G Protein-coupled receptors
|
Rhodopsin family
|
Acetylcholine (muscarinic)
|
CHRM [HSA:1128 1129 1131 1132 1133] [KO:K04129 K04130 K04131 K04132 K04133]
|
D08389 Pirenzepine (USAN/INN)
D01297 Pirenzepine hydrochloride (USAN)
D05276 Pirenzepine hydrochloride hydrate (JP18) <JP>
D08160 Mebeverine (INN)
D04868 Mebeverine hydrochloride (USAN)
D07821 Dihexyverine (INN)
D03824 Dihexyverine hydrochloride (USAN)
D07079 Difemerine (INN)
D08382 Piperidolate (INN)
D01165 Piperidolate hydrochloride (JAN) <JP>
D03088 Benzilonium bromide (USAN/INN)
D07081 Penthienate bromide (NF XIII)
D00481 Propantheline bromide (JP18/USP/INN) <JP>
D07083 Otilonium bromide (INN)
D00721 Methanthelinium bromide (INN)
D05535 Poldine methylsulfate (USAN)
D00720 Mepenzolate bromide (JP18/INN) <JP>
D01532 Bevonium methylsulfate (JAN)
D07084 Pipenzolate bromide (INN)
D01201 Tiemonium iodide (JAN/INN)
D01377 Prifinium bromide (JAN/INN)
D02535 Timepidium bromide hydrate (JP18) <JP>
D07070 Fenpiverinium bromide (INN)
D01538 Valethamate bromide (JAN)
D00113 Atropine (USP) <US>
D02069 Atropine sulfate (JP18/USP) <JP/US>
D00147 Hyoscyamine (USP)
D00719 Hyoscyamine sulfate (USP)
D01648 Hyoscyamine methylbromide (JAN)
D04479 Hyoscyamine hydrobromide (USP)
D01451 Scopolamine butylbromide (JP18) <JP>
D01077 Methylatropine nitrate (USAN)
D03814 Atropine methylbromide (JAN)
D01976 N-Methylscopolamine methylsulfate (JAN)
D07951 Fentonium bromide (INN)
D07099 Cimetropium bromide (JAN/INN)
D02070 Homatropine methylbromide (USP)
D00138 Scopolamine (INN) <US>
D02071 Scopolamine hydrobromide (USP)
D10939 Glycopyrronium tosylate (USAN) <JP/US>
D00465 Oxybutynin (USAN/INN) <US>
D00722 Oxybutynin chloride (USP) <JP/US>
D08441 Propiverine (INN)
D01007 Propiverine hydrochloride (JP18) <JP>
D00765 Rocuronium bromide (JAN/USP/INN) <JP/US>
D08418 Pridinol (INN)
D02064 Pridinol mesilate (JAN) <JP>
D08419 Pridinol hydrochloride
D08638 Trihexyphenidyl (INN)
D00787 Trihexyphenidyl hydrochloride (JP18/USP) <JP/US>
D00779 Biperiden (JAN/USP/INN)
D02246 Biperiden hydrochloride (JP18/USP) <JP>
D02247 Biperiden lactate (JAN/USP) <JP>
D08209 Metixene (INN)
D01871 Methixene hydrochloride (USAN)
D08425 Procyclidine (INN)
D00782 Procyclidine hydrochloride (USP)
D08426 Profenamine (INN)
D01118 Profenamine hydrochloride (JAN)
D03276 Profenamine hibenzate (JAN)
D03711 Dexetimide (USAN/INN)
D07804 Dexetimide hydrochloride
D07301 Phenglutarimide (INN)
D08157 Mazaticol (INN)
D03264 Mazaticol hydrochloride hydrate (JAN)
D07302 Bornaprine (INN)
D07303 Tropatepine (INN)
D08653 Tropatepine hydrochloride
D07511 Benzatropine (INN)
D00778 Benztropine mesylate (USP) <US>
D04087 Ethybenztropine (USAN)
D00270 Chlorpromazine (USP/INN)
D00789 Chlorpromazine hydrochloride (JP18/USP) <JP/US>
D03274 Chlorpromazine hibenzate (JAN)
D04034 Chlorpromazine phenolphthalinate (JAN) <JP>
D09819 Chlorpromazine tannate (JAN)
D11383 Blarcamesine (USAN/INN)
D11549 Blarcamesine hydrochloride (USAN)
D00524 Carbachol (JAN/USP/INN) <US>
D01000 Bethanechol chloride (JP18/USP) <JP/US>
D07349 Choline alfoscerate (INN)
D02212 Ipratropium bromide (USP) <JP/US>
D01946 Oxitropium bromide (JAN/INN)
D08837 Aclidinium bromide (JAN/USAN/INN) <JP/US>
D10181 Umeclidinium bromide (JAN/USAN) <JP/US>
D00999 Acetylcholine chloride (JP18/USP/INN) <JP/US>
D07759 Cyclopentolate (INN)
D01002 Cyclopentolate hydrochloride (JP18/USP) <JP/US>
D01004 Homatropine hydrobromide (JP18/USP)
D00397 Tropicamide (JP18/USP/INN) <JP/US>
D04970 Methacholine chloride (JAN/USP/INN) <JP/US>
D00232 Anisotropine methylbromide (USAN)
D00715 Methscopolamine bromide (USP) <US>
D00716 Clidinium bromide (USP/INN)
D01175 Carpronium chloride (JAN/INN) <JP>
D01231 Piroheptine hydrochloride (JAN) <JP>
D01315 Methylbenactyzium bromide (JP18/INN)
D01318 Diphenidol hydrochloride (USAN) <JP>
D01359 Etomidoline (JAN/INN)
D01463 Diponium bromide (JAN/INN)
D01491 Butropium bromide (JP18/INN)
D01521 Pipethanate hydrochloride (JAN)
D01600 Diphenylpiperidinomethyldioxolan iodide (JAN)
D01815 Oxapium iodide (JP18/INN)
D01955 Aclatonium napadisilate (JAN)
D01987 Pipethanate ethobromide (JAN)
D02417 Flutropium bromide (JAN)
D02603 Diethazine hydrochloride
D03011 Atropine oxide hydrochloride (USAN)
D03076 Benapryzine hydrochloride (USAN)
D03087 Benzetimide hydrochloride (USAN)
D03858 Diphenidol (USAN/INN)
D03859 Diphenidol pamoate (USAN)
D03970 Elantrine (USAN)
D03979 Elucaine (USAN)
D04116 Eucatropine hydrochloride (USP XXXII)
D04434 Heteronium bromide (USAN/INN)
D05012 Metoquizine (USAN/INN)
D05035 Milameline hydrochloride (USAN)
D05360 Parapenzolate bromide (USAN/INN)
D05418 Pentapiperium methylsulfate (USAN)
D05452 Phencarbamide (USAN)
D05628 Propenzolate hydrochloride (USAN)
D05703 Rapacuronium bromide (USAN/INN)
D06015 Tazomeline citrate (USAN)
D06061 Tematropium methylsulfate (USAN)
D06175 Tofenacin hydrochloride (USAN)
D06192 Toquizine (USAN)
D06217 Triampyzine sulfate (USAN)
D07477 Atropine oxide (INN)
D07513 Benzetimide (INN)
D07823 Diethazine (INN)
D08384 Pipethanate (INN)
D08395 Piroheptine (INN)
D08595 Tiemonium methylsulfate
D09402 Darotropium bromide (USAN/INN)
D09752 Carpronium chloride hydrate (JAN) <JP>
D10180 Umeclidinium (USAN)
D10545 Batefenterol (USAN)
D10546 Batefenterol succinate (USAN)
|
CHRM1 [HSA:1128] [KO:K04129]
|
D08325 Oxyphencyclimine (INN)
D01006 Oxyphencyclimine hydrochloride (JAN)
D07820 Dicycloverine (INN)
D00717 Dicyclomine hydrochloride (JAN/USP) <US>
D06877 Oxyphenonium bromide (INN)
D00723 Tridihexethyl chloride (BAN)
D06273 Imidafenacin (JAN/INN) <JP>
D02750 Aceclidine (USAN/INN)
D13152 Aceclidine hydrochloride <US>
D02876 Alvameline maleate (USAN)
D04057 Esoxybutynin chloride (USAN)
D05779 Sabcomeline hydrochloride (USAN)
D06000 Talsaclidine fumarate (USAN)
D06330 Xanomeline (USAN)
D06331 Xanomeline tartrate (USAN)
D11098 Telenzepine hydrochloride hydrate (JAN)
|
CHRM2 [HSA:1129] [KO:K04130]
|
D08325 Oxyphencyclimine (INN)
D01006 Oxyphencyclimine hydrochloride (JAN)
D07820 Dicycloverine (INN)
D00717 Dicyclomine hydrochloride (JAN/USP) <US>
D00723 Tridihexethyl chloride (BAN)
D07853 Dimetindene (INN)
D01103 Trospium chloride (JAN/USP/INN) <US>
D07226 Fesoterodine (INN)
D08923 Fesoterodine fumarate (JAN/USAN) <JP/US>
D02292 Gallamine triethiodide (USP)
D00525 Pilocarpine (JAN/USP)
D02200 Pilocarpine hydrochloride (JP18/USP) <JP/US>
D05478 Pilocarpine nitrate (USP)
D08376 Pilocarpine borate
D02876 Alvameline maleate (USAN)
D04057 Esoxybutynin chloride (USAN)
|
CHRM3 [HSA:1131] [KO:K04131]
|
D08325 Oxyphencyclimine (INN)
D01006 Oxyphencyclimine hydrochloride (JAN)
D07078 Rociverine (INN)
D07820 Dicycloverine (INN)
D00717 Dicyclomine hydrochloride (JAN/USP) <US>
D00540 Glycopyrrolate (USP) <JP/US>
D00723 Tridihexethyl chloride (BAN)
D01005 Isopropamide iodide (JAN/USP/INN)
D01003 Hexocyclium metilsulfate (INN)
D06878 Diphemanil metilsulfate (INN)
D00193 Dexpanthenol (USP/INN) <JP>
D10938 Glycopyrronium (USAN)
D10989 Sofpironium bromide (JAN/USAN/INN) <JP/US>
D00646 Tolterodine (USAN/INN)
D01148 Tolterodine tartrate (JAN/USP) <US>
D08522 Solifenacin (INN)
D01269 Solifenacin succinate (JAN/USAN/INN) <JP/US>
D01103 Trospium chloride (JAN/USP/INN) <US>
D03654 Darifenacin (USAN/INN)
D01699 Darifenacin hydrobromide (JAN/USAN) <US>
D07226 Fesoterodine (INN)
D08923 Fesoterodine fumarate (JAN/USAN) <JP/US>
D10853 Desfesoterodine (INN)
D06273 Imidafenacin (JAN/INN) <JP>
D00525 Pilocarpine (JAN/USP)
D02200 Pilocarpine hydrochloride (JP18/USP) <JP/US>
