination) (JAN); Somatrogon-ghla; Ngenla (TN) (P) unclassified
D10994  Upadacitinib (USAN/INN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D10995  Upadacitinib tartrate (USAN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D10999  Valbenazine tosylate (USAN); Valbenazine tosilate (JAN); Valbenazine ditosylate; Ingrezza (TN); Dysval (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D11000  Vamorolone (USAN/INN); Agamree (TN) (P) Enzyme: CYP3A4 / Target: NR3C1 / CYP induction: CYP3A4
D11009  Indacaterol acetate (JAN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D11012  Lorlatinib (JAN/USAN/INN); Lorbrena (TN) (P) unclassified
D11022  Lemborexant (JAN/USAN/INN); Dayvigo (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D11023  Evogliptin (INN) (P) unclassified
D11029  Andexanet alfa (USAN/INN); Andexanet alfa (genetical recombination) (JAN); Andexxa (TN); Ondexxya (TN) (P) unclassified
D11034  Insulin glargine and lixisenatide; Insulin glargine (genetical recombination) and lixisenatide; Soliqua (TN) (P) unclassified
D11036  Glycopyrrolate and formoterol; Bevespi (TN) (P) unclassified
D11040  Apalutamide (JAN/INN); Erleada (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D11043  Ertugliflozin pidolate; Ertugliflozin L-pyroglutamic acid; Steglatro (TN) (P) unclassified
D11045  Darolutamide (JAN/USAN/INN); Nebeqa (TN) (P) unclassified
D11048  Upadacitinib hydrate (JAN); Upadacitinib hemihydrate; Rinvoq (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D11053  Encorafenib (JAN/USAN/INN); Braftovi (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D11056  Mirtazapine hydrate (JAN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D11061  Osilodrostat (USAN/INN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D11062  Osilodrostat phosphate (JAN/USAN); Isturisa (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D11063  Evocalcet (JAN/INN); Orkedia (TN) (P) unclassified
D11064  Sitagliptin and ipragliflozin; Sujanu (TN) (P) unclassified
D11066  Ertugliflozin and sitagliptin; Steglujan (TN) (P) unclassified
D11067  Ertugliflozin and metformin; Segluromet (TN) (P) unclassified
D11070  Tirabrutinib hydrochloride (JAN/USAN); Velexbru (TN) (P) unclassified
D11072  Siponimod fumarate (USAN); Siponimod fumaric acid (JAN); Mayzent (TN) (P) unclassified
D11073  Tepotinib hydrochloride (USAN); Tepotinib hydrochloride hydrate (JAN); Tepmetko (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D11093  Avacopan (JAN/USAN/INN); Tavneos (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D11095  Atorvastatin calcium propylene glycol solvate (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D11109  Anagliptin and Metformin hydrochloride (P) unclassified
D11114  Esomeprazole magnesium dihydrate (P) unclassified
D11138  Larotrectinib sulfate (JAN/USAN); Vitrakvi (TN) (P) unclassified
D11150  Cenobamate (USAN/INN); Xcopri (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D11158  Leniolisib (USAN/INN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D11159  Leniolisib phosphate (USAN); Joenja (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D11160  Caplacizumab (USAN/INN); Caplacizumab (genetical recombination) (JAN); Caplacizumab-yhdp; Cablivi (TN) (P) unclassified
D11194  Somapacitan (USAN/INN); Somapacitan (genetical recombination) (JAN); Somapacitan-beco; Sogroya (TN) (P) unclassified
D11222  Selinexor (USAN/INN); Xpovio (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D11252  Fexinidazole (USAN/INN); Fexinidazole (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D11270  Pexidartinib (USAN/INN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D11271  Pexidartinib hydrochloride (JAN/USAN); Turalio (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D11280  Bivalirudin trifluoroacetate (USAN); Angiomax (TN) (P) unclassified
D11282  Dolutegravir sodium and rilpivirine hydrochloride; Juluca (TN) (CI) unclassified
D11296  Fedratinib hydrochloride (USAN); Fedratinib hydrochloride hydrate (JAN); Fedratinib dihydrochloride monohydrate; Inrebic (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D11313  Atogepant (USAN); Qulipta (TN); Aquipta (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D11330  Voxelotor (USAN); Oxbryta (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D11342  Dorzagliatin (USAN) (P) unclassified
D11360  Tirzepatide (JAN/USAN); Mounjaro (TN) (P) unclassified
D11370  Fosnetupitant chloride hydrochloride (JAN/USAN); Arokaris (TN) (P) unclassified
