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Drug interaction list


Query:
D00211  Rifampin (USP); Rifampicin (JP18/INN); Rifadin (TN); Rimactane (TN)

Interactions: 2069 hits    [ ATC classification | Therapeutic category ]

C00304  Kanamycin (P) unclassified
C04227  Octopamine; 1-(4-Hydroxyphenyl)-2-aminoethanol; p-Hydroxyphenylethanolamine (P) unclassified
C04931  Argatroban; (2R,4R)-4-Methyl-1[Nalpha-[(3-methyl-1,2,3,4-tetrahydro-8-quinolinyl)sulfonyl]-L-arginyl]-2-piperadinecarboxylic acid (P) unclassified
C06174  Codeine; (5alpha,6alpha)-7,8-Didehydro-4,5-epoxy-3-methoxy-17-methylmorphinan-6-ol (P) unclassified
C06921  Clorazepate; Clorazepic acid (P) unclassified
C07005  Flunisolide; Flunisolide anhydrous (P) unclassified
C07051  Indinavir (CI,P) unclassified
C07370  Prednisone; 1,2-Dehydrocortisone; 17,21-Dihydroxypregna-1,4-diene-3,11,20-trione (P) unclassified
C07533  Prenalterol (P) unclassified
C08859  Cymarin; Strophanthidin 3-O-beta-D-cymaroside (P) unclassified
D00058  gamma-Aminobutyric acid (JAN); Gammalon (TN) (P) unclassified
D00059  Levodopa (JP18/USP/INN); Dopar (TN) (P) unclassified
D00066  Progesterone (JP18/USP/INN); Crinone (TN); Prometrium (TN) (P) CYP induction: CYP3A4
D00067  Estrone (JAN/USP/INN); Estrone (TN) (P) CYP induction: CYP3A4
D00076  Noradrenaline (JP18); Norepinephrine (INN); Nor adrenalin (TN) (P) unclassified
D00088  Hydrocortisone (JP18/USP/INN); HC; Acticort (TN); Anusol HC (TN); Colocort (TN); Cortef (TN); Hytone (TN); Plenadren (TN) (P) unclassified
D00094  Tretinoin (JAN/USP/INN); Avita (TN); Renova (TN); Retin A (TN); Tretinoin (TN) (CI,P) unclassified
D00095  Epinephrine (USP/INN); Adrenaline (JP18); Adrenalin (TN); Auvi-q (TN); Epipen (TN) (P) unclassified
D00104  Chloramphenicol (JP18/USP/INN); Amphicol (TN); Chloromycetin (TN); Econochlor (TN) (P) unclassified
D00105  Estradiol (JAN/USP/INN); Climara (TN); Divigel (TN); Estrace (TN); Estraderm (TN); Estrasorb (TN); Estring (TN); Estrogel (TN); Innofem (TN); Vagifem (TN); Vivelle (TN) (P) CYP induction: CYP3A4
D00107  Tacrolimus (USP/INN); Tacrolimus hydrate (JP18); Prograf (TN); Protopic (TN) (P) CYP induction: CYP3A4
D00112  G-Strophanthin (JAN); Ouabain octahydrate (P) unclassified
D00124  Ephedrine (USP); Ephedrine (TN) (P) unclassified
D00125  Etoposide (JP18/USP/INN); Vepesid (TN) (CI,P) unclassified
D00135  Capreomycin sulfate (JAN/USP); Capastat sulfate (TN) (P) unclassified
D00136  Haloperidol (JP18/USP/INN); Haldol (TN) (P) CYP induction: CYP3A4
D00138  Scopolamine (INN); Transderm scop (TN) (P) unclassified
D00142  Methotrexate (JP18/USP/INN); Otrexup (TN); Xatmep (TN) (CI,P) unclassified
D00144  Pyrazinamide (JP18/USP/INN); Pyrazinamide (TN) (P) unclassified
D00155  Pentostatin (JAN/USAN/INN); Nipent (TN) (CI,P) unclassified
D00161  Mercaptopurine (USP); Mercaptopurine hydrate (JP18); Purinethol (TN); Purixan (TN) (CI,P) unclassified
D00162  Aminosalicylic acid (USP); Pamisyl (TN); Paser (TN) (P) unclassified
D00165  Hydrocortisone acetate (JP18/USP); Cortifoam (TN); U-cort (TN) (P) unclassified
D00168  Cytarabine (JP18/USP/INN); ARA-C; Depocyt (TN) (CI,P) unclassified
D00178  Octopamine hydrochloride (JAN) (P) unclassified
D00181  Argatroban (USP); Argatroban hydrate (JP18); Novastan (TN) (P) CYP induction: CYP3A4
D00184  Cyclosporine (USP); Ciclosporin (JP18); Gengraf (TN); Neoral (TN); Restasis (TN); Sandimmune (TN) (P) CYP induction: CYP3A4
D00195  Codeine (USP); Codeine hydrate (P) unclassified
D00197  Reserpine (JP18/USP/INN); Apoplon (TN); Serpalan (TN) (P) unclassified
D00198  Rescinnamine (JAN/INN); Tsuruselpi S (TN) (P) unclassified
D00199  Ajmaline (JP18); Ajimalin (TN) (P) unclassified
D00208  Mitomycin (USP/INN); Mitomycin C (JP18); MMC; Jelmyto (TN); Mitomycin (TN); Muamycin (TN) (CI,P) unclassified
D00211  Rifampin (USP); Rifampicin (JP18/INN); Rifadin (TN); Rimactane (TN) (P) unclassified
D00214  Dactinomycin (USP); Actinomycin D (JP18); Cosmegen (TN) (CI,P) unclassified
D00216  Acarbose (JAN/USAN/INN); Precose (TN) (P) unclassified
D00217  Acetaminophen (JP18/USP); Paracetamol (INN); Tylenol (TN) (P) unclassified
D00219  Acetohexamide (JP18/USP/INN); Dymelor (TN) (P) unclassified
D00225  Alprazolam (JP18/USP/INN); Xanax (TN) (P) unclassified
D00231  Inamrinone (USP); Amrinone (JAN/INN); Amcoral (TN) (P) unclassified
D00235  Atenolol (JP18/USP/INN); Tenormin (TN) (P) unclassified
D00236  Atovaquone (JAN/USP/INN); Mepron (TN) (P) unclassified
D00244  Betamethasone (JP18/USP/INN); Celestone (TN); Rinderon (TN) (P) unclassified
D00246  Budesonide (JP18/USP/INN); Entocort EC (TN); Pulmicort (TN); Rhinocort (TN); Uceris (TN) (P) CYP induction: CYP3A4
D00248  Busulfan (JP18/USP/INN); Myleran (TN) (CI,P) unclassified
D00252  Carbamazepine (JP18/USP/INN); Equetro (TN); Tegretol (TN) (P) CYP induction: CYP3A4
D00253  Carbidopa hydrate and levodopa; Parcopa (TN); Sinemet (TN) (P) unclassified
D00254  Carmustine (JAN/USP/INN); Bicnu (TN); Gliadel (TN) (CI,P) unclassified
D00255  Carvedilol (JP18/USP/INN); Artist (TN); Coreg (TN) (P) CYP induction: CYP3A4
D00265  Chloral hydrate (JP18/USP); Noctec (TN) (P) unclassified
D00266  Chlorambucil (JAN/USP/INN); Leukeran (TN) (CI,P) unclassified
D00267  Chlordiazepoxide (JP18/USP/INN); Libritabs (TN) (P) unclassified
D00271  Chlorpropamide (JP18/USP/INN); Diabinese (TN) (P) unclassified
D00275  Cisplatin (JP18/USP/INN); Platinol (TN) (CI,P) unclassified
D00276  Clarithromycin (JP18/USP/INN); Biaxin (TN) (P) CYP induction: CYP3A4
D00279  Clofibrate (JP18/USP/INN); Atromid-S (TN) (P) unclassified
D00280  Clonazepam (JP18/USP/INN); Klonopin (TN) (P) unclassified
D00281  Clonidine (JAN/USP/INN); Catarpres-TTS (TN) (P) unclassified
D00282  Clotrimazole (JP18/USP/INN); Lotrimin (TN); Mycelex (TN) (P) unclassified
D00283  Clozapine (JAN/USP/INN); Clozaril (TN) (P) CYP induction: CYP3A4
D00287  Cyclophosphamide (USP); Cyclophosphamide hydrate (JP18); Cytoxan (TN); Neosar (TN) (CI,P) CYP induction: CYP3A4
D00288  Dacarbazine (JAN/USP/INN); DTIC-Dome (TN) (CI,P) unclassified
D00292  Dexamethasone (JP18/USP/INN); Decadron (TN); Maxidex (TN) (P) CYP induction: CYP3A4
D00293  Diazepam (JP18/USP/INN); Diastat (TN); Valium (TN) (P) CYP induction: CYP3A4
D00294  Diazoxide (JAN/USP/INN); Hyperstat (TN); Proglycem (TN) (P) unclassified
D00296  Didanosine (JAN/USP/INN); Videx (TN) (CI,P) unclassified
D00297  Digitoxin (JAN/USP/INN); Crystodigin (TN) (P) Transporter induction: ABCB1
D00298  Digoxin (JP18/USP); Lanoxicaps (TN); Lanoxin (TN) (P) Transporter induction: ABCB1
D00302  Dipyridamole (JP18/USP/INN); Persantine (TN) (P) unclassified
D00303  Disopyramide (JP18/USAN/INN); Rythmodan P (TN) (P) CYP induction: CYP3A4
D00304  Divalproex sodium (USP); Valproate semisodium (INN); Depakote (TN) (P) unclassified
D00311  Estazolam (JP18/USP/INN); ProSom (TN) (P) unclassified
D00312  Estrone sodium sulfate; Sodium estrone sulfate (P) CYP induction: CYP3A4
D00319  Felodipine (JP18/USP/INN); Plendil (TN) (P) CYP induction: CYP3A4
D00320  Fentanyl (JAN/USP/INN); Duragesic (TN); Subsys (TN) (P) CYP induction: CYP3A4
D00321  Finasteride (JAN/USP/INN); Propecia (TN); Proscar (TN) (P) CYP induction: CYP3A4
D00322  Fluconazole (JP18/USP/INN); Diflucan (TN) (P) unclassified
D00324  Flunisolide (JAN/USP); Aerospan (TN); Nasalide (TN) (P) CYP induction: CYP3A4
D00325  Fluocinonide (JP18/USP/INN); Lidex (TN); Vanos (TN) (P) unclassified
D00328  Flurandrenolide (USP); Fludroxycortide (JAN/INN); Cordran (TN) (P) unclassified
D00329  Flurazepam (JAN/INN); Insumin (TN) (P) unclassified
D00335  Glipizide (USP/INN); Glucotrol (TN) (P) unclassified
D00336  Glyburide (USP); Glibenclamide (JP18/INN); Diabeta (TN); Glynase (TN); Micronase (TN) (P) CYP induction: CYP3A4
D00338  Halazepam (USAN/INN); Paxipam (TN) (P) unclassified
D00341  Hydroxyurea (USP); Hydroxycarbamide (JAN/INN); Droxia (TN); Hydrea (TN); Siklos (TN) (CI,P) unclassified
D00343  Ifosfamide (JAN/USP/INN); Ifex (TN) (CI,P) CYP induction: CYP3A4
D00346  Isoniazid (JP18/USP/INN); Laniazid (TN) (P) unclassified
D00349  Isradipine (USP/INN); Dynacirc (TN) (P) unclassified
D00350  Itraconazole (JP18/USP); Itrizole (TN); Sporanox (TN) (P) CYP induction: CYP3A4
D00351  Ketoconazole (JP18/USP); Nizoral (TN); Xolegel (TN) (P) CYP induction: CYP3A4
D00353  Lamivudine (JAN/USP/INN); Epivir (TN) (CI,P) unclassified
D00354  Lamotrigine (JAN/USP/INN); Lamictal (TN) (P) unclassified
D00355  Lansoprazole (JP18/USP/INN); Prevacid (TN) (P) CYP induction: CYP3A4
D00358  Lidocaine (JP18/USP/INN); Dentipatch (TN); Xylocaine (TN) (P) CYP induction: CYP3A4
D00359  Lovastatin (USP/INN); MK-803; ML-530B; Mevacor (TN) (P) CYP induction: CYP3A4
D00363  Lomustine (USP/INN); Gleostine (TN) (CI,P) unclassified
D00364  Loratadine (JAN/USP/INN); Claritin (TN) (P) CYP induction: CYP3A4
D00365  Lorazepam (JP18/USP/INN); Ativan (TN) (P) unclassified
D00369  Melphalan (JP18/USP/INN); Alkeran (TN) (CI,P) unclassified
D00370  Temazepam (USP/INN); Restoril (TN) (P) unclassified
D00371  Theophylline (JP18); Elixophyllin (TN); Quibron-t (TN); Theo-24 (TN); Theodur G (TN); Theolair (TN); Uniphyl (TN) (P) unclassified
D00372  Thiabendazole (USP); Tiabendazole (JAN/INN); Mintezol (TN) (P) unclassified
D00375  Mephenytoin (USP/INN); Mesantoin (TN) (P) unclassified
D00376  Meprobamate (JAN/USP/INN); Equanil (TN); Miltown (TN) (P) unclassified
D00378  Timolol (USAN); Timolol hemihydrate; Betimol (TN) (P) unclassified
D00379  Tolazamide (JAN/USP/INN); Tolinase (TN) (P) unclassified
D00380  Tolbutamide (JP18/USP/INN); Orinase (TN) (P) unclassified
D00385  Triamcinolone (JP18/USP/INN); Aristocort (TN); Kenacort (TN) (P) unclassified
D00387  Triazolam (JP18/USP/INN); Halcion (TN) (P) CYP induction: CYP3A4
D00388  Triclofos sodium (JP18/USAN); Tricloryl (TN) (P) unclassified
D00392  Trimethadione (JP18/INN); Tridione (TN) (P) unclassified
D00395  Troglitazone (JAN/USAN/INN); Rezulin (TN) (P) unclassified
D00399  Valproic acid (USP); Depakene (TN) (P) unclassified
D00404  Methsuximide (USP); Mesuximide (INN); Celontin (TN) (P) unclassified
D00405  Methyldopa (USP); Methyldopa hydrate (JP18); Aldomet (TN) (P) unclassified
D00407  Methylprednisolone (JP18/USP/INN); Medrol (TN) (P) CYP induction: CYP3A4
D00412  Zalcitabine (JAN/USP/INN); Hivid (TN) (CI,P) unclassified
D00413  Zidovudine (JP18/USP/INN); Azidothymidine; Retrovir (TN) (CI,P) unclassified
D00416  Miconazole (JP18/USP/INN); Monistat (TN); Oravig (TN) (P) unclassified
D00417  Milrinone (JAN/USP/INN); Milrila (TN) (P) Enzyme induction: UGT
D00418  Minoxidil (JAN/USP/INN); Loniten (TN); Riup (TN); Rogaine (TN) (P) unclassified
D00420  Mitotane (JAN/USP/INN); Lysodren (TN) (CI,P) unclassified
D00424  Rifabutin (JAN/USP/INN); Mycobutin (TN) (P) CYP induction: CYP3A4
D00426  Risperidone (JP18/USP/INN); Risperdal (TN) (P) CYP induction: CYP3A4
D00427  Ritonavir (JAN/USP/INN); Norvir (TN) (CI,P) unclassified
D00429  Saquinavir (JAN/USP/INN); Fortovase (TN) (CI,P) CYP induction: CYP3A4 / Transporter induction: ABCB1
D00430  Secobarbital (USP/INN); Seconal (TN) (P) unclassified
D00432  Nadolol (JP18/USP/INN); Corgard (TN) (P) unclassified
D00434  Simvastatin (JP18/USP/INN); MK-733; Zocor (TN) (P) CYP induction: CYP3A4 / Transporter inhibition: SLCO1B1
D00435  Nevirapine (JAN/USP/INN); Viramune (TN) (CI,P) CYP induction: CYP3A4
D00437  Nifedipine (JP18/USP/INN); Adalat (TN); Afeditab CR (TN); Procardia (TN) (P) CYP induction: CYP3A4
D00438  Nimodipine (USP/INN); Nimotop (TN); Nymalize (TN) (P) CYP induction: CYP3A4
D00445  Stavudine (USAN/INN); Sanilvudine (JAN); Zerit (TN) (CI,P) unclassified
D00453  Ofloxacin (JP18/USP/INN); Floxin (TN) (P) CYP induction: CYP3A4
D00454  Olanzapine (JAN/USP/INN); Zyprexa (TN) (P) unclassified
D00455  Omeprazole (JP18/USP/INN); Prilosec (TN) (P) unclassified
D00456  Ondansetron (JAN/USP/INN); Zofran ODT (TN) (P) CYP induction: CYP3A4
D00457  Quazepam (JAN/USP/INN); Doral (TN) (P) CYP induction: CYP3A4
D00458  Quetiapine fumarate (JP18/USP); Seroquel (TN) (P) CYP induction: CYP3A4
D00464  Oxazepam (JAN/USP/INN); Serax (TN) (P) unclassified
D00465  Oxybutynin (USAN/INN); Anturol (TN); Oxytrol (TN) (P) CYP induction: CYP3A4
D00467  Pipobroman (JAN/USAN/INN); Vercyte (TN) (CI,P) unclassified
D00468  Plicamycin (USAN/INN); Mithracin (TN) (CI,P) unclassified
D00470  Prazepam (JP18/USAN/INN); Centrax (TN) (P) unclassified
D00471  Praziquantel (JAN/USP/INN); Biltricide (TN) (CI,P) CYP induction: CYP3A4
D00472  Prednisolone (JP18/USP/INN); Delta-cortef (TN) (P) unclassified
D00473  Prednisone (USP); Prednisone monohydrate; Deltasone (TN); Meticorten (TN); Rayos (TN) (P) unclassified
D00474  Primidone (JP18/USP/INN); Mysoline (TN) (P) unclassified
D00477  Procainamide hydrochloride (JP18/USP); Procan SR (TN); Procanbid (TN); Pronestyl (TN) (P) unclassified
D00478  Procarbazine hydrochloride (JP18/USP); Matulane (TN) (CI,P) unclassified
D00483  Propranolol hydrochloride (JP18/USP); Inderal (TN); Innopran XL (TN) (P) unclassified
D00491  Paclitaxel (JAN/USP/INN); Abraxane (TN); Taxol (TN) (CI,P) CYP induction: CYP3A4
D00495  Paramethadione (INN); Paradione (TN) (P) unclassified
D00499  Pentobarbital (USP/INN); Nembutal (TN) (P) unclassified
D00500  Pentobarbital sodium (JAN/USP); Nembutal sodium (TN) (P) unclassified
D00502  Pergolide mesylate (USP); Pergolide mesilate (JAN); Permax (TN) (P) unclassified
D00504  Phenacemide (JAN/INN); Phenurone (TN) (P) unclassified
D00506  Phenobarbital (JP18/USP/INN); Luminal (TN) (P) unclassified
D00508  Phensuximide (USP/INN); Milontin (TN) (P) unclassified
D00511  Phenylephrine hydrochloride (JP18/USP); Neo-synephrine (TN) (P) unclassified
D00512  Phenytoin (JP18/USP/INN); Dilantin (TN) (P) unclassified
D00513  Pindolol (JP18/USP/INN); Blocklin-L (TN); Carvisken (TN); Visken (TN) (P) unclassified
D00514  Dexmedetomidine (USAN/INN); Dexdor (TN); Precedex (TN) (P) unclassified
D00528  Caffeine (USP); Anhydrous caffeine (JP18); Anhydrous caffeine (TN); Respia (TN) (P) unclassified
D00529  Montelukast sodium (JP18/USP); Singulair (TN) (P) CYP induction: CYP3A4
D00530  Zaleplon (JAN/USP/INN); Sonata (TN) (P) CYP induction: CYP3A4
D00531  Nitrazepam (JP18/USAN/INN); Benzalin (TN); Nitrazepam (TN) (P) unclassified
D00532  Glutethimide (JAN/INN); Doriden (TN) (P) unclassified
D00533  Oxcarbazepine (JAN/USP/INN); Oxtellar (TN); Trileptal (TN) (P) unclassified
D00535  Vigabatrin (JAN/USP/INN); Sabril (TN) (P) unclassified
D00536  Felbamate (USPINN); Felbatol (TN) (P) unclassified
D00537  Topiramate (JAN/USP/INN); Topamax (TN); Trokendi xr (TN) (P) CYP induction: CYP3A4
D00538  Zonisamide (JP18/USP/INN); Excegran (TN) (P) unclassified
D00539  Ethosuximide (JP18/USP/INN); Zarontin (TN) (P) CYP induction: CYP3A4
D00542  Halothane (JP18/USP/INN); Fluothane (TN) (P) CYP induction: CYP3A4
D00544  Methoxyflurane (USP/INN); Penthrane (TN) (P) CYP induction: CYP3A4
D00550  Midazolam (JAN/USP/INN); Dormicum (TN); Buccolam (TN); Nayzilam (TN) (P) CYP induction: CYP3A4
D00553  Prilocaine (USP/INN); Propitocaine (JAN) (P) unclassified
D00554  Ethinyl estradiol (USP); Ethinylestradiol (JP18/INN); Estinyl (TN) (P) CYP induction: CYP3A4
D00555  Amobarbital (JP18/INN); Isomytal (TN) (P) unclassified
D00557  Methaqualone (JAN/USAN/INN) (P) unclassified
D00558  Carbidopa (USP); Carbidopa hydrate (JP18); Lodosyn (TN) (P) unclassified
D00559  Pramipexole dihydrochloride (USP); Pramipexole hydrochloride hydrate (JAN); Pramipexole dihydrochloride monohydrate; Mirapex (TN) (P) unclassified
D00560  Pimozide (JP18/USP/INN); Orap (TN) (P) CYP induction: CYP3A4
D00563  Mirtazapine (JAN/USP/INN); Remeron (TN); Reflex (TN) (P) CYP induction: CYP3A4
D00564  Warfarin sodium (USP); Coumadin (TN); Jantoven (TN) (P) unclassified
D00567  Celecoxib (JP18/USP/INN); Celebrex (TN); Onsenal (TN) (CI,P) unclassified
D00570  Colchicine (JP18/USP); Colchicine (TN) (P) CYP induction: CYP3A4 / Transporter induction: ABCB1
D00578  Voriconazole (JP18/USP/INN); Vfend (TN) (CI,P) unclassified
D00583  Thiotepa (JAN/USP/INN); Thioplex (TN); Tepadina (TN); Rethio (TN) (CI,P) unclassified
D00584  Fluorouracil (JP18/USP/INN); 5-FU (TN); Adrucil (TN); Carac (TN); Fluoroplex (TN) (CI,P) unclassified
D00585  Mifepristone (JAN/USAN/INN); Korlym (TN); Mifeprex (TN) (P) CYP induction: CYP3A4
D00588  Levofloxacin (USP); Levofloxacin hydrate (JP18); Levofloxacin hemihydrate; Iquix (TN); Levaquin (TN); Quixin (TN) (P) unclassified
D00591  Ethionamide (JP18/USP/INN); Trecator (TN) (P) unclassified
D00592  Dapsone (USP); Diaphenylsulfone (JAN); Aczone (TN) (P) CYP induction: CYP3A4
D00593  Glimepiride (JP18/USP/INN); Amaryl (TN) (P) unclassified
D00594  Repaglinide (JAN/USP/INN); Prandin (TN); Surepost (TN) (P) unclassified
D00595  Buformin (USAN/INN) (P) unclassified
D00596  Rosiglitazone maleate (JAN/USP); Avandia (TN) (P) unclassified
D00597  Acebutolol hydrochloride (JP18/USP); Sectral (TN) (P) unclassified
D00598  Betaxolol hydrochloride (JP18/USP); Betoptic (TN); Kerlone (TN) (P) unclassified
D00599  Carteolol hydrochloride (JP18/USP); Cartrol (TN); Ocupress (TN) (P) unclassified
D00601  Metoprolol tartrate (JP18/USP); Lopressor (TN) (P) unclassified
D00602  Penbutolol sulfate (JP18/USP); Levatol (TN) (P) unclassified
D00603  Timolol maleate (JP18/USP); Blocadren (TN); Istalol (TN); Timoptic (TN) (P) unclassified
D00604  Clonidine hydrochloride (JP18/USP); Nexiclon (TN); Kapvay (TN); Duraclon (TN); Catapres (TN) (P) unclassified
D00606  Guanfacine hydrochloride (JAN/USP); Intuniv (TN); Tenex (TN) (P) CYP induction: CYP3A4
D00608  Doxazosin mesylate (USP); Doxazosin mesilate (JP18); Cardura (TN) (P) unclassified
D00609  Prazosin hydrochloride (JP18/USP); Minipress (TN) (P) unclassified
D00611  Mecamylamine hydrochloride (USP); Inversine (TN) (P) unclassified
D00612  Trimetaphan camsilate (JAN/INN); Trimetaphan camsylate; Arfonad (TN) (P) unclassified
D00614  Sodium nitroprusside (USP); Sodium nitroprusside hydrate (JAN); Nitropress (TN) (P) unclassified
D00615  Amlodipine besylate (USP); Amlodipine besilate (JP18); Norvasc (TN) (P) CYP induction: CYP3A4
D00616  Diltiazem hydrochloride (JP18/USP); Cardizem (TN); Cartia XT (TN); Dilacor XR (TN); Dilt-CD (TN) (P) CYP induction: CYP3A4
D00617  Nicardipine hydrochloride (JP18/USAN); Cardene (TN) (P) CYP induction: CYP3A4
D00618  Nisoldipine (JAN/USAN/INN); Sular (TN) (P) CYP induction: CYP3A4
D00619  Verapamil hydrochloride (JP18/USP); Calan (TN); Covera-hs (TN); Vasolan (TN); Verelan (TN) (P) CYP induction: CYP3A4 / Transporter induction: ABCB1
D00621  Enalapril maleate (JP18/USP); Renivace (TN); Vasotec (TN) (P) unclassified
D00625  Miglitol (JP18/USAN/INN); Glyset (TN) (P) unclassified
D00629  Nitrendipine (JP18/USAN/INN); Baypress (TN) (P) CYP induction: CYP3A4
D00631  Bepridil hydrochloride (USAN); Bepridil hydrochloride hydrate (JAN); Vascor (TN) (P) CYP induction: CYP3A4
D00632  Dobutamine hydrochloride (JP18/USP); Dobutrex (TN) (P) unclassified
D00633  Dopamine hydrochloride (JP18/USP); Actopamin (TN); Intropin (TN) (P) unclassified
D00634  Bisoprolol fumarate (JP18/USP); Zebeta (TN) (P) unclassified
D00635  Metoprolol succinate (USP); Toprol XL (TN) (P) unclassified
D00636  Amiodarone hydrochloride (JP18/USP); Ancaron (TN); Cordarone (TN); Nexterone (TN) (P) CYP induction: CYP3A4
D00637  Disopyramide phosphate (JAN/USP); Norpace (TN) (P) CYP induction: CYP3A4
D00638  Flecainide acetate (JP18/USP); Tambocor (TN) (P) unclassified
D00639  Mexiletine hydrochloride (JP18/USP); Mexitil (TN) (P) unclassified
D00640  Propafenone hydrochloride (JP18/USP); Rythmol (TN) (P) CYP induction: CYP3A4
D00642  Quinidine gluconate (USP); Quinaglute (TN) (P) unclassified
D00643  Quinidine polygalacturonate; Cardioquin (TN) (P) unclassified
D00644  Esmolol hydrochloride (JAN/USP); Brevibloc (TN) (P) unclassified
D00645  Bretylium tosylate (USP); Bretylium tosilate (INN); Bretylol (TN) (P) unclassified
D00646  Tolterodine (USAN/INN) (P) CYP induction: CYP3A4
D00647  Dofetilide (JAN/USP/INN); Tikosyn (TN) (P) unclassified
D00648  Ibutilide fumarate (USP); Corvert (TN) (P) unclassified