D05478 Pilocarpine nitrate (USP)
D08376 Pilocarpine borate
D07667 Cevimeline (INN)
D00661 Cevimeline hydrochloride (USAN) <JP/US>
D01929 Tiotropium bromide hydrate (JAN) <JP/US>
D10978 Revefenacin (USAN/INN) <US>
D01875 Tiquizium bromide (JAN/INN) <JP>
D02876 Alvameline maleate (USAN)
D04057 Esoxybutynin chloride (USAN)
D11900 Navafenterol (USAN)
D11901 Navafenterol saccharinate (USAN)
|
CHRM4 [HSA:1132] [KO:K04132]
|
D06330 Xanomeline (USAN)
D06331 Xanomeline tartrate (USAN)
D12468 Emraclidine (USAN/INN)
D13221 Direclidine (USAN/INN)
D13222 Direclidine citrate (USAN)
|
Adrenaline
|
ADRA1 [HSA:148 147 146] [KO:K04135 K04136 K04137]
|
D00095 Epinephrine (USP/INN) <JP/US>
D00996 Epinephrine hydrochloride (JAN)
D02149 Epinephrine bitartrate (USP) <US>
D02774 Adrenalone (USAN/INN)
D07560 Adrenalone hydrochloride
D02910 Amiodarone (USAN/INN)
D00636 Amiodarone hydrochloride (JP18/USP) <JP/US>
D02537 Dronedarone (INN)
D03914 Dronedarone hydrochloride (USP) <US>
D07931 Etilefrine (INN)
D01573 Etilefrine hydrochloride (JP18) <JP>
D00076 Noradrenaline (JP18) <JP>
D05206 Norepinephrine bitartrate (USP) <US>
D08284 Norepinephrine hydrochoride
D09794 Norepinephrine hydrochloride (JAN)
D08286 Norfenefrine (INN)
D01405 Norfenefrine hydrochloride (JAN)
D08365 Phenylephrine (INN)
D00511 Phenylephrine hydrochloride (JP18/USP) <JP/US>
D08366 Phenylephrine tartrate
D08966 Phenylephrine bitartrate (USP)
D08192 Metaraminol (INN)
D01019 Metaraminol bitartrate (JAN/USP)
D08201 Methoxamine (BAN)
D01020 Methoxamine hydrochloride (JAN)
D08220 Midodrine (INN)
D01307 Midodrine hydrochloride (JAN/USP) <JP/US>
D00124 Ephedrine (USP)
D01386 Ephedrine hydrochloride (JP18/USP) <JP>
D04018 Ephedrine sulfate (USP) <US>
D01277 Droxidopa (JP18/USAN/INN) <JP/US>
D08411 Prazosin (INN)
D00609 Prazosin hydrochloride (JP18/USP) <JP/US>
D04531 Indoramin (USAN/INN)
D04532 Indoramin hydrochloride (USAN)
D08212 Trimazosin (INN)
D06234 Trimazosin hydrochloride (USAN)
D07874 Doxazosin (INN)
D00608 Doxazosin mesylate (USP) <JP/US>
D01333 Urapidil (JP18/INN) <JP>
D08662 Urapidil hydrochloride
D08362 Phentolamine (INN)
D00509 Phentolamine mesylate (USP) <JP/US>
D08614 Tolazoline (INN)
D00997 Tolazoline hydrochloride (JAN/USP)
D02268 Ergoloid mesylates (USP)
D01290 Nicergoline (JP18/USAN/INN) <JP>
D08271 Nicergoline tartrate
D07834 Dihydroergocristine (BAN)
D07833 Dihydroergocristine mesilate (BAN)
D08358 Phenoxybenzamine (INN)
D00507 Phenoxybenzamine hydrochloride (USP) <US>
D08239 Moxisylyte (INN)
D01571 Moxisylyte hydrochloride (JAN)
D08064 Ifenprodil (INN)
D01445 Ifenprodil tartrate (JP18) <JP>
D01369 Bevantolol hydrochloride (JAN/USAN) <JP>
D08106 Labetalol (INN)
D00600 Labetalol hydrochloride (JP18/USP) <JP/US>
D00255 Carvedilol (JP18/USP/INN) <JP/US>
D03415 Carvedilol phosphate (USAN) <US>
D08207 Methylergometrine (INN)
D00680 Methylergonovine maleate (USP) <JP/US>
D07906 Ergotamine (INN)
D07905 Ergometrine (INN)
D01163 Ergonovine maleate (USP)
D08560 Tamsulosin (INN)
D01024 Tamsulosin hydrochloride (JP18/USP) <JP/US>
D08569 Terazosin (INN)
D00610 Terazosin hydrochloride (USP) <JP/US>
D11585 Terazosin hydrochloride anhydrous <US>
D00679 Ergotamine tartrate (JP18/USP) <US>
D01485 Propericiazine (JAN) <JP>
D00308 Droperidol (JP18/USP/INN) <JP/US>
D00454 Olanzapine (JAN/USP/INN) <JP/US>
D06623 Olanzapine pamoate (USAN) <US>
D08257 Nefazodone (INN)
D00819 Nefazodone hydrochloride (USP) <US>
D08578 Tetryzoline (INN)
D00756 Tetrahydrozoline nitrate (JAN)
D01023 Tetrahydrozoline hydrochloride (JAN/USP)
D08684 Xylometazoline (INN)
D00757 Xylometazoline hydrochloride (USP)
D08253 Naphazoline (INN)
D00743 Naphazoline hydrochloride (JP18/USP)
D01021 Naphazoline nitrate (JP18) <JP>
D08624 Tramazoline (INN)
D01347 Tramazoline hydrochloride (JAN/USAN) <JP>
D08368 Phenylpropanolamine (INN)
D01224 Phenylpropanolamine hydrochloride (JAN/USP)
D05466 Phenylpropanolamine polistirex (USAN)
D08449 Pseudoephedrine (INN)
D00485 Pseudoephedrine hydrochloride (USP)
D05648 Pseudoephedrine polistirex (USAN)
D05649 Pseudoephedrine sulfate (USP)
D02349 Dipivefrin (USAN)
D01017 Dipivefrin hydrochloride (USP)
D08115 Levobunolol (INN)
D01025 Levobunolol hydrochloride (JAN/USP) <JP/US>
D07775 Dapiprazole (INN)
D03648 Dapiprazole hydrochloride (USAN) <US>
D00607 Guanadrel sulfate (USAN)
D01171 Monatepil maleate (JAN/USAN)
D01444 Bunitrolol hydrochloride (JAN)
D01469 Amosulalol hydrochloride (JP18) <JP>
D01674 Naftopidil (JP18/INN) <JP>
D01691 Nipradilol (JAN/INN) <JP>
D01830 Arotinolol hydrochloride (JP18) <JP>
D01887 Bunazosin hydrochloride (JP18) <JP>
D01952 L-Methylephedrine hydrochloride (JAN)
D02109 dl-Methylephedrine hydrochloride (JP18) <JP>
D02568 Flesinoxan (INN)
D02901 Amidephrine mesylate (USAN)
D03887 Domazoline fumarate (USAN)
D04026 Epinephryl borate (USP)
D05228 Octodrine (USAN/INN)
D05395 Pelanserin hydrochloride (USAN)
D05637 Propylhexedrine (USP/INN)
D05688 Racepinephrine (USP/INN)
D05689 Racepinephrine hydrochloride (USP)
D07451 Amosulalol (INN)
D07465 Arotinolol (INN)
D07550 Bunazosin (INN)
D08029 Guanadrel (INN)
D08206 Methylephedrine (BAN)
D08444 Propylhexedrine hydrochloride
D08982 Racephedrine hydrochloride (USAN)
D09842 dl-Methylephedrine saccharinate (JAN)
D12934 Dibutepinephrine (USAN/INN)
D12935 Dibutepinephrine hydrochloride (USAN)
|
ADRA1A [HSA:148] [KO:K04135]
|
D07097 Isometheptene mucate (USP)
D08322 Oxymetazoline (INN)
D01022 Oxymetazoline hydrochloride (JAN/USP) <US>
D07124 Alfuzosin (INN)
D01692 Alfuzosin hydrochloride (JAN/USAN) <US>
D01965 Silodosin (JP18/INN) <JP/US>
D04184 Fiduxosin hydrochloride (USAN)
D06380 Zolertine hydrochloride (USAN)
D06394 Dabuzalgron hydrochloride (USAN)
D09784 Garomefrine hydrochloride (JAN)
|
ADRA1D [HSA:146] [KO:K04137]
|
D06380 Zolertine hydrochloride (USAN)
|
ADRA2 [HSA:150 151 152] [KO:K04138 K04139 K04140]
|
D00095 Epinephrine (USP/INN) <JP/US>
D00996 Epinephrine hydrochloride (JAN)
D02149 Epinephrine bitartrate (USP) <US>
D07931 Etilefrine (INN)
D01573 Etilefrine hydrochloride (JP18) <JP>
D00076 Noradrenaline (JP18) <JP>
D05206 Norepinephrine bitartrate (USP) <US>
D08284 Norepinephrine hydrochoride
D09794 Norepinephrine hydrochloride (JAN)
D08192 Metaraminol (INN)
D01019 Metaraminol bitartrate (JAN/USP)
D00124 Ephedrine (USP)
D01386 Ephedrine hydrochloride (JP18/USP) <JP>
D04018 Ephedrine sulfate (USP) <US>
D01277 Droxidopa (JP18/USAN/INN) <JP/US>
D08205 Methyldopa (INN)
D00405 Methyldopa (USP) <JP/US>
D00281 Clonidine (JAN/USP/INN) <US>
D00604 Clonidine hydrochloride (JP18/USP) <JP/US>
D05087 Moxonidine (USAN/INN)
D08482 Rilmenidine (INN)
D01603 Bethanidine sulfate (JAN/USAN)
D08362 Phentolamine (INN)
D00509 Phentolamine mesylate (USP) <JP/US>
D08614 Tolazoline (INN)
D00997 Tolazoline hydrochloride (JAN/USP)
D02268 Ergoloid mesylates (USP)
D07834 Dihydroergocristine (BAN)
D07833 Dihydroergocristine mesilate (BAN)
D08358 Phenoxybenzamine (INN)
D00507 Phenoxybenzamine hydrochloride (USP) <US>
D07540 Brimonidine (INN)
D02076 Brimonidine tartrate (JAN/USAN) <JP/US>
D08207 Methylergometrine (INN)
D00680 Methylergonovine maleate (USP) <JP/US>
D07905 Ergometrine (INN)
D01163 Ergonovine maleate (USP)
D08685 Yohimbine (DCF)
D06671 Yohimbine hydrochloride (USP)
D08611 Tizanidine (INN)
D00776 Tizanidine hydrochloride (JP18/USP) <JP/US>
D00270 Chlorpromazine (USP/INN)
D00789 Chlorpromazine hydrochloride (JP18/USP) <JP/US>
D03274 Chlorpromazine hibenzate (JAN)
D04034 Chlorpromazine phenolphthalinate (JAN) <JP>
D09819 Chlorpromazine tannate (JAN)