D11371  Capivasertib (JAN/USAN); Truqap (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D11382  Darunavir, cobicistat, emtricitabine and tenofovir alafenamide; Symtuza (TN) (P) unclassified
D11389  Dutasteride and tamsulosin; Jalyn (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D11403  Asciminib (USAN/INN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D11404  Asciminib hydrochloride (JAN/USAN); Scemblix (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D11406  Risdiplam (JAN/USAN/INN); Evrysdi (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D11417  Pemigatinib (JAN/USAN/INN); Pemazyre (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D11441  Aprocitentan (USAN/INN); Tryvio (TN) (P) unclassified
D11453  Nirogacestat hydrobromide (USAN); Ogsiveo (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D11454  Repotrectinib (JAN/USAN); Augtyro (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D11460  Siponimod (USAN/INN) (P) unclassified
D11485  Tazemetostat hydrobromide (JAN/USAN); Tazverik (TN) (P) unclassified
D11490  Pitolisant hydrochloride (USAN); Wakix (TN) (P) unclassified
D11553  Lidocaine and tetracaine; Pliaglis (TN); Synera (TN) (P) unclassified
D11564  Upacicalcet sodium hydrate (JAN); Upasita (TN) (P) unclassified
D11567  Insulin degludec and liraglutide; Xultophy (TN) (P) unclassified
D11568  Edoxaban tosylate (USAN) (P) unclassified
D11572  Beclomethasone dipropionate monohydrate; Beconase aq (TN) (P) Enzyme: CYP3A4 / Target: NR3C1 / CYP induction: CYP3A4
D11573  Oxycodone and ibuprofen (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D11576  Naproxen and esomeprazole magnesium; Vimovo (TN) (P) unclassified
D11584  Budesonide, glycopyrronium bromide and formoterol fumarate; Budesonide, glycopyrrolate and formoterol fumarate; Breztri (TN) (P) unclassified
D11603  Leriglitazone (USAN/INN); 1-Hydroxypioglitazone (P) unclassified
D11604  Leriglitazone hydrochloride (USAN) (P) unclassified
D11616  Aspirin and omeprazole; Yosprala (TN) (P) unclassified
D11617  Eletriptan hydrobromide monohydrate (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D11619  Desvenlafaxine succinate anhydrous; Desvenlafaxine succinate (TN) (P) unclassified
D11628  Benzhydrocodone and acetaminophen; Apadaz (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D11631  Lefamulin (USAN/INN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D11632  Lefamulin acetate (USAN); Xenleta (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D11652  Tenapanor (USAN/INN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D11653  Tenapanor hydrochloride (JAN/USAN); Ibsrela (TN); Phozevel (TN); Xphozah (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D11656  Azelastine hydrochloride and fluticasone propionate; Dymista (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D11659  Tolvaptan sodium phosphate (JAN); Samtasu (TN) (P) unclassified
D11662  Valemetostat tosilate (JAN); Valemetostat tosylate; Ezharmia (TN) (P) unclassified
D11671  Elacestrant (USAN/INN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D11672  Elacestrant hydrochloride (USAN); Elacestrant dihydrochloride; Orserdu (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D11674  Berotralstat hydrochloride (JAN/USAN); Orladeyo (TN) (P) CYP inhibition: CYP3A4
D11706  Omeprazole and sodium bicarbonate; Zegerid (TN) (P) unclassified
D11710  Phentermine and topiramate; Qsymia (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D11711  Dapagliflozin, metformin and saxagliptin; Qternmet xr (TN) (P) unclassified
D11713  Selpercatinib (JAN/USAN/INN); Retevmo (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D11717  Tepotinib (USAN/INN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D11725  Futibatinib (JAN/USAN/INN); Lytgobi (TN) (P) unclassified
D11757  Inebilizumab (USAN/INN); Inebilizumab (genetical recombination) (JAN); Inebilizumab-cdon; Uplizna (TN) (P) unclassified
D11768  Pacritinib (USAN/INN); Vonjo (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D11784  Vonoprazan (USAN/INN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D11785  Oteseconazole (USAN/INN); Vivijoa (TN) (P) unclassified
D11793  Zuranolone (JAN/USAN/INN); Zurzuvae (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D11804  Aspirin and vonoprazan; Cabpirin (TN) (P) unclassified
D11807  Imeglimin hydrochloride (JAN); Twymeeg (TN) (P) unclassified
D11816  Belumosudil mesylate (USAN); Belumosudil mesilate (JAN); Rezurock (TN) (P) unclassified
D11851  Butalbital, acetaminophen, caffeine and codeine phosphate (P) unclassified