D00653  Dorzolamide hydrochloride (JP18/USP); Trusopt (TN) (P) CYP induction: CYP3A4
D00661  Cevimeline hydrochloride (USAN); Cevimeline hydrochloride hydrate (JAN); Evoxac (TN); Saligren (TN) (P) CYP induction: CYP3A4
D00670  Donepezil hydrochloride (JP18/USP); Aricept (TN) (P) CYP induction: CYP3A4
D00672  Hydroxyzine hydrochloride (JP18/USP); Hydroxyzine dihydrochloride; Atarax (TN); Vistaril (TN) (P) unclassified
D00674  Naratriptan hydrochloride (JAN/USP); Amerge (TN) (P) CYP induction: CYP3A4
D00677  Granisetron hydrochloride (JAN/USP); Kytril (TN) (P) CYP induction: CYP3A4
D00678  Ondansetron hydrochloride hydrate (JAN/USP); Ondansetron hydrochloride; Zofran (TN) (P) CYP induction: CYP3A4
D00679  Ergotamine tartrate (JP18/USP); Ergomar (TN) (P) CYP induction: CYP3A4
D00680  Methylergonovine maleate (USP); Methylergometrine maleate (JP18); Methergine (TN) (P) CYP induction: CYP3A4
D00687  Salmeterol xinafoate (JAN/USP); Serevent (TN) (P) CYP induction: CYP3A4
D00689  Beclomethasone dipropionate (USP); Beclometasone dipropionate (JP18); Beclovent (TN); Qnasl (TN); Vanceril (TN) (P) CYP induction: CYP3A4
D00690  Mometasone furoate (JAN/USP); Asmanex (TN); Elocon (TN) (P) CYP induction: CYP3A4
D00693  Chlordiazepoxide hydrochloride (JAN/USP); Librium (TN) (P) unclassified
D00694  Clorazepate dipotassium (JP18/USP); Tranxene (TN) (P) unclassified
D00695  Flurazepam hydrochloride (USP); Flurazepam dihydrochloride; Dalmane (TN) (P) unclassified
D00696  Midazolam hydrochloride (USAN); Versed (TN) (P) CYP induction: CYP3A4
D00698  Aprobarbital (INN); Alurate (TN) (P) unclassified
D00700  Mephobarbital (JAN/USP); Methylphenobarbital (INN); Mebaral (TN) (P) unclassified
D00701  Phenobarbital sodium (JAN/USP/INN); Luminal sodium (TN) (P) unclassified
D00702  Buspirone hydrochloride (USP); Buspar (TN) (P) unclassified
D00704  Ethchlorvynol (JAN/USP/INN); Placidyl (TN) (P) unclassified
D00705  Paraldehyde (USP); Paral (TN) (P) unclassified
D00706  Zolpidem tartrate (JP18/USP); Ambien (TN); Intermezzo (TN) (P) CYP induction: CYP3A4
D00708  Ethotoin (JAN/USP/INN); Accenon (TN); Peganone (TN) (P) unclassified
D00709  Levetiracetam (JAN/USP/INN); Keppra (TN); E keppra (TN) (P) unclassified
D00710  Valproate sodium (USAN); Sodium valproate (JP18); Depakene (TN); Selenica (TN) (P) unclassified
D00712  Methohexital sodium (USP); Brevital sodium (TN) (P) unclassified
D00714  Thiopental sodium (JP18/USP/INN); Pentothal (TN) (P) unclassified
D00722  Oxybutynin chloride (USP); Oxybutynin hydrochloride (JP18); Ditropan (TN); Gelnique (TN) (P) CYP induction: CYP3A4
D00724  Rabeprazole sodium (JP18/USP); Aciphex (TN); Pariet (TN) (P) CYP induction: CYP3A4
D00725  Dolasetron mesylate (USP); Anzemet (TN) (P) unclassified
D00726  Metoclopramide (JP18/INN); Elieten (TN); Terperan (TN) (P) unclassified
D00729  Loperamide hydrochloride (JAN/USP); Imodium (TN) (P) CYP induction: CYP3A4 / Transporter induction: ABCB1
D00749  Leflunomide (JAN/USP/INN); Arava (TN) (P) CYP induction: CYP3A4
D00751  Methylprednisolone sodium succinate (JAN/USP); A-methapred (TN); Solu-medrol (TN) (P) CYP induction: CYP3A4
D00752  Mycophenolate mofetil (JAN/USP); Cellcept (TN) (P) unclassified
D00753  Sirolimus (JAN/USAN/INN); Rapamune (TN); Rapamycin (TN) (CI,P) CYP induction: CYP3A4 / Transporter induction: ABCB1
D00762  Metyrosine (USP); Metirosine (JAN/INN); Demser (TN) (P) unclassified
D00769  Clopidogrel bisulfate (USP); Clopidogrel sulfate (JP18); Clopidogrel sulfate tablets (JP18); Clopidogrel hydrogen sulphate; Isocover (TN); Plavix (TN) (P) unclassified
D00776  Tizanidine hydrochloride (JP18/USP); Zanaflex (TN) (P) unclassified
D00777  Amantadine hydrochloride (JP18/USP); Symmetrel (TN); Gocovri (TN); Osmolex er (TN) (P) unclassified
D00779  Biperiden (JAN/USP/INN); Akineton (TN) (P) unclassified
D00780  Bromocriptine mesylate (USP); Bromocriptine mesilate (JP18); Parlodel (TN) (P) CYP induction: CYP3A4
D00781  Entacapone (JP18/USP/INN); Comtan (TN) (P) unclassified
D00784  Ropinirole hydrochloride (JAN/USP); Requip (TN) (P) unclassified
D00785  Selegiline hydrochloride (JAN/USP); Eldepryl (TN) (P) CYP induction: CYP3A4
D00786  Tolcapone (JAN/USP/INN); Tasmar (TN) (P) unclassified
D00787  Trihexyphenidyl hydrochloride (JP18/USP); Artane (TN) (P) unclassified
D00794  Loxapine succinate (USP); Loxitane (TN) (P) CYP induction: CYP3A4
D00804  Ivermectin (JAN/USP/INN); Sklice (TN); Soolantra (TN); Stromectol (TN) (P) CYP induction: CYP3A4 / Transporter induction: ABCB1
D00809  Amitriptyline hydrochloride (JP18/USP); Elavil (TN) (P) CYP induction: CYP3A4
D00811  Clomipramine hydrochloride (JP18/USP); Anafranil (TN) (P) CYP induction: CYP3A4
D00815  Imipramine hydrochloride (JP18/USP); Tofranil (TN) (P) CYP induction: CYP3A4
D00816  Nortriptyline hydrochloride (JP18/USP/INN); Pamelor (TN) (P) unclassified
D00820  Trazodone hydrochloride (JAN/USP); Desyrel (TN) (P) CYP induction: CYP3A4
D00821  Venlafaxine hydrochloride (JAN/USP); Effexor (TN) (P) unclassified
D00822  Citalopram hydrobromide (USP); Celexa (TN) (P) CYP induction: CYP3A4 / Transporter induction: ABCB1
D00825  Sertraline hydrochloride (JAN/USP); Zoloft (TN) (P) CYP induction: CYP3A4
D00829  Eflornithine hydrochloride (USAN); Iwilfin (TN); Vaniqa (TN) (CI,P) unclassified
D00831  Mefloquine hydrochloride (JP18/USP); Lariam (TN) (P) unclassified
D00836  Buprenorphine hydrochloride (JP18/USP); Buprenex (TN) (P) CYP induction: CYP3A4
D00840  Levomethadyl acetate hydrochloride (USAN); Orlaam (TN) (P) CYP induction: CYP3A4
D00847  Oxycodone hydrochloride (USP); Oxecta (TN); Oxycontin (TN); Roxicodone (TN) (P) CYP induction: CYP3A4
D00866  Kanamycin sulfate (USP); Kanamycin monosulfate (JP18); Kantrex (TN) (P) unclassified
D00875  Aminosalicylate sodium (USP); Parasal sodium (TN) (P) unclassified
D00877  Cycloserine (JP18/USP/INN); Seromycin (TN) (P) unclassified
D00878  Ethambutol hydrochloride (JP18/USP); Myambutol (TN) (P) unclassified
D00879  Rifapentine (USAN/INN); Priftin (TN) (P) unclassified
D00880  Butoconazole nitrate (USP); Femstat (TN); Gynazole-1 (TN) (P) unclassified
D00881  Econazole nitrate (JAN/USP); Ecoza (TN); Spectazole (TN) (P) unclassified
D00882  Miconazole nitrate (JP18/USP); Micatin (TN); Monistat (TN) (P) unclassified
D00885  Oxiconazole nitrate (JAN/USAN); Oxistat (TN) (P) unclassified
D00886  Sulconazole nitrate (JAN/USP); Exelderm (TN) (P) unclassified
D00887  Atorvastatin calcium anhydorous; Lipitor (TN) (P) CYP induction: CYP3A4 / Transporter inhibition: SLCO1B1 SLCO1B3 / Transporter induction: ABCB1
D00888  Terconazole (USP/INN); Terazol 3 (TN) (P) unclassified
D00889  Cerivastatin sodium (JAN/USAN); Baycol (TN) (P) CYP induction: CYP3A4
D00890  Tioconazole (JAN/USP/INN); Vagistat-1 (TN) (P) unclassified
D00891  Abacavir sulfate (JAN/USP); Ziagen (TN) (CI,P) unclassified
D00892  Fluvastatin sodium (JAN/USP); Lescol (TN) (P) CYP induction: CYP3A4 / Transporter inhibition: SLCO1B1
D00894  Amprenavir (JAN/USAN/INN); Agenerase (TN) (CI,P) CYP induction: CYP3A4
D00895  Delavirdine mesylate (USAN); Delavirdine mesilate (JAN); Rescriptor (TN) (CI,P) unclassified
D00896  Efavirenz (JAN/USP/INN); Sustiva (TN) (CI,P) CYP induction: CYP3A4
D00897  Indinavir sulfate (USP); Crixivan (TN) (CI,P) CYP induction: CYP3A4
D00899  Nelfinavir mesylate (USAN/INN); Nelfinavir mesilate (JAN); Viracept (TN) (CI,P) CYP induction: CYP3A4
D00944  Metformin hydrochloride (JP18/USP); Glucophage (TN) (P) unclassified
D00945  Pioglitazone hydrochloride (JP18/USP); Actos (TN) (P) unclassified
D00947  Linezolid (JAN/USAN/INN); Zyvox (TN) (P) unclassified
D00948  Estropipate (USP); Piperazine estrone sulfate; Ogen (TN) (P) CYP induction: CYP3A4
D00950  Levonorgestrel (JAN/USP/INN); Mirena (TN); Norplant (TN); Skyla (TN) (P) unclassified
D00963  Exemestane (JAN/USP/INN); Aromasin (TN) (P) CYP induction: CYP3A4
D00964  Letrozole (JAN/USP/INN); Femara (TN) (P) CYP induction: CYP3A4
D00966  Tamoxifen citrate (JP18/USP); Nolvadex (TN); Soltamox (TN) (P) CYP induction: CYP3A4
D00967  Toremifene citrate (JAN/USAN); Fareston (TN) (P) CYP induction: CYP3A4
D00969  Meloxicam (JAN/USP/INN); Mobic (TN) (P) unclassified
D00972  Betamethasone sodium phosphate (JP18/USP); Celestone (TN) (P) unclassified
D00973  Cortisone acetate (JP18/USP); Cortone acetate (TN) (P) unclassified
D00975  Dexamethasone sodium phosphate (JAN/USP); Dalalone (TN); Maxidex (TN) (P) CYP induction: CYP3A4
D00976  Hydrocortisone cypionate (P) unclassified
D00977  Hydrocortisone sodium phosphate (JP18/USP); Hydrocortone phosphate (TN) (P) unclassified
D00978  Hydrocortisone sodium succinate (JP18/USP); A-hydrocort (TN); Solu-cortef (TN) (P) unclassified
D00979  Methylprednisolone acetate (JAN/USP); Depo-medrol (TN) (P) CYP induction: CYP3A4
D00980  Prednisolone acetate (JP18/USP/INN); Econopred (TN); Pred forte (TN) (P) unclassified
D00981  Prednisolone sodium phosphate (JP18/USP); Pediapred (TN) (P) unclassified
D00982  Prednisolone tebutate (JAN/USP); Hydeltra-TBA (TN) (P) unclassified
D00983  Triamcinolone acetonide (JP18/USP); Azmacort (TN); Kenalog (TN); Nasacort (TN) (P) unclassified
D00984  Triamcinolone diacetate (JAN/USP); Aristocort (TN) (P) unclassified
D00985  Triamcinolone hexacetonide (USP/INN); Aristospan (TN) (P) unclassified
D00986  Fludrocortisone acetate (JP18/USP); Florinef acetate (TN) (P) unclassified
D00987  Cabergoline (JP18/USP/INN); Cabaser (TN); Dostinex (TN) (P) CYP induction: CYP3A4
D00996  Epinephrine hydrochloride (JAN); Adrenalin chloride (TN) (P) unclassified
D01007  Propiverine hydrochloride (JP18); Bup-4 (TN); Mictonorm (TN) (P) CYP induction: CYP3A4
D01018  Mephentermine sulfate; Wyamine sulfate (TN) (P) unclassified
D01019  Metaraminol bitartrate (JAN/USP); Aramine (TN) (P) unclassified
D01020  Methoxamine hydrochloride (JAN); Vasoxyl (TN) (P) unclassified
D01025  Levobunolol hydrochloride (JAN/USP); Betagan (TN) (P) unclassified
D01026  Sotalol hydrochloride (JAN/USP); Betapace (TN); Sorine (TN) (P) unclassified
D01041  Sparteine (INN) (P) unclassified
D01055  Emivirine (USAN/INN); Coactinon (TN) (CI,P) unclassified
D01056  Benzbromarone (JP18/USAN/INN); Uroleap (TN) (P) unclassified
D01059  Nimustine hydrochloride (JAN); Nidran (TN) (CI,P) unclassified
D01061  Irinotecan hydrochloride (USP); Irinotecan hydrochloride hydrate (JP18); Irinotecan hydrochloride trihydrate; CPT 11; CPT-11; Campto (TN); Camptosar (TN); Onivyde (TN) (CI,P) unclassified
D01064  Raltitrexed (JAN/USAN/INN); Tomudex (TN) (CI,P) unclassified
D01068  Vinblastine sulfate (JP18/USP); Exal (TN); Velban (TN) (CI,P) CYP induction: CYP3A4
D01071  Hexobarbital (JAN/INN) (P) unclassified
D01072  Chloramphenicol palmitate (JP18/USP); Chloromycetin palmitate (TN) (P) unclassified
D01092  Lanoconazole (JP18/INN); Latoconazole; Astat (TN) (P) unclassified
D01096  Hydroxyzine pamoate (JP18/USP); Atarax-P (TN); Vistaril pamoate (TN) (P) unclassified
D01098  Maxacalcitol (JAN/USAN/INN); Oxarol (TN); Prezios (TN) (P) CYP induction: CYP3A4
D01101  Bromperidol (JAN/USAN/INN); Impromen (TN) (P) CYP induction: CYP3A4
D01104  Barnidipine hydrochloride (JAN); Hypoca (TN) (P) CYP induction: CYP3A4
D01111  Nateglinide (JP18/USP/INN); Starsis (TN) (P) unclassified
D01115  Eplerenone (JP18/USAN/INN); Inspra (TN) (P) CYP induction: CYP3A4
D01121  Rebamipide (JP18/INN); Mucosta (TN) (P) CYP induction: CYP3A4
D01131  Lafutidine (JP18/INN); Protecadin (TN) (P) CYP induction: CYP3A4
D01133  Pimobendan (JAN/USAN/INN); Acardi (TN) (P) unclassified
D01145  Azelnidipine (JP18/INN); Calblock (TN) (P) CYP induction: CYP3A4
D01148  Tolterodine tartrate (JAN/USP); Detrol (TN); Detrusitol (TN) (P) CYP induction: CYP3A4
D01150  Methyprylon (JAN/INN); Noludar (TN) (P) unclassified
D01155  Gemcitabine hydrochloride (JAN/USP); Gemzar (TN) (CI,P) unclassified
D01160  Saquinavir mesylate (USP); Saquinavir mesilate (JAN); Invirase (TN) (CI,P) CYP induction: CYP3A4 / Transporter induction: ABCB1
D01161  Fulvestrant (JAN/USP/INN); Faslodex (TN) (P) CYP induction: CYP3A4
D01163  Ergonovine maleate (USP); Ergometrine maleate (JP18); Ergometrine (TN) (P) CYP induction: CYP3A4
D01164  Aripiprazole (JAN/USP/INN); Abilify (TN) (P) CYP induction: CYP3A4
D01173  Cilnidipine (JP18/INN); Atelec (TN) (P) CYP induction: CYP3A4
D01176  Blonanserin (JAN/INN); AD 5423 (P) CYP induction: CYP3A4
D01182  Alprenolol hydrochloride (JP18/USAN); Regletin (TN) (P) unclassified
D01190  Ethylphenacemide (JAN); Pheneturide (INN) (P) unclassified
D01195  Prothionamide (JP18); Protionamide (INN); Trevintix (TN) (P) unclassified
D01198  Toborinone (JAN/USAN/INN) (P) unclassified
D01199  Emtricitabine (JAN/USAN/INN); Emtriva (TN) (CI,P) unclassified
D01205  Dexmedetomidine hydrochloride (JAN/USP); Igalmi (TN); Precedex (TN) (P) unclassified
D01207  Omeprazole sodium (USAN); Losec sodium (TN) (P) unclassified
D01208  Aluminum clofibrate (JAN/INN); Alfibrate (TN) (P) unclassified
D01213  Tolvaptan (JAN/USAN/INN); Samsca (TN) (P) CYP induction: CYP3A4 / Transporter induction: ABCB1
D01217  Dydrogesterone (JP18/USP/INN); Duphaston (TN); Gynorest (TN) (P) CYP induction: CYP3A4
D01223  Capecitabine (JAN/USP/INN); Xeloda (TN) (CI,P) unclassified
D01227  Bosentan (USAN); Bosentan hydrate (JAN); Tracleer (TN) (P) CYP induction: CYP3A4
D01229  Paramethasone acetate (JAN/USAN); Haldrone (TN) (P) unclassified
D01230  Flunitrazepam (JP18/USAN/INN); Rohypnol (TN) (P) unclassified
D01231  Piroheptine hydrochloride (JAN); Trimol (TN) (P) unclassified
D01238  Bucladesine sodium (JAN); Actosin (TN) (P) unclassified
D01239  Prednisolone sodium succinate (JP18/USP); Kohakusanin (TN) (P) unclassified
D01240  Deslanoside (JP18/USP/INN); Cedilanid-d (TN) (P) unclassified
D01243  Prilocaine hydrochloride (USP); Propitocaine hydrochloride (JAN); Citanest (TN) (P) unclassified
D01244  Tegafur (JP18/USAN/INN); Atillon (TN) (CI,P) unclassified
D01245  Bromazepam (JP18/USAN/INN); Lectopam (TN) (P) unclassified
D01253  Clobazam (JAN/USAN/INN); Mystan (TN); Onfi (TN) (P) CYP induction: CYP3A4
D01254  Tofisopam (JP18/INN); Emandaxin (TN) (P) unclassified
D01264  Daunorubicin hydrochloride (JP18/USP); Cerubidine (TN) (CI,P) unclassified
D01266  Difluprednate (JAN/USAN/INN); Durezol (TN) (P) unclassified
D01268  Cloxazolam (JP18/INN); Sepazon (TN) (P) unclassified
D01269  Solifenacin succinate (JAN/USAN/INN); Vesicare (TN) (P) CYP induction: CYP3A4
D01270  Carboquone (JAN/INN); Esquinon (TN) (CI,P) unclassified
D01272  Clobetasol propionate (JP18/USP); Clobex (TN); Cormax (TN); Olux (TN) (P) unclassified
D01273  Clobetasone butyrate (JAN/USAN); Kindavate (TN) (P) unclassified
D01275  Doxorubicin hydrochloride (JP18/USP); Adriacin (TN); Adriamycin (TN); Doxil (TN); Rubex (TN) (CI,P) unclassified
D01276  Atazanavir sulfate (JAN/USAN); Reyataz (TN) (CI,P) unclassified
D01277  Droxidopa (JP18/USAN/INN); Dops (TN); Northera (TN) (P) unclassified
D01278  Oxazolam (JP18/INN); Serenal (TN) (P) unclassified
D01279  Flutoprazepam (JP18/INN); Restas (TN) (P) unclassified
D01280  Warfarin potassium (JP18); Athrombin-K (TN) (P) unclassified
D01285  Lofepramine hydrochloride (JAN/USAN); Amplit (TN) (P) unclassified
D01286  Flutazolam (JAN/INN); Coreminal (TN) (P) unclassified
D01287  Levobupivacaine hydrochloride (JAN/USAN); Chirocaine (TN) (P) CYP induction: CYP3A4
D01292  Medazepam (JP18/INN); Pamnace (TN) (P) unclassified
D01293  Ethyl loflazepate (JP18/INN); Meilax (TN) (P) CYP induction: CYP3A4
D01302  Hydralazine hydrochloride (JP18/USP); Apresoline (TN) (P) unclassified
D01303  Flunarizine hydrochloride (JAN/USAN) (P) unclassified
D01304  Amezinium metilsulfate (JAN); Risumic (TN) (P) unclassified
D01307  Midodrine hydrochloride (JAN/USP); Pro-Amatine (TN) (P) unclassified
D01308  Halcinonide (JAN/USP/INN); Halog (TN) (P) unclassified
D01310  Secobarbital sodium (JAN/USP); Seconal sodium (TN) (P) unclassified
D01316  Mexazolam (JAN/INN); Melex (TN) (P) CYP induction: CYP3A4
D01322  Troleandomycin (USAN/INN); Triacetyloleandomycin (JAN); TAO; Tao (TN) (P) CYP induction: CYP3A4
D01326  Aprindine hydrochloride (JP18/USAN); Aspenon (TN) (P) unclassified
D01327  Diflorasone diacetate (JP18/USP); Florone (TN); Psorcon (TN) (P) unclassified
D01328  Clotiazepam (JP18/INN); Rize (TN) (P) unclassified
D01333  Urapidil (JP18/INN); Ebrantil (TN) (P) unclassified
D01350  Streptomycin sulfate (JP18/USP); Streptomycin sulfate (TN) (P) unclassified
D01354  Fludiazepam (JP18/INN); Erispan (TN) (P) unclassified
D01355  Tramadol hydrochloride (JP18/USP); Ultram (TN) (P) CYP induction: CYP3A4
D01356  Glymidine sodium (JAN/USAN/INN) (P) unclassified
D01357  Betamethasone valerate (JP18/USP); Beta-Val (TN); Luxiq (TN); Rinderon-V (TN) (P) unclassified
D01358  Mianserin hydrochloride (JAN/USAN); Tetramide (TN) (P) CYP induction: CYP3A4
D01363  Carboplatin (JP18/USP/INN); Paraplatin (TN) (CI,P) unclassified
D01367  Fluorometholone (JP18/USP/INN); NSC 33001; Fluor-op (TN); Fml (TN); Oxylone (TN) (P) unclassified
D01370  Cladribine (JAN/USP/INN); Leustatin (TN); Mavenclad (TN) (CI,P) unclassified
D01372  Zopiclone (JP18/INN); Amoban (TN); Zopiclone (TN) (P) CYP induction: CYP3A4
D01379  Proscillaridin (JAN/USAN/INN); Talusin (TN) (P) unclassified
D01382  Metharbital (JAN/INN); Gemonil (TN) (P) unclassified
D01386  Ephedrine hydrochloride (JP18/USP); Ephedrine hydrochloride (TN) (P) unclassified
D01387  Amcinonide (JAN/USP/INN); Cyclocort (TN) (P) unclassified
D01390  Isoproterenol hydrochloride (USP); dl-Isoprenaline hydrochloride (JAN); Isuprel (TN); Proternol-S (TN) (P) unclassified
D01391  Bromovalerylurea (JP18); Bromisoval (INN); Bromisovalum; Bromovalerylurea (TN); Bromural (TN); Brovarin (TN) (P) unclassified
D01399  Fentanyl citrate (JP18/USP); Abstral (TN); Fentora (TN); Lazanda (TN); Oralet (TN) (P) CYP induction: CYP3A4
D01402  Betamethasone acetate (JAN/USP) (P) unclassified
D01405  Norfenefrine hydrochloride (JAN); Zondel (TN) (P) unclassified
D01408  Flurazepam hydrochloride (JP18); Flurazepam monohydrochloride; Dalmate (TN) (P) unclassified
D01413  Estradiol valerate (JAN/USP/INN); Deladumone (TN) (P) CYP induction: CYP3A4
D01418  Tamibarotene (JAN/USAN/INN); Am 80; Amnoid (TN) (P) CYP induction: CYP3A4
D01425  Lopinavir (JAN/USP/INN) (CI,P) unclassified
D01429  Fosfluconazole (JAN/INN); Prodif (TN) (P) unclassified
D01434  Deprodone propionate (JAN); Allomidon (TN) (P) unclassified
D01441  Imatinib mesylate (USAN); Imatinib mesilate (JAN); Gleevec (TN); Glivec (TN) (CI,P) CYP induction: CYP3A4
D01442  Hydrocortisone succinate (JP18) (P) unclassified
D01450  Bupivacaine hydrochloride (USP); Bupivacaine hydrochloride hydrate (JP18); Marcaine (TN) (P) CYP induction: CYP3A4
D01453  Caffeine hydrate (JP18); Caffeine monohydrate; Caffeine (TN) (P) unclassified
D01454  Bupranolol hydrochloride (JP18) (P) unclassified
D01455  Cifenline succinate (USAN); Cibenzoline succinate (JP18); Cibenol (TN); Cipralan (TN) (P) CYP induction: CYP3A4
D01464  Flumethasone pivalate (USP); Flumetasone pivalate (JAN/BAN); Locorten (TN) (P) unclassified
D01468  Nemonapride (JAN/INN); Emilace (TN) (P) CYP induction: CYP3A4
D01471  Esatenolol (JAN/INN); (S)-Atenolol (P) unclassified
D01478  Ebastine (JP18/USAN/INN); Kestine (TN) (P) CYP induction: CYP3A4
D01480  Isoconazole nitrate (JAN); Adestan-G (TN) (P) unclassified
D01481  Dihydrocodeine phosphate (JP18); Dihydro (TN) (P) unclassified
D01492  Bucumolol hydrochloride (JP18) (P) unclassified
D01501  Isoniazid calcium pyruvinate (JAN); Pyruvic acid calcium isoniazid (P) unclassified
D01504  Bufetolol hydrochloride (JP18); Adobiol (TN) (P) unclassified
D01510  Dexamethasone metasulfobenzoate sodium (JAN); Dexamethazone metasulfobenzoate sodium; Dexapos; Santeson (TN) (P) CYP induction: CYP3A4
D01512  Befunolol hydrochloride (JAN); Bentos (TN) (P) unclassified
D01514  Etizolam (JP18/INN); Sedekopan (TN) (P) CYP induction: CYP3A4
D01516  Tretinoin tocoferil (JAN); Tocoretinate (CI,P) unclassified
D01546  Dothiepin hydrochloride (USAN); Dosulepin hydrochloride (JAN); Dosulepin (TN) (P) unclassified
D01553  Manidipine hydrochloride (JP18); Manidipine dihydrochloride; Calslot (TN) (P) CYP induction: CYP3A4