D00283 Clozapine (JAN/USP/INN) <JP/US>
D00514 Dexmedetomidine (USAN/INN)
D01205 Dexmedetomidine hydrochloride (JAN/USP) <JP/US>
D08216 Mianserin (INN)
D01358 Mianserin hydrochloride (JAN/USAN) <JP>
D00563 Mirtazapine (JAN/USP/INN) <JP/US>
D11056 Mirtazapine hydrate (JAN)
D08141 Lofexidine (INN)
D04765 Lofexidine hydrochloride (USAN) <US>
D08684 Xylometazoline (INN)
D00757 Xylometazoline hydrochloride (USP)
D08624 Tramazoline (INN)
D01347 Tramazoline hydrochloride (JAN/USAN) <JP>
D08368 Phenylpropanolamine (INN)
D01224 Phenylpropanolamine hydrochloride (JAN/USP)
D05466 Phenylpropanolamine polistirex (USAN)
D08449 Pseudoephedrine (INN)
D00485 Pseudoephedrine hydrochloride (USP)
D05648 Pseudoephedrine polistirex (USAN)
D05649 Pseudoephedrine sulfate (USP)
D02349 Dipivefrin (USAN)
D01017 Dipivefrin hydrochloride (USP)
D07461 Apraclonidine (INN)
D01008 Apraclonidine hydrochloride (JAN/USP) <JP/US>
D00605 Guanabenz acetate (JP18/USP) <JP>
D00607 Guanadrel sulfate (USAN)
D01952 L-Methylephedrine hydrochloride (JAN)
D02034 Setiptiline maleate (JAN) <JP>
D02109 dl-Methylephedrine hydrochloride (JP18) <JP>
D02388 Levonordefrin (USP)
D02407 Lidamidine hydrochloride (USAN)
D02569 Sunepitron hydrochloride (USAN)
D02972 Aptazapine maleate (USAN)
D03002 Atipamezole (USAN/INN)
D03672 Delequamine hydrochloride (USAN)
D03702 Detomidine hydrochloride (USAN)
D03887 Domazoline fumarate (USAN)
D04026 Epinephryl borate (USP)
D04124 Fadolmidine hydrochloride (USAN)
D04223 Fluparoxan hydrochloride (USAN)
D04375 Guanabenz (USAN/INN)
D04883 Medetomidine hydrochloride (USAN)
D05119 Napamezole hydrochloride (USAN)
D05228 Octodrine (USAN/INN)
D05637 Propylhexedrine (USP/INN)
D05688 Racepinephrine (USP/INN)
D05689 Racepinephrine hydrochloride (USP)
D06344 Xylazine hydrochloride (USP)
D07795 Detomidine (INN)
D08029 Guanadrel (INN)
D08126 Lidamidine (INN)
D08165 Medetomidine (INN)
D08206 Methylephedrine (BAN)
D08444 Propylhexedrine hydrochloride
D08487 Romifidine (INN)
D08511 Setiptiline (INN)
D08683 Xylazine (USP/INN)
D08982 Racephedrine hydrochloride (USAN)
D09842 dl-Methylephedrine saccharinate (JAN)
D11320 Vatinoxan (USAN)
D11321 Vatinoxan hydrochloride (USAN)
D12934 Dibutepinephrine (USAN/INN)
D12935 Dibutepinephrine hydrochloride (USAN)
|
ADRA2A [HSA:150] [KO:K04138]
|
D08031 Guanfacine (INN)
D00606 Guanfacine hydrochloride (JAN/USP) <JP/US>
D00560 Pimozide (JP18/USP/INN) <US>
|
ADRA2B [HSA:151] [KO:K04139]
|
D04514 Imiloxan hydrochloride (USAN)
|
ADRB [HSA:153 154 155] [KO:K04141 K04142 K04143]
|
D00095 Epinephrine (USP/INN) <JP/US>
D00996 Epinephrine hydrochloride (JAN)
D02149 Epinephrine bitartrate (USP) <US>
D07931 Etilefrine (INN)
D01573 Etilefrine hydrochloride (JP18) <JP>
D08090 Isoprenaline (INN)
D01390 Isoproterenol hydrochloride (USP) <JP/US>
D02066 Isoproterenol sulfate (USP)
D02150 l-Isoprenaline hydrochloride (JP18) <JP>
D00076 Noradrenaline (JP18) <JP>
D05206 Norepinephrine bitartrate (USP) <US>
D08284 Norepinephrine hydrochoride
D09794 Norepinephrine hydrochloride (JAN)
D02976 Arbutamine hydrochloride (USAN)
D00124 Ephedrine (USP)
D01386 Ephedrine hydrochloride (JP18/USP) <JP>
D04018 Ephedrine sulfate (USP) <US>
D01277 Droxidopa (JP18/USAN/INN) <JP/US>
D07156 Alprenolol (INN)
D01182 Alprenolol hydrochloride (JP18/USAN)
D08318 Oxprenolol (INN)
D01806 Oxprenolol hydrochloride (JP18/USP)
D00513 Pindolol (JP18/USP/INN) <US>
D08443 Propranolol (INN)
D00483 Propranolol hydrochloride (JP18/USP) <JP/US>
D07181 Mepindolol (INN)
D07624 Carteolol (INN)
D00599 Carteolol hydrochloride (JP18/USP) <JP/US>
D07182 Tertatolol (INN)
D08572 Tertatolol hydrochloride
D07537 Bopindolol (INN)
D01794 Bopindolol malonate (JAN)
D07590 Bupranolol (INN)
D01454 Bupranolol hydrochloride (JP18)
D08074 Penbutolol (INN)
D00602 Penbutolol sulfate (JP18/USP)
D07183 Cloranolol (INN)
D07184 Talinolol (INN)
D08368 Phenylpropanolamine (INN)
D01224 Phenylpropanolamine hydrochloride (JAN/USP)
D05466 Phenylpropanolamine polistirex (USAN)
D08449 Pseudoephedrine (INN)
D00485 Pseudoephedrine hydrochloride (USP)
D05648 Pseudoephedrine polistirex (USAN)
D05649 Pseudoephedrine sulfate (USP)
D02349 Dipivefrin (USAN)
D01017 Dipivefrin hydrochloride (USP)
D08115 Levobunolol (INN)
D01025 Levobunolol hydrochloride (JAN/USP) <JP/US>
D02374 Metipranolol (USAN/INN)
D02081 Metipranolol hydrochloride
D07496 Befunolol (INN)
D01512 Befunolol hydrochloride (JAN)
D01444 Bunitrolol hydrochloride (JAN)
D01504 Bufetolol hydrochloride (JP18)
D01691 Nipradilol (JAN/INN) <JP>
D01795 Tilisolol hydrochloride (JAN)
D01906 Dilevalol hydrochloride (JAN/USAN)
D01952 L-Methylephedrine hydrochloride (JAN)
D02109 dl-Methylephedrine hydrochloride (JP18) <JP>
D02765 Adaprolol maleate (USAN)
D02834 Alprenoxime hydrochloride (USAN)
D03502 Cimaterol (USAN/INN)
D03729 Dexpropranolol hydrochloride (USAN)
D03759 Diacetolol hydrochloride (USAN)
D04026 Epinephryl borate (USP)
D04120 Exaprolol hydrochloride (USAN)
D04190 Flestolol sulfate (USAN)
D04888 Medroxalol (USAN/INN)
D04889 Medroxalol hydrochloride (USAN)
D05228 Octodrine (USAN/INN)
D05345 Pamatolol sulfate (USAN)
D05688 Racepinephrine (USP/INN)
D05689 Racepinephrine hydrochloride (USP)
D06014 Tazolol hydrochloride (USAN)
D06162 Tiprenolol hydrochloride (USAN)
D06176 Tolamolol (USAN/INN)
D08206 Methylephedrine (BAN)
D08598 Tilisolol (INN)
D08982 Racephedrine hydrochloride (USAN)
D09842 dl-Methylephedrine saccharinate (JAN)
D09843 Beradilol monoethyl maleate (JAN)
D12934 Dibutepinephrine (USAN/INN)
D12935 Dibutepinephrine hydrochloride (USAN)
|
ADRB1 [HSA:153] [KO:K04141]
|
D02910 Amiodarone (USAN/INN)
D00636 Amiodarone hydrochloride (JP18/USP) <JP/US>
D02537 Dronedarone (INN)
D03914 Dronedarone hydrochloride (USP) <US>
D03879 Dobutamine (USAN/INN)
D00632 Dobutamine hydrochloride (JP18/USP) <JP/US>
D03880 Dobutamine lactobionate (USAN)
D03881 Dobutamine tartrate (USAN)
D06328 Xamoterol (USAN)
D06329 Xamoterol fumarate (USAN)
D08600 Timolol (INN)
D00378 Timolol (USAN) <US>
D00603 Timolol maleate (JP18/USP) <JP/US>
D08525 Sotalol (INN)
D01026 Sotalol hydrochloride (JAN/USP) <JP/US>
D00432 Nadolol (JP18/USP/INN) <JP/US>
D05587 Practolol (USAN)
D02358 Metoprolol (USAN/INN)
D00601 Metoprolol tartrate (JP18/USP) <JP/US>
D00635 Metoprolol succinate (USP) <US>
D05011 Metoprolol fumarate (USP)
D00235 Atenolol (JP18/USP/INN) <JP/US>
D02338 Acebutolol (USAN/INN)
D00597 Acebutolol hydrochloride (JP18/USP) <US>
D07526 Betaxolol (INN)
D00598 Betaxolol hydrochloride (JP18/USP) <JP/US>
D01369 Bevantolol hydrochloride (JAN/USAN) <JP>
D02342 Bisoprolol (JAN/USAN/INN) <JP>
D00634 Bisoprolol fumarate (JP18/USP) <JP/US>
D07660 Celiprolol (INN)
D01741 Celiprolol hydrochloride (JAN/USAN) <JP>
D07916 Esmolol (INN)
D00644 Esmolol hydrochloride (JAN/USP) <JP/US>
D06646 Epanolol (USAN/INN)
D01471 Esatenolol (JAN/INN)
D05127 Nebivolol (USAN/INN)
D06622 Nebivolol hydrochloride (USAN) <US>
D01847 Landiolol hydrochloride (JAN/USAN) <JP/US>
D12410 Landiolol (USAN/INN)
D08106 Labetalol (INN)
D00600 Labetalol hydrochloride (JP18/USP) <JP/US>
D00255 Carvedilol (JP18/USP/INN) <JP/US>
D03415 Carvedilol phosphate (USAN) <US>
D01469 Amosulalol hydrochloride (JP18) <JP>
D01492 Bucumolol hydrochloride (JP18)
D01830 Arotinolol hydrochloride (JP18) <JP>
D01903 Docarpamine (JAN/INN) <JP>
D01958 Indenolol hydrochloride (JP18)
D02389 Primidolol (USAN/INN)
D02614 Denopamine (JAN/INN) <JP>
D03177 Bunolol hydrochloride (USAN)
D03195 Butopamine (USAN/INN)
D03449 Cetamolol hydrochloride (USAN)