D11856  Empagliflozin, linagliptin and metformin hydrochloride; Trijardy xr (TN) (P) unclassified
D11860  Butalbital, aspirin, caffeine and codeine; Fiorinal with codeine (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D11861  Indacaterol acetate, glycopyrronium bromide and mometasone furoate; Enerzair (TN) (P) unclassified
D11862  Indacaterol and mometasone furoate; Atectura (TN) (P) unclassified
D11863  Human papillomavirus 9-valent vaccine, recombinant; Recombinant adsorbed 9-valent human papillomavirus virus-like particle vaccine (yeast origin); Gardasil 9 (TN); Silgard 9 (TN) (P) unclassified
D11881  Amlodipine benzoate; Katerzia (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D11886  Daridorexant (USAN/INN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D11910  Danuglipron (USAN) (P) unclassified
D11911  Danuglipron tromethamine (USAN) (P) unclassified
D11920  Pimitespib (JAN); Jeselhy (TN) (P) unclassified
D11923  Lobeglitazone (INN) (P) unclassified
D11924  Beinaglutide (INN) (P) unclassified
D11954  Belzutifan (JAN/USAN/INN); Welireg (TN) (P) unclassified
D11968  Teneligliptin hydrobromide (JAN) (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D11970  Ritlecitinib tosylate (USAN); Ritlecitinib tosilate (JAN); Litfulo (TN) (P) unclassified
D12005  Treprostinil palmitil (USAN/INN) (P) unclassified
D12055  Sotorasib (JAN/USAN); Lumakras (TN) (P) unclassified
D12130  Drospirenone, ethinyl estradiol and levomefolate calcium; Beyaz (TN); Safyral (TN); Tydemy (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D12162  Lenacapavir sodium (JAN/USAN); Sunlenca (TN) (P) unclassified
D12205  Pneumococcal 15-valent conjugate vaccine; Vaxneuvance (TN) (P) unclassified
D12225  Mazdutide (USAN) (P) unclassified
D12265  Mavacamten (JAN/USAN/INN); Camzyos (TN) (P) unclassified
D12269  Nirmatrelvir and ritonavir; Paxlovid (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D12294  Sitagliptin phosphate (JAN) (P) unclassified
D12301  Adagrasib (USAN/INN); Krazati (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D12311  Bortezomib hydrate (JAN) (P) unclassified
D12312  Codeine phosphate and chlorpheniramine maleate; Tuxarin (TN) (P) unclassified
D12313  Chlorpheniramine polistirex and codeine polistirex; Tuzistra (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D12326  Opelconazole (USAN/INN) (P) unclassified
D12341  Vurolenatide (USAN/INN) (P) unclassified
D12353  Ensitrelvir fumarate (USAN); Ensitrelvir fumaric acid (JAN); Xocova (TN) (P) unclassified
D12358  Insulin icodec (USAN/INN); Insulin icodec (genetical recombination) (JAN) (P) unclassified
D12403  Venlafaxine besylate monohydrate; Venlafaxine besylate (TN) (P) unclassified
D12444  Nilotinib hydrochloride dihydrate (JAN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D12446  Anpocogin (USAN) (P) unclassified
D12483  Olutasidenib (USAN/INN); Rezlidhia (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D12484  Carfloglitazar (INN) (P) unclassified
D12486  Finasteride and tadalafil; Entadfi (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D12497  Drospirenone and estradiol; Angeliq (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D12529  Orforglipron calcium (USAN) (P) unclassified
D12536  Orforglipron (USAN) (P) unclassified
D12544  Vortioxetine hemihydrobromide (USAN) (P) unclassified
D12555  Lotiglipron (USAN) (P) unclassified
D12586  Mifepristone and misoprostol; Mefeego (TN) (CI,P) unclassified
D12595  Aspirin trelamine (USAN) (P) unclassified
D12596  Aspirin trelamine hydrochloride (USAN) (P) unclassified
D12609  Dasatinib laurylsulfate (USAN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D12629  Treprostinil phosphate (USAN); Treprostinil biphosphate (P) unclassified
D12637  Darunavir hydrate (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D12703  Linagliptin hydrate (JAN); Linagliptin hemihydrate (P) unclassified
D12735  Lotiglipron tromethamine (USAN) (P) unclassified
D12752  Darunavir propylene glycolate (P) Enzyme: CYP3A4 / CYP inhibition: CYP3A4 / CYP induction: CYP3A4
D12756  Vonoprazan and amoxicillin; Voquezna (TN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D12816  Dexlansoprazole sesquihydrate (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D12854  Nilotinib laurylsulfate (USAN) (P) Enzyme: CYP3A4 / CYP induction: CYP3A4
D12861  Pemvidutide (USAN/INN) (P) unclassified
D12874  Live attenuated influenza virus vaccine, intranasal; Flumist (TN) (CI) unclassified