D01554  Pilsicainide hydrochloride hydrate (JP18); Pilsicainide hydrochloride; SUN 1165 (TN); Sunrythm (TN) (P) unclassified
D01562  Aranidipine (JAN/INN); Sapresta (TN) (P) CYP induction: CYP3A4
D01564  Rilmazafone hydrochloride hydrate (JP18); Rilmazafone hydrochloride dihydrate; Rilmazafone hydrochloride; Rhythmy (TN) (P) CYP induction: CYP3A4
D01573  Etilefrine hydrochloride (JP18); Etilefrine hydrochloride (TN) (P) unclassified
D01593  Nimetazepam (JAN/INN); Erimin (TN) (P) unclassified
D01599  Gliclazide (JP18/INN); Glimicron (TN) (P) unclassified
D01603  Bethanidine sulfate (JAN/USAN); Tenathan (TN) (P) unclassified
D01604  Efonidipine hydrochloride ethanolate (JAN); Efonidipine hydrochloride ethanol; Efonidipine hydrochloride; NZ 105 ethanolate; Landel (TN) (P) unclassified
D01613  Azasetron hydrochloride (JAN); Serotone (TN) (P) unclassified
D01615  Dexamethasone palmitate (JAN); Dexamethasone 21-palmitate; Limethason (TN) (P) CYP induction: CYP3A4
D01617  Estradiol dipropionate (JAN); Ovahormon (TN) (P) CYP induction: CYP3A4
D01619  Hydrocortisone butyrate (JP18/USP); Locoid (TN) (P) unclassified
D01620  Neticonazole hydrochloride (JAN); Atolant (TN) (P) unclassified
D01624  Sarpogrelate hydrochloride (JP18); Anplag (TN) (P) CYP induction: CYP3A4
D01632  Dexamethasone dipropionate (USAN); Dexamethasone propionate (JAN); Hifmeta (TN) (P) CYP induction: CYP3A4
D01637  Betamethasone dipropionate (JP18/USP); Diprolene (TN); Rinderon-DP (TN); Sernivo (TN) (P) unclassified
D01643  Aluminoparaaminosalicylate calcium hydrate (JAN); Aluminoparaaminosalicylate calcium pentahydrate; Aluminoparaaminosalicylate calcium; Alumino nippas calcium (TN) (P) unclassified
D01656  Brovincamine fumarate (JAN); Sabromin (TN) (P) unclassified
D01657  Lormetazepam (JAN/USAN/INN); Loramet (TN) (P) unclassified
D01663  Quinine ethylcarbonate (JP18); Quinine ethylcarbonate (TN) (P) CYP induction: CYP3A4 / Transporter induction: ABCB1
D01664  Omoconazole nitrate (JAN/USAN) (P) unclassified
D01665  Voglibose (JP18/USAN/INN); Basen (TN) (P) unclassified
D01689  Loteprednol etabonate (JAN/USAN); Lotemax (TN) (P) unclassified
D01690  Vesnarinone (JAN/USAN/INN); Arkin Z (TN) (P) unclassified
D01692  Alfuzosin hydrochloride (JAN/USAN); Uroxatral (TN) (P) CYP induction: CYP3A4
D01697  Colforsin daropate hydrochloride (JAN); Nkh 477; Adehl (TN) (P) unclassified
D01699  Darifenacin hydrobromide (JAN/USAN); Enablex (TN) (P) CYP induction: CYP3A4
D01703  Ciclesonide (JAN/USAN/INN); Alvesco (TN); Omnaris (TN); Zetonna (TN) (P) CYP induction: CYP3A4
D01708  Fluticasone propionate (JAN/USP); Cutivate (TN); Flonase (TN); Flovent (TN) (P) CYP induction: CYP3A4
D01712  Theophylline sodium acetate (JAN) (P) unclassified
D01740  Barbital (JP18/INN); Barbital (TN) (P) unclassified
D01741  Celiprolol hydrochloride (JAN/USAN); Selectol (TN) (P) unclassified
D01744  Brotizolam (JP18/USAN/INN); Lendormin (TN) (P) CYP induction: CYP3A4
D01745  Domperidone (JP18/USAN/INN); Motilium (TN) (P) CYP induction: CYP3A4
D01747  Idarubicin hydrochloride (JP18/USP); Idamycin (TN) (CI,P) unclassified
D01758  Haloxazolam (JP18/INN); Somelin (TN) (P) unclassified
D01760  Ranimustine (JAN/INN); Cymerin (TN) (CI,P) unclassified
D01764  Diflucortolone valerate (JP18); Afusona (TN) (P) unclassified
D01769  Vindesine sulfate (JAN/USAN); Fildesin (TN) (CI,P) unclassified
D01775  Bifonazole (JP18/USAN/INN); Mycospor (TN) (P) unclassified
D01784  Carmofur (JP18/INN); Mifurol (TN) (CI,P) unclassified
D01785  Pirmenol hydrochloride hydrate (JAN); Pimenol (TN) (P) unclassified
D01787  Sulthiame (USAN); Sultiame (JP18); Ospolot (TN) (P) unclassified
D01790  Oxaliplatin (JAN/USP/INN); Eloxatin (TN) (CI,P) unclassified
D01794  Bopindolol malonate (JAN); Sandonorm (TN) (P) unclassified
D01795  Tilisolol hydrochloride (JAN); Selecal (TN) (P) unclassified
D01799  Glyclopyramide (JAN/INN); Deamelin-S (TN) (P) unclassified
D01804  Cadralazine (JP18/INN); Cadral (TN) (P) unclassified
D01806  Oxprenolol hydrochloride (JP18/USP); Okuspurecol (TN) (P) unclassified
D01807  Mebutamate (JAN/USAN); Capla (TN); Dormate (TN) (P) unclassified
D01820  Alclometasone dipropionate (JAN/USP); Aclovate (TN) (P) unclassified
D01825  Fluocinolone acetonide (JP18/USP/INN); Fluocet (TN); Retisert (TN); Synalar (TN) (P) unclassified
D01830  Arotinolol hydrochloride (JP18); Almarl (TN) (P) unclassified
D01832  Modafinil (JAN/USP/INN); Provigil (TN) (P) CYP induction: CYP3A4
D01847  Landiolol hydrochloride (JAN/USAN); ONO 1101 hydrochloride; Onoact (TN) (P) unclassified
D01849  Lercanidipine hydrochloride (JAN/USAN); Cardiovasc (TN) (P) unclassified
D01854  Mitiglinide calcium hydrate (JP18); Mitiglinide calcium dihydrate; Glufast (TN) (P) Enzyme induction: UGT
D01855  Mozavaptane hydrochloride (JAN) (P) CYP induction: CYP3A4
D01856  Nifekalant hydrochloride (JAN); MS 551; Shinbit (TN) (P) unclassified
D01862  Pitavastatin calcium (JAN); NK 104; Livalo (TN) (P) unclassified
D01872  Doxapram hydrochloride (USP); Doxapram hydrochloride hydrate (JP18); Dopram (TN) (P) CYP induction: CYP3A4
D01885  Pirarubicin (JP18/INN); Therarubicin (TN) (CI,P) unclassified
D01886  Hydrocortisone probutate (USAN); Hydrocortisone butyrate propionate (JAN); Hydrocortisone buteprate; Pandel (TN) (P) unclassified
D01887  Bunazosin hydrochloride (JP18); Detantol (TN) (P) unclassified
D01896  Cilostazol (JP18/USP/INN); Pletal (TN) (P) CYP induction: CYP3A4
D01898  Haloperidol decanoate (JAN/USP); Halomonth (TN) (P) CYP induction: CYP3A4
D01903  Docarpamine (JAN/INN); Tanadopa (TN) (P) unclassified
D01907  Fludarabine phosphate (JAN/USP); Fludara (TN) (CI,P) unclassified
D01908  Nilvadipine (JP18/USAN/INN); Nivadil (TN) (P) CYP induction: CYP3A4
D01911  Aclarubicin hydrochloride (JP18); Aclacinon (TN) (CI,P) unclassified
D01933  Vatanidipine hydrochloride (JAN); AE 0047; Calbren (TN) (P) unclassified
D01935  Vinorelbine tartrate (USP); Vinorelbine ditartrate (JAN); KW 2307; Navelbine (TN) (CI,P) CYP induction: CYP3A4
D01948  Dexamethasone valerate (JAN); Dexamethasone 17-valerate; DV-17; Voalla ointment (TN) (P) CYP induction: CYP3A4
D01953  Estradiol benzoate (JP18/USP); Ovahormon (TN) (P) CYP induction: CYP3A4
D01958  Indenolol hydrochloride (JP18) (P) unclassified
D01965  Silodosin (JP18/INN); KMD 3213; Rapaflo (TN); Urief (TN) (P) CYP induction: CYP3A4 / Enzyme induction: UGT
D01969  Gallopamil hydrochloride (JAN) (P) unclassified
D01972  Lanatoside C (JAN/INN); Digilanogen C (TN) (P) unclassified
D01973  Eletriptan hydrobromide (JAN/USAN); Relpax (TN) (P) CYP induction: CYP3A4
D01977  Gefitinib (JP18/USAN/INN); Iressa (TN) (CI,P) unclassified
D01980  Luliconazole (JAN/USAN/INN); Lulicon (TN); Luzu (TN) (P) unclassified
D01982  Tenofovir disoproxil fumarate (JAN/USAN); Viread (TN) (CI,P) unclassified
D01984  Esomeprazole magnesium (USP); Esomeprazole magnesium hydrate (JAN); Esomeprazole magnesium trihydrate; Nexium (TN) (P) unclassified
D01994  Mosapride citrate hydrate (JP18); Mosapride citrate dihydrate; Gasmotin (TN) (P) CYP induction: CYP3A4
D01998  Prednisolone farnesylate (JAN); PNF 21; Farnerate (TN) (P) unclassified
D02002  Isoniazid sodium methanesulfonate hydrate (JAN); Isoniazid sodium methanesulfonate monohydrate; Isoniazid sodium methanesulfonate; IHMS; Neoiscotin (TN) (P) unclassified
D02004  Apomorphine hydrochloride (USP); Apomorphine hydrochloride hydrate (JAN); Apokyn (TN); Ixense (TN); Uprima (TN) (P) unclassified
D02008  Tadalafil (JAN/USP/INN); Adcirca (TN); Cialis (TN); Zalutia (TN) (CI,P) CYP induction: CYP3A4
D02016  Ramosetron hydrochloride (JAN); YM 060; Nasea (TN); Irribow (TN) (P) unclassified
D02020  Mitobronitol (JAN/INN) (CI,P) unclassified
D02032  Betamethasone butyrate propionate (JAN); Antebate (TN) (P) unclassified
D02041  Tropisetron hydrochloride (JAN); Navoban (TN) (P) unclassified
D02042  Olprinone hydrochloride hydrate (JAN); Coretec (TN) (P) unclassified
D02045  Benidipine hydrochloride (JP18); KW 3049; Coniel (TN) (P) CYP induction: CYP3A4
D02066  Isoproterenol sulfate (USP); Isoprenaline sulfate (JAN); Luf-Iso (TN); Medihaler-Iso (TN) (P) unclassified
D02071  Scopolamine hydrobromide (USP); Scopolamine hydrobromide hydrate (JP18); Scopolamine hydrobromide trihydrate; Hysco (TN); Isopto hyoscine (TN) (P) unclassified
D02081  Metipranolol hydrochloride; Optipranolol (TN) (P) unclassified
D02084  Inamrinone ethylenelactate; Amrinone ethylenelactate; Inocor (TN) (P) unclassified
D02085  Milrinone lactate; Primacor (TN) (P) Enzyme induction: UGT
D02086  Lidocaine hydrochloride (JAN/USP); Dalcaine (TN); Xylocaine (TN) (P) CYP induction: CYP3A4
D02087  Moricizine hydrochloride (USP); Ethmozine (TN) (P) unclassified
D02088  Tocainide hydrochloride (USP); Tonocard (TN) (P) unclassified
D02096  Fosphenytoin sodium (USP); Cerebyx (TN); Sesquient (TN) (P) unclassified
D02097  Tiagabine hydrochloride (USP); Gabitril (TN) (P) unclassified
D02101  Codeine phosphate (USP); Codeine phosphate hydrate (JP18); Codeine (TN) (P) unclassified
D02102  Methadone hydrochloride (JAN/USP); Dolophine hydrochloride (TN) (P) CYP induction: CYP3A4 / Transporter induction: ABCB1
D02103  Phenytoin sodium (USP); Phenytoin sodium for injection (JP18); Aleviatin (TN); Dilantin (TN) (P) unclassified
D02106  Arsenic trioxide (JP18/USAN); Trisenox (TN) (CI,P) unclassified
D02114  Hydroxychloroquine sulfate (JAN/USP); Plaquenil (TN) (P) CYP induction: CYP3A4
D02115  Methotrexate sodium; Trexall (TN); Rasuvo (TN) (CI,P) unclassified
D02129  Doxycycline hyclate (USP); Doxycycline hydrochloride hydrate (JP18); Doryx (TN); Lymepak (TN); Periostat (TN); Vibra-tabs (TN) (P) unclassified
D02130  Tropisetron (INN); Navoban (TN) (P) unclassified
D02131  Tegafur and uracil; Uftoral (TN) (CI,P) unclassified
D02135  Levodopa and benserazide hydrochloride; Madopar (TN) (P) unclassified
D02149  Epinephrine bitartrate (JAN/USP); Asmatane mist (TN); Medihaler-epi (TN) (P) unclassified
D02150  l-Isoprenaline hydrochloride (JP18); Proternol-L (TN) (P) unclassified
D02156  Prednisolone hemisuccinate (USP); Prednisolone succinate (JP18) (P) unclassified
D02165  Docetaxel (USP); Docetaxel hydrate (JP18); Docetaxel trihydrate; Taxotere (TN) (CI,P) CYP induction: CYP3A4
D02166  Mitoxantrone hydrochloride (JAN/USP); Novantron (TN) (CI,P) unclassified
D02168  Topotecan hydrochloride (USAN); Nogitecan hydrochloride (JAN); Hycamtin (TN); Potactasol (TN) (CI,P) Transporter induction: ABCB1
D02169  Croconazole hydrochloride (JP18); Pilzcin (TN) (P) unclassified
D02173  Galantamine hydrobromide (JAN/USP); Razadyne (TN); Reminyl (TN) (P) CYP induction: CYP3A4
D02174  Dexamethasone acetate (JAN/USP); Decadronal (TN) (P) CYP induction: CYP3A4
D02175  Compound oxycodone (JP18); Pavinal (TN) (P) CYP induction: CYP3A4
D02177  Bleomycin sulfate (JP18/USP); Blenoxane (TN) (CI,P) unclassified
D02185  Chloramphenicol sodium succinate (JP18/USP); Chloromycetin succinate (TN) (P) unclassified
D02197  Vincristine sulfate (JP18/USP); VCR; Marqibo (TN); Oncovin (TN); Vincasar (TN); Vincrex (TN) (CI,P) unclassified
D02205  Ethylmorphine hydrochloride hydrate (JP18); Ethylmorphine hydrochloride dihydrate; Ethylmorphine hydrochloride (TN) (P) CYP induction: CYP3A4
D02206  Buformin hydrochloride (JP18); Dibetos-B (TN) (P) unclassified
D02211  Dihydroergotamine mesylate (USP); Dihydroergotamine mesilate (JP18); Migranal (TN); Trudhesa (TN) (P) CYP induction: CYP3A4
D02213  Metoclopramide hydrochloride (JAN); Metoclopramide dihydrochloride monohydrate; Primperan (TN); Reglan (TN) (P) unclassified
D02214  Epirubicin hydrochloride (JP18/USP); EPI; Ellence (TN) (CI,P) unclassified
D02219  Terbinafine hydrochloride (JP18/USP); Lamisil (TN) (P) CYP induction: CYP3A4
D02229  Sildenafil citrate (JAN/USP); Revatio (TN); Viagra (TN) (P) CYP induction: CYP3A4
D02237  Guanethidine sulfate (USAN) (P) unclassified
D02239  Sparteine sulfate (JAN/USAN); Sparteine sulfate pentahydrate (P) unclassified
D02246  Biperiden hydrochloride (JP18/USP); Tasmolin (TN) (P) unclassified
D02247  Biperiden lactate (JAN/USP); Tasmolin (TN) (P) unclassified
D02252  Amobarbital sodium (JAN/USP); Amytal sodium (TN) (P) unclassified
D02253  Pentobarbital calcium (JP18); Ravona (TN) (P) unclassified
D02258  Atorvastatin calcium (USP); Atorvastatin calcium hydrate (JP18); Atorvastatin calcium trihydrate; Atorvaliq (TN); Lipitor (TN) (P) CYP induction: CYP3A4 / Transporter inhibition: SLCO1B1 SLCO1B3 / Transporter induction: ABCB1
D02260  Paroxetine hydrochloride hemihydrate (USP); Paroxetine hydrochloride hydrate (JP18); Paxil (TN) (P) unclassified
D02261  Quinine hydrochloride hydrate (JP18); Quinine hydrochloride dihydrate; Quinine hydrochloride (TN) (P) CYP induction: CYP3A4 / Transporter induction: ABCB1
D02262  Quinine sulfate (USP); Quinine sulfate hydrate (JP18); Quinine hydrogen sulfate; Coco-quinine (TN) (P) CYP induction: CYP3A4 / Transporter induction: ABCB1
D02268  Ergoloid mesylates (USP); Dihydroergotoxine mesilate (JP18); Circanol (TN); Hydergine (TN); Inorter (TN) (P) CYP induction: CYP3A4
D02272  Quinidine sulfate (USP); Quinidine sulfate hydrate (JP18); Quinidex (TN) (P) unclassified
D02286  Betamethasone benzoate (USP); Uticort (TN) (P) unclassified
D02287  Clocortolone pivalate (USP); Cloderm (TN) (P) unclassified
D02288  Hydrocortisone valerate (USP); Westcort (TN) (P) unclassified
D02289  Medrysone (USAN); HMS (TN) (P) unclassified
D02297  Emtricitabine and tenofovir disoproxil; Truvada (TN) (CI,P) unclassified
D02321  Amsacrine (USAN/INN); Amsidyl (TN) (CI,P) unclassified
D02323  Tolrestat (USAN/INN); Alredase (TN) (P) unclassified
D02338  Acebutolol (USAN/INN) (P) unclassified
D02340  Loxapine (USAN/INN); Adasuve (TN) (P) CYP induction: CYP3A4
D02342  Bisoprolol (JAN/USAN/INN) (P) unclassified
D02356  Verapamil (USAN/INN) (P) CYP induction: CYP3A4 / Transporter induction: ABCB1
D02358  Metoprolol (USAN/INN) (P) unclassified
D02360  Sertraline (INN) (P) CYP induction: CYP3A4
D02361  Propiomazine (USAN/INN) (P) unclassified
D02363  Ketanserin (USAN/INN) (P) unclassified
D02368  Gemcitabine (USAN/INN) (CI,P) unclassified
D02374  Metipranolol (USAN/INN) (P) unclassified
D02375  Terbinafine (USAN/INN); Lamasil (TN) (P) CYP induction: CYP3A4
D02389  Primidolol (USAN/INN) (P) unclassified
D02398  Estramustine phosphate sodium (USAN); Emcyt (TN) (CI,P) unclassified
D02404  Procaterol hydrochloride (USAN); Pro-Air (TN) (P) CYP induction: CYP3A4
D02425  Carbutamide (INN); Invenol (TN) (P) unclassified
D02427  Glibornuride (USAN/INN); Glutril (TN) (P) unclassified
D02430  Gliquidone (INN); Glurenorm (TN) (P) unclassified
D02472  Atovaquone and proguanil hydrochloride; Malarone (TN) (P) unclassified
D02484  Artemether and lumefantrine; Coartem (TN) (CI) unclassified
D02497  Fosamprenavir (INN) (CI,P) CYP induction: CYP3A4
D02498  Lopinavir and ritonavir; Kaletra (TN) (CI,P) unclassified
D02499  Enfuvirtide (USAN/INN); Fuzeon (TN) (CI,P) unclassified
D02501  Caspofungin acetate (JAN/USAN); Cancidas (TN) (P) unclassified
D02537  Dronedarone (INN) (P) unclassified
D02549  Rifamycin (USAN/INN); Rifamycin SV (P) unclassified
D02550  Rifalazil (USAN/INN); RLZ (P) unclassified
D02551  Rifametane (USAN/INN) (P) unclassified
D02552  Rifamexil (USAN/INN) (P) unclassified
D02553  Rifamide (USAN) (P) unclassified
D02554  Rifaximin (JAN/USAN/INN); Xifaxan (TN) (P) CYP induction: CYP3A4 / Transporter inhibition: SLCO1B1 SLCO1B3 / Transporter induction: ABCB1
D02555  Posaconazole (JAN/USAN/INN); Noxafil (TN) (P) Transporter induction: ABCB1
D02556  Ravuconazole (prop.INN) (P) unclassified
D02557  Chlormidazole (INN) (P) unclassified
D02562  Rasagiline mesylate (USAN); Rasagiline mesilate (JAN); Azilect (TN) (P) unclassified
D02564  Pargyline hydrochloride (USAN); Eutonyl (TN) (P) unclassified
D02567  Escitalopram oxalate (JAN/USP); Lexapro (TN) (P) CYP induction: CYP3A4
D02570  Desvenlafaxine succinate (USAN); Desvenlafaxine succinate hydrate (JAN); Desvenlafaxine succinate monohydrate; Pristiq (TN) (P) CYP induction: CYP3A4 / Enzyme induction: UGT
D02577  Flibanserin (USAN/INN); Addyi (TN) (P) CYP induction: CYP3A4
D02582  Fenticonazole (INN) (P) unclassified
D02583  Fenticonazole nitrate (USAN); Lomexin (TN) (P) unclassified
D02584  Aliconazole (INN) (P) unclassified
D02585  Vibunazole; Bay N-7133 (P) unclassified
D02586  Alteconazole (INN) (P) unclassified
D02587  Metildigoxin (JP18); Lanirapid (TN) (P) Transporter induction: ABCB1
D02591  Dexamethasone acefurate (USAN/INN) (P) CYP induction: CYP3A4
D02592  Dexamethasone beloxil (USAN) (P) CYP induction: CYP3A4
D02593  Pantoprazole sodium (USP); Pantoprazole sodium hydrate (JAN); Protonix (TN) (P) unclassified
D02600  Demoxepam (USAN/INN) (P) unclassified
D02614  Denopamine (JAN/INN); Kalgut (TN) (P) unclassified
D02615  Chlorpromazine hydrochloride, promethazine hydrochloride and phenobarbital; Vegetamin (TN) (P) unclassified
D02618  Butobarbital (BAN); Butethal; Neonal (TN) (P) unclassified
D02619  Carbromal (INN); Adalin (TN) (P) unclassified
D02624  Eszopiclone (JAN/USP/INN); Estorra (TN); Lunesta (TN) (P) CYP induction: CYP3A4
D02626  Bromperidol decanoate (USAN) (P) CYP induction: CYP3A4
D02629  Fluspirilene (USAN/INN); Imap (TN) (P) unclassified
D02630  Penfluridol (USAN/INN); Semap (TN) (P) unclassified
D02632  Indisetron hydrochloride (JAN); Sinseron (TN) (P) unclassified
D02633  Lomerizine hydrochloride (JAN); Terranas (TN) (P) unclassified
D02666  Iloperidone (USAN/INN); Fanapt (TN) (P) CYP induction: CYP3A4
D02689  Ramelteon (JAN/USAN/INN); Rozerem (TN) (P) unclassified
D02697  Valrubicin (USP/INN); Valstar (TN) (CI,P) unclassified
D02698  Teniposide (USP/INN); Vumon (TN) (CI,P) unclassified
D02714  Everolimus (JAN/USAN/INN); Afinitor (TN); Votubia (TN); Zortress (TN) (CI,P) CYP induction: CYP3A4 / Transporter induction: ABCB1
D02717  Valnoctamide (USAN/INN); Axiquel (TN) (P) unclassified
D02731  Vardenafil dihydrochoride (USAN); Levitra (TN) (P) CYP induction: CYP3A4
D02732  Pranlukast hydrate (JP18); Onon (TN) (P) CYP induction: CYP3A4
D02734  Abacavir succinate (USAN) (CI,P) unclassified
D02740  Lidocaine and prilocaine; Lidocaine and propitocaine; Emla (TN); Oraqix (TN); Lidocaine and prilocaine (TN) (P) CYP induction: CYP3A4
D02746  Acecainide hydrochloride (USAN) (P) unclassified
D02756  Aclarubicin (USAN/INN); Aclacinomycin A; ACM (CI,P) unclassified
D02763  Actodigin (USAN/INN) (P) unclassified
D02765  Adaprolol maleate (USAN) (P) unclassified
D02766  Valpromide (INN); Depamide (TN) (P) unclassified
D02770  Adinazolam (USAN/INN) (P) unclassified
D02771  Adinazolam mesylate (USAN) (P) unclassified
D02815  Alitretinoin (USAN); Panretin (TN) (CI,P) unclassified
D02817  Allobarbital (USAN/INN) (P) unclassified
D02824  Almotriptan (USAN) (P) CYP induction: CYP3A4
D02825  Almotriptan malate (USP); Axert (TN) (P) CYP induction: CYP3A4
D02829  Alosetron hydrochloride (USAN); Lotrpnex (TN) (P) unclassified
D02834  Alprenoxime hydrochloride (USAN) (P) unclassified
D02841  Altretamine (USP/INN); Hexalen (TN) (CI,P) unclassified
D02861  Indinavir sulfate ethanolate (JAN); Crixivan (TN) (CI,P) CYP induction: CYP3A4
D02867  Fosamprenavir calcium hydrate (JAN); Lexiva (TN) (CI,P) CYP induction: CYP3A4
D02890  Amdoxovir (USAN/INN) (CI,P) unclassified
D02901  Amidephrine mesylate (USAN); Amidefrine mesilate (INN) (P) unclassified
D02908  Aminolevulinic acid hydrochloride (JAN/USAN); 5-Aminolevulinic acid hydrochloride; Levulan (TN); Ameluz (TN); Gleolan (TN) (CI,P) unclassified
D02910  Amiodarone (USAN/INN) (P) CYP induction: CYP3A4
D02914  Amlodipine maleate (USAN); Amvaz (TN) (P) CYP induction: CYP3A4
D02933  Anagrelide hydrochloride (USP); Agrylin (TN); Xagrid (TN) (CI,P) unclassified
D02964  Apaxifylline (USAN/INN) (P) unclassified
D02968  Aprepitant (JAN/USP/INN); Aponvie (TN); Emend (TN); Cinvanti (TN) (P) CYP induction: CYP3A4
D02969  Aprindine (USAN/INN) (P) unclassified
D02976  Arbutamine hydrochloride (USAN); Genesa (TN) (P) unclassified