D03490 Cicloprolol hydrochloride (USAN)
D04708 Levdobutamine lactobionate (USAN)
D04710 Levobetaxolol hydrochloride (USAN)
D07451 Amosulalol (INN)
D07465 Arotinolol (INN)
D08078 Indenolol (INN)
|
ADRB2 [HSA:154] [KO:K04142]
|
D03891 Dopexamine (USAN/INN)
D03892 Dopexamine hydrochloride (USAN)
D08092 Isoxsuprine (INN)
D01748 Isoxsuprine hydrochloride (JP18/USP) <JP>
D08093 Isoxsuprine lactate
D08600 Timolol (INN)
D00378 Timolol (USAN) <US>
D00603 Timolol maleate (JP18/USP) <JP/US>
D08525 Sotalol (INN)
D01026 Sotalol hydrochloride (JAN/USP) <JP/US>
D00432 Nadolol (JP18/USP/INN) <JP/US>
D08106 Labetalol (INN)
D00600 Labetalol hydrochloride (JP18/USP) <JP/US>
D00255 Carvedilol (JP18/USP/INN) <JP/US>
D03415 Carvedilol phosphate (USAN) <US>
D02359 Ritodrine (USAN/INN)
D01263 Ritodrine hydrochloride (JP18/USP) <JP>
D04157 Fenoterol (USAN/INN)
D01428 Fenoterol hydrobromide (JAN) <JP>
D08300 Orciprenaline (INN)
D00685 Metaproterenol sulfate (USP)
D04954 Metaproterenol polistirex (USAN)
D02147 Albuterol (USP)
D00683 Albuterol sulfate (USP) <JP/US>
D08570 Terbutaline (INN)
D00688 Terbutaline sulfate (JP18/USP) <JP/US>
D05730 Rimiterol hydrobromide (USAN)
D08039 Hexoprenaline (INN)
D02396 Hexoprenaline sulfate (USAN)
D04625 Isoetharine (USP)
D02093 Isoetharine hydrochloride (USP)
D04626 Isoetharine mesylate (USP)
D08387 Pirbuterol (INN)
D00686 Pirbuterol acetate (USAN)
D01349 Pirbuterol hydrochloride (JAN/USAN)
D08629 Tretoquinol (INN)
D01978 Trimetoquinol hydrochloride
D05037 Trimetoquinol hydrochloride hydrate (JP18) <JP>
D03402 Carbuterol hydrochloride (USAN)
D02151 Tulobuterol (JP18/INN) <JP>
D01362 Tulobuterol hydrochloride (JP18) <JP>
D05792 Salmeterol (USAN/INN)
D00687 Salmeterol xinafoate (JAN/USP) <JP/US>
D07990 Formoterol (INN)
D01373 Formoterol fumarate (USP) <US>
D05277 Formoterol fumarate hydrate (JP18) <JP/US>
D07713 Clenbuterol (INN)
D01360 Clenbuterol hydrochloride (JAN/USP) <JP>
D08474 Reproterol (INN)
D05718 Reproterol hydrochloride (USAN)
D08424 Procaterol (INN)
D02404 Procaterol hydrochloride (USAN)
D05366 Procaterol hydrochloride hydrate (JP18) <JP>
D07534 Bitolterol (INN)
D00684 Bitolterol mesylate (USAN)
D09318 Indacaterol (USAN/INN)
D09319 Indacaterol maleate (JAN/USAN) <JP>
D11009 Indacaterol acetate (JAN)
D10145 Olodaterol (USAN/INN)
D10020 Olodaterol hydrochloride (JAN/USAN) <US>
D01635 Methoxyphenamine hydrochloride (JAN)
D07377 Bambuterol (INN)
D07489 Bambuterol hydrochloride
D01469 Amosulalol hydrochloride (JP18) <JP>
D01492 Bucumolol hydrochloride (JP18)
D01589 Mabuterol hydrochloride (JAN)
D01830 Arotinolol hydrochloride (JP18) <JP>
D01835 Clorprenaline hydrochloride (JAN/USAN)
D01958 Indenolol hydrochloride (JP18)
D02281 Levalbuterol hydrochloride (USP) <US>
D02981 Arformoterol tartrate (USAN) <US>
D03170 Bucindolol hydrochloride (USAN)
D03177 Bunolol hydrochloride (USAN)
D03198 Butoxamine hydrochloride (USAN)
D03587 Colterol mesylate (USAN)
D04072 Etafedrine hydrochloride (USAN)
D04701 Levalbuterol sulfate (USAN)
D04703 Levalbuterol tartrate (USAN) <US>
D04953 Metalol hydrochloride (USAN)
D05476 Picumeterol fumarate (USAN)
D05691 Ractopamine hydrochloride (USP)
D05832 Sibenadet hydrochloride (USAN)
D05902 Soterenol hydrochloride (USAN)
D06374 Zinterol hydrochloride (USAN)
D06562 Bedoradrine sulfate (USAN)
D07451 Amosulalol (INN)
D07463 Arformoterol (INN)
D07465 Arotinolol (INN)
D07608 Carazolol (INN)
D08078 Indenolol (INN)
D08124 Levosalbutamol (INN)
D08945 Milveterol hydrochloride (USAN)
D09696 Vilanterol (USAN/INN)
D09697 Vilanterol trifenatate (JAN/USAN)
D10219 Abediterol (USAN/INN)
D10220 Abediterol napadisylate (USAN)
D10545 Batefenterol (USAN)
D10546 Batefenterol succinate (USAN)
D11900 Navafenterol (USAN)
D11901 Navafenterol saccharinate (USAN)
|
ADRB3 [HSA:155] [KO:K04143]
|
D09535 Mirabegron (JAN/USAN/INN) <JP/US>
D10433 Vibegron (JAN/USAN/INN) <JP/US>
D02702 Talibegron hydrochloride (USAN)
D05879 Solabegron hydrochloride (USAN)
D08850 Amibegron (USAN/INN)
D08851 Amibegron hydrochloride (USAN)
D09344 Fasobegron (INN)
D09732 Ritobegron ethyl hydrochloride (JAN)
|
Dopamine
|
DRD [HSA:1812 1813 1814 1815 1816] [KO:K04144 K04145 K04146 K04147 K05840]
|
D07870 Dopamine (INN)
D00633 Dopamine hydrochloride (JP18/USP) <JP/US>
D03891 Dopexamine (USAN/INN)
D03892 Dopexamine hydrochloride (USAN)
D00059 Levodopa (JP18/USP/INN) <JP/US>
D02676 Oxiperomide (USAN/INN)
D04097 Etilevodopa (USAN/INN)
D09886 Dexpramipexole (USAN/INN)
D09887 Dexpramipexole dihydrochloride (USAN)
D11839 Foslevodopa (JAN/USAN/INN)
|
DRD1 [HSA:1812] [KO:K04144]
|
D04488 Ibopamine (USAN/INN)
D08057 Ibopamine hydrochloride
D07946 Fenoldopam (INN)
D00613 Fenoldopam mesylate (USP)
D07460 Apomorphine (BAN)
D02004 Apomorphine hydrochloride (USP) <JP/US>
D08339 Pergolide (INN)
D00502 Pergolide mesylate (USP) <JP>
D07065 Acepromazine (INN)
D02604 Acepromazine maleate (USP)
D00788 Acetophenazine maleate (USAN)
D08385 Pipotiazine (INN)
D02680 Pipotiazine palmitate (USAN)
D01044 Flupentixol (INN)
D02236 Flupentixol dihydrochloride (JAN)
D07976 Flupentixol decanoate
D02613 Clopenthixol (USAN)
D00790 Chlorprothixene (JAN/USAN/INN)
D02162 Chlorprothixene hydrochloride (JAN)
D07686 Chlorprothixene acetate
D07687 Chlorprothixene citrate
D03556 Zuclopenthixol (INN)
D08691 Zuclopenthixol acetate
D08692 Zuclopenthixol decanoate
D08693 Zuclopenthixol dihydrochloride
D01903 Docarpamine (JAN/INN) <JP>
D02641 Butaclamol hydrochloride (USAN)
D02644 Carphenazine maleate (USAN)
D02775 Adrogolide hydrochloride (USAN)
D03494 Ciladopa hydrochloride (USAN)
D03937 Ecopipam hydrochloride (USAN)
D10329 Zicronapine (USAN/INN)
D10495 Zicronapine succinate (USAN)
D11431 Tavapadon (USAN/INN)
D11822 Mevidalen hydroxybenzoate (USAN)
D11826 Mevidalen (USAN)
D12766 Razpipadon (USAN/INN)
D13239 Glovadalen (USAN/INN)
|
DRD2 [HSA:1813] [KO:K04145]
|
D00726 Metoclopramide (JP18/INN) <JP>
D02213 Metoclopramide hydrochloride (JAN) <JP>
D05008 Metoclopramide hydrochloride (USP) <US>
D01745 Domperidone (JP18/USAN/INN) <JP>
D07868 Domperidone maleate
D07101 Bromopride (INN)
D07102 Alizapride (INN)
D07563 Alizapride hydrochloride
D03534 Clebopride (USAN)
D01742 Clebopride malate (JP18)
D08094 Itopride (INN)
D02729 Itopride hydrochloride (JAN) <JP>
D05010 Metopimazine (USAN/INN)
D04488 Ibopamine (USAN/INN)
D08057 Ibopamine hydrochloride
D03165 Bromocriptine (USAN/INN)
D00780 Bromocriptine mesylate (USP) <JP/US>
D08132 Lisuride (INN)
D01462 Lisuride maleate (JAN)
D00987 Cabergoline (JP18/USP/INN) <JP/US>
D07217 Quinagolide (INN/BAN)
D08457 Quinagolide hydrochloride (BAN)
D01348 Terguride (JAN/INN)
D07460 Apomorphine (BAN)
D02004 Apomorphine hydrochloride (USP) <JP/US>
D08339 Pergolide (INN)
D00502 Pergolide mesylate (USP) <JP>
D07836 Dihydroergocryptine mesilate
D08489 Ropinirole (USAN/INN)
D00784 Ropinirole hydrochloride (JAN/USP) <JP/US>
D05575 Pramipexole (USAN/INN)
D00559 Pramipexole dihydrochloride (USP) <JP/US>
D07305 Piribedil (INN)
D05768 Rotigotine (JAN/USAN/INN) <JP/US>
D00270 Chlorpromazine (USP/INN)
D00789 Chlorpromazine hydrochloride (JP18/USP) <JP/US>
D03274 Chlorpromazine hibenzate (JAN)
D04034 Chlorpromazine phenolphthalinate (JAN) <JP>
D09819 Chlorpromazine tannate (JAN)
D00403 Methotrimeprazine (USP)
D01520 Levomepromazine hydrochloride (JAN/USAN)
D02248 Levomepromazine maleate (JP18/USAN) <JP>
D08430 Promazine (INN)
D00797 Promazine hydrochloride (USP)
D07065 Acepromazine (INN)
D02604 Acepromazine maleate (USP)
D00390 Triflupromazine (USP/INN)
D00800 Triflupromazine hydrochloride (JAN/USP)
D07977 Fluphenazine (INN)
D00791 Fluphenazine hydrochloride (JAN/USP) <US>
D00792 Fluphenazine enanthate (JP18/USP)
D00793 Fluphenazine decanoate (JAN/USP) <JP/US>
D02163 Fluphenazine maleate (JAN) <JP>
D00503 Perphenazine (JP18/USP/INN) <JP/US>
D02037 Perphenazine maleate (JP18) <JP>
D04038 Perphenazine fendizoate (JAN) <JP>
D04965 Perphenazine hydrochloride <JP>
D08341 Perphenazine decanoate
D08342 Perphenazine enantate
D00493 Prochlorperazine (JAN/USP/INN) <US>
D00479 Prochlorperazine maleate (JP18/USP) <JP/US>
D02022 Prochlorperazine mesilate (JAN) <JP>
D02609 Prochlorperazine edisylate (USP) <US>
D08636 Trifluoperazine (INN)
D00799 Trifluoperazine hydrochloride (JAN/USP) <US>
D01448 Trifluoperazine maleate (JAN)
D00788 Acetophenazine maleate (USAN)
D08585 Thioproperazine (INN)
D01447 Thioproperazine mesilate (JAN)
D01412 Perazine maleate (JAN)
D01860 Perazine dimalonate (JAN)
D02608 Perazine fendizoate (JAN)
D01485 Propericiazine (JAN) <JP>
D00373 Thioridazine (USP/INN)
D00798 Thioridazine hydrochloride (JP18/USP) <US>
D02671 Mesoridazine (USAN/INN)
D00795 Mesoridazine besylate (USP)
D08385 Pipotiazine (INN)
D02680 Pipotiazine palmitate (USAN)
D00136 Haloperidol (JP18/USP/INN) <JP/US>
D01898 Haloperidol decanoate (JAN/USP) <JP/US>
D08035 Haloperidol lactate <US>
D02625 Trifluperidol (USAN/INN)
D08637 Trifluperidol hydrochloride
D07309 Melperone (INN)
D08172 Melperone hydrochloride
D02623 Moperone (INN)
D01105 Moperone hydrochloride (JAN)
D02622 Pipamperone (USAN/INN)
D01482 Pipamperone hydrochloride (JAN) <JP>
D01101 Bromperidol (JAN/USAN/INN) <JP>
D02626 Bromperidol decanoate (USAN)
D02627 Benperidol (USAN/INN)
D00308 Droperidol (JP18/USP/INN) <JP/US>
D11169 Lumateperone (USAN/INN)
D11170 Lumateperone tosylate (USAN) <US>
D08226 Molindone (INN)
D00796 Molindone hydrochloride (USP) <US>
D00561 Sertindole (USAN/INN)
D08687 Ziprasidone (INN)
D01939 Ziprasidone hydrochloride (USP) <US>
D02100 Ziprasidone mesylate (USAN) <US>
D04820 Lurasidone hydrochloride (JAN/USAN) <JP/US>
D01044 Flupentixol (INN)
D02236 Flupentixol dihydrochloride (JAN)
D07976 Flupentixol decanoate
D02613 Clopenthixol (USAN)
D00790 Chlorprothixene (JAN/USAN/INN)
D02162 Chlorprothixene hydrochloride (JAN)
D07686 Chlorprothixene acetate
D07687 Chlorprothixene citrate
D00374 Thiothixene (USP) <US>
D02612 Thiothixene hydrochloride (USP)
D03556 Zuclopenthixol (INN)
D08691 Zuclopenthixol acetate
D08692 Zuclopenthixol decanoate
D08693 Zuclopenthixol dihydrochloride
D00560 Pimozide (JP18/USP/INN) <US>
D02340 Loxapine (USAN/INN)
D00794 Loxapine succinate (USP) <US>
D08148 Loxapine hydrochloride
D00454 Olanzapine (JAN/USP/INN) <JP/US>
D06623 Olanzapine pamoate (USAN) <US>
D08456 Quetiapine (INN)
D00458 Quetiapine fumarate (JP18/USP) <JP/US>
D11769 Asenapine (INN) <US>
D02995 Asenapine maleate (JAN/USAN) <JP/US>
D01226 Sulpiride (JP18/USAN/INN) <JP>
D08549 Sultopride (INN)
D02208 Sultopride hydrochloride (JAN) <JP>
D08590 Tiapride (INN)
D01522 Tiapride hydrochloride (JP18) <JP>
D02682 Remoxipride (USAN)
D02683 Remoxipride hydrochloride (USAN)
D07310 Amisulpride (INN) <US>
D07312 Levosulpiride (INN)
D00426 Risperidone (JP18/USP/INN) <JP/US>
D08235 Mosapramine (INN)
D01548 Mosapramine hydrochloride (JAN) <JP>
D01321 Zotepine (JAN/INN) <JP>
D01164 Aripiprazole (JP18/USP/INN) <JP/US>
D10355 Aripiprazole cavoxil (USAN)
D10364 Aripiprazole lauroxil (USAN) <US>
D10516 Aripiprazole hydrate (JAN) <JP/US>
D05339 Paliperidone (JAN/USP/INN) <JP/US>
D05340 Paliperidone palmitate (JAN/USAN) <JP/US>
D02666 Iloperidone (USAN/INN) <US>
D09997 Cariprazine (USAN/INN)
D09876 Cariprazine hydrochloride (JAN/USAN) <US>
D10309 Brexpiprazole (JAN/USAN/INN) <JP/US>
D13183 Brexpiprazole fumarate hydrate (JAN)
D07593 Buspirone (INN)
D00702 Buspirone hydrochloride (USP) <US>
D08297 Opipramol (INN)
D01477 Opipramol hydrochloride (JAN/USAN)
D09953 Pridopidine (USAN/INN)
D09954 Pridopidine hydrochloride (USAN)
D02354 Thiethylperazine (USAN/INN)
D01130 Thiethylperazine maleate (JAN/USP)
D02610 Thiethylperazine malate (JAN)
D01051 Spiperone (JAN/USAN) <JP>
D01176 Blonanserin (JAN/INN) <JP>
D01468 Nemonapride (JAN/INN) <JP>
D01505 Talipexole hydrochloride (JAN)
D02035 Timiperone (JAN) <JP>
D02371 Clocapramine hydrochloride hydrate (JP18) <JP>
D02372 Perospirone hydrochloride hydrate (JAN) <JP>
D02605 Methoxypromazine maleate
D02634 Alentemol hydrobromide (USAN)
D02641 Butaclamol hydrochloride (USAN)
D02644 Carphenazine maleate (USAN)
D02645 Carvotroline hydrochloride (USAN)
D02670 Mazapertine succinate (USAN)
D02675 Ocaperidone (USAN)
D02681 Piquindone hydrochloride (USAN)
D02688 Tiospirone hydrochloride (USAN)
D03214 Aplindore fumarate (USAN)
D03494 Ciladopa hydrochloride (USAN)
D04693 Lergotrile (USAN/INN)
D04694 Lergotrile mesylate (USAN)
D05124 Naxagolide hydrochloride (USAN)
D05677 Quinelorane hydrochloride (USAN)
D05682 Quinpirole hydrochloride (USAN)
D05690 Raclopride C11 (USAN)
D05804 Sarizotan hydrochloride (USAN)
D05832 Sibenadet hydrochloride (USAN)
D06566 Bifeprunox (USAN/INN)
D06567 Bifeprunox mesylate (USAN)
D07718 Clocapramine (INN)
D07835 Dihydroergocryptine
D08558 Talipexole (INN)
D09366 Pardoprunox hydrochloride (USAN)
D09397 Pardoprunox (USAN/INN)
D10329 Zicronapine (USAN/INN)
D10495 Zicronapine succinate (USAN)
D11982 Trazpiroben (USAN/INN)
D12733 Dordaviprone (USAN/INN)
D12734 Dordaviprone hydrochloride (JAN/USAN) <US>
D12813 Brilaroxazine (USAN/INN)
D12814 Brilaroxazine hydrochloride (USAN)
D13099 Milsaperidone (USAN)
|
DRD3 [HSA:1814] [KO:K04146]
|
D08132 Lisuride (INN)
D01462 Lisuride maleate (JAN)
D08489 Ropinirole (USAN/INN)
D00784 Ropinirole hydrochloride (JAN/USP) <JP/US>
D05575 Pramipexole (USAN/INN)
D00559 Pramipexole dihydrochloride (USP) <JP/US>
D07305 Piribedil (INN)
D00374 Thiothixene (USP) <US>
D02612 Thiothixene hydrochloride (USP)
D00454 Olanzapine (JAN/USP/INN) <JP/US>
D06623 Olanzapine pamoate (USAN) <US>
D07310 Amisulpride (INN) <US>
D01164 Aripiprazole (JP18/USP/INN) <JP/US>
D10355 Aripiprazole cavoxil (USAN)
D10364 Aripiprazole lauroxil (USAN) <US>
D10516 Aripiprazole hydrate (JAN) <JP/US>
D07316 Captodiame (BAN)
D01176 Blonanserin (JAN/INN) <JP>
D03214 Aplindore fumarate (USAN)
D05682 Quinpirole hydrochloride (USAN)
D09366 Pardoprunox hydrochloride (USAN)
D09397 Pardoprunox (USAN/INN)
D11982 Trazpiroben (USAN/INN)
|
DRD4 [HSA:1815] [KO:K04147]
|
D08132 Lisuride (INN)
D01462 Lisuride maleate (JAN)
D08489 Ropinirole (USAN/INN)
D00784 Ropinirole hydrochloride (JAN/USP) <JP/US>
D05575 Pramipexole (USAN/INN)
D00559 Pramipexole dihydrochloride (USP) <JP/US>
D00283 Clozapine (JAN/USP/INN) <JP/US>
D00454 Olanzapine (JAN/USP/INN) <JP/US>
D06623 Olanzapine pamoate (USAN) <US>
D02656 Fananserin (USAN/INN)
D05891 Sonepiprazole mesylate (USAN)
|
DRD5 [HSA:1816] [KO:K05840]
|
D03937 Ecopipam hydrochloride (USAN)
D11431 Tavapadon (USAN/INN)
D12766 Razpipadon (USAN/INN)
|
Histamine
|
HRH1 [HSA:3269] [KO:K04149]
|
D08587 Thonzylamine (INN)
D01801 Thonzylamine hydrochloride (JAN/USAN)
D08183 Mepyramine (INN)
D05660 Pyrilamine maleate (USP)
D07194 Thenalidine (INN)
D08645 Tripelennamine (INN)
D02091 Tripelennamine hydrochloride (USP)
D06246 Tripelennamine citrate
D07195 Chloropyramine (INN)
D07679 Chloropyramine hydrochloride
D00494 Promethazine (JAN/INN)
D00480 Promethazine hydrochloride (JP18/USP) <JP/US>
D01242 Promethazine teoclate (JAN/INN)
D03290 Promethazine methylenedisalicylate (JAN) <JP>
D08432 Promethazine maleate
D08768 Promethazine hibenzate <JP>