D02994  Rituximab (USAN/INN); Rituximab (genetical recombination) (JAN); Rituximab (genetical recombination) [Rituximab biosimilar 1] (JAN); Rituximab (genetical recombination) [Rituximab biosimilar 2] (JAN); Rituximab-abbs; Rituximab-pvvr; Rituximab-arrx; Rituxan (TN); Riabni (TN); Truximab (TN) (CI,P) unclassified
D02997  Asparaginase (USAN); L-Asparaginase (JAN); Asparaginase Erwinia chrysanthemi (USAN); Asparaginase erwinia chrysanthemi (recombinant)-rywn; Elspar (TN); Erwinaze (TN); Rylaze (TN) (CI,P) unclassified
D03001  Atevirdine mesylate (USAN) (CI,P) unclassified
D03021  Azacitidine (JAN/USAN/INN); Vidaza (TN) (CI,P) unclassified
D03023  Azaconazole (USAN/INN) (P) unclassified
D03037  Azimilide dihydrochloride (USAN) (P) unclassified
D03046  Cytarabine ocfosfate hydrate (JAN); Cytarabine ocfosphate hydrate; Fosteabine sodium monohydrate; Starasid (TN) (CI,P) unclassified
D03060  Batanopride hydrochloride (USAN) (P) unclassified
D03067  Belfosdil (USAN/INN) (P) unclassified
D03072  Bemarinone hydrochloride (USAN) (P) unclassified
D03075  Bemoradan (USAN/INN) (P) unclassified
D03083  Bentazepam (USAN/INN) (P) unclassified
D03089  Benzoctamine hydrochloride (USAN) (P) unclassified
D03106  Bexarotene (JAN/USAN/INN); Targretin (TN) (CI,P) unclassified
D03150  Bortezomib (JAN/USAN/INN); Velcade (TN) (CI,P) unclassified
D03164  Bromindione (USAN/INN) (P) unclassified
D03165  Bromocriptine (USAN/INN) (P) CYP induction: CYP3A4
D03170  Bucindolol hydrochloride (USAN) (P) unclassified
D03177  Bunolol hydrochloride (USAN) (P) unclassified
D03195  Butopamine (USAN/INN) (P) unclassified
D03198  Butoxamine hydrochloride (USAN) (P) unclassified
D03208  Aliskiren (USAN/INN); Rasilez (TN) (P) CYP induction: CYP3A4 / Transporter induction: ABCB1
D03213  Apixaban (JAN/USAN/INN); Eliquis (TN) (P) CYP induction: CYP3A4 / Transporter induction: ABCB1
D03215  Armodafinil (USAN/INN); Nuvigil (TN) (P) CYP induction: CYP3A4
D03217  Avanafil (USAN/INN); Stendra (TN); Spedra (TN) (P) CYP induction: CYP3A4
D03218  Axitinib (JAN/USAN); Inlyta (TN) (CI,P) CYP induction: CYP3A4
D03225  Belotecan hydrochloride (USAN) (CI,P) unclassified
D03229  Bleomycin hydrochloride (JP18); BLM; Bleo (TN) (CI,P) unclassified
D03230  Insulin human (USP/INN); Insulin human (genetical recombination) (JP18); Insulin human (biosynthesis) (JAN); Insulin human (synthesis) (JAN); Humulin (TN) (P) unclassified
D03250  Insulin glargine (USAN/INN); Insulin glargine (genetical recombination) (JP18); Insulin glargine (genetical recombination) [Insulin glargin biosimilar 1] (JAN); Insulin glargine (genetical recombination) [Insulin glargin biosimilar 2] (JAN); Lantus (TN) (P) unclassified
D03252  Bosutinib (USAN) (CI,P) CYP induction: CYP3A4
D03253  Brecanavir (USAN) (CI,P) unclassified
D03257  Trastuzumab (USAN/INN); Trastuzumab (genetical recombination) (JAN); Trastuzumab (genetical recombination) [Trastuzumab biosimilar 1] (JAN); Trastuzumab (genetical recombination) [Trastuzumab biosimilar 2] (JAN); Trastuzumab (genetical recombination) [Trastuzumab biosimilar 3] (JAN); Trastuzumab-pkrb; Trastuzumab-anns; Trastuzumab-dkst; Trastuzumab-dttb; Trastuzumab-qyyp; Trastuzumab-anns; Herceptin (TN); Herzuma (TN); Kanjinti (TN); Ogivri (TN); Ontruzant (TN) (CI,P) unclassified
D03259  Gemtuzumab ozogamicin (USAN); Gemtuzumab ozogamicin (genetical recombination) (JAN); Gemtuzumab (INN); Mylotarg (TN) (CI,P) CYP induction: CYP3A4
D03260  Vardenafil hydrochloride hydrate (JAN); Vardenafil monohydrochloride trihydrate; Levitra (TN); Staxyn (TN) (P) CYP induction: CYP3A4
D03262  Kanamycin sulfate (JP18); Kanamycin sulfate (TN) (P) unclassified
D03264  Mazaticol hydrochloride hydrate (JAN); Mazaticol hydrochloride; Pentona (TN) (P) unclassified
D03278  Enviomycin sulfate (JP18); Tuberactin (TN) (P) unclassified
D03301  Prednisolone valerate acetate (JAN); PDL; Spirazon (TN) (P) unclassified
D03325  Mometasone furoate hydrate (JAN); Mometasone furoate monohydrate; Nasonex (TN) (P) CYP induction: CYP3A4
D03327  Porfimer sodium (JAN/USAN/INN); Photofrin II; Photofrin (TN) (CI,P) unclassified
D03368  Calcium para-aminosalicylate (JP18); Nippas calcium (TN) (P) unclassified
D03371  Capravirine (USAN/INN) (CI,P) unclassified
D03415  Carvedilol phosphate (USAN); Carvedilol phosphate hydrate (JAN); Coreg CR (TN) (P) CYP induction: CYP3A4
D03449  Cetamolol hydrochloride (USAN) (P) unclassified
D03455  Cetuximab (USAN/INN); Cetuximab (genetical recombination) (JAN); Erbitux (TN) (CI,P) unclassified
D03461  Chloramphenicol pantothenate complex (USAN/INN); Pantofenicol (TN) (P) unclassified
D03485  Ciclafrine hydrochloride (USAN) (P) unclassified
D03490  Cicloprolol hydrochloride (USAN) (P) unclassified
D03492  Cifenline (USAN); Cibenzoline (INN) (P) CYP induction: CYP3A4
D03495  Cilansetron (USAN/INN) (P) unclassified
D03496  Cilansetron hydrochloride (USAN) (P) unclassified
D03504  Cinacalcet (USAN) (P) CYP induction: CYP3A4
D03505  Cinacalcet hydrochloride (JAN/USAN); Sensipar (TN); Mimpara (TN) (P) CYP induction: CYP3A4
D03526  Cisconazole (USAN/INN) (P) unclassified
D03536  Clentiazem maleate (JAN/USAN) (P) unclassified
D03541  Clocortolone acetate (USAN) (P) unclassified
D03546  Clofarabine (JAN/USAN/INN); Clolar (TN) (CI,P) unclassified
D03561  Cloprednol (USAN/INN); Cloradryn (TN) (P) unclassified
D03562  Clorazepate monopotassium (USAN) (P) unclassified
D03579  Codeine polistirex (USAN) (P) unclassified
D03580  Codeine sulfate (USP); Codeine sulfate trihydrate; Codeine sulfate (TN) (P) unclassified
D03594  Cortivazol (USAN) (P) unclassified
D03631  Cyprazepam (USAN/INN) (P) unclassified
D03637  Cytarabine hydrochloride (USAN) (CI,P) unclassified
D03654  Darifenacin (USAN/INN) (P) CYP induction: CYP3A4
D03655  Darodipine (USAN/INN) (P) unclassified
D03656  Darunavir (USAN/INN) (CI,P) CYP induction: CYP3A4
D03657  Dasantafil (USAN/INN) (P) unclassified
D03658  Dasatinib (JAN/INN) (CI,P) CYP induction: CYP3A4 / Enzyme induction: UGT
D03662  Dazopride fumarate (USAN) (P) unclassified
D03664  Debrisoquin sulfate (USAN); Declinax (TN) (P) unclassified
D03665  Decitabine (USAN/INN); Dacogen (TN) (CI,P) unclassified
D03669  Deferasirox (JAN/USAN/INN); Exjade (TN); Jadenu (TN) (P) unclassified
D03671  Deflazacort (USAN/INN); Emflaza (TN) (P) CYP induction: CYP3A4 / Transporter induction: ABCB1
D03682  Denileukin diftitox (USAN/INN); Denileukin difitox (genetical recombination) (JAN); Ontak (TN); Remitoro (TN) (CI,P) unclassified
D03696  Desonide (USP/INN); Desowen (TN); Verdeso (TN) (P) unclassified
D03697  Desoximetasone (USP/INN); Topicort (TN) (P) unclassified
D03725  Hydrocodone bitartrate (USP); Hydrocodone bitartrate hemipentahydrate; Dicodid (TN) (P) CYP induction: CYP3A4
D03729  Dexpropranolol hydrochloride (USAN) (P) unclassified
D03731  Selegiline (USAN/INN); Emsam (TN) (P) CYP induction: CYP3A4
D03732  Dexsotalol hydrochloride (USAN) (P) unclassified
D03737  Dextofisopam (USAN/INN) (P) unclassified
D03759  Diacetolol hydrochloride (USAN) (P) unclassified
D03783  Oxycodone terephthalate (USP) (P) CYP induction: CYP3A4
D03785  Dichloralphenazone (USP) (P) unclassified
D03798  Dicumarol (USAN); Dicoumarol (INN); Dicumarol (TN) (P) unclassified
D03799  Dienogest (JAN/USAN/INN); Endometrion (TN) (P) CYP induction: CYP3A4
D03812  Diflucortolone (USAN) (P) unclassified
D03813  Diflucortolone pivalate (USAN) (P) unclassified
D03819  Digitalis (USP); Digiglusin (TN) (P) unclassified
D03820  Dutasteride (JAN/USP/INN); Avodart (TN) (P) CYP induction: CYP3A4
D03825  Dihydrocodeine bitartrate (USP) (P) unclassified
D03828  Pemetrexed disodium (USAN); Alimta (TN) (CI,P) unclassified
D03830  Diltiazem malate (USAN); Tiamate (TN) (P) CYP induction: CYP3A4
D03833  Indinavir (USAN); Indinavir hydrate (CI,P) CYP induction: CYP3A4
D03835  Fosamprenavir calcium (USAN); Lexiva (TN); Telzir (TN) (CI,P) CYP induction: CYP3A4
D03837  Fosamprenavir sodium (USAN) (CI,P) CYP induction: CYP3A4
D03839  Droxinavir hydrochloride (USAN) (CI,P) unclassified
D03840  Palinavir (USAN/INN) (CI,P) unclassified
D03842  Telinavir (USAN/INN) (CI,P) unclassified
D03843  Tipranavir disodium (USAN) (CI,P) unclassified
D03844  Phenytoin, phenobarbital and caffeine and sodium benzoate; Hydantol F (TN) (P) unclassified
D03852  Droperidol and fentanyl citrate; Innovar (TN) (P) CYP induction: CYP3A4
D03879  Dobutamine (USAN/INN) (P) unclassified
D03880  Dobutamine lactobionate (USAN) (P) unclassified
D03881  Dobutamine tartrate (USAN) (P) unclassified
D03883  Doconazole (USAN/INN) (P) unclassified
D03891  Dopexamine (USAN/INN) (P) unclassified
D03892  Dopexamine hydrochloride (USAN); Dopacard (TN) (P) unclassified
D03899  Doxorubicin (USAN/INN); ADR; Adriblastina (TN) (CI,P) unclassified
D03914  Dronedarone hydrochloride (USP); Multaq (TN) (P) unclassified
D03917  Drospirenone (JAN/USP/INN); Slynd (TN) (P) CYP induction: CYP3A4
D03936  Econazole (USAN/INN) (P) unclassified
D03958  Edrecolomab (USAN/INN); Panorex (TN) (CI,P) unclassified
D03961  Efaproxiral (USAN/INN) (CI,P) unclassified
D03962  Efaproxiral sodium (USAN) (CI,P) unclassified
D03975  Allylisopropylacetylurea; Apronal; Apronalide (P) unclassified
D03981  Elvucitabine (USAN/INN) (CI,P) unclassified
D03991  Encainide hydrochloride (USAN) (P) unclassified
D03994  Endralazine mesylate (USAN); Endralazine monomethanesulfonate; Migranal (TN) (P) unclassified
D03997  Enilconazole (USAN/INN) (P) unclassified
D04004  Enoximone (USAN/INN); Perfan (TN) (P) unclassified
D04018  Ephedrine sulfate (USP); Akovaz (TN); Corphedra (TN); Emerphed (TN) (P) unclassified
D04023  Erlotinib hydrochloride (JAN/USAN); Tarceva (TN) (CI,P) CYP induction: CYP3A4
D04024  Lapatinib ditosylate (USAN); Lapatinib tosilate hydrate (JAN); Lapatinib ditosylate monohydrate; Tykerb (TN); Tyverb (TN) (CI,P) CYP induction: CYP3A4 / Transporter induction: ABCB1
D04048  Ropivacaine hydrochloride (USP); Ropivacaine hydrochloride hydrate (JAN); Anapeine (TN) (P) CYP induction: CYP3A4
D04052  Epinephrine and lidocaine hydrochloride; Adrenaline and lidocaine hydrochloride; Xylocaine (TN) (P) CYP induction: CYP3A4
D04056  Esomeprazole sodium (USAN); Nexium IV (TN) (P) unclassified
D04061  Estradiol acetate (USAN); Femring (TN) (P) CYP induction: CYP3A4
D04063  Estradiol cypionate (USP); Depo-estradiol (TN) (P) CYP induction: CYP3A4
D04064  Estradiol enanthate (USAN) (P) CYP induction: CYP3A4
D04065  Estradiol undecylate (USAN/INN); Delestrec (TN) (P) CYP induction: CYP3A4
D04066  Estramustine (USAN/INN) (CI,P) unclassified
D04070  Estrogens, conjugated (JAN/USP); Conjugated estrogens; Premarin (TN) (P) CYP induction: CYP3A4
D04107  Etoposide phosphate (USAN); Etopophos (TN) (CI,P) unclassified
D04112  Etravirine (JAN/USAN/INN); Intelence (TN) (CI,P) CYP induction: CYP3A4
D04121  Exenatide (JAN/USAN/INN); Byetta (TN) (P) unclassified
D04148  Fenfluramine hydrochloride (JAN/USAN); Fintepla (TN); Pondimin (TN) (P) CYP induction: CYP3A4
D04190  Flestolol sulfate (USAN) (P) unclassified
D04193  Flordipine (USAN/INN) (P) unclassified
D04197  Floxuridine (USP/INN); FUDR (TN) (CI,P) unclassified
D04201  Flucloronide (USAN); Fluclorolone acetonide (INN) (P) unclassified
D04208  Flumethasone (USAN); Flumetasone (INN) (P) unclassified
D04214  Flunisolide acetate (USAN) (P) CYP induction: CYP3A4
D04217  Fluocortin butyl (USAN) (P) unclassified
D04218  Fluocortolone (USAN/INN) (P) unclassified
D04219  Fluocortolone caproate (USAN) (P) unclassified
D04221  Fluorometholone acetate (USP); Fluorometholone 17-acetate; Flarex (TN) (P) unclassified
D04225  Fluperolone acetate (USAN); Methral (TN) (P) unclassified
D04244  Formocortal (USAN/INN); Deflamene (TN) (P) unclassified
D04248  Fosazepam (USAN/INN) (P) unclassified
D04260  Fostedil (USAN/INN) (P) unclassified
D04265  Reserpine, hydralazine hydrochloride and hydrochlorothiazide (P) unclassified
D04266  Benzylhydrochlorothiazide, Reserpine and Carbazochrome; Behyd RA (TN) (P) unclassified
D04292  Galantamine (USAN/INN); Reminyl (TN) (P) CYP induction: CYP3A4
D04300  Ganaxolone (USAN/INN); Ztalmy (TN) (P) CYP induction: CYP3A4
D04313  Dihydrocodeine phosphate, dl-methylephedrine hydrochloride and Chlorpheniramine maleate; Huscode (TN) (P) unclassified
D04314  Gepirone hydrochloride (USAN); Exxua (TN) (P) CYP induction: CYP3A4
D04338  Dihydrocodeine phosphate, ephedrine hydrochloride and ammmonium chloride; Sekicode (TN) (P) unclassified
D04340  Dextromethorphan hydrobromide and potassium cresolsulfonate; Medicon (TN) (P) CYP induction: CYP3A4
D04370  Granisetron (JAN/USAN/INN); Sancuso (TN) (P) CYP induction: CYP3A4
D04382  Guanethidine monosulfate (USP); Guanethidine sulfate (JP18); Ismelin (TN) (P) unclassified
D04386  Guanoclor sulfate (USAN); Vatensol (TN) (P) unclassified
D04398  Guanoxabenz (USAN/INN) (P) unclassified
D04399  Guanoxan sulfate (USAN); Envacar (TN) (P) unclassified
D04403  Guar gum (NF) (P) unclassified
D04409  Halobetasol propionate (USP); Ulobetasol propionate; Ultravate (TN) (P) unclassified
D04446  Betamethasone acetate and betamethasone sodium phosphate; Celestone soluspan (TN); Rinderon (TN) (P) CYP induction: CYP3A4
D04447  Betamethasone and d-chlorpheniramine maleate; Celestamine (TN) (P) CYP induction: CYP3A4
D04457  Hydroxyprogesterone caproate and estradiol dipropionate; EP Hormone (TN) (P) unclassified
D04458  Hydralazine polistirex (USAN) (P) unclassified
D04459  Progesterone and estradiol; Lutes (TN) (P) unclassified
D04460  Ethinylestradiol and ethynodiol diacetate; Edulen (TN); Zovia (TN) (P) unclassified
D04461  Hydrocodone polistirex (USAN) (P) CYP induction: CYP3A4
D04462  Norethisterone and mestranol; Necon (TN) (P) unclassified
D04463  Norgestrel and ethinylestradiol tablets (JP18); Low-ogestrel (TN); Planovar (TN) (P) CYP induction: CYP3A4
D04464  Chlormadinone acetate and mestranol; Lutedion (TN) (P) unclassified
D04465  Hydroxyprogesterone caproate and estradiol benzoate; Lutes (TN) (P) unclassified
D04466  Mestranol and lynestrenol; Lo-Lyndiol (TN) (P) unclassified
D04467  Hydrocortisone hemisuccinate (USP) (P) unclassified
D04475  Insulin aspart (USP/INN); Insulin aspart (genetical recombination) (JP18); Insulin aspart (genetical recombination) [Insulin aspart biosimilar 1] (JAN); Insulin X 14; NovoRapid (TN); Novolog (TN) (P) unclassified
D04477  Insulin lispro (USP/INN); Insulin lispro (genetical recombination) (JAN); Insulin lispro (genetical recombination) [Insulin lispro Biosimilar 1] (JAN); Insulin lispro-aabc; Humalog (TN); Lyumjev (TN) (P) unclassified
D04482  Ethinylestradiol and levonorgestrel; Ange (TN); Levora (TN); Lo/ovral (TN); Seasonique (TN); Triphasil-21 (TN); Trivora (TN) (P) unclassified
D04483  Ethinylestradiol and norethisterone; Norethindrone and ethinyl estradiol; Synphase T28 (TN) (P) unclassified
D04484  Desogestrel and ethinylestradiol; Marvelon21 (TN); Ortho-cept (TN) (P) unclassified
D04488  Ibopamine (USAN/INN) (P) unclassified
D04508  Imazodan hydrochloride (USAN) (P) unclassified
D04529  Indolidan (USAN/INN) (P) unclassified
D04531  Indoramin (USAN/INN) (P) unclassified
D04532  Indoramin hydrochloride (USAN) (P) unclassified
D04539  Insulin detemir (USAN/INN); Insulin detemir (genetical recombination) (JAN); Levemir (TN) (P) unclassified
D04540  Insulin glulisine (USAN/INN); Insulin glulisine (genetical recombination) (JAN); Apidra (TN) (P) unclassified
D04548  Insulin, neutral (USAN); Neutral insulin injection (INN) (P) unclassified
D04603  Ipilimumab (USAN/INN); Ipilimumab (genetical recombination) (JAN); Yervoy (TN) (CI,P) unclassified
D04624  Isoconazole (USAN/INN) (P) unclassified
D04641  Istradefylline (JAN/USAN/INN); Nourianz (TN); Nouriast (TN) (P) CYP induction: CYP3A4
D04642  Itasetron (USAN/INN) (P) unclassified
D04645  Ixabepilone (JAN/USAN/INN); Ixempra (TN) (CI,P) CYP induction: CYP3A4
D04650  Ketazolam (USAN/INN) (P) unclassified
D04657  Lacidipine (USAN/INN); Motens (TN) (P) unclassified
D04708  Levdobutamine lactobionate (USAN) (P) unclassified
D04710  Levobetaxolol hydrochloride (USAN); Betaxon (TN) (P) unclassified
D04716  Levomethadyl acetate (USAN); Levacetylmethadol (INN) (P) CYP induction: CYP3A4
D04720  Levosimendan (USAN/INN); Simdax (TN) (P) unclassified
D04721  Levotofisopam (USAN/INN) (P) unclassified
D04733  Lidoflazine (USAN/INN); Angex (TN) (P) unclassified
D04768  Lonafarnib (JAN/USAN/INN); Zokinvy (TN) (P) unclassified
D04774  Lorajmine hydrochloride (USAN) (P) unclassified
D04778  Lorcainide hydrochloride (USAN) (P) unclassified
D04786  Loviride (USAN/INN) (CI,P) unclassified
D04813  Lidocaine hydrochloride and epinephrine bitartrate; Lidocaine hydrochloride and adrenaline bitartrate; Ora (TN); Lidosite (TN) (P) CYP induction: CYP3A4
D04820  Lurasidone hydrochloride (JAN/USAN); SM 13496; Latuda (TN) (CI,P) CYP induction: CYP3A4
D04859  Maribavir (JAN/USAN/INN); Camvia (TN); Livtencity (TN) (P) CYP induction: CYP3A4
D04862  Masoprocol (USAN/INN); meso-Nordihydroguaiaretic acid; Actinex (TN) (CI,P) unclassified
D04872  Mechlorethamine hydrochloride (USP); Chlormethine hydrochloride; Mustargen (TN); Valchlor (TN) (CI,P) unclassified
D04882  Medazepam hydrochloride (USAN); Nobrium (TN) (P) unclassified
D04884  Medorinone (USAN/INN) (P) unclassified
D04888  Medroxalol (USAN/INN) (P) unclassified
D04889  Medroxalol hydrochloride (USAN) (P) unclassified
D04931  Mercaptopurine (INN); Mercaptopurine anhydrous; Purinethol (TN) (CI,P) unclassified
D04955  Sematilide hydrochloride (USAN) (P) unclassified
D04966  Metformin (USAN/INN) (P) unclassified
D04985  Methohexital (USP/INN) (P) unclassified
D04988  Methyl aminolevulinate hydrochloride (USAN); Metvixia (TN) (CI,P) unclassified
D05000  Methylprednisolone hemisuccinate (USP); Methylprednisolone succinate (JP18) (P) CYP induction: CYP3A4
D05001  Methylprednisolone sodium phosphate (USAN) (P) CYP induction: CYP3A4
D05002  Methylprednisolone suleptanate (USAN/INN) (P) CYP induction: CYP3A4
D05008  Metoclopramide hydrochloride (USP); Metoclopramide monohydrochloride monohydrate; Clopra (TN); Reglan (TN) (P) unclassified
D05011  Metoprolol fumarate (USP); Lopressor (TN) (P) unclassified
D05024  Mibefradil dihydrochloride (USAN); Posicor (TN) (P) unclassified
D05028  Midazolam maleate (USAN) (P) CYP induction: CYP3A4
D05029  Midostaurin (JAN/USAN/INN); Rydapt (TN) (CI,P) CYP induction: CYP3A4
D05077  Moricizine (USAN); Moracizine (INN) (P) unclassified
D05087  Moxonidine (USAN/INN); Cynt (TN) (P) unclassified
D05127  Nebivolol (USAN/INN) (P) unclassified
D05134  Nelarabine (JAN/USAN/INN); Nelzarabine (USAN); Arranon (TN) (CI,P) unclassified
D05206  Norepinephrine bitartrate (USP); Levophed (TN) (P) unclassified
D05216  Oblimersen sodium (USAN); Genasense (TN) (CI,P) unclassified
D05259  Omeprazole magnesium (USP); Prilosec OTC (TN) (P) unclassified
D05261  Omeprazole sodium injection (JAN); Omeprazole sodium hydrate; Omepral (TN) (P) unclassified
D05268  Orconazole nitrate (USAN) (P) unclassified
D05312  Oxycodone (USAN/INN) (P) CYP induction: CYP3A4
D05333  Paclitaxel poliglumex (USAN/INN) (CI,P) CYP induction: CYP3A4
D05343  Palonosetron hydrochloride (JAN/USP); Aloxi (TN) (P) CYP induction: CYP3A4
D05345  Pamatolol sulfate (USAN) (P) unclassified
D05348  Pancopride (USAN/INN) (P) unclassified
D05350  Panitumumab (USAN/INN); Panitumumab (genetical recombination) (JAN); Vectibix (TN) (CI,P) unclassified
D05353  Pantoprazole (USAN/INN) (P) unclassified
D05366  Procaterol hydrochloride hydrate (JP18); Meptin (TN) (P) CYP induction: CYP3A4
D05367  Parconazole hydrochloride (USAN) (P) unclassified
D05380  Pazopanib hydrochloride (JAN/USAN); Votrient (TN) (CI,P) unclassified
D05387  Pegaspargase (JAN/USAN/INN); Oncaspar (TN) (CI,P) unclassified
D05403  Pelrinone hydrochloride (USAN) (P) unclassified
D05429  Aminophylline hydrate (JP18) (P) unclassified
D05442  Perhexiline maleate (USAN) (P) unclassified
D05446  Pertuzumab (USAN/INN); Pertuzumab (genetical recombination) (JAN); Perjeta (TN) (CI,P) unclassified
D05457  Phenprocoumon (USAN/INN); Liquamar (TN) (P) unclassified
D05460  Phenyl aminosalicylate (USAN); Fenamisal (INN); Pheny-Pas-Tebamin (TN) (P) unclassified
D05462  Oxycodone hydrochloride hydrate (JP18) (P) CYP induction: CYP3A4
D05482  Pinacidil (USAN); Pinacidil hydrate; Pindac (TN) (P) unclassified
D05522  Pixantrone (USAN/INN); Pixuvri (TN) (CI,P) unclassified
D05538  Mozenavir (INN) (CI,P) unclassified
D05575  Pramipexole (USAN/INN) (P) unclassified
D05587  Practolol (USAN) (P) unclassified
D05589  Pralatrexate (JAN/USAN/INN); 10-Propargyl-10-deazaaminopterin; Folotyn (TN) (CI,P) unclassified
D05594  Pramlintide (USAN/INN) (P) unclassified
D05595  Pramlintide acetate (USAN); Symlin (TN) (P) unclassified
D05601  Prednicarbate (USP/INN); Dermatop (TN) (P) unclassified
D05602  Prednimustine (USAN/INN) (CI,P) unclassified
D05606  Prenalterol hydrochloride (USAN) (P) unclassified
D05612  Prinoxodan (USAN/INN) (P) unclassified
D05621  Progabide (USAN/INN); Gabren (TN) (P) unclassified
D05681  Quinine ascorbate (USAN); Quinine biascorbate (P) CYP induction: CYP3A4 / Transporter induction: ABCB1
D05705  Rauwolfia serpentina (USP); Rauwolfia extract; Himolfia (TN) (P) unclassified
D05710  Reclazepam (USAN/INN) (P) unclassified
D05719  Resocortol butyrate (USAN) (P) unclassified
D05729  Rimexolone (USP/INN); Vexol (TN) (P) unclassified
D05744  Roflumilast (JAN/USAN/INN); Daliresp (TN); Zoryve (TN) (P) CYP induction: CYP3A4
D05768  Rotigotine (JAN/USAN/INN); Neupro (TN) (P) unclassified
D05775  Rufinamide (JAN/USP/INN); Banzel (TN) (P) unclassified
D05792  Salmeterol (USAN/INN) (P) CYP induction: CYP3A4
D05800  Saperconazole (USAN/INN) (P) unclassified
D05807  Satraplatin (USAN/INN) (CI,P) unclassified
D05822  Semustine (USAN/INN) (CI,P) unclassified
D05928  Stiripentol (JAN/USAN/INN); Diacomit (TN) (P) CYP induction: CYP3A4
D05932  Streptozocin (JAN/USAN/INN); Streptozotocin; Zanosar (TN) (CI,P) unclassified
D05942  Sulazepam (USAN/INN) (P) unclassified
D05987  Synthetic conjugated estrogens, B (USAN); Enjuvia (TN) (P) CYP induction: CYP3A4
D06060  Teludipine hydrochloride (USAN) (P) unclassified
D06066  Temoporfin (USAN/INN) (CI,P) unclassified
D06067  Temozolomide (JP18/USAN/INN); Temodal (TN); Temodar (TN) (CI,P) unclassified
D06068  Temsirolimus (JAN/USAN/INN); Torisel (TN) (CI,P) CYP induction: CYP3A4
D06074  Tenofovir (USAN); Tenofovir hydrate (CI,P) unclassified
D06103  Theophylline (USP); Theophylline monohydrate; Accurbron (TN) (P) unclassified
D06104  Theophylline sodium glycinate (USP); Asbron (TN) (P) unclassified
D06109  Thioguanine (USP); Thioguanine hydrate; Tabloid (TN); Thioguanine (TN) (CI,P) unclassified
D06129  Tiapamil hydrochloride (USAN) (P) unclassified
D06130  Tiazofurin (USAN); Tiazofurine (INN) (CI,P) unclassified
D06162  Tiprenolol hydrochloride (USAN) (P) unclassified
D06171  Tixocortol pivalate (USAN) (P) unclassified
D06172  Tocainide (USAN/INN) (P) unclassified
D06176  Tolamolol (USAN/INN) (P) unclassified
D06177  Tolbutamide sodium, sterile; Orinase diagnostic (TN) (P) unclassified
D06199  Trabectedin (JAN/USAN/INN); Yondelis (TN) (CI,P) CYP induction: CYP3A4
D06213  Treprostinil (JAN/USAN/INN); Remodulin (TN) (P) unclassified
D06216  Triamcinolone acetonide sodium phosphate (USAN) (P) unclassified
D06231  Triflubazam (USAN/INN) (P) unclassified
D06234  Trimazosin hydrochloride (USAN); Trimazosin hydrochloride monohydrate (P) unclassified
D06253  Tropanserin hydrochloride (USAN) (P) unclassified
D06265  Uracil mustard (USAN); Uramustine (INN); Uracil mustard (TN) (CI,P) unclassified
D06272  Sorafenib tosylate (USAN); Sorafenib tosilate (JAN); Nexavar (TN) (CI,P) unclassified
D06273  Imidafenacin (JAN/INN); Uritos (TN); Staybla (TN) (P) CYP induction: CYP3A4
D06304  Vindesine (USAN/INN) (CI,P) unclassified
D06315  Fluticasone furoate (JAN/USAN/INN); Veramyst (TN) (P) CYP induction: CYP3A4
D06320  Vorinostat (JAN/USAN); Zolinza (TN) (CI,P) Enzyme induction: UGT
D06328  Xamoterol (USAN) (P) unclassified
D06329  Xamoterol fumarate (USAN) (P) unclassified
D06353  Zacopride hydrochloride (USAN) (P) unclassified
D06363  Ziconotide (USAN/INN); Prialt (TN) (P) unclassified
D06373  Zinoconazole hydrochloride (USAN) (P) unclassified
D06386  Zorubicin hydrochloride (USAN) (CI,P) unclassified
D06396  Renzapride (INN) (P) unclassified
D06397  Estramustine phosphate sodium hydrate (JAN); Estramustine phosphate sodium monohydrate; Estracyt (TN); Emcyt (TN) (CI,P) unclassified
D06399  Tegafur, gimeracil and oteracil potassium; Ts-1 (TN); Teysuno (TN) (CI,P) unclassified
D06402  Sunitinib malate (JAN/USAN); Sutent (TN) (CI,P) CYP induction: CYP3A4
D06404  Liraglutide (USAN/INN); Liraglutide (genetical recombination) (JAN); Victoza (TN) (P) unclassified
D06405  Nalfurafine hydrochloride (JAN/USAN) (P) CYP induction: CYP3A4
D06407  Vandetanib (JAN/USAN/INN); Caprelsa (TN) (CI,P) CYP induction: CYP3A4
D06409  Bevacizumab (USAN); Bevacizumab (genetical recombination) (JAN); Bevacizumab (genetical recombination) [Bevacizumab biosimilar 1] (JAN); Bevacizumab (genetical recombination) [Bevacizumab biosimilar 2] (JAN); Bevacizumab (genetical recombination) [Bevacizumab biosimilar 3] (JAN); Bevacizumab (genetical recombination) [Bevacizumab biosimilar 4] (JAN); Bevacizumab-awwb; Bevacizumab-bvzr; Bevacizumab-maly; Bevacizumab-adcd; Avastin (TN); Alymsys (TN); Mvasi (TN); Vegzelma (TN); Zirabev (TN) (CI,P) unclassified
D06412  Aliskiren fumarate (JAN/USAN); Aliskiren hemifumarate; Tekturna (TN) (P) CYP induction: CYP3A4 / Transporter induction: ABCB1
D06413  Nilotinib hydrochloride hydrate (JAN); Nilotinib monohydrochloride monohydrate; Tasigna (TN) (CI,P) CYP induction: CYP3A4 / Transporter induction: ABCB1
D06414  Dasatinib (USAN); Dasatinib hydrate (JAN); Sprycel (TN) (CI,P) CYP induction: CYP3A4 / Enzyme induction: UGT
D06478  Darunavir ethanolate (JAN); Prezista (TN) (CI,P) CYP induction: CYP3A4
D06503  Pemetrexed sodium hydrate (JAN); Pemetrexed disodium heptahydrate; Alimta (TN) (CI,P) unclassified
D06517  Pirmenol hydrochloride (USAN); Pirmavar (TN) (P) unclassified
D06553  Alogliptin benzoate (JAN/USAN); Vipidia (TN); Nesina (TN) (P) unclassified
D06573  Carisbamate (USAN) (P) unclassified
D06580  Dexelvucitabine (USAN/INN); Reverset (TN) (CI,P) unclassified
D06597  Fosaprepitant dimeglumine (USAN); Fosaprepitant meglumine (JAN); Proemend (TN) (P) CYP induction: CYP3A4
D06622  Nebivolol hydrochloride (USAN); Bystolic (TN) (P) unclassified
D06623  Olanzapine pamoate (USAN); Olanzapine pamoate monohydrate; Zyprexa (TN) (P) unclassified
D06630  Pramiconazole (USAN/INN) (P) unclassified
D06637  Romidepsin (JAN/USAN/INN); Istodax (TN) (CI,P) unclassified
D06645  Sitagliptin phosphate (USAN); Sitagliptin phosphate hydrate (JP18); Sitagliptin phosphate monohydrate; Januvia (TN) (P) unclassified
D06646  Epanolol (USAN/INN) (P) unclassified
D06652  Tedisamil (USAN) (P) unclassified
D06653  Tedisamil sesquifumarate (USAN) (P) unclassified
D06657  Tremelimumab (USAN/INN); Tremelimumab (genetical recombination) (JAN); Tremelimumab-actl; CP 675206; Imjudo (TN) (CI,P) unclassified
D06665  Vernakalant hydrochloride (USAN) (P) unclassified
D06670  Maraviroc (JAN/INN); Selzentry (TN) (CI,P) CYP induction: CYP3A4
D06673  Meprednisone (USP/INN) (P) unclassified
D06676  Raltegravir (INN); MK-0518 (CI,P) unclassified
D06677  Elvitegravir (JAN/USAN); Vitekta (TN) (CI,P) unclassified
D06699  Japanese valerian (JP18); Powdered japanese valerian (JP18); Valerianae radix (TN) (P) unclassified
D06876  Hydrocortisone aceponate (INN); Efficort (TN) (P) unclassified
D06881  Acetyldigitoxin (INN); Acylanid (TN) (P) unclassified
D06883  Sertaconazole (INN) (P) unclassified
D06887  Talbutal (INN); Lotusate (TN) (P) unclassified
D07057  Abacavir (INN) (CI,P) unclassified
D07064  Acenocoumarol (INN); Acenocoumarin; Mini-sintrom (TN) (P) unclassified
D07071  Mannosulfan (INN) (CI,P) unclassified
D07073  Dexamethasone cipecilate (JAN/INN) (P) CYP induction: CYP3A4
D07077  Ambrisentan (JAN/INN); Letairis (TN); Volibris (TN) (P) unclassified
D07080  Vildagliptin (JAN/USAN/INN); Equa (TN); Galvus (TN) (P) unclassified
D07082  Dabigatran etexilate mesylate (USAN); Dabigatran etexilate methanesulfonate (JAN); Dabigatran etexilate mesilate; Pradaxa (TN) (P) Transporter induction: ABCB1
D07085  Bendamustine hydrochloride (JAN/USAN); Treanda (TN); Ribomustin (TN) (CI,P) unclassified
D07086  Rivaroxaban (JAN/USAN/INN); Xarelto (TN) (P) CYP induction: CYP3A4 / Transporter induction: ABCB1
D07100  Amrubicin hydrochloride (JAN/USAN); Calsed (TN) (CI,P) unclassified
D07113  Loperamide oxide (INN) (P) CYP induction: CYP3A4 / Transporter induction: ABCB1
D07116  Alclometasone (INN) (P) unclassified
D07117  Metahexamide (INN) (P) unclassified
D07118  Glisoxepide (INN) (P) unclassified
D07124  Alfuzosin (INN); Xatral (TN) (P) CYP induction: CYP3A4
D07129  Alosetron (INN) (P) unclassified
D07131  Ethyl biscoumacetate (INN) (P) unclassified
D07132  Buprenorphine (JAN/INN); Temgesic (TN) (P) CYP induction: CYP3A4
D07133  Raltegravir potassium (JAN/USAN); Isentress (TN) (CI,P) unclassified
D07135  Clorindione (INN); G-25766 (P) unclassified
D07136  Diphenadione (INN) (P) unclassified
D07137  Tioclomarol (INN) (P) unclassified
D07139  Cloricromen (INN) (P) unclassified
D07147  Gitoformate (INN) (P) unclassified
D07148  Oxedrine (BAN); (+/-)-Synephrine (P) unclassified
D07149  Dimetofrine (INN) (P) unclassified
D07150  Gepefrine (INN) (P) unclassified
D07151  Cafedrine (BAN) (P) unclassified
D07155  Theodrenaline (INN) (P) unclassified
D07156  Alprenolol (INN) (P) unclassified
D07165  Ivabradine (USAN/INN) (P) CYP induction: CYP3A4
D07166  Methoserpidine (INN) (P) unclassified
D07167  Bietaserpine (prop.INN) (P) unclassified
D07168  Tolonidine (INN) (P) unclassified
D07169  Guanazodine (INN) (P) unclassified
D07170  Dihydralazine (INN) (P) unclassified
D07171  Sitaxentan (USAN/INN) (P) unclassified
D07175  Palonosetron (INN); Aloxi (TN) (P) CYP induction: CYP3A4
D07181  Mepindolol (INN) (P) unclassified
D07182  Tertatolol (INN) (P) unclassified
D07183  Cloranolol (INN) (P) unclassified
D07184  Talinolol (INN) (P) unclassified
D07185  Fendiline (INN) (P) unclassified
D07192  Benfluorex (INN/BAN); Mediaxal (TN) (P) unclassified
D07193  Flutrimazole (INN) (P) unclassified
D07201  Fluprednidene (INN) (P) unclassified
D07202  Halometasone (INN) (P) unclassified
D07203  Methylprednisolone aceponate (INN); Advantan (TN) (P) CYP induction: CYP3A4
D07218  Metergoline (INN) (P) unclassified
D07226  Fesoterodine (INN) (P) CYP induction: CYP3A4
D07230  Prednylidene (INN) (P) unclassified
D07246  Tiocarlide (INN) (P) unclassified
D07247  Terizidone (INN); Terivalidin (TN) (P) unclassified
D07248  Morinamide (INN) (P) unclassified
D07252  Trofosfamide (INN) (CI,P) unclassified
D07253  Treosulfan (USAN/INN); Ovastat (TN) (CI,P) unclassified
D07254  Triaziquone (INN) (CI,P) unclassified
D07255  Fotemustine (INN/BAN); Muphoran (TN) (CI,P) unclassified
D07256  Etoglucid (INN) (CI,P) unclassified
D07257  Lonidamine (INN); Doridamina (TN) (CI,P) unclassified
D07258  Mitoguazone (INN) (CI,P) unclassified
D07283  Esketamine (USAN/INN) (P) CYP induction: CYP3A4 / Enzyme induction: UGT
D07298  Barbexaclone (INN); Maliasin (TN) (P) unclassified
D07299  Lacosamide (JAN/USAN/INN); Erlosamide; Vimpat (TN) (P) CYP induction: CYP3A4
D07300  Beclamide (INN) (P) unclassified
D07314  Pinazepam (INN); Domar (TN) (P) unclassified
D07315  Camazepam (INN) (P) unclassified
D07316  Captodiame (BAN) (P) unclassified
D07317  Emylcamate (INN) (P) unclassified
D07318  Mephenoxalone (INN); Dorsiflex (TN) (P) unclassified
D07319  Gedocarnil (INN) (P) unclassified
D07320  Etifoxine (INN/BAN) (P) unclassified
D07321  Vinylbital (INN); Vinylbitone (P) unclassified
D07322  Vinbarbital (INN) (P) unclassified
D07323  Cyclobarbital (INN); Ciclobarbital (TN) (P) unclassified
D07324  Proxibarbal (INN); Centralgol (TN) (P) unclassified
D07325  Chloralodol (INN); Chlorhexadol (P) unclassified
D07326  Loprazolam (INN); Dormonoct (TN) (P) unclassified
D07327  Doxefazepam (INN) (P) unclassified
D07328  Cinolazepam (INN); Gerodorm (TN) (P) unclassified
D07329  Pyrithyldione (INN) (P) unclassified
D07330  Clomethiazole (INN); Distraneurine (TN) (P) unclassified
D07331  Hexapropymate (INN); Merinax (TN) (P) unclassified
D07332  Methylpentynol (INN); Meparfynol; Methylparafynol; Atemorin (TN) (P) unclassified
D07333  Niaprazine (INN); Nopron (TN) (P) unclassified
D07402  Levocetirizine (USAN/INN); Xazal (TN) (P) CYP induction: CYP3A4
D07407  Rupatadine (INN) (P) CYP induction: CYP3A4
D07428  Bunaftine (INN) (P) unclassified
D07441  Amantadine (INN) (P) unclassified
D07448  Amitriptyline (INN); Laroxyl (TN) (P) CYP induction: CYP3A4
D07450  Amlodipine (USP/INN); Norvasc (TN) (P) CYP induction: CYP3A4
D07455  Anagrelide (INN/BAN) (CI,P) unclassified
D07457  Anisindione (INN); Miradon (TN) (P) unclassified
D07460  Apomorphine (BAN); Uprima (TN) (P) unclassified
D07464  Paramethasone (INN); Dillar (TN) (P) unclassified
D07465  Arotinolol (INN) (P) unclassified
D07471  Atazanavir (INN); Reyataz (TN) (CI,P) unclassified
D07472  Pemetrexed (INN); Alimta (TN); Pemetrexed (TN); Pemfexy (TN) (CI,P) unclassified
D07474  Atorvastatin (INN); Lipitor (TN); Sortis (TN) (P) CYP induction: CYP3A4 / Transporter inhibition: SLCO1B1 SLCO1B3 / Transporter induction: ABCB1
D07481  Azasetron (INN) (P) unclassified
D07494  Barnidipine (INN); Vasexten (TN) (P) CYP induction: CYP3A4
D07495  Beclometasone (INN); Beclometason (TN) (P) unclassified
D07496  Befunolol (INN) (P) unclassified
D07501  Bendamustine (INN); Treanda (TN) (CI,P) unclassified
D07507  Zidovudine and lamivudine; Combivir (TN); Lamivudine zidovudine (TN) (CI,P) unclassified
D07508  Benfluorex hydrochloride; Mediator (TN) (P) unclassified
D07509  Benidipine (INN) (P) CYP induction: CYP3A4
D07520  Bepridil (INN); Bepadin (TN) (P) CYP induction: CYP3A4
D07526  Betaxolol (INN); Betaxolol (TN) (P) unclassified
D07535  Bleomycin (INN); BLM; Bleomycin Hexal (TN) (CI,P) unclassified
D07537  Bopindolol (INN); Sandonorm (TN) (P) unclassified
D07538  Bosentan (INN) (P) CYP induction: CYP3A4
D07545  Brovincamine (INN); Sarbromin (TN) (P) unclassified
D07546  Bucladesine (INN) (P) unclassified
D07552  Bupivacaine (USAN/INN); Bucaine (TN); Exparel (TN) (P) CYP induction: CYP3A4
D07555  Acetyldigoxin; Cedigossima (TN) (P) unclassified
D07556  beta-Acetyldigoxin; Acetyldigoxin beta isomer; Corotal (TN) (P) unclassified
D07567  Aminolevulinic acid (CI,P) unclassified
D07569  Candesartan cilexetil and anmlodipine besylate (JP18); Unisia (TN) (P) CYP induction: CYP3A4
D07583  Phenytoin and phenobarbital; Aleviatin with phenobarbital (TN) (P) unclassified
D07585  Isopropylantipyrine, ergotamine tartrate and anhydrous caffeine; Cleamine A (TN) (P) CYP induction: CYP3A4
D07590  Bupranolol (INN) (P) unclassified
D07593  Buspirone (INN); Gen-Buspirone (TN) (P) unclassified
D07595  Fosphenytoin sodium hydrate (JAN); Fostoin (TN) (P) unclassified
D07598  Butoconazole (INN); Gynofort (TN) (P) unclassified
D07603  Caffeine citrate (USP); Cafcit (TN) (P) unclassified
D07607  Capreomycin (INN) (P) unclassified
D07608  Carazolol (INN); Conducton (TN); Suacron [veterinary] (TN) (P) unclassified
D07624  Carteolol (INN) (P) unclassified
D07660  Celiprolol (INN); Celiprolol PCH (TN) (P) unclassified
D07661  Cerivastatin (INN) (P) CYP induction: CYP3A4
D07667  Cevimeline (INN) (P) CYP induction: CYP3A4
D07671  Chlormethine (INN); Mechlorethamine (CI,P) unclassified
D07674  Chloramphenicol stearate; Quemicetina (TN) (P) unclassified
D07675  Chloramphenicol succinate; Chloramphenicol ICN (TN) (P) unclassified
D07676  Chlormidazole hydrochloride; Unfungicid (TN) (P) unclassified
D07682  Clazosentan sodium (JAN/USAN); Pivlaz (TN) (P) unclassified
D07704  Citalopram (USP/INN); Citadur (TN) (P) CYP induction: CYP3A4 / Transporter induction: ABCB1
D07705  Citalopram hydrochloride; Seropram (TN) (P) CYP induction: CYP3A4 / Transporter induction: ABCB1
D07710  Clarithromycin lactobionate; Klacid (TN) (P) CYP induction: CYP3A4
D07714  Climazolam (INN); Climasol [veterinary] (TN) (P) unclassified
D07715  Clobetasol (INN); Clobecort Amex (TN) (P) unclassified
D07717  Clobetasone (INN) (P) unclassified
D07719  Clocortolone (INN) (P) unclassified
D07724  Magnesium clofibrate (INN); Clofibric acid magnesium salt; Clofibrate Magnesico Chobet (TN) (P) unclassified
D07725  Clomethiazole edisilate; Heminevrin (TN) (P) unclassified
D07727  Clomipramine (INN); Anafranil (TN) (P) CYP induction: CYP3A4
D07729  Clopidogrel (USP/INN); Clopidogrel (TN); Plavix (TN) (P) unclassified
D07736  Cloricromen hydrohloride; Proendotel (TN) (P) unclassified
D07740  Codeine hydrochloride; Bisoltus (TN) (P) unclassified
D07749  Cortisone (INN); Cortisone (TN) (P) unclassified
D07752  Croconazole (INN) (P) unclassified
D07757  Cyclobarbital calcium (BAN); Phanodorn calcium (TN) (P) unclassified
D07760  Cyclophosphamide (INN); Cyclophosphamide (TN); Cytoxan (TN) (CI,P) CYP induction: CYP3A4
D07772  Dacarbazine citrate (CI,P) unclassified
D07776  Daunorubicin (INN); DM; DaunoXome (TN) (CI,P) unclassified
D07782  Delavirdine (INN) (CI,P) unclassified
D07784  Delorazepam (INN); Dadumir (TN) (P) unclassified
D07793  Desvenlafaxine (INN); Khedezla (TN) (P) CYP induction: CYP3A4 / Enzyme induction: UGT
D07796  Dexamethasone 21-acetate; Dexamethasone acetate anhydrous; Decaject-L.A. (TN) (P) CYP induction: CYP3A4
D07797  Dexamethasone isonicotinate; Dexamethasone 21-isonicotinate; Voren [veterinary] (TN) (P) CYP induction: CYP3A4
D07798  Dexamethasone sodium hemisulfate; Dexamethasone 21-sodium sulfate; Colircusi Dexametasona (TN) (P) CYP induction: CYP3A4
D07799  Dexamethasone 21-tebutate; Dexamethasone tertiary butyl acetate; Dexamedium [veterinary] (TN) (P) CYP induction: CYP3A4
D07800  Dexamethasone 21-valerate; Voalla (TN); Zalucs (TN) (P) CYP induction: CYP3A4
D07801  Dexamethasone phenylpropionate; Dexafort [veterinary] (TN) (P) CYP induction: CYP3A4
D07802  Dexamethasone phosphate; Decadron-phosphate (TN) (P) CYP induction: CYP3A4
D07827  Diflorasone (INN); Murode (TN) (P) unclassified
D07830  Dihydralazine sulfate; Dihydralazine hydrogen sulfate; Nepresol (TN) (P) unclassified
D07831  Dihydrocodeine (INN); Remedacen (TN) (P) unclassified
D07832  Dihydrocodeine thiocyanate; Paracodin (TN) (P) unclassified
D07837  Dihydroergotamine (INN); Neomigran (TN) (P) CYP induction: CYP3A4
D07838  Dihydroergotamine tartrate; Divegal (TN) (P) CYP induction: CYP3A4
D07839  Dihydroergotoxine; Co-Dergocrin (TN) (P) CYP induction: CYP3A4
D07845  Diltiazem (INN); Surazem (TN) (P) CYP induction: CYP3A4
D07866  Docetaxel (JAN/INN); Docetaxel (TN); Taxotere (TN) (CI,P) CYP induction: CYP3A4
D07867  Dolasetron (INN) (P) unclassified
D07868  Domperidone maleate; Domperidone (TN) (P) CYP induction: CYP3A4
D07869  Donepezil (JAN/INN); Donaz (TN); Allydone (TN) (P) CYP induction: CYP3A4
D07870  Dopamine (INN); Medopa (TN) (P) unclassified
D07871  Dorzolamide (INN); Trusopt (TN) (P) CYP induction: CYP3A4
D07873  Doxapram (INN); Docatone (TN) (P) CYP induction: CYP3A4
D07874  Doxazosin (INN); Cardura XL (TN) (P) unclassified
D07882  Eberconazole (INN) (P) unclassified
D07883  Eflornithine (INN) (CI,P) unclassified
D07884  Eberconazole nitrate; Ebernet (TN) (P) unclassified
D07886  Efonidipine (INN) (P) unclassified
D07887  Eletriptan (INN) (P) CYP induction: CYP3A4
D07894  Encainide (INN) (P) unclassified
D07897  Enviomycin (INN) (P) unclassified
D07901  Epirubicin (INN); Farmorubicin (TN) (CI,P) unclassified
D07905  Ergometrine (INN) (P) CYP induction: CYP3A4
D07906  Ergotamine (INN) (P) CYP induction: CYP3A4
D07907  Erlotinib (INN) (CI,P) CYP induction: CYP3A4
D07913  Escitalopram (INN); Esertia (TN) (P) CYP induction: CYP3A4
D07916  Esmolol (INN) (P) unclassified
D07917  Esomeprazole (INN); Inexium paranova (TN) (P) unclassified
D07918  Estradiol hemihydrate; Estrasorb (TN); Vagifem (TN) (P) CYP induction: CYP3A4
D07919  Estradiol 17 beta-hemisuccinate; 17beta-Estradiol hemisuccinate; Eutocol (TN) (P) CYP induction: CYP3A4
D07925  Ethambutol (INN); Servambutol (TN) (P) unclassified
D07928  Ethinylestradiol propanesulfonate; Turisteron (TN) (P) CYP induction: CYP3A4