D07196 Tolpropamine (INN)
D07853 Dimetindene (INN)
D01343 Dimethindene maleate (USAN)
D03535 Clemastine (USAN)
D00666 Clemastine fumarate (JP18/USP) <JP/US>
D07197 Bamipine (INN)
D07492 Bamipine dihydrochloride
D07493 Bamipine lactate
D08355 Pheniramine (INN)
D01174 Pheniramine maleate (JAN/USP)
D08091 Isothipendyl (INN)
D01143 Isothipendyl hydrochloride (JAN)
D00300 Diphenhydramine (JP18/INN) <JP>
D00669 Diphenhydramine hydrochloride (JP18/USP) <JP/US>
D02419 Diphenhydramine salicylate (JAN)
D03285 Diphenhydramine tannate (JP18)
D03360 Diphenhydramine laurylsulfate (JAN)
D03854 Diphenhydramine citrate (USP)
D07198 Chlorphenoxamine (INN)
D07684 Chlorphenoxamine hydrochloride
D07875 Doxepin (INN)
D00814 Doxepin hydrochloride (USP) <US>
D00774 Orphenadrine citrate (USP) <US>
D07854 Dimetotiazine (INN)
D01902 Fonazine mesylate (USAN) <JP>
D02599 Orphenadrine hydrochloride
D00270 Chlorpromazine (USP/INN)
D00789 Chlorpromazine hydrochloride (JP18/USP) <JP/US>
D03274 Chlorpromazine hibenzate (JAN)
D04034 Chlorpromazine phenolphthalinate (JAN) <JP>
D09819 Chlorpromazine tannate (JAN)
D00454 Olanzapine (JAN/USP/INN) <JP/US>
D06623 Olanzapine pamoate (USAN) <US>
D08054 Hydroxyzine (INN)
D00672 Hydroxyzine hydrochloride (JP18/USP) <JP/US>
D01096 Hydroxyzine pamoate (JP18/USP) <JP/US>
D08297 Opipramol (INN)
D01477 Opipramol hydrochloride (JAN/USAN)
D08216 Mianserin (INN)
D01358 Mianserin hydrochloride (JAN/USAN) <JP>
D07522 Betahistine (INN)
D01592 Betahistine mesilate (JP18) <JP>
D03102 Betahistine hydrochloride (USP)
D01295 Cinnarizine (JAN/USAN/INN)
D07734 Cinnarizine dihydrochloride
D08117 Levocabastine (INN)
D01717 Levocabastine hydrochloride (JAN/USP) <JP>
D07483 Azelastine (INN)
D00659 Azelastine hydrochloride (JP18/USP) <JP/US>
D07458 Antazoline (INN)
D02950 Antazoline phosphate (USP)
D07459 Antazoline hydrochloride
D08293 Olopatadine (INN)
D01192 Olopatadine hydrochloride (JP18/USP) <JP/US>
D03166 Bromodiphenhydramine hydrochloride (USP)
D07862 Diphenylpyraline (INN)
D01172 Diphenylpyraline hydrochloride (JAN)
D01627 Diphenylpyraline teoclate (JAN)
D07617 Carbinoxamine (INN)
D01336 Carbinoxamine maleate (JAN/USP) <US>
D09808 Carbinoxamine diphenyldisulfonate (JAN)
D07878 Doxylamine (INN)
D02327 Doxylamine succinate (USP)
D00520 Dimenhydrinate (JP18/USP/INN) <JP/US>
D07543 Brompheniramine (INN)
D00663 Brompheniramine maleate (USP)
D07803 Dexchlorpheniramine (INN)
D00668 Dexchlorpheniramine maleate (USP) <JP/US>
D07398 Chlorphenamine (INN)
D00665 Chlorpheniramine maleate (JP18/USP) <JP>
D03475 Chlorpheniramine polistirex (USAN)
D03704 Dexbrompheniramine maleate (USP)
D07400 Histapyrrodine (INN)
D07125 Alimemazine (INN)
D02245 Trimeprazine tartrate (USP) <JP>
D04979 Methdilazine (INN)
D04980 Methdilazine hydrochloride (USP)
D01324 Mequitazine (JP18/INN) <JP>
D07401 Oxomemazine (INN)
D07547 Buclizine (INN)
D02089 Buclizine hydrochloride (USAN)
D03621 Cyclizine (INN)
D02090 Cyclizine lactate (BAN)
D03622 Cyclizine hydrochloride (USP)
D08163 Meclozine (BAN)
D01317 Meclizine hydrochloride (JAN/USP) <US>
D07662 Cetirizine (INN)
D00664 Cetirizine hydrochloride (JP18/USP) <JP/US>
D07402 Levocetirizine (USAN/INN)
D08118 Levocetirizine dihydrochloride (USP) <JP/US>
D07765 Cyproheptadine (INN)
D02234 Cyproheptadine hydrochloride (JP18/USP) <JP/US>
D08353 Phenindamine (INN)
D02148 Phenindamine tartrate (USAN)
D08648 Triprolidine (INN)
D01782 Triprolidine hydrochloride (USP)
D07403 Pyrrobutamine (BAN)
D07482 Azatadine (INN)
D00662 Azatadine maleate (USP)
D00234 Astemizole (JAN/USP/INN)
D00521 Terfenadine (JAN/USAN/INN)
D00364 Loratadine (JAN/USP/INN) <JP/US>
D08161 Mebhydrolin (INN)
D01786 Mebhydrolin napadisilate (JAN)
D07404 Deptropine (INN)
D07790 Deptropine citrate
D08105 Ketotifen (INN)
D01332 Ketotifen fumarate (JP18/USAN) <JP>
D02760 Acrivastine (USAN/INN)
D01478 Ebastine (JP18/USAN/INN) <JP>
D07406 Pimethixene (INN)
D07900 Epinastine (INN)
D01713 Epinastine hydrochloride (JAN) <JP/US>
D01117 Mizolastine (JAN/INN)
D07958 Fexofenadine (INN)
D00671 Fexofenadine hydrochloride (JP18/USP) <JP>
D03693 Desloratadine (JAN/USP/INN) <JP/US>
D07407 Rupatadine (USAN/INN)
D08497 Rupatadine fumarate (JAN/USAN) <JP>
D09570 Bilastine (JAN/INN) <JP>
D10230 Quifenadine (INN)
D10510 Sequifenadine
D07890 Emedastine (INN)
D02249 Emedastine difumarate (JP18/USP) <JP>
D06552 Alcaftadine (JAN/USAN/INN) <US>
D04445 Histamine phosphate (USP) <US>
D01460 Homochlorcyclizine hydrochloride (JP18)
D01654 Bepotastine besylate (USAN) <JP/US>
D01701 Difeterol hydrochloride (JAN)
D02067 Diphenylimidazole (JAN)
D03056 Barmastine (USAN/INN)
D03491 Cidoxepin hydrochloride (USAN)
D03568 Closiramine aceturate (USAN)
D03620 Cycliramine maleate (USAN)
D03893 Dorastine hydrochloride (USAN)
D03963 Efletirizine dihydrochloride (USAN)
D04055 Esmirtazapine maleate (USAN)
D04494 Icotidine (USAN)
D05196 Noberastine (USAN/INN)
D05664 Pyroxamine maleate (USAN)
D05742 Rocastine hydrochloride (USAN)
D05769 Rotoxamine (USAN/INN)
D06012 Tazifylline hydrochloride (USAN)
D06021 Tecastemizole (USAN/INN)
D06063 Temelastine (USAN/INN)
D06084 Tesmilifene hydrochloride (USAN)
D06376 Zolamine hydrochloride (USAN)
D07532 Bisulepin
D07533 Bisulepin hydrochloride
D07860 Dioxopromethazine hydrochloride
D07889 Embramine (INN)
D08040 Histamine (DCF)
D08041 Homochlorcyclizine (INN)
D08305 Orphenadrine (INN)
D08967 Phenyltoloxamine citrate (USP)
D09705 Bepotastine (USAN/INN)
D09747 Difeterol phosphate (JAN)
D09748 Difeterol (JAN/INN)
D09838 Broizine (JAN)
|
HRH2 [HSA:3274] [KO:K04150]
|
D00295 Cimetidine (JP18/USP/INN) <JP/US>
D03503 Cimetidine hydrochloride (USP) <US>
D00422 Ranitidine (USAN/INN)
D00673 Ranitidine hydrochloride (JP18/USP) <US>
D00318 Famotidine (JP18/USP/INN) <JP/US>
D00440 Nizatidine (JP18/USP/INN) <JP/US>
D07072 Niperotidine (INN)
D08494 Roxatidine (INN)
D01467 Roxatidine acetate hydrochloride (JP18/USAN) <JP>
D08495 Roxatidine acetate (BAN)
D05699 Ranitidine bismuth citrate (USAN)
D01131 Lafutidine (JP18/INN) <JP>
D00721 Methanthelinium bromide (INN)
D01187 Betazole hydrochloride (JAN)
D04445 Histamine phosphate (USP) <US>
D01193 Osutidine (JAN/INN)
D01698 Dalcotidine (JAN/INN)
D01861 Pibutidine hydrochloride (JAN)
D03889 Donetidine (USAN)
D04098 Etintidine hydrochloride (USAN)
D04494 Icotidine (USAN)
D04517 Impromidine hydrochloride (USAN)
D04680 Lavoltidine succinate (USAN)
D04794 Lupitidine hydrochloride (USAN)
D05004 Metiamide (USAN/INN)
D05306 Oxmetidine hydrochloride (USAN)
D05307 Oxmetidine mesylate (USAN)
D05939 Sufotidine (USAN/INN)
D06157 Tiotidine (USAN/INN)
D06355 Zaltidine hydrochloride (USAN)
D08040 Histamine (DCF)
|
HRH3 [HSA:11255] [KO:K04151]
|
D07522 Betahistine (INN)
D01592 Betahistine mesilate (JP18) <JP>
D03102 Betahistine hydrochloride (USP)
D10749 Pitolisant (USAN/INN)
D11490 Pitolisant hydrochloride (JAN/USAN) <US>
D04445 Histamine phosphate (USP) <US>
D03518 Cipralisant maleate (USAN)
D08040 Histamine (DCF)
D09870 Bavisant (USAN/INN)
D09871 Bavisant dihydrochloride (USAN)
D10128 Irdabisant (USAN)
D10129 Irdabisant hydrochloride (USAN)
|
HRH4 [HSA:59340] [KO:K04152]
|
D08040 Histamine (DCF)
D10735 Toreforant (USAN/INN)
D10736 Toreforant tartrate (USAN)
D11819 Adriforant (USAN/INN)
|
Serotonin
|
HTR1 [HSA:3350 3351 3352 3354 3355] [KO:K04153]
|
D07700 Cinitapride (INN)
D07701 Cinitapride tartrate
D05523 Pizotyline (USAN)
D08397 Pizotifen malate
D01321 Zotepine (JAN/INN) <JP>
D07765 Cyproheptadine (INN)
D02234 Cyproheptadine hydrochloride (JP18/USP) <JP/US>