D07929  Ethylmorphine (BAN) (P) CYP induction: CYP3A4
D07930  Etifoxine hydrochloride; Stresam (TN) (P) unclassified
D07931  Etilefrine (INN); Corcanfol (TN) (P) unclassified
D07933  Etofylline (INN); Oxyphyllin (TN) (P) unclassified
D07943  Fendiline hydrochloride; Sensit (TN) (P) unclassified
D07945  Fenfluramine (INN); Ponderax (TN) (P) CYP induction: CYP3A4
D07962  Flecainide (INN) (P) unclassified
D07966  Fludarabine (INN); Fluradosa (TN) (CI,P) unclassified
D07967  Fludrocortisone (INN); Astonin-H (TN) (P) unclassified
D07969  Fluindione (INN); Previsccan (TN) (P) unclassified
D07971  Flunarizine (INN); Sibelium (TN) (P) unclassified
D07972  Fluocortin (INN) (P) unclassified
D07973  Fluocortolone 21-pivalate; Fluocortolone pivalate; Ultradil (TN) (P) unclassified
D07974  Fluorouracil sodium salt; Fluorouracil (TN) (CI,P) unclassified
D07980  Fluprednidene acetate; Fluprednidene 21-acetate; Decoderm (TN) (P) unclassified
D07981  Fluticasone (INN); Fluticaps (TN) (P) CYP induction: CYP3A4
D07983  Fluvastatin (INN); Fluvas (TN) (P) CYP induction: CYP3A4 / Transporter inhibition: SLCO1B1
D07993  Fosphenytoin (INN) (P) unclassified
D08009  Gallopamil (INN) (P) unclassified
D08020  Lorcainide (INN) (P) unclassified
D08024  Vosaroxin (USAN); Voreloxin (CI,P) unclassified
D08030  Guanethidine (INN) (P) unclassified
D08031  Guanfacine (INN); Estulic (TN) (P) CYP induction: CYP3A4
D08035  Haloperidol lactate; Haldol (TN) (P) CYP induction: CYP3A4
D08044  Hydralazine (INN); Hidral (TN) (P) unclassified
D08045  Hydrocodone (INN); Dihydrocodeinone (P) CYP induction: CYP3A4
D08046  Hydrocodone hydrochloride; Dihydrocodeinone hydrochloride; Dicodid (TN) (P) CYP induction: CYP3A4
D08048  Hydroquinidine (DCF); Dihydroquinidine (P) unclassified
D08049  Hydroquinidine hydrochloride; Idrochinidine (TN); Serecor (TN) (P) unclassified
D08050  Hydroxychloroquine (INN); Polirreumin (TN) (P) CYP induction: CYP3A4
D08054  Hydroxyzine (INN); Marex (TN) (P) unclassified
D08057  Ibopamine hydrochloride; Scandine (TN) (P) unclassified
D08060  Ibutilide (INN) (P) unclassified
D08062  Idarubicin (INN); Zavedos (TN) (CI,P) unclassified
D08066  Imatinib (INN); Glamox (TN) (CI,P) CYP induction: CYP3A4
D08070  Imipramine (INN); Tofranil (TN) (P) CYP induction: CYP3A4
D08071  Imipramine pamoate (USP); Imipramine embonate; Tofranil-pm (TN) (P) CYP induction: CYP3A4
D08074  Penbutolol (INN) (P) unclassified
D08078  Indenolol (INN) (P) unclassified
D08086  Irinotecan (INN); Biotecan (TN) (CI,P) unclassified
D08090  Isoprenaline (INN) (P) unclassified
D08095  Ivabradine hydrochloride (JAN/USAN); Ivabrandine hydrochloride; Corlanor (TN); Corlentor (TN); Coralan (TN) (P) CYP induction: CYP3A4
D08099  Ketanserin tartrate; Sufrexal (TN) (P) unclassified
D08108  Lapatinib (INN) (CI,P) CYP induction: CYP3A4 / Transporter induction: ABCB1
D08111  Lercanidipine (INN); Lercanil (TN) (P) unclassified
D08115  Levobunolol (INN) (P) unclassified
D08116  Levobupivacaine (INN); Novabupi (TN) (P) CYP induction: CYP3A4
D08118  Levocetirizine dihydrochloride (USP); Levocetirizine hydrochloride (JAN); Xyzal (TN) (P) CYP induction: CYP3A4
D08120  Levofloxacin (INN); Cravit (TN); Levaquin (TN) (P) unclassified
D08127  Lidocaine hydrochloride monohydrate; Lidocaine (TN); Zingo (TN) (P) CYP induction: CYP3A4
D08144  Loperamide (INN); Diamide (TN) (P) CYP induction: CYP3A4 / Transporter induction: ABCB1
D08145  Loprazolam mesilate; Loprazolam mesylate; Loprazolam methanesulfonate; Havlane (TN) (P) unclassified
D08147  Loteprednol (INN) (P) unclassified
D08148  Loxapine hydrochloride; Desconex (TN) (P) CYP induction: CYP3A4
D08155  Manidipine (INN); Manidipine 6300; Artedil (TN) (P) CYP induction: CYP3A4
D08157  Mazaticol (INN) (P) unclassified
D08170  Melatonin (JAN); Melatonina (TN); Melatobel (TN) (P) unclassified
D08173  Melphalan hydrochloride; Alkeran (TN); Evomela (TN) (CI,P) unclassified
D08180  Mephentermine (INN) (P) unclassified
D08192  Metaraminol (INN) (P) unclassified
D08194  Deserpidine (INN); Halmonyl (TN) (P) unclassified
D08195  Methadone (BAN) (P) CYP induction: CYP3A4 / Transporter induction: ABCB1
D08201  Methoxamine (BAN) (P) unclassified
D08204  Methyl aminolevulinate (CI,P) unclassified
D08205  Methyldopa (INN); Aldomet (TN) (P) unclassified
D08207  Methylergometrine (INN); Ergotyl (TN) (P) CYP induction: CYP3A4
D08212  Trimazosin (INN) (P) unclassified
D08215  Mexiletine (INN) (P) unclassified
D08216  Mianserin (INN); Tolvon (TN) (P) CYP induction: CYP3A4
D08217  Mibefradil (INN) (P) unclassified
D08220  Midodrine (INN) (P) unclassified
D08224  Mitoxantrone (INN); Misostol (TN) (CI,P) unclassified
D08227  Mometasone (INN) (P) CYP induction: CYP3A4
D08229  Montelukast (INN); Brondilat (TN) (P) CYP induction: CYP3A4
D08236  Mosapride (INN); Mosart (TN) (P) CYP induction: CYP3A4
D08254  Endralazine (INN) (P) unclassified
D08255  Naratriptan (INN); Naramig (TN) (P) CYP induction: CYP3A4
D08259  Nelfinavir (INN); Viracept (TN) (CI,P) CYP induction: CYP3A4
D08270  Nicardipine (INN); Cardene (TN) (P) CYP induction: CYP3A4
D08276  Nimustine (INN) (CI,P) unclassified
D08283  Nordazepam (INN); Calmday (TN) (P) CYP induction: CYP3A4
D08284  Norepinephrine hydrochoride; (-)-Noradrenaline hydrochloride; Arterenol (TN) (P) unclassified
D08286  Norfenefrine (INN) (P) unclassified
D08290  Oblimersen (INN) (CI,P) unclassified
D08291  Ofloxacin hydrochloride; Tarivid (TN) (P) CYP induction: CYP3A4
D08294  Olprinone (INN) (P) unclassified
D08296  Omoconazole (INN) (P) unclassified
D08308  Oxedrine tartrate; Dacryoboraline (TN) (P) unclassified
D08309  Oxedrine hydrochloride; Ocuton (TN) (P) unclassified
D08313  Oxiconazole (INN) (P) unclassified
D08315  Oxilofrine hydrochloride; Carnigen (TN) (P) unclassified
D08318  Oxprenolol (INN); Oxprenolol (TN) (P) unclassified
D08339  Pergolide (INN); Permax (TN) (P) unclassified
D08340  Perhexiline (INN) (P) unclassified
D08351  Phenformin (BAN) (P) unclassified
D08352  Phenformin hydrochloride; Debei (TN) (P) unclassified
D08354  Phenindione (INN); Hedulin (TN) (P) unclassified
D08356  Phenobarbital diethylamine; Gratusminal (TN) (P) unclassified
D08365  Phenylephrine (INN); Phenylephrine Minims (TN) (P) unclassified
D08366  Phenylephrine tartrate; L-Phenylephrine tartrate; Boraline (TN) (P) unclassified
D08377  Pilsicainide (INN) (P) unclassified
D08378  Pioglitazone (INN); Actos (TN) (P) unclassified
D08386  Pirarubicin hydrochloride; Pinorubin (TN); Therarubicin (TN) (CI,P) unclassified
D08394  Pirmenol (INN) (P) unclassified
D08395  Piroheptine (INN) (P) unclassified
D08408  Pranlukast (INN); Azlaire (TN) (P) CYP induction: CYP3A4
D08411  Prazosin (INN); Minipress (TN) (P) unclassified
D08412  Prednisolone pivalate; Prednisolone 21-pivalate; Ultracortenol (TN) (P) unclassified
D08413  Prednisolone sodium metazoate (USAN); Prednisolone metasulfobenzoate sodium; Prednisolone 21-(sodium 3-sulfobenzoate); Predenema (TN) (P) unclassified
D08414  Prednisolone 21-(sodium tetrahydrophthalate); Prednisolone sodium tetrahydrophthalate; Fenicort (TN) (P) unclassified
D08415  Prednisolone steaglate (BAN); Prednisolone 21-steaglate; Sintisone (TN) (P) unclassified
D08416  Prednisone acetate; Prednisone 21-acetate (P) unclassified
D08421  Procainamide (INN) (P) unclassified
D08423  Procarbazine (INN) (CI,P) unclassified
D08424  Procaterol (INN); Meptin (TN) (P) CYP induction: CYP3A4
D08435  Propafenone (INN); Propafenon hexal (TN) (P) CYP induction: CYP3A4
D08439  Propiomazine maleate; Propavan (TN) (P) unclassified
D08441  Propiverine (INN) (P) CYP induction: CYP3A4
D08443  Propranolol (INN); Propranolol (TN) (P) unclassified
D08453  Pargyline (INN) (P) unclassified
D08456  Quetiapine (INN); Norsic (TN) (P) CYP induction: CYP3A4
D08458  Quinidine (BAN); Kinidin (TN) (P) unclassified
D08459  Quinidine phenylethylbarbiturate; Quinidine 5-ethyl 5-phenyl barbiturate; Natisedine (TN) (P) unclassified
D08460  Quinine (BAN); Kinder Quinina (TN) (P) CYP induction: CYP3A4 / Transporter induction: ABCB1
D08461  Quinine dihydrochloride; Quinine (TN) (P) CYP induction: CYP3A4 / Transporter induction: ABCB1
D08463  Rabeprazole (INN); Eraloc (TN) (P) CYP induction: CYP3A4
D08466  Ramosetron (INN) (P) unclassified
D08469  Rasagiline (USAN/INN); Azilect (TN) (P) unclassified
D08476  Resocortol (INN) (P) unclassified
D08479  Rifampicin sodium; Rifadine (TN) (P) unclassified
D08480  Rifamycin sodium (USAN); Rifamycin SV sodium salt; Aemcolo (TN); Otofa (TN); Rifocina (TN) (P) unclassified
D08481  Rilmazafone (INN) (P) CYP induction: CYP3A4
D08482  Rilmenidine (INN); Hyperium (TN) (P) unclassified
D08488  Amlodipine besilate and atorvastatin calcium; Caduet (TN) (P) CYP induction: CYP3A4
D08489  Ropinirole (USAN/INN); Ropitor (TN) (P) unclassified
D08490  Ropivacaine (INN); Naropin (TN) (P) CYP induction: CYP3A4
D08491  Rosiglitazone (INN); Gaudil (TN) (P) unclassified
D08493  Dorzolamide hydrochloride and timolol maleate (JP18); Cosopt (TN) (P) CYP induction: CYP3A4
D08497  Rupatadine fumarate (JAN); Rinialer (TN); Rupafin (TN) (P) CYP induction: CYP3A4
D08508  Sarpogrelate (INN) (P) CYP induction: CYP3A4
D08510  Sertaconazole nitrate; Ertaczo (TN); Zalain (TN) (P) unclassified
D08514  Sildenafil (INN); Aphrodil (TN) (P) CYP induction: CYP3A4
D08516  Sitagliptin (USAN/INN) (P) unclassified
D08517  Sitaxentan sodium (USAN); Thelin (TN) (P) unclassified
D08522  Solifenacin (INN) (P) CYP induction: CYP3A4
D08524  Sorafenib (USAN/INN) (CI,P) unclassified
D08525  Sotalol (INN); Darob mite (TN) (P) unclassified
D08531  Streptomycin (INN); Streptomycin (TN) (P) unclassified
D08535  Sulconazole (INN) (P) unclassified
D08552  Sunitinib (INN) (CI,P) CYP induction: CYP3A4
D08556  Tacrolimus (INN); Prograf (TN) (P) CYP induction: CYP3A4
D08559  Tamoxifen (INN); Tamoxifen (TN); Tamoplex (TN) (P) CYP induction: CYP3A4
D08572  Tertatolol hydrochloride; Artex (TN) (P) unclassified
D08575  Tetrabenazine (JAN/INN); Nitoman (TN); Xenazine (TN) (P) unclassified
D08584  Thioacetazone (INN); Amithiozone; Citazone (TN) (P) unclassified
D08588  Tiagabine (INN); Gabitril (TN) (P) unclassified
D08598  Tilisolol (INN) (P) unclassified
D08600  Timolol (INN); Timolol (TN); Betimol (TN) (P) unclassified
D08603  Tioguanine (INN); Lanvis (TN) (CI,P) unclassified
D08605  Tipranavir (INN); Aptivus (TN) (CI,P) unclassified
D08610  Tixocortol (INN) (P) unclassified
D08616  Teneligliptin (INN) (P) CYP induction: CYP3A4
D08618  Topotecan (BAN); Hycamtin (TN) (CI,P) Transporter induction: ABCB1
D08620  Toremifene (INN); Fareston (TN) (P) CYP induction: CYP3A4
D08623  Tramadol (INN); Amanda (TN) (P) CYP induction: CYP3A4
D08626  Trazodone (INN); Trittico (TN) (P) CYP induction: CYP3A4
D08628  Treprostinil monosodium salt; Treprostinil sodium; Trepulmix (TN) (P) unclassified
D08634  Triclofos (INN); Neguvon [veterinary] (TN) (P) unclassified
D08638  Trihexyphenidyl (INN); Apo-trihex (TN) (P) unclassified
D08660  Ulobetasol (INN); Halobetasol (P) unclassified
D08662  Urapidil hydrochloride; Ebrantil (TN) (P) unclassified
D08667  Calcium valproate; Valproic acid calcium salt; Convulsofin (TN) (P) unclassified
D08668  Vardenafil (USAN/INN); Levitra (TN) (P) CYP induction: CYP3A4
D08670  Venlafaxine (INN); Efectin (TN) (P) unclassified
D08675  Vinblastine (INN); Vinblastina (TN) (CI,P) CYP induction: CYP3A4
D08679  Vincristine (INN); Tecnocris (TN) (CI,P) unclassified
D08680  Vinorelbine (INN); Navelbine (TN) (CI,P) CYP induction: CYP3A4
D08682  Warfarin (INN); Warfarine; Choice (TN) (P) unclassified
D08686  Ziconotide acetate; Prialt (TN) (P) unclassified
D08690  Zolpidem (INN); Sanval (TN) (P) CYP induction: CYP3A4
D08695  dl-Methylephedrine hydrochloride, dihydrocodeine phosphate, diprophylline, diphenhydramine salicylate, acetaminophen and bromovalerylurea; Coughcode N (TN) (P) unclassified
D08697  Platycodon fluidextract, glycyrrhiza extract, plantago herb extract, peony root extract and dihydrocodeine phosphate; Opisezol codeine (TN) (P) unclassified
D08699  Salmeterol xinafoate and fluticasone propionate; Adoair diskus (TN); Aerivio Spiromax (TN) (P) CYP induction: CYP3A4
D08774  Amoxicillin hydrate, clarithromycin and lansoprazole; Lansap (TN); Prevpac (TN) (P) CYP induction: CYP3A4
D08775  Abacavir sulfate and lamivudine; Epzicom (TN) (CI,P) unclassified
D08843  Albiglutide (USAN); Albiglutide (genetical recombination) (JAN); Tanzeum (TN) (P) unclassified
D08854  Amrubicin (USAN/INN) (CI,P) unclassified
D08856  Anamorelin hydrochloride (JAN/USAN); Adlumiz (TN) (P) CYP induction: CYP3A4
D08860  Apremilast (JAN/USAN); Otezla (TN) (P) unclassified
D08870  Belinostat (USAN/INN); Beleodaq (TN) (CI,P) CYP induction: CYP3A4
D08879  Brivaracetam (JAN/USAN/INN); Briviact (TN) (P) unclassified
D08880  Carfilzomib (JAN/USAN/INN); Kyprolis (TN) (CI,P) unclassified
D08881  Cediranib (USAN/INN) (CI,P) unclassified
D08883  Cediranib maleate (JAN/USAN) (CI,P) unclassified
D08892  Clevidipine (USAN/INN); Clevidipine butyrate; Cleviprex (TN) (P) unclassified
D08897  Dapagliflozin (JAN/USAN/INN); Forxiga (TN) (P) unclassified
D08900  Ridaforolimus (JAN/USAN/INN); Deforolimus (CI,P) unclassified
D08903  Dexlansoprazole (INN/USAN); Dexilant (TN) (P) CYP induction: CYP3A4
D08914  Eribulin mesylate (USAN); Eribulin mesilate (JAN); Halaven (TN) (CI,P) CYP induction: CYP3A4
D08923  Fesoterodine fumarate (JAN/USAN); Toviaz (TN) (P) CYP induction: CYP3A4
D08933  Inotuzumab ozogamicin (USAN/INN); Inotuzumab ozogamicin (genetical recombination) (JAN); Besponsa (TN) (CI,P) unclassified
D08950  Neratinib (USAN/INN) (CI,P) unclassified
D08953  Nilotinib (USAN/INN) (CI,P) CYP induction: CYP3A4 / Transporter induction: ABCB1
D08956  Omacetaxine mepesuccinate (USAN); Homoharringtonine; Synribo (TN) (CI,P) unclassified
D08964  Perampanel (USAN); Fycompa (TN) (P) unclassified
D08966  Phenylephrine bitartrate (USP) (P) unclassified
D08969  Pimavanserin tartrate (USAN); Nuplazide (TN) (P) CYP induction: CYP3A4
D08976  Pomalidomide (JAN/USAN/INN); Pomalyst (TN) (P) CYP induction: CYP3A4
D08988  Rolapitant hydrochloride (USAN); Varubi (TN) (P) CYP induction: CYP3A4
D08996  Saxagliptin (USAN/INN) (P) CYP induction: CYP3A4
D09012  Telaprevir (JAN/USAN/INN); Incivek (TN); Incivo (TN) (P) CYP induction: CYP3A4
D09013  Teplizumab (USAN/INN); Teplizumab-mzwv; Tzield (TN) (P) unclassified
D09017  Ticagrelor (JAN/USAN/INN); Brilinta (TN) (CI,P) Transporter induction: ABCB1
D09032  Vinflunine ditartrate (USAN); Javlor (TN) (CI,P) unclassified
D09033  Voclosporin (JAN/USAN/INN); Lupkynis (TN) (P) CYP induction: CYP3A4
D09187  Estradiol and levonorgestrel; Wellnara (TN); Climara pro (TN) (P) CYP induction: CYP3A4
D09188  Estradiol and norethindrone; Menoaid (TN); Activella (TN); Combipatch (TN); Estradiol and norethindrone acetate (TN) (P) CYP induction: CYP3A4
D09207  Catumaxomab (INN); Removab (TN) (CI,P) unclassified
D09215  Eslicarbazepine (USAN/INN) (P) unclassified
D09217  Sitimagene ceradenovec (INN) (CI,P) unclassified
D09314  Ofatumumab (USAN/INN); Ofatumumab (genetical recombination) (JAN); Arzerra (TN); Kesimpta (TN) (CI,P) unclassified
D09318  Indacaterol (USAN/INN) (P) CYP induction: CYP3A4 / Transporter induction: ABCB1
D09319  Indacaterol maleate (JAN/USAN); Arcapta neohaler (TN) (P) CYP induction: CYP3A4 / Transporter induction: ABCB1
D09321  Obinutuzumab (USAN/INN); Obinutuzumab (genetical recombination) (JAN); Gazyva (TN) (CI,P) unclassified
D09325  Blinatumomab (USAN/INN); Blinatumomab (genetical recombination) (JAN); Blincyto (TN) (CI,P) unclassified
D09337  Elotuzumab (USAN); Elotuzumab (genetical recombination) (JAN); Empliciti (TN) (CI,P) unclassified
D09338  Entinostat (JAN/USAN/INN) (CI,P) unclassified
D09339  Esomeprazole potassium (USAN) (P) unclassified
D09347  Fostamatinib (USAN) (P) CYP induction: CYP3A4
D09348  Fostamatinib disodium (USAN); Fostamatinib sodium hydrate (JAN); Fostamatinib disodium hexahydrate; Tavalisse (TN) (P) CYP induction: CYP3A4
D09365  Palovarotene (JAN/USAN/INN); Sohonos (TN) (P) CYP induction: CYP3A4
D09371  Ramucirumab (USAN); Ramucirumab (genetical recombination) (JAN); Cyramza (TN) (CI,P) unclassified
D09388  Tasimelteon (USAN/INN); Hetlioz (TN) (P) CYP induction: CYP3A4
D09535  Mirabegron (JAN/USAN/INN); Myrbetriq (TN) (P) CYP induction: CYP3A4
D09544  Ozenoxacin (JAN/USAN/INN); Xepi (TN) (P) CYP induction: CYP3A4
D09566  Linagliptin (JAN/USAN/INN); Tradjenta (TN) (P) unclassified
D09569  Ezogabine (USAN); Retigabine (INN); Potiga (TN) (P) unclassified
D09572  Riociguat (JAN/USAN/INN); Adempas (TN) (P) Transporter induction: ABCB1
D09574  Aflibercept (USAN/INN); Aflibercept (genetical recombination) (JAN); Aflibercept (genetical recombination) [Aflibercept biosimilar 1] (JAN); Ziv-aflibercept; Eylea (TN); Zaltrap (TN) (CI,P) unclassified
D09587  Brentuximab vedotin (USAN/INN); Brentuximab vedotin (genetical recombination) (JAN); Adcetris (TN) (CI,P) unclassified
D09592  Canagliflozin (USAN/INN); Canagliflozin hydrate (JAN); Invokana (TN) (P) Transporter induction: ABCB1
D09594  Olmesartan medoxomil and azelnidipine; Rezaltas (TN) (P) CYP induction: CYP3A4
D09595  Budesonide and formoterol fumarate dihydrate; Symbicort (TN); Budeforu (TN) (P) CYP induction: CYP3A4 / Enzyme induction: UGT
D09612  Eslicarbazepine acetate (USAN); Zebinix (TN); Aptiom (TN) (P) unclassified
D09621  Gisadenafil (USAN/INN) (P) unclassified
D09622  Gisadenafil besylate (USAN) (P) unclassified
D09629  Imetelstat (USAN/INN) (CI,P) unclassified
D09630  Imetelstat sodium (USAN) (CI,P) unclassified
D09634  Lersivirine (USAN/INN) (CI,P) unclassified
D09637  Lomitapide (USAN/INN) (P) CYP induction: CYP3A4
D09638  Lomitapide mesylate (USAN); Lomitapide mesilate (JAN); Juxtapid (TN); Lojuxta (TN) (P) CYP induction: CYP3A4
D09654  Pixantrone dimaleate (USAN); Pixuvri (TN) (CI,P) unclassified
D09666  Selumetinib (USAN/INN) (CI,P) CYP induction: CYP3A4
D09676  Tecarfarin (USAN/INN) (P) unclassified
D09677  Tecarfarin sodium (USAN) (P) unclassified
D09683  Tivozanib (USAN/INN) (CI,P) CYP induction: CYP3A4
D09692  Veliparib (JAN/USAN/INN) (CI,P) unclassified
D09698  Vilazodone (USAN/INN) (P) CYP induction: CYP3A4
D09699  Vilazodone hydrochloride (USAN); Viibryd (TN) (P) CYP induction: CYP3A4
D09701  Abiraterone acetate (JAN/USP); Zytiga (TN) (P) CYP induction: CYP3A4
D09702  Albaconazole (USAN/INN) (P) unclassified
D09720  Rilpivirine (JAN/USAN/INN); Rekambys (TN) (CI,P) unclassified
D09724  Afatinib (USAN/INN) (CI,P) Transporter induction: ABCB1
D09727  Insulin degludec (USAN/INN); Insulin degludec (genetical recombination) (JAN); Tresiba (TN) (P) unclassified
D09728  Bosutinib hydrate (JAN); Bosutinib monohydrate; Bosulif (TN) (CI,P) CYP induction: CYP3A4
D09729  Lixisenatide (JAN/USAN/INN); Adlyxin (TN); Lyxumia (TN) (P) unclassified
D09730  Olaparib (JAN/USAN/INN); Lynparza (TN) (CI,P) unclassified
D09731  Crizotinib (JAN/USAN/INN); Xalkori (TN) (CI,P) CYP induction: CYP3A4
D09733  Afatinib dimaleate (USAN); Afatinib maleate (JAN); Gilotrif (TN); Giotrif (TN) (CI,P) Transporter induction: ABCB1
D09741  Drospirenone and ethinylestradiol; Drospirenone and ethinylestradiol betadex; Angeliq (TN); Yaz (TN); Flexyess (TN) (P) CYP induction: CYP3A4
D09742  Lansoprazole, amoxicillin hydrate and metronidazole; Lampion (TN) (P) CYP induction: CYP3A4
D09743  Telmisartan and amlodipine besilate (JP18); Telmisartan and amlodipine besylate; Micamlo (TN); Twynsta (TN) (P) CYP induction: CYP3A4 / Enzyme induction: UGT
D09744  Pioglitazone hydrochloride and metformin hydrochloride (JP18); Pioglitazone and metformin; Metact (TN) (P) unclassified
D09745  Valsartan and amlodipine besilate; Exforge (TN) (P) CYP induction: CYP3A4
D09749  Itasetron hydrochloride hydrate (JAN) (P) unclassified
D09753  Saxagliptin hydrate (JAN); Onglyza (TN) (P) CYP induction: CYP3A4
D09755  Cabazitaxel (USAN/INN); Jevtana (TN) (CI,P) unclassified
D09756  Teneligliptin hydrobromide hydrate (JAN) (P) CYP induction: CYP3A4
D09761  Mogamulizumab (USAN); Mogamulizumab (genetical recombination) (JAN); Mogamulizumab-kpkc; Poteligeo (TN) (CI,P) unclassified
D09763  Dapagliflozin propanediol (USAN); Dapagliflozin propylene glycolate hydrate (JAN); Dapagliflozin propandiol monohydrate; Forxiga (TN); Farxiga (TN) (P) unclassified
D09765  Vorapaxar (USAN/INN) (P) CYP induction: CYP3A4
D09766  Vorapaxar sulfate (JAN/USAN); Zontivity (TN) (P) CYP induction: CYP3A4
D09773  Isoniazid glucuronate sodium (JAN) (P) unclassified
D09783  Tofacitinib citrate (JAN/USAN); Tasocitinib citrate; Xeljanz (TN) (P) CYP induction: CYP3A4
D09785  Delamanid (JAN/USAN); Deltyba (TN) (P) CYP induction: CYP3A4
D09789  Kirenidipine hydrochloride (JAN) (P) unclassified
D09794  Norepinephrine hydrochloride (JAN); (+/-)-Noradrenaline hydrochloride (P) unclassified
D09796  Hydrocortisone caproate (JAN) (P) unclassified
D09799  Carotegrast methyl (JAN); Carogra (TN) (P) Transporter inhibition: SLCO1B1 SLCO1B3
D09807  Difethiarol (JAN); Difethialone (P) unclassified
D09843  Beradilol monoethyl maleate (JAN); TZC-5665 (P) unclassified
D09847  Metildigoxin (INN); Medigoxin (BAN) (P) Transporter induction: ABCB1
D09848  Pioglitazone hydrochloride and glimepiride tablets (JP18); Pioglitazone and glimepiride; Duetact; Sonias (TN) (P) unclassified
D09872  Bedaquiline (USAN/INN) (P) CYP induction: CYP3A4
D09873  Bedaquiline fumarate (JAN/USAN); Sirturo (TN) (P) CYP induction: CYP3A4
D09876  Cariprazine hydrochloride (JAN/USAN); Vraylar (TN) (P) CYP induction: CYP3A4
D09883  Dacomitinib (INN) (CI,P) unclassified
D09889  Dulaglutide (USAN/INN); Dulaglutide (genetical recombination) (JAN); Trulicity (TN) (P) unclassified
D09893  Eliglustat (USAN/INN) (P) Transporter induction: ABCB1
D09894  Eliglustat tartrate (JAN/USAN); Eliglustat hemitartrate; Cerdelga (TN) (P) Transporter induction: ABCB1
D09906  Fosdevirine (USAN/INN) (CI,P) unclassified
D09919  Lenvatinib (USAN/INN) (CI,P) Transporter induction: ABCB1
D09920  Lenvatinib mesylate (USAN); Lenvatinib mesilate (JAN); Lenvima (TN) (CI,P) Transporter induction: ABCB1
D09932  Moxetumomab pasudotox (USAN/INN); Moxetumomab pasudotox-tdfk; Lumoxiti (TN) (CI,P) unclassified
D09935  Navitoclax (JAN/USAN/INN) (CI,P) unclassified
D09936  Navitoclax dihydrochloride (USAN) (CI,P) unclassified
D09939  Olaratumab (USAN/INN); Olaratumab (genetical recombination) (JAN); Lartruvo (TN) (CI,P) unclassified
D09950  Ponatinib (USAN/INN) (CI,P) unclassified
D09951  Ponatinib hydrochloride (JAN/USAN); Iclusig (TN) (CI,P) unclassified
D09955  Quizartinib (USAN/INN) (CI,P) unclassified
D09956  Quizartinib dihydrochloride (USAN); Quizartinib hydrochloride (JAN); Vanflyta (TN) (CI,P) unclassified
D09958  Rilpivirine hydrochloride (JAN/USAN); Edurant (TN) (CI,P) unclassified
D09959  Ruxolitinib (USAN/INN) (CI,P) CYP induction: CYP3A4
D09960  Ruxolitinib phosphate (JAN/USAN); Jakafi (TN); Jakavi (TN); Opzelura (TN) (CI,P) CYP induction: CYP3A4
D09966  Talimogene laherparepvec (USAN); Talminogene laherparepvec; Imlygic (TN); Oncovex (TN) (CI,P) unclassified
D09970  Tofacitinib (USAN); Tasocitinib (P) CYP induction: CYP3A4
D09980  Trastuzumab emtansine (USAN/INN); Trastuzumab emtansine (genetical recombination) (JAN); Ado-trastuzumab emtansine; Kadcyla (TN) (CI,P) unclassified
D09989  Vardenafil hydrochloride (USP) (P) CYP induction: CYP3A4
D09992  Vismodegib (USAN/INN); Erivedge (TN) (CI,P) unclassified
D09994  Selexipag (JAN/USAN/INN); Uptravi (TN) (P) CYP induction: CYP3A4
D09996  Vemurafenib (JAN/USAN/INN); Zelboraf (TN) (CI,P) unclassified
D09997  Cariprazine (USAN/INN) (P) CYP induction: CYP3A4
D09999  Tramadol hydrochloride and acetaminophen; Tramcet (TN) (P) CYP induction: CYP3A4
D10018  Necitumumab (USAN/INN); Necitumumab (genetical recombination) (JAN); Portrazza (TN) (CI,P) unclassified
D10019  Panobinostat lactate (JAN); Farydak (TN) (CI,P) CYP induction: CYP3A4
D10021  Efinaconazole (JAN/USAN/INN); Clenafin (TN); Jublia (TN) (P) unclassified
D10024  Selumetinib sulfate (JAN/USAN); Koselugo (TN) (CI,P) CYP induction: CYP3A4
D10025  Semaglutide (USAN/INN); Semaglutide (genetical recombination) (JAN); Ozempic (TN) (P) unclassified
D10027  Udenafil (USAN/INN) (P) unclassified
D10062  Cabozantinib (USAN); Cabometyx (TN); Cometriq (TN) (CI,P) unclassified
D10064  Dabrafenib (USAN) (CI,P) CYP induction: CYP3A4
D10065  Daclatasvir (USAN) (P) CYP induction: CYP3A4 / Transporter induction: ABCB1
D10066  Dolutegravir (USAN); Tivicay (TN) (CI,P) unclassified
D10079  Rucaparib (USAN/INN) (CI,P) unclassified
D10082  Suvorexant (JAN/USAN); MK-4305; Belsomra (TN) (P) unclassified
D10095  Cabozantinib s-malate (USAN); Cabozantinib malate (JAN); Cometriq (TN); Cabometyx (TN) (CI,P) unclassified
D10104  Dabrafenib mesylate (USAN); Dabrafenib mesilate (JAN); Tafinlar (TN) (CI,P) CYP induction: CYP3A4
D10105  Daclatasvir dihydrochloride (USAN); Daclatasvir hydrochloride (JAN); Daklinza (TN) (P) CYP induction: CYP3A4 / Transporter induction: ABCB1
D10113  Dolutegravir sodium (JAN/USAN); Tivicay (TN) (CI,P) unclassified
D10119  Sonidegib (USAN/INN); Erismodegib (CI,P) unclassified
D10120  Esomeprazole strontium (USAN); Esomeprazole strontium tetrahydrate; Esomeprazole strontium (TN) (P) unclassified
D10130  Ixazomib (USAN) (CI,P) unclassified
D10131  Ixazomib citrate (JAN/USAN); Ninlaro (TN) (CI,P) unclassified
D10135  Macitentan (JAN/USAN); Opsumit (TN) (CI,P) CYP induction: CYP3A4
D10137  Regorafenib hydrate (JAN); Stivarga (TN) (CI,P) CYP induction: CYP3A4 / Transporter induction: ABCB1
D10138  Regorafenib (USAN/INN); Stivarga (TN) (CI,P) CYP induction: CYP3A4 / Transporter induction: ABCB1
D10140  Niraparib (USAN) (CI,P) unclassified
D10157  Rucaparib phosphate (USAN) (CI,P) unclassified
D10158  Safinamide (USAN/INN) (P) unclassified
D10159  Alogliptin benzoate and pioglitazone hydrochloride; Liovel (TN); Oseni (TN); Incresync (TN) (P) unclassified
D10170  Tedatioxetine (USAN) (P) unclassified
D10171  Tedatioxetine hydrobromide (USAN) (P) unclassified
D10175  Trametinib (USAN) (CI,P) unclassified
D10176  Trametinib dimethyl sulfoxide (JAN/USAN); Mekinist (TN); Spexotras (TN) (CI,P) unclassified
D10184  Vortioxetine (USAN); Brintellix (TN) (P) unclassified
D10185  Vortioxetine hydrobromide (JAN/USAN); Brintellix (TN); Trintellix (TN) (P) unclassified
D10188  Naldemedine (USAN/INN) (P) CYP induction: CYP3A4
D10190  Tivozanib hydrochloride (USAN); Tivozanib hydrochloride monohydrate; Fotivda (TN) (CI,P) CYP induction: CYP3A4
D10191  Safinamide mesylate (USAN); Safinamide mesilate (JAN); Safinamide methanesulfonate; Xadago (TN); Equfina (TN) (P) unclassified
D10194  Remimazolam besylate (USAN); Remimazolam besilate (JAN); Anerem (TN); Byfavo (TN) (P) unclassified
D10195  Luseogliflozin hydrate (JAN); Lusefi (TN) (P) unclassified
D10196  Ipragliflozin (INN) (P) unclassified
D10200  Ipragliflozin L-proline (JAN); Suglat (TN) (P) unclassified
D10218  Enzalutamide (JAN/USAN); Xtandi (TN) (P) unclassified
D10222  Gemcitabine elaidate (USAN/INN) (CI,P) unclassified
D10223  Ibrutinib (JAN/USAN); Imbruvica (TN) (CI,P) unclassified
D10229  Masitinib (INN) (CI,P) unclassified
D10243  Irbesartan and amlodipine besilate (JP18); Aimix (TN) (P) CYP induction: CYP3A4
D10244  Metformin hydrochloride and rosiglitazone maleate; Avandamet (TN) (P) unclassified
D10246  Omeprazole, clarithromycin and amoxicillin; Omeclamox-pak (TN) (P) CYP induction: CYP3A4
D10251  Glimepiride and rosiglitazone maleate; Avandaryl (TN) (P) unclassified
D10253  Alogliptin benzoate and metformin hydrochloride; Kazano (TN); Vipdomet (TN) (P) unclassified
D10255  Anagrelide hydrochloride hydrate (JAN); Anagrelide hydrochloride monohydrate; Agrylin (TN) (CI,P) unclassified
D10258  Simvastatin and sitagliptin phosphate; Juvisync (TN) (P) unclassified
D10261  Metformin hydrochloride and sitagliptin phosphate; Janumet (TN) (P) unclassified
D10262  Saxagliptin hydrochloride; Onglyza (TN) (P) CYP induction: CYP3A4
D10263  Metformin hydrochloride and saxagliptin hydrochloride; Kombiglyze (TN) (P) CYP induction: CYP3A4
D10264  Linagliptin and metformin hydrochloride; Jentaduet (TN) (P) Transporter induction: ABCB1
D10265  Glipizide and metformin hydrochloride; Metaglip (TN) (P) unclassified
D10266  Glyburide and metformin hydrochloride; Glibenclamide and metformin hydrochloride; Glucovance (TN) (P) unclassified
D10267  Methyldopa and hydrochlorothiazide; Methyldopa and hydrochlorothiazide (TN) (P) unclassified
D10293  Carbidopa, levodopa and entacapone; Stalevo (TN) (P) unclassified
D10306  Avatrombopag (USAN/INN) (P) CYP induction: CYP3A4
D10307  Avatrombopag maleate (JAN/USAN); Doptelet (TN) (P) CYP induction: CYP3A4
D10309  Brexpiprazole (JAN/USAN/INN); Rexulti (TN) (P) CYP induction: CYP3A4
D10313  Ertugliflozin (USAN/INN) (P) unclassified
D10315  Momelotinib (USAN/INN) (CI,P) CYP induction: CYP3A4
D10316  Nivolumab (USAN/INN); Nivolumab (genetical recombination) (JAN); Opdivo (TN) (CI,P) unclassified
D10319  Panobinostat (USAN/INN); Farydak (TN) (CI,P) CYP induction: CYP3A4
D10355  Aripiprazole cavoxil (USAN) (P) CYP induction: CYP3A4
D10358  Momelotinib dihydrochloride (USAN) (CI,P) CYP induction: CYP3A4
D10364  Aripiprazole lauroxil (USAN); Aristada (TN) (P) CYP induction: CYP3A4
D10366  Sofosbuvir (JAN/USAN/INN); Sovaldi (TN) (CI) Transporter induction: ABCB1
D10367  Etirinotecan pegol (USAN/INN) (CI,P) unclassified
D10372  Palbociclib (JAN/USAN); Ibrance (TN) (CI,P) unclassified
D10385  Ezetimibe and atorvastatin; Atozet (TN); Liptruzet (TN) (P) CYP induction: CYP3A4
D10396  Nintedanib esylate (USAN); Nintedanib ethanesulfonate (JAN); Ofev (TN) (CI,P) Transporter induction: ABCB1 / Enzyme induction: UGT
D10405  Cobimetinib (USAN/INN) (CI,P) unclassified
D10422  Etirinotecan pegol tetrahydrochloride (USAN) (CI,P) unclassified
D10427  Etirinotecan pegol tetratriflutate (USAN) (CI,P) unclassified
D10428  Tenofovir alafenamide (USAN/INN) (CI,P) Transporter induction: ABCB1
D10430  Treprostinil diolamine (USAN); Orenitram (TN) (P) unclassified
D10433  Vibegron (JAN/USAN/INN); Beova (TN); Gemtesa (TN) (P) CYP induction: CYP3A4 / Transporter induction: ABCB1
D10434  Vintafolide (USAN/INN) (CI,P) unclassified
D10446  Margetuximab (USAN/INN); Margetuximab-cmkb; Margenza (TN) (CI,P) unclassified
D10450  Alectinib hydrochloride (JAN); Alecensa (TN) (CI,P) CYP induction: CYP3A4
D10452  Cabazitaxel acetonate (JAN); Cabazitaxel acetone; Jevtana (TN) (CI,P) unclassified
D10459  Empagliflozin (JAN/USAN/INN); Jardiance (TN) (P) Transporter induction: ABCB1
D10461  Dienogest and estradiol valerate; Natazia (TN) (P) unclassified
D10466  Vonoprazan fumarate (JAN/USAN); Takecab (TN); Voquezna (TN) (P) CYP induction: CYP3A4
D10478  Naldemedine tosylate (JAN/USAN); Naldemedine tosilate; Symproic (TN) (P) CYP induction: CYP3A4
D10481  Nintedanib (USAN/INN); Ofev (TN) (CI,P) Transporter induction: ABCB1 / Enzyme induction: UGT
D10500  Metformin hydrochloride and repaglinide; Prandimet (TN) (P) unclassified
D10501  Fluticasone furoate and vilanterol trifenatate; Breo ellipta (TN); Relvar ellipita (TN) (P) CYP induction: CYP3A4
D10502  Gemigliptin (INN) (P) unclassified
D10503  Ethacizine (P) unclassified
D10505  Glycopyrronium bromide and indacaterol maleate; Ultibro (TN) (P) CYP induction: CYP3A4 / Transporter induction: ABCB1
D10506  Fluticasone propionate and formoterol fumarate hydrate; Flutiform (TN) (P) CYP induction: CYP3A4 / Enzyme induction: UGT
D10512  Brinzolamide and timolol maleate; Azorga (TN) (P) CYP induction: CYP3A4
D10513  Clopidogrel sulfate and aspirin; Clopidogrel and acetylsalicyclic acid; Complavin (TN) (P) CYP induction: CYP3A4
D10514  Dacomitinib (USAN); Dacomitinib hydrate (JAN); Vizimpro (TN) (CI,P) unclassified
D10516  Aripiprazole hydrate (JAN); Aripiprazole monohydrate; Abilify maintena (TN) (P) CYP induction: CYP3A4
D10517  Crisantaspase (JAN/INN); Enrylaze (TN); Erwinase (TN) (CI,P) unclassified
D10519  Rabeprazole, amoxicillin and clarithromycin; Rabecure (TN) (P) CYP induction: CYP3A4
D10520  Rabeprazole, amoxicillin and metronidazole; Rabefine (TN) (P) CYP induction: CYP3A4
D10524  Azilsartan and amlodipine besilate; Zacras (TN) (P) CYP induction: CYP3A4
D10525  Valsartan and cilnidipine; Atedio (TN) (P) CYP induction: CYP3A4
D10526  Trifluridine and tipiracil hydrochloride; Lonsurf (TN) (CI,P) unclassified
D10527  Acetylsalicylic acid and lansoprazole; Acetylsalicylic acid and lansoprazole; Takelda (TN) (P) CYP induction: CYP3A4
D10528  Aldosterone (INN) (P) unclassified
D10533  Umeclidinium bromide and vilanterol; Anoro (TN) (P) CYP induction: CYP3A4
D10542  Alectinib (USAN/INN) (CI,P) CYP induction: CYP3A4
D10548  Cabotegravir (JAN/USAN/INN); Vocabria (TN); Apretude (TN) (CI,P) unclassified
D10549  Cabotegravir sodium (JAN/USAN); Vocabria (TN) (CI,P) unclassified
D10551  Ceritinib (JAN/USAN/INN); Zykadia (TN) (CI,P) unclassified
D10555  Duvelisib (USAN/INN) (CI,P) unclassified
D10559  Dinutuximab (USAN/INN); Dinutuximab (genetical recombination) (JAN); Unituxin (TN) (CI,P) unclassified
D10560  Idelalisib (JAN/USAN/INN); Zydelig (TN) (CI,P) unclassified
D10561  Fabomotizole (INN) (P) unclassified
D10564  Amenamevir (JAN/INN); Amenalief (TN) (CI,P) unclassified
D10568  Pitavastatin calcium hydrate (JP18); Livalo (TN) (P) unclassified
D10570  Insulin degludec (genetical recombination) and insulin aspart (genetical recombination); Ryzodeg (TN) (P) unclassified
D10571  Rilpivirine hydrochloride, tenofovir disoproxil fumarate and emtricitabine; Complera (TN); Eviplera (TN) (CI,P) unclassified
D10572  Fosnetupitant and palonosetron hydrochloride; Netupitant and palonosetron hydrochloride; Akynzeo (TN) (P) CYP induction: CYP3A4
D10574  Pembrolizumab (USAN); Pembrolizumab (genetical recombination) (JAN); Keytruda (TN) (CI,P) unclassified
D10578  Ledipasvir and sofosbuvir; Harvoni (TN) (CI) Transporter induction: ABCB1
D10586  Dapagliflozin and metformin; Xigduo xr (TN) (P) unclassified
D10587  Canagliflozin and metformin; Invokamet (TN) (P) unclassified
D10588  Empagliflozin and linagliptin; Glyxambi (TN) (P) Transporter induction: ABCB1
D10590  Norgestimate and ethinyl estradiol; Mononessa (TN); Trinessa (TN) (P) unclassified
D10591  Clonidine and chlorthalidone; Clorpres (TN) (P) unclassified
D10596  Pemetrexed sodium hemipentahydrate (JAN); Pemetrexed disodium hemipentahydrate; Pemetrexed accord (TN) (CI,P) unclassified
D10600  Dolutegravir, abacavir and lamivudine; Triumeq (TN) (CI,P) unclassified
D10604  Binimetinib (JAN/USAN/INN); Mektovi (TN) (CI,P) unclassified
D10605  Tenofovir alafenamide fumarate (JAN/USAN); Vemlidy (TN) (CI,P) Transporter induction: ABCB1
D10612  Benzhydrocodone (USAN/INN) (P) CYP induction: CYP3A4
D10615  Cobimetinib fumarate (USAN); Cobimetinib hemifumarate; Cotellic (TN) (CI,P) unclassified
D10624  Doravirine (JAN/USAN/INN); Pifeltro (TN) (CI,P) unclassified
D10627  Esketamine hydrochloride (JAN/USAN); Spravato (TN) (P) CYP induction: CYP3A4 / Enzyme induction: UGT
D10630  Fedratinib (USAN/INN) (CI,P) CYP induction: CYP3A4
D10633  Finerenone (JAN/USAN/INN); Kerendia (TN) (P) CYP induction: CYP3A4
D10636  Glasdegib (USAN/INN) (CI,P) unclassified
D10642  Irinotecan sucrosofate (USAN) (CI,P) unclassified
D10643  Isavuconazonium sulfate (JAN/USAN); Cresemba (TN) (CI) unclassified
D10652  Palbociclib isethionate (USAN) (CI,P) unclassified
D10662  Rimegepant (USAN/INN) (P) CYP induction: CYP3A4
D10663  Rimegepant sulfate (USAN); Nurtec odt (TN); Vydura (TN) (P) CYP induction: CYP3A4
D10669  Sotagliflozin (USAN/INN); Inpefa (TN) (P) unclassified
D10673  Ubrogepant (USAN/INN); Ubrelvy (TN) (P) CYP induction: CYP3A4
D10675  Valbenazine (USAN/INN) (P) CYP induction: CYP3A4
D10679  Venetoclax (JAN/USAN/INN); Venclexta (TN) (CI,P) unclassified
D10688  Abemaciclib (JAN/USAN/INN); Verzenio (TN) (CI,P) unclassified
D10692  Benzhydrocodone hydrochloride (USAN) (P) CYP induction: CYP3A4
D10696  Capmatinib (USAN/INN) (CI,P) CYP induction: CYP3A4
D10709  Gilteritinib (USAN/INN) (CI,P) CYP induction: CYP3A4 / Transporter induction: ABCB1
D10711  Pemafibrate (JAN); Parmodia (TN) (CI,P) Transporter inhibition: SLCO1B1 SLCO1B3
D10722  Pretomanid (USAN/INN); Pretomanid (TN) (P) unclassified
D10729  Sonidegib phosphate (USAN); Sonidegib diphosphate; Odomzo (TN) (CI,P) unclassified
D10732  Talazoparib (USAN/INN) (CI,P) unclassified
D10733  Talazoparib tosylate (USAN); Talazoparib tosilate (JAN); Talzenna (TN) (CI,P) unclassified
D10742  Rolapitant (USAN/INN); Varubi (TN) (P) CYP induction: CYP3A4
D10743  Vildagliptin and metformin hydrochloride (P) unclassified
D10745  Ombitasvir, paritaprevir and ritonavir; Technivie (TN) (P) CYP induction: CYP3A4 / Transporter inhibition: SLCO1B1 SLCO1B3 / Transporter induction: ABCB1
D10749  Pitolisant (USAN/INN); Wakix (TN); Ozawade (TN) (P) unclassified
D10750  Isavuconazole (INN); Cresemba (TN) (P) unclassified
D10752  Empagliflozin and metformin; Synjardy (TN) (P) unclassified
D10753  Atazanavir and cobicistat; Evotaz (TN) (CI,P) CYP induction: CYP3A4
D10754  Lamivudine and raltegravir; Lamivudine and raltegravir potassium; Dutrebis (TN) (CI,P) unclassified
D10755  Elvitegravir, cobicistat, emtricitabine and tenofovir alafenamide; Genvoya (TN) (CI,P) unclassified
D10756  Elvitegravir, cobicistat, emtricitabine and tenofovir disoproxil; Stribild (TN) (CI,P) unclassified
D10761  Polatuzumab vedotin (USAN); Polatuzumab vedotin (genetical recombination) (JAN); Polatuzumab vedotin-piiq; Polivy (TN) (CI,P) unclassified
D10762  Fosravuconazole L-lysine ethanolate (JAN) (P) unclassified
D10766  Osimertinib mesylate (USAN); Osimertinib mesilate (JAN); Tagrisso (TN) (CI,P) unclassified
D10772  Lascufloxacin hydrochloride (JAN); Lasvic (TN) (P) unclassified
D10773  Atezolizumab (USAN/INN); Atezolizumab (genetical recombination) (JAN); Tecentriq (TN) (CI,P) unclassified
D10774  Vonoprazan, amoxicillin and metronidazole; Vonopion (TN) (P) CYP induction: CYP3A4
D10775  Vonoprazan, amoxicillin and clarithromycin; Vonosap (TN); Voquenza (TN) (P) CYP induction: CYP3A4
D10777  Daratumumab (USAN); Daratumumab (genetical recombination) (JAN); Darzalex (TN) (CI,P) unclassified
D10780  Perampanel hydrate (JAN); Fycompa (TN) (P) unclassified
D10787  Daunorubicin citrate; Daunoxome (TN) (CI,P) unclassified
D10797  Copanlisib hydrochloride (USAN) (CI,P) unclassified
D10798  Copanlisib hydrochloride hydrate (JAN); Aliqopa (TN) (CI,P) unclassified
D10800  Gilteritinib fumarate (JAN/USAN); Xospata (TN) (CI,P) CYP induction: CYP3A4 / Transporter induction: ABCB1
D10801  Letermovir (JAN/USAN/INN); Prevymis (TN) (P) Transporter inhibition: SLCO1B1 SLCO1B3
D10805  Telmisartan, amlodipine and hydrochlorothiazide; Micatrio (TN) (P) CYP induction: CYP3A4 / Enzyme induction: UGT
D10808  Durvalumab (USAN/INN); Durvalumab (genetical recombination) (JAN); Imfinzi (TN) (CI,P) unclassified
D10811  Fentanyl hydrochloride (JAN); Ionsys (TN) (P) CYP induction: CYP3A4
D10817  Avelumab (USAN/INN); Avelumab (genetical recombination) (JAN); Bavencio (TN) (CI,P) unclassified
D10823  Clopidogrel hydrochloride; Clopidogrel (TN) (P) unclassified
D10824  Clopidogrel besilate; Clopidogrel besylate; Clopidogrel (TN) (P) unclassified
D10825  Opicapone (JAN/USAN/INN); Ongentys (TN) (P) unclassified
D10826  Saxagliptin and dapagliflozin; Qtern (TN) (P) unclassified
D10827  Sofosbuvir and velpatasvir; Epclusa (TN) (CI,P) CYP induction: CYP3A4 / Transporter induction: ABCB1
D10829  Rasagiline tartrate; Rasagiline (TN) (P) unclassified
D10832  Darunavir and cobicistat; Prezcobix (TN); Rezolsta (TN) (CI,P) unclassified
D10834  Tenofovir disoproxil phosphate (CI,P) unclassified
D10835  Emtricitabine and tenofovir alafenamide; Descovy (TN) (CI,P) Transporter induction: ABCB1
D10836  Emtricitabine, rilpivirine and tenofovir alafenamide; Odefsey (TN) (CI,P) Transporter induction: ABCB1
D10838  Abacavir, lamivudine and zidovudine; Trizivir (TN) (CI,P) unclassified
D10839  Norelgestromin and ethinyl estradiol; Evra (TN); Xulane (TN); Zafemy (TN) (P) unclassified
D10851  Efavirenz, emtricitabine and tenofovir disoproxil; Atripla (TN) (CI,P) unclassified
D10858  Rociletinib (USAN/INN) (CI,P) unclassified
D10859  Olmutinib (USAN/INN) (CI,P) unclassified