D04533 Indorenate hydrochloride (USAN)
|
HTR1A [HSA:3350] [KO:K04153]
|
D07906 Ergotamine (INN)
D02577 Flibanserin (USAN/INN) <US>
D00679 Ergotamine tartrate (JP18/USP) <US>
D02357 Methysergide (USAN/INN)
D00681 Methysergide maleate (USP)
D08385 Pipotiazine (INN)
D02680 Pipotiazine palmitate (USAN)
D02995 Asenapine maleate (JAN/USAN) <JP/US>
D01164 Aripiprazole (JP18/USP/INN) <JP/US>
D10355 Aripiprazole cavoxil (USAN)
D10364 Aripiprazole lauroxil (USAN) <US>
D10516 Aripiprazole hydrate (JAN) <JP/US>
D09997 Cariprazine (USAN/INN)
D09876 Cariprazine hydrochloride (JAN/USAN) <US>
D10309 Brexpiprazole (JAN/USAN/INN) <JP/US>
D13183 Brexpiprazole fumarate hydrate (JAN)
D07593 Buspirone (INN)
D00702 Buspirone hydrochloride (USP) <US>
D04314 Gepirone hydrochloride (USAN) <US>
D09698 Vilazodone (USAN/INN)
D09699 Vilazodone hydrochloride (USAN) <US>
D10184 Vortioxetine (USAN)
D10185 Vortioxetine hydrobromide (JAN/USAN) <JP/US>
D12544 Vortioxetine hemihydrobromide (USAN)
D06327 Xaliproden (USAN)
D01537 Xaliproden hydrochloride (JAN)
D01992 Tandospirone citrate (JAN/USAN) <JP>
D02568 Flesinoxan (INN)
D02569 Sunepitron hydrochloride (USAN)
D02576 Eptapirone (INN)
D02688 Tiospirone hydrochloride (USAN)
D02767 Adatanserin hydrochloride (USAN)
D03121 Binospirone mesylate (USAN)
D04611 Ipsapirone hydrochloride (USAN)
D04683 Lecozotan hydrochloride (USAN)
D05804 Sarizotan hydrochloride (USAN)
D06354 Zalospirone hydrochloride (USAN)
D06566 Bifeprunox (USAN/INN)
D06567 Bifeprunox mesylate (USAN)
D08561 Tandospirone (INN)
D09358 Naluzotan (USAN/INN)
D09359 Naluzotan hydrochloride (USAN)
D09366 Pardoprunox hydrochloride (USAN)
D09397 Pardoprunox (USAN/INN)
D12474 Ulotaront (USAN/INN)
D12475 Ulotaront hydrochloride (JAN/USAN)
|
HTR1B [HSA:3351] [KO:K04153]
|
D07906 Ergotamine (INN)
D07837 Dihydroergotamine (INN)
D02211 Dihydroergotamine mesylate (USP) <US>
D07838 Dihydroergotamine tartrate
D00679 Ergotamine tartrate (JP18/USP) <US>
D00451 Sumatriptan (JAN/USP/INN) <JP/US>
D00676 Sumatriptan succinate (JAN/USP) <JP/US>
D08255 Naratriptan (INN)
D00674 Naratriptan hydrochloride (JAN/USP) <JP/US>
D00415 Zolmitriptan (JAN/USP/INN) <JP/US>
D08485 Rizatriptan (INN)
D00675 Rizatriptan benzoate (JAN/USP) <JP/US>
D05740 Rizatriptan sulfate (USAN)
D02824 Almotriptan (USAN)
D02825 Almotriptan malate (USP) <US>
D07887 Eletriptan (INN)
D01973 Eletriptan hydrobromide (JAN/USAN) <JP/US>
D11617 Eletriptan hydrobromide monohydrate
D07997 Frovatriptan (INN)
D04264 Frovatriptan succinate (USAN) <US>
D02826 Alniditan dihydrochloride (USAN)
D03014 Avitriptan fumarate (USAN)
D03982 Elzasonan citrate (USAN)
D03983 Elzasonan hydrochloride (USAN)
|
HTR1D [HSA:3352] [KO:K04153]
|
D07945 Fenfluramine (INN)
D04148 Fenfluramine hydrochloride (JAN/USAN) <JP/US>
D07906 Ergotamine (INN)
D07837 Dihydroergotamine (INN)
D02211 Dihydroergotamine mesylate (USP) <US>
D07838 Dihydroergotamine tartrate
D00679 Ergotamine tartrate (JP18/USP) <US>
D00451 Sumatriptan (JAN/USP/INN) <JP/US>
D00676 Sumatriptan succinate (JAN/USP) <JP/US>
D08255 Naratriptan (INN)
D00674 Naratriptan hydrochloride (JAN/USP) <JP/US>
D00415 Zolmitriptan (JAN/USP/INN) <JP/US>
D08485 Rizatriptan (INN)
D00675 Rizatriptan benzoate (JAN/USP) <JP/US>
D05740 Rizatriptan sulfate (USAN)
D02824 Almotriptan (USAN)
D02825 Almotriptan malate (USP) <US>
D07887 Eletriptan (INN)
D01973 Eletriptan hydrobromide (JAN/USAN) <JP/US>
D11617 Eletriptan hydrobromide monohydrate
D07997 Frovatriptan (INN)
D04264 Frovatriptan succinate (USAN) <US>
D02826 Alniditan dihydrochloride (USAN)
D03014 Avitriptan fumarate (USAN)
D03982 Elzasonan citrate (USAN)
D03983 Elzasonan hydrochloride (USAN)
|
HTR1F [HSA:3355] [KO:K04153]
|
D10338 Lasmiditan (USAN/INN)
D10424 Lasmiditan succinate (JAN/USAN) <JP/US>
|
HTR2 [HSA:3356 3357 3358] [KO:K04157]
|
D07700 Cinitapride (INN)
D07701 Cinitapride tartrate
D02577 Flibanserin (USAN/INN) <US>
D02357 Methysergide (USAN/INN)
D00681 Methysergide maleate (USP)
D05523 Pizotyline (USAN)
D08397 Pizotifen malate
D07854 Dimetotiazine (INN)
D01902 Fonazine mesylate (USAN) <JP>
D00270 Chlorpromazine (USP/INN)
D00789 Chlorpromazine hydrochloride (JP18/USP) <JP/US>
D03274 Chlorpromazine hibenzate (JAN)
D04034 Chlorpromazine phenolphthalinate (JAN) <JP>
D09819 Chlorpromazine tannate (JAN)
D01485 Propericiazine (JAN) <JP>
D00454 Olanzapine (JAN/USP/INN) <JP/US>
D06623 Olanzapine pamoate (USAN) <US>
D02666 Iloperidone (USAN/INN) <US>
D08297 Opipramol (INN)
D01477 Opipramol hydrochloride (JAN/USAN)
D08626 Trazodone (INN)
D00820 Trazodone hydrochloride (JAN/USP) <JP/US>
D00563 Mirtazapine (JAN/USP/INN) <JP/US>
D11056 Mirtazapine hydrate (JAN)
D07765 Cyproheptadine (INN)
D02234 Cyproheptadine hydrochloride (JP18/USP) <JP/US>
D02675 Ocaperidone (USAN)
D02686 Setoperone (USAN/INN)
D02688 Tiospirone hydrochloride (USAN)
D02767 Adatanserin hydrochloride (USAN)
D04320 Glemanserin (USAN/INN)
D05015 Metrenperone (USAN/INN)
D05395 Pelanserin hydrochloride (USAN)
D05829 Sergolexole maleate (USAN)
D06253 Tropanserin hydrochloride (USAN)
D06343 Xylamidine tosylate (USAN)
D12707 Brolamfetamine (INN)
D13099 Milsaperidone (USAN)
|
HTR2A [HSA:3356] [KO:K04157]
|
D00274 Cisapride (USP/INN)
D02092 Cisapride (JAN)
D07945 Fenfluramine (INN)
D04148 Fenfluramine hydrochloride (JAN/USAN) <JP/US>
D02363 Ketanserin (USAN/INN)
D08099 Ketanserin tartrate
D08244 Naftidrofuryl (INN)
D05107 Nafronyl oxalate (USAN)
D07307 Cyamemazine (INN)
D07756 Cyamemazine tartrate
D02671 Mesoridazine (USAN/INN)
D00795 Mesoridazine besylate (USP)
D08385 Pipotiazine (INN)
D02680 Pipotiazine palmitate (USAN)
D11169 Lumateperone (USAN/INN)
D11170 Lumateperone tosylate (USAN) <US>
D00561 Sertindole (USAN/INN)
D08687 Ziprasidone (INN)
D01939 Ziprasidone hydrochloride (USP) <US>
D02100 Ziprasidone mesylate (USAN) <US>
D04820 Lurasidone hydrochloride (JAN/USAN) <JP/US>
D02340 Loxapine (USAN/INN)
D00794 Loxapine succinate (USP) <US>
D08148 Loxapine hydrochloride
D00283 Clozapine (JAN/USP/INN) <JP/US>
D08456 Quetiapine (INN)
D00458 Quetiapine fumarate (JP18/USP) <JP/US>
D11769 Asenapine (INN) <US>
D02995 Asenapine maleate (JAN/USAN) <JP/US>
D00426 Risperidone (JP18/USP/INN) <JP/US>
D08235 Mosapramine (INN)
D01548 Mosapramine hydrochloride (JAN) <JP>
D01164 Aripiprazole (JP18/USP/INN) <JP/US>
D10355 Aripiprazole cavoxil (USAN)
D10364 Aripiprazole lauroxil (USAN) <US>
D10516 Aripiprazole hydrate (JAN) <JP/US>
D05339 Paliperidone (JAN/USP/INN) <JP/US>
D05340 Paliperidone palmitate (JAN/USAN) <JP/US>
D09997 Cariprazine (USAN/INN)
D09876 Cariprazine hydrochloride (JAN/USAN) <US>
D10309 Brexpiprazole (JAN/USAN/INN) <JP/US>
D13183 Brexpiprazole fumarate hydrate (JAN)
D08969 Pimavanserin tartrate (USAN) <US>
D08216 Mianserin (INN)
D01358 Mianserin hydrochloride (JAN/USAN) <JP>
D08257 Nefazodone (INN)
D00819 Nefazodone hydrochloride (USP) <US>
D01176 Blonanserin (JAN/INN) <JP>
D01624 Sarpogrelate hydrochloride (JP18) <JP>
D02372 Perospirone hydrochloride hydrate (JAN) <JP>
D02656 Fananserin (USAN/INN)
D02836 Altanserin tartrate (USAN)
D02893 Amesergide (USAN/INN)
D03005 Atiprosin maleate (USAN)
D04055 Esmirtazapine maleate (USAN)
D04788 Lubazodone hydrochloride (USAN)
D05738 Ritanserin (USAN/INN)
D06632 Pruvanserin (USAN/INN)
D06633 Pruvanserin hydrochloride (USAN)
D08508 Sarpogrelate (INN)
D09645 Nelotanserin (USAN/INN)
D09976 Temanogrel (USAN/INN)
D09977 Temanogrel hydrochloride (USAN)
D10006 Eplivanserin (USAN/INN)
D10329 Zicronapine (USAN/INN)
D10495 Zicronapine succinate (USAN)