D10865  Bexagliflozin (USAN); Brenzavvy (TN) (P) unclassified
D10866  Brigatinib (JAN/USAN); Alunbrig (TN) (CI,P) CYP induction: CYP3A4
D10867  Copanlisib (USAN/INN) (CI,P) unclassified
D10874  Daprodustat (JAN/USAN/INN); Duvroq (TN); Jesduvroq (TN) (P) unclassified
D10883  Ribociclib (USAN/INN) (CI,P) CYP induction: CYP3A4
D10888  Relugolix (JAN/USAN/INN); Orgovyx (TN) (P) Transporter induction: ABCB1
D10889  Momelotinib hydrochloride hydrate (JAN); Momelotinib dihydrochloride monohydrate; Ojjaara (TN); Omjjara (TN) (CI,P) CYP induction: CYP3A4
D10891  Capmatinib hydrochloride (USAN); Capmatinib hydrochloride hydrate (JAN); Tabrecta (TN) (CI,P) CYP induction: CYP3A4
D10892  Esaxerenone (JAN/INN) (P) unclassified
D10893  Acalabrutinib (JAN/USAN/INN); Calquence (TN) (CI,P) unclassified
D10895  Fosaprepitant (INN) (P) CYP induction: CYP3A4
D10897  Teneligliptin and canagliflozin; Teneligliptin and canagliflozin; Canalia (TN) (P) CYP induction: CYP3A4 / Transporter induction: ABCB1
D10898  Neratinib maleate; Nerlynx (TN) (CI,P) unclassified
D10901  Enasidenib (USAN/INN) (CI,P) unclassified
D10909  Bictegravir (USAN/INN) (CI,P) unclassified
D10910  Bictegravir sodium (JAN/USAN) (CI,P) unclassified
D10915  Cannabidiol (USAN/INN); CBD; Epidiolex (TN) (P) CYP induction: CYP3A4 / Transporter induction: ABCB1
D10926  Entrectinib (JAN/USAN/INN); Rozlytrek (TN) (CI,P) CYP induction: CYP3A4
D10927  Erdafitinib (JAN/USAN/INN); Balversa (TN) (CI,P) CYP induction: CYP3A4 / Transporter induction: ABCB1
D10930  Etrasimod (USAN) (P) CYP induction: CYP3A4 / Enzyme induction: UGT
D10931  Etrasimod arginine (USAN); Etrasimod L-arginine (JAN); Velsipity (TN) (P) CYP induction: CYP3A4 / Enzyme induction: UGT
D10954  Mirvetuximab soravtansine (USAN/INN); Mirvetuximab soravtansine-gynx; Elahere (TN) (CI,P) CYP induction: CYP3A4
D10960  Nirogacestat (USAN/INN) (P) CYP induction: CYP3A4
D10973  Padeliporfin (USAN/INN) (CI,P) unclassified
D10979  Ribociclib succinate (USAN); Kisqali (TN) (CI,P) CYP induction: CYP3A4
D10982  Rucaparib camsylate (USAN); Rubraca (TN) (CI,P) unclassified
D10985  Sacituzumab govitecan (USAN/INN); Sacituzumab govitecan (genetical recombination) (JAN); Sacituzumab govitecan-hziy; Trodelvy (TN) (CI,P) unclassified
D10994  Upadacitinib (USAN/INN) (P) CYP induction: CYP3A4
D10995  Upadacitinib tartrate (USAN) (P) CYP induction: CYP3A4
D10999  Valbenazine tosylate (USAN); Valbenazine tosilate (JAN); Valbenazine ditosylate; Ingrezza (TN); Dysval (TN) (P) CYP induction: CYP3A4
D11000  Vamorolone (USAN/INN); Agamree (TN) (P) CYP induction: CYP3A4
D11009  Indacaterol acetate (JAN) (P) CYP induction: CYP3A4 / Transporter induction: ABCB1
D11011  Alpelisib (JAN/USAN/INN); Piqray (TN) (CI,P) unclassified
D11012  Lorlatinib (JAN/USAN/INN); Lorbrena (TN) (CI,P) unclassified
D11014  Glecaprevir and pibrentasvir; Mavyret (TN) (CI) Transporter inhibition: SLCO1B1 SLCO1B3 / Transporter induction: ABCB1
D11022  Lemborexant (JAN/USAN/INN); Dayvigo (TN) (P) CYP induction: CYP3A4
D11023  Evogliptin (INN) (P) unclassified
D11032  Plitidepsin (INN) (CI,P) unclassified
D11034  Insulin glargine and lixisenatide; Insulin glargine (genetical recombination) and lixisenatide; Soliqua (TN) (P) unclassified
D11039  Bictegravir, emtricitabine and tenofovir alafenamide; Biktarvy (TN) (CI,P) unclassified
D11040  Apalutamide (JAN/INN); Erleada (TN) (P) CYP induction: CYP3A4
D11043  Ertugliflozin pidolate; Ertugliflozin L-pyroglutamic acid; Steglatro (TN) (P) unclassified
D11044  Enasidenib mesylate (USAN); Idhifa (TN) (CI,P) unclassified
D11045  Darolutamide (JAN/USAN/INN); Nebeqa (TN) (P) unclassified
D11048  Upadacitinib hydrate (JAN); Upadacitinib hemihydrate; Rinvoq (TN) (P) CYP induction: CYP3A4
D11049  Epacadostat (JAN/USAN/INN) (CI,P) unclassified
D11050  Isatuximab (USAN/INN); Isatuximab (genetical recombination) (JAN); Isatuximab-irfc; Sarclisa (TN) (CI,P) unclassified
D11053  Encorafenib (JAN/USAN/INN); Braftovi (TN) (CI,P) CYP induction: CYP3A4
D11056  Mirtazapine hydrate (JAN) (P) CYP induction: CYP3A4
D11061  Osilodrostat (USAN/INN) (P) CYP induction: CYP3A4 / Enzyme induction: UGT
D11062  Osilodrostat phosphate (JAN/USAN); Isturisa (TN) (P) CYP induction: CYP3A4 / Enzyme induction: UGT
D11066  Ertugliflozin and sitagliptin; Steglujan (TN) (P) unclassified
D11067  Ertugliflozin and metformin; Segluromet (TN) (P) unclassified
D11070  Tirabrutinib hydrochloride (JAN/USAN); Velexbru (TN) (P) unclassified
D11072  Siponimod fumarate (USAN); Siponimod fumaric acid (JAN); Mayzent (TN) (P) unclassified
D11073  Tepotinib hydrochloride (USAN); Tepotinib hydrochloride hydrate (JAN); Tepmetko (TN) (CI,P) CYP induction: CYP3A4
D11090  Ivosidenib (JAN/USAN/INN); Tibsovo (TN) (CI,P) unclassified
D11093  Avacopan (JAN/USAN/INN); Tavneos (TN) (P) CYP induction: CYP3A4
D11095  Atorvastatin calcium propylene glycol solvate (P) CYP induction: CYP3A4 / Transporter inhibition: SLCO1B1 SLCO1B3 / Transporter induction: ABCB1
D11107  Glasdegib maleate (JAN); Daurismo (TN) (CI,P) unclassified
D11108  Cemiplimab (USAN); Cemiplimab (genetical recombination) (JAN); Cemiplimab-rwlc; Libtayo (TN) (CI,P) unclassified
D11114  Esomeprazole magnesium dihydrate (P) unclassified
D11115  Olmutinib hydrochloride (USAN) (CI,P) unclassified
D11137  Larotrectinib (USAN/INN) (CI,P) unclassified
D11138  Larotrectinib sulfate (JAN/USAN); Vitrakvi (TN) (CI,P) unclassified
D11140  Sitravatinib (USAN/INN) (CI,P) unclassified
D11141  Tucatinib (USAN/INN); Tukysa (TN) (CI,P) unclassified
D11144  Axicabtagene ciloleucel (USAN); Yescarta (TN) (CI,P) unclassified
D11146  Tabelecleucel (USAN); Ebvallo (TN) (CI,P) unclassified
D11150  Cenobamate (USAN/INN); Xcopri (TN) (P) CYP induction: CYP3A4
D11158  Leniolisib (USAN/INN) (P) CYP induction: CYP3A4
D11159  Leniolisib phosphate (USAN); Joenja (TN) (P) CYP induction: CYP3A4
D11222  Selinexor (USAN/INN); Xpovio (TN) (CI,P) CYP induction: CYP3A4 / Enzyme induction: UGT
D11246  Dapivirine (USAN/INN) (CI,P) unclassified
D11251  Icotinib (CI,P) unclassified
D11252  Fexinidazole (USAN/INN); Fexinidazole (TN) (P) CYP induction: CYP3A4
D11253  Bermekimab (USAN) (CI,P) unclassified
D11270  Pexidartinib (USAN/INN) (CI,P) CYP induction: CYP3A4
D11271  Pexidartinib hydrochloride (JAN/USAN); Turalio (TN) (CI,P) CYP induction: CYP3A4
D11279  Avapritinib (USAN/INN); Ayvakit (TN); Ayvakyt (TN) (CI,P) unclassified
D11282  Dolutegravir sodium and rilpivirine hydrochloride; Juluca (TN) (CI,P) unclassified
D11296  Fedratinib hydrochloride (USAN); Fedratinib hydrochloride hydrate (JAN); Fedratinib dihydrochloride monohydrate; Inrebic (TN) (CI,P) CYP induction: CYP3A4
D11313  Atogepant (USAN); Qulipta (TN); Aquipta (TN) (P) CYP induction: CYP3A4
D11322  Umbralisib (USAN/INN) (CI,P) unclassified
D11323  Umbralisib tosylate (USAN); Ukoniq (TN) (CI,P) unclassified
D11330  Voxelotor (USAN); Oxbryta (TN) (P) CYP induction: CYP3A4
D11338  Loncastuximab tesirine (USAN); Loncastuximab tesirine (genetical recombination) (JAN); Loncastuximab tesirine-lpyl; Zynlonta (TN) (CI,P) unclassified
D11342  Dorzagliatin (USAN) (P) unclassified
D11353  Ripretinib (USAN); Qinlock (TN) (CI,P) unclassified
D11358  Tagraxofusp (USAN/INN); Tagraxofusp-erzs; Elzonris (TN) (CI,P) unclassified
D11360  Tirzepatide (JAN/USAN); Mounjaro (TN) (P) unclassified
D11366  Dostarlimab (USAN); Dostarlimab-gxly; Jemperli (TN) (CI,P) unclassified
D11370  Fosnetupitant chloride hydrochloride (JAN/USAN); Arokaris (TN) (P) unclassified
D11371  Capivasertib (JAN/USAN); Truqap (TN) (CI,P) CYP induction: CYP3A4
D11375  Trastuzumab duocarmazine (USAN/INN) (CI,P) unclassified
D11382  Darunavir, cobicistat, emtricitabine and tenofovir alafenamide; Symtuza (TN) (CI,P) unclassified
D11386  Tisagenlecleucel-T (USAN); Tisagenlecleucel (INN); Kymriah (TN) (CI,P) unclassified
D11389  Dutasteride and tamsulosin; Jalyn (TN) (P) CYP induction: CYP3A4
D11390  Daunorubicin and cytarabine; Vyxeos (TN) (CI,P) unclassified
D11391  Tenofovir disoproxil maleate (CI,P) unclassified
D11392  Efavirenz, lamivudine and tenofovir disoproxil fumarate; Symfi (TN) (CI,P) unclassified
D11393  Rituximab and hyaluronidase; Rituxan hycela (TN) (CI,P) unclassified
D11395  Lamivudine and tenofovir disoproxil; Cimduo (TN); Temixys (TN) (CI,P) unclassified
D11396  Doravirine, lamivudine and tenofovir disoproxil; Delstrigo (TN) (CI,P) unclassified
D11400  Abrocitinib (JAN/USAN); Cibinqo (TN) (P) unclassified
D11403  Asciminib (USAN/INN) (CI,P) CYP induction: CYP3A4
D11404  Asciminib hydrochloride (JAN/USAN); Scemblix (TN) (CI,P) CYP induction: CYP3A4
D11406  Risdiplam (JAN/USAN/INN); Evrysdi (TN) (P) CYP induction: CYP3A4
D11416  Naxitamab (USAN); Naxitamab-gqgk; Danyelza (TN) (CI,P) unclassified
D11417  Pemigatinib (JAN/USAN/INN); Pemazyre (TN) (CI,P) CYP induction: CYP3A4
D11422  Zanubrutinib (JAN/USAN/INN); Brukinsa (TN) (CI,P) unclassified
D11426  Pamiparib (USAN/INN) (CI,P) unclassified
D11437  Parsaclisib (USAN/INN) (CI,P) unclassified
D11441  Aprocitentan (USAN/INN); Tryvio (TN) (P) unclassified
D11444  Tazemetostat (USAN/INN) (CI,P) Transporter induction: ABCB1
D11453  Nirogacestat hydrobromide (USAN); Ogsiveo (TN) (P) CYP induction: CYP3A4
D11454  Repotrectinib (JAN/USAN); Augtyro (TN) (P) CYP induction: CYP3A4
D11460  Siponimod (USAN/INN) (P) unclassified
D11463  Mosunetuzumab (USAN/INN); Mosunetuzumab (genetical recombination) (JAN); Mosunetuzumab-axgb; Lunsumio (TN) (CI,P) unclassified
D11485  Tazemetostat hydrobromide (JAN/USAN); Tazverik (TN) (CI,P) Transporter induction: ABCB1
D11487  Tislelizumab (USAN/INN); Tislelizumab (genetical recombination) (JAN); Tislelizumab-jsgr; Tevimbra (TN) (CI,P) unclassified
D11490  Pitolisant hydrochloride (USAN); Wakix (TN) (P) unclassified
D11506  Parsaclisib hydrochloride (JAN/USAN) (CI,P) unclassified
D11521  Lamivudine, nevirapine and zidovudine (CI,P) Enzyme induction: UGT
D11522  Dolutegravir and lamivudine; Dovato (TN) (CI,P) unclassified
D11525  Enfortumab vedotin (USAN); Enfortumab vedotin (genetical recombination) (JAN); Enfortumab vedotin-ejfv; Padcev (TN) (CI,P) unclassified
D11529  Trastuzumab deruxtecan (USAN/INN); Trastuzumab deruxtecan (genetical recombination) (JAN); Fam-trastuzumab deruxtecan-nxki; Enhertu (TN) (CI,P) unclassified
D11541  Sitravatinib malate (USAN) (CI,P) unclassified
D11553  Lidocaine and tetracaine; Pliaglis (TN); Synera (TN) (P) unclassified
D11556  Idecabtagene vicleucel (USAN); Abecma (TN) (CI,P) unclassified
D11560  Trastuzumab and hyaluronidase; Trastuzumab and hyaluronidase-oysk; Herceptin hylecta (TN) (CI,P) unclassified
D11567  Insulin degludec and liraglutide; Xultophy (TN) (P) unclassified
D11572  Beclomethasone dipropionate monohydrate; Beconase aq (TN) (P) CYP induction: CYP3A4
D11573  Oxycodone and ibuprofen (P) CYP induction: CYP3A4
D11576  Naproxen and esomeprazole magnesium; Vimovo (TN) (P) unclassified
D11589  Infigratinib (USAN/INN) (CI,P) unclassified
D11595  Belantamab mafodotin (USAN); Belantamab mafodotin (genetical recombination) (JAN); Belantamab mafodotin-blmf; Blenrep (TN) (CI,P) unclassified
D11601  Tafasitamab (USAN/INN); Tafasitamab (genetical recombination) (JAN); Tafasitamab-cxix; Monjuvi (TN); Minjuvi (TN) (CI,P) unclassified
D11611  Infigratinib phosphate (USAN); Truseltiq (TN) (CI,P) unclassified
D11616  Aspirin and omeprazole; Yosprala (TN) (P) unclassified
D11617  Eletriptan hydrobromide monohydrate (P) CYP induction: CYP3A4
D11619  Desvenlafaxine succinate anhydrous; Desvenlafaxine succinate (TN) (P) Enzyme induction: UGT
D11628  Benzhydrocodone and acetaminophen; Apadaz (TN) (P) CYP induction: CYP3A4
D11631  Lefamulin (USAN/INN) (P) CYP induction: CYP3A4
D11632  Lefamulin acetate (USAN); Xenleta (TN) (P) CYP induction: CYP3A4
D11644  Lurbinectedin (USAN/INN); Zepzelca (TN) (CI,P) unclassified
D11652  Tenapanor (USAN/INN) (P) CYP induction: CYP3A4
D11653  Tenapanor hydrochloride (JAN/USAN); Ibsrela (TN); Phozevel (TN); Xphozah (TN) (P) CYP induction: CYP3A4
D11656  Azelastine hydrochloride and fluticasone propionate; Dymista (TN) (P) CYP induction: CYP3A4
D11658  Duvelisib hydrate (JAN); Copiktra (TN) (CI,P) unclassified
D11659  Tolvaptan sodium phosphate (JAN); Samtasu (TN) (P) unclassified
D11661  Bendamustine hydrochloride hydrate (JAN); Bendamustine hydrochloride monohydrate; Treakisym (TN) (CI,P) unclassified
D11662  Valemetostat tosilate (JAN); Valemetostat tosylate; Ezharmia (TN) (P) unclassified
D11671  Elacestrant (USAN/INN) (P) CYP induction: CYP3A4
D11672  Elacestrant hydrochloride (USAN); Elacestrant dihydrochloride; Orserdu (TN) (P) CYP induction: CYP3A4
D11706  Omeprazole and sodium bicarbonate; Zegerid (TN) (P) unclassified
D11710  Phentermine and topiramate; Qsymia (TN) (P) CYP induction: CYP3A4
D11711  Dapagliflozin, metformin and saxagliptin; Qternmet xr (TN) (P) unclassified
D11712  Pralsetinib (USAN/INN); Gavreto (TN) (CI,P) unclassified
D11713  Selpercatinib (JAN/USAN/INN); Retevmo (TN) (CI,P) CYP induction: CYP3A4
D11717  Tepotinib (USAN/INN) (CI,P) CYP induction: CYP3A4
D11720  Acalabrutinib maleate (USAN) (CI,P) unclassified
D11725  Futibatinib (JAN/USAN/INN); Lytgobi (TN) (CI,P) unclassified
D11768  Pacritinib (USAN/INN); Vonjo (TN) (CI,P) CYP induction: CYP3A4
D11784  Vonoprazan (USAN/INN) (P) CYP induction: CYP3A4
D11785  Oteseconazole (USAN/INN); Vivijoa (TN) (P) unclassified
D11788  Remimazolam (USAN/INN); Byfavo (TN) (P) unclassified
D11793  Zuranolone (JAN/USAN/INN); Zurzuvae (TN) (P) CYP induction: CYP3A4
D11807  Imeglimin hydrochloride (JAN); Twymeeg (TN) (P) unclassified
D11814  Tisotumab vedotin (USAN/INN); Tisotumab vedotin (genetical recombination) (JAN); Tisotumab vedotin-tftv; Tivdak (TN) (CI,P) unclassified
D11827  Retifanlimab (USAN); Retifanlimab-dlwr; Zynyz (TN) (CI,P) unclassified
D11833  Glofitamab (USAN/INN); Glofitamab-gxbm; Columvi (TN) (CI,P) unclassified
D11848  Decitabine and cedazuridine; Inqovi (TN) (CI,P) unclassified
D11851  Butalbital, acetaminophen, caffeine and codeine phosphate (P) unclassified
D11856  Empagliflozin, linagliptin and metformin hydrochloride; Trijardy xr (TN) (P) unclassified
D11860  Butalbital, aspirin, caffeine and codeine; Fiorinal with codeine (TN) (P) CYP induction: CYP3A4
D11865  Melphalan flufenamide (USAN/INN) (CI,P) unclassified
D11870  Melphalan flufenamide hydrochloride (USAN); Pepaxto (TN); Pepaxti (TN) (CI,P) unclassified
D11880  Brexucabtagene autoleucel (USAN); Tecartus (TN) (CI,P) unclassified
D11881  Amlodipine benzoate; Katerzia (TN) (P) CYP induction: CYP3A4
D11885  Surufatinib (USAN/INN) (CI,P) unclassified
D11886  Daridorexant (USAN/INN) (P) CYP induction: CYP3A4
D11887  Daridorexant hydrochloride (JAN/USAN); Quviviq (TN) (P) unclassified
D11894  Amivantamab (USAN/INN); Amivantamab (genetical recombination) (JAN); Amivantamab-vmjw; Rybrevant (TN) (CI,P) unclassified
D11895  Niraparib tosilate hydrate (JAN); Niraparib tosylate monohydrate; Zejula (TN) (CI,P) unclassified
D11913  Oportuzumab monatox (USAN) (CI,P) unclassified
D11923  Lobeglitazone (INN) (P) unclassified
D11924  Beinaglutide (INN) (P) unclassified
D11934  Pertuzumab, trastuzumab and hyaluronidase; Pertuzumab (genetical recombination), trastuzumab (genetical recombination) and vorhyaluronidase alfa (genetical recombination); Pertuzumab, trastuzumab and hyaluronidase-zzxf; Phesgo (TN) (CI,P) unclassified
D11954  Belzutifan (JAN/USAN/INN); Welireg (TN) (CI,P) unclassified
D11967  Daratumumab and hyaluronidase; Daratumumab (genetical recombination) and vorhyaluronidase alfa (genetical recombination); Daratumumab and hyaluronidase-fihj; Darzalex faspro (TN); Darzquro (TN) (CI,P) unclassified
D11968  Teneligliptin hydrobromide (JAN) (P) CYP induction: CYP3A4
D11969  Mobocertinib succinate (JAN); Exkivity (TN) (CI,P) unclassified
D11977  Fruquintinib (JAN/USAN); Fruzaqla (TN) (CI,P) unclassified
D11980  Lazertinib (USAN) (CI,P) unclassified
D11990  Lisocabtagene maraleucel (USAN/INN); Breyanzi (TN) (CI,P) unclassified
D12001  Mobocertinib (USAN/INN) (CI,P) unclassified
D12005  Treprostinil palmitil (USAN/INN) (P) unclassified
D12050  Pirtobrutinib (JAN/USAN); Jaypirca (TN) (CI,P) unclassified
D12055  Sotorasib (JAN/USAN); Lumakras (TN) (CI,P) unclassified
D12130  Drospirenone, ethinyl estradiol and levomefolate calcium; Beyaz (TN); Safyral (TN); Tydemy (TN) (P) CYP induction: CYP3A4
D12160  Orelabrutinib (USAN/INN) (CI,P) unclassified
D12162  Lenacapavir sodium (JAN/USAN); Sunlenca (TN) (CI) Transporter induction: ABCB1
D12164  Sabatolimab (USAN/INN); Sabatolimab (genetical recombination) (JAN) (CI,P) unclassified
D12177  Teclistamab (USAN/INN); Teclistamab (genetical recombination) (JAN); Teclistamab-cqyv; Tecvayli (TN) (CI,P) unclassified
D12180  Talquetamab (USAN/INN); Talquetamab-tgvs; Talvey (TN) (CI,P) unclassified
D12202  Toripalimab (USAN/INN); Toripalimab-tpzi; Loqtorzi (TN) (CI,P) unclassified
D12245  Lazertinib mesilate hydrate (JAN) (CI,P) unclassified
D12258  Aumolertinib (USAN/INN) (CI,P) unclassified
D12259  Aumolertinib mesylate (USAN) (CI,P) unclassified
D12265  Mavacamten (JAN/USAN/INN); Camzyos (TN) (P) unclassified
D12269  Nirmatrelvir and ritonavir; Paxlovid (TN) (CI,P) CYP induction: CYP3A4
D12294  Sitagliptin phosphate (JAN) (P) unclassified
D12296  Tebentafusp (USAN/INN); Tebentafusp-tebn; Kimmtrak (TN) (CI,P) unclassified
D12301  Adagrasib (USAN/INN); Krazati (TN) (CI,P) CYP induction: CYP3A4
D12311  Bortezomib hydrate (JAN) (CI,P) unclassified
D12312  Codeine phosphate and chlorpheniramine maleate; Tuxarin (TN) (P) unclassified
D12313  Chlorpheniramine polistirex and codeine polistirex; Tuzistra (TN) (P) CYP induction: CYP3A4
D12315  Ciltacabtagene autoleucel (USAN/INN); Carvykti (TN); Carvykti (TN) (CI,P) unclassified
D12326  Opelconazole (USAN/INN) (P) unclassified
D12334  Nivolumab and relatlimab; Nivolumab and relatlimab-rmbw; Opdualag (TN) (CI,P) unclassified
D12353  Ensitrelvir fumarate (USAN); Ensitrelvir fumaric acid (JAN); Xocova (TN) (CI,P) unclassified
D12354  Pralsetinib hydrate (JAN) (CI,P) unclassified
D12358  Insulin icodec (USAN/INN); Insulin icodec (genetical recombination) (JAN) (P) unclassified
D12368  Epcoritamab (USAN/INN); Epcoritamab (genetical recombination) (JAN); Epcoritamab-bysp; Epkinly (TN); Tepkinly (TN) (CI,P) unclassified
D12403  Venlafaxine besylate monohydrate; Venlafaxine besylate (TN) (P) unclassified
D12410  Landiolol (USAN/INN) (P) unclassified
D12438  Pitavastatin calcium and ezetimibe; Livazebe (TN) (P) unclassified
D12442  Tucatinib ethanolate (JAN); Tucatinib hemiethanolate (CI,P) unclassified
D12444  Nilotinib hydrochloride dihydrate (JAN) (CI,P) CYP induction: CYP3A4 / Transporter induction: ABCB1
D12483  Olutasidenib (USAN/INN); Rezlidhia (TN) (P) CYP induction: CYP3A4
D12484  Carfloglitazar (INN) (P) unclassified
D12486  Finasteride and tadalafil; Entadfi (TN) (P) CYP induction: CYP3A4
D12497  Drospirenone and estradiol; Angeliq (TN) (P) CYP induction: CYP3A4
D12531  Nadofaragene firadenovec (USAN/INN); Nadofaragene firadenovec-vncg; Adstiladrin (TN) (CI,P) unclassified
D12544  Vortioxetine hemihydrobromide (USAN) (P) unclassified
D12586  Mifepristone and misoprostol; Mefeego (TN) (CI,P) unclassified
D12609  Dasatinib laurylsulfate (USAN) (CI,P) CYP induction: CYP3A4 / Enzyme induction: UGT
D12629  Treprostinil phosphate (USAN); Treprostinil biphosphate (P) unclassified
D12637  Darunavir hydrate (CI,P) CYP induction: CYP3A4
D12653  Niraparib and abiraterone; Akeega (TN) (CI,P) unclassified
D12703  Linagliptin hydrate (JAN); Linagliptin hemihydrate (P) unclassified
D12704  Acalabrutinib maleate hydrate (JAN); Acalabrutinib maleate monohydrate (CI,P) unclassified
D12750  Sugemalimab (INN) (CI,P) unclassified
D12751  Serplulimab (INN) (CI,P) unclassified
D12752  Darunavir propylene glycolate (CI,P) CYP induction: CYP3A4
D12756  Vonoprazan and amoxicillin; Voquezna (TN) (P) CYP induction: CYP3A4
D12816  Dexlansoprazole sesquihydrate (P) CYP induction: CYP3A4
D12833  Lifileucel (USAN/INN); Amtagvi (TN) (CI,P) unclassified
D12854  Nilotinib laurylsulfate (USAN) (CI,P) CYP induction: CYP3A4 / Transporter induction: ABCB1