D12881 Psilocybin (USAN)
D13135 Deupsilocin besylate (USAN)
D13136 Deupsilocin (USAN/INN)
D13141 Dimethyltryptamine (USAN/INN)
|
HTR2C [HSA:3358] [KO:K04157]
|
D07945 Fenfluramine (INN)
D04148 Fenfluramine hydrochloride (JAN/USAN) <JP/US>
D06613 Lorcaserin hydrochloride (USAN)
D11566 Lorcaserin hydrochloride hemihydrate
D07307 Cyamemazine (INN)
D07756 Cyamemazine tartrate
D00283 Clozapine (JAN/USP/INN) <JP/US>
D02995 Asenapine maleate (JAN/USAN) <JP/US>
D08969 Pimavanserin tartrate (USAN) <US>
D07316 Captodiame (BAN)
D08216 Mianserin (INN)
D01358 Mianserin hydrochloride (JAN/USAN) <JP>
D08257 Nefazodone (INN)
D00819 Nefazodone hydrochloride (USP) <US>
D02578 Agomelatine (INN)
D02893 Amesergide (USAN/INN)
D05738 Ritanserin (USAN/INN)
D06660 Vabicaserin hydrochloride (USAN)
D10170 Tedatioxetine (USAN)
D10171 Tedatioxetine hydrobromide (USAN)
D10710 Idalopirdine (USAN/INN)
D13035 Bexicaserin (USAN/INN)
D13036 Bexicaserin hydrochloride (USAN)
|
HTR4 [HSA:3360] [KO:K04160]
|
D00274 Cisapride (USP/INN)
D02092 Cisapride (JAN)
D07700 Cinitapride (INN)
D07701 Cinitapride tartrate
D08236 Mosapride (INN)
D01994 Mosapride citrate hydrate (JP18) <JP>
D09205 Prucalopride (USAN/INN)
D10152 Prucalopride succinate (USAN) <US>
D06056 Tegaserod (USAN/INN)
D02730 Tegaserod maleate (USAN)
D01838 Fabesetron hydrochloride (JAN)
D05471 Piboserod hydrochloride (USAN)
D05941 Sulamserod hydrochloride (USAN)
D06396 Renzapride (INN)
D09693 Velusetrag (USAN/INN)
D09694 Velusetrag hydrochloride (USAN)
D09933 Naronapride (USAN/INN)
D09934 Naronapride dihydrochloride (USAN)
D11220 Relenopride (USAN/INN)
D11221 Relenopride hydrochloride (USAN)
D12157 Felcisetrag (USAN/INN)
|
HTR6 [HSA:3362] [KO:K04162]
|
D00454 Olanzapine (JAN/USP/INN) <JP/US>
D06623 Olanzapine pamoate (USAN) <US>
D02995 Asenapine maleate (JAN/USAN) <JP/US>
D02688 Tiospirone hydrochloride (USAN)
D10099 Cerlapirdine (USAN)
D10100 Cerlapirdine hydrochloride (USAN)
D10710 Idalopirdine (USAN/INN)
D10747 Idalopirdine hydrochloride (JAN)
|
HTR7 [HSA:3363] [KO:K04163]
|
D02357 Methysergide (USAN/INN)
D00681 Methysergide maleate (USP)
D02995 Asenapine maleate (JAN/USAN) <JP/US>
|
Trace amine
|
TAAR [HSA:134864 9287 9038 319100 83551 134860] [KO:K05051]
|
D11830 Ralmitaront (USAN/INN)
|
TAAR1 [HSA:134864] [KO:K05051]
|
D12474 Ulotaront (USAN/INN)
D12475 Ulotaront hydrochloride (JAN/USAN)
D12707 Brolamfetamine (INN)
|
Anaphylatoxin
|
C5AR1 (CD88) [HSA:728] [KO:K04010]
|
D11093 Avacopan (JAN/USAN/INN) <JP/US>
|
Angiotensin
|
AGTR1 [HSA:185] [KO:K04166]
|
D02939 Angiotensin amide (USAN)
D00150 Angiotensin II (INN)
D02014 Angiotensin II (USAN)
D11142 Angiotensin II acetate (USAN) <US>
D08146 Losartan (INN)
D00357 Losartan potassium (JP18/USP) <JP/US>
D04040 Eprosartan (USAN/INN)
D02082 Eprosartan mesylate (USAN)
D00400 Valsartan (JP18/USP/INN) <JP/US>
D00523 Irbesartan (JP18/USP/INN) <JP/US>
D06010 Tasosartan (USAN/INN)
D00522 Candesartan (USAN/INN)
D00626 Candesartan cilexetil (JP18/USP) <JP/US>
D00627 Telmisartan (JP18/USP/INN) <JP/US>
D01204 Olmesartan medoxomil (JP18/USP) <JP/US>
D08067 Azilsartan medoxomil (USAN)
D08865 Azilsartan kamedoxomil (USAN) <US>
D10556 Fimasartan (INN)
D10226 Sacubitril valsartan sodium hydrate (JAN) <JP/US>
D11776 Sparsentan (JAN/USAN/INN) <US>
D01922 Pratosartan (JAN/INN)
D04126 Saralasin acetate (USAN)
D04243 Forasartan (USAN/INN)
D05246 Olmesartan (USAN/INN)
D05801 Saprisartan potassium (USAN)
D08864 Azilsartan (JAN/USAN/INN) <JP>
D12942 Talfirastide (USAN/INN)
D13133 Buloxibutid (USAN/INN)
D13134 Buloxibutid sodium (USAN)
|
AGTR2 [HSA:186] [KO:K04167]
|
D02939 Angiotensin amide (USAN)
D00150 Angiotensin II (INN)
D02014 Angiotensin II (USAN)
D11142 Angiotensin II acetate (USAN) <US>
D04126 Saralasin acetate (USAN)
D13133 Buloxibutid (USAN/INN)
D13134 Buloxibutid sodium (USAN)
|
Bradykinin
|
BDKRB2 [HSA:624] [KO:K03916]
|
D04492 Icatibant acetate (JAN/USAN) <JP/US>
D03677 Deltibant (USAN/INN)
D08937 Labradimil (INN/USAN)
D12618 Deucrictibant (USAN/INN)
|
Cholecystokinin
|
CCKAR [HSA:886] [KO:K04194]
|
D03442 Ceruletide (USAN/INN)
D03443 Ceruletide diethylamine (USAN)
D01113 Loxiglumide (JAN/INN)
D01858 Panazepide (JAN)
D02693 Devazepide (USAN/INN)
D02710 Tarazepide (INN)
|
CCKBR [HSA:887] [KO:K04195]
|
D01818 Proglumide (JP18/USAN/INN)
D01631 Pentagastrin (JAN/USAN/INN)
D01858 Panazepide (JAN)
|
Endothelin
|
EDNR [HSA:1909 1910] [KO:K04197 K04198]
|
D11974 Centhaquine (USAN)
D11975 Centhaquine citrate (USAN)
D11441 Aprocitentan (USAN/INN) <US>
D07538 Bosentan (INN)
D01227 Bosentan (USAN) <JP/US>
D10135 Macitentan (JAN/USAN) <JP/US>
|
EDNRA [HSA:1909] [KO:K04197]
|
D07077 Ambrisentan (JAN/INN) <JP/US>
D07171 Sitaxentan (USAN/INN)
D08517 Sitaxentan sodium (USAN)
D11664 Clazosentan (USAN/INN)
D07682 Clazosentan sodium (JAN/USAN) <JP>
D11776 Sparsentan (JAN/USAN/INN) <US>
D03009 Atrasentan hydrochloride (USAN) <US>
D03953 Edonentan (USAN)
D04128 Fandosentan potassium (USAN)
D07741 Zibotentan (JAN/USAN/INN)
|
EDNRB [HSA:1910] [KO:K04198]
|
D11964 Sovatelitide (USAN)
|
Follicle stimulating hormone
|
FSHR [HSA:2492] [KO:K04247]
|
D06457 Gonadotropin, chorionic (USP) <JP/US>
D02692 Menotropins (USAN) <JP>
D06459 Purified human menopausal gonadotrophin (JAN) <JP>
D05258 Serum gonadotrophin (JAN)
D06269 Urofollitropin (USAN/INN)
D04429 Follitropin alfa (genetical recombination) (JAN) <JP/US>
D04430 Follitropin beta (genetical recombination) (JAN) <JP/US>
D08895 Corifollitropin alfa (INN/USAN)
D06400 Follitropin delta (USAN) <JP>
D01281 Cyclofenil (JAN/INN) <JP>
|
Ghrelin
|
GHSR [HSA:2693] [KO:K04284]
|
D10563 Macimorelin (USAN)
D10562 Macimorelin acetate (USAN) <US>
D02040 Pralmorelin dihydrochloride (USAN) <JP>
D03373 Capromorelin tartrate (USAN)
D05734 Rismorelin porcine (USAN)
D08856 Anamorelin hydrochloride (JAN/USAN) <JP>
D09981 Ulimorelin (USAN/INN)
D09982 Ulimorelin hydrochloride (USAN)
D10660 Relamorelin (USAN/INN)
|
Gonadotropin-releasing hormone
|
GNRHR [HSA:2798] [KO:K04280]
|
D08027 Gonadorelin (INN)
D00988 Gonadorelin hydrochloride (USP)
D03267 Gonadorelin diacetate (JP18) <JP>
D04361 Gonadorelin acetate (USP)
D08241 Nafarelin (INN)
D00990 Nafarelin acetate (USAN) <JP/US>
D08010 Ganirelix (INN)
D04302 Ganirelix acetate (JAN/USAN) <JP/US>
D07665 Cetrorelix (INN)
D01685 Cetrorelix acetate (JAN/USAN) <JP/US>
D09335 Elagolix (USAN/INN)
D09336 Elagolix sodium (USAN) <US>
D11608 Linzagolix (USAN/INN)
D11609 Linzagolix choline (JAN/USAN)
D07259 Buserelin (INN)
D01831 Buserelin acetate (JAN/USAN) <JP>
D08113 Leuprolide (USAN)
D00989 Leuprolide acetate (USP) <JP/US>
D12337 Leuprolide mesylate (USAN) <US>
D04405 Goserelin (USAN/INN)
D00573 Goserelin acetate (JP18/USP) <JP/US>
D06247 Triptorelin (USAN/INN)
D06248 Triptorelin pamoate (USAN) <US>
D08649 Triptorelin acetate
D02369 Histrelin (USAN/INN)
D02116 Histrelin acetate <US>
D02738 Abarelix (USAN/INN)
D08901 Degarelix (INN/USAN)
D08635 Degarelix acetate (USAN)
D09400 Degarelix acetate (JAN) <JP/US>
D10888 Relugolix (JAN/USAN/INN) <JP/US>
D04644 Iturelix (USAN/INN)
D04823 Lutrelin acetate (USAN)
D05599 Prazarelix acetate (USAN)
D07957 Fertirelin (INN)
D11351 Opigolix (USAN/INN)
|
Lutropin-choriogonadotropic hormone
|
LHCGR [HSA:3973] [KO:K04248]
|
D06457 Gonadotropin, chorionic (USP) <JP/US>
D02692 Menotropins (USAN) <JP>
D06459 Purified human menopausal gonadotrophin (JAN) <JP>
D05258 Serum gonadotrophin (JAN)
D04824 Lutropin alfa (USAN/INN)
D03478 Choriogonadotropin alfa (USAN/INN) <JP/US>
D01281 Cyclofenil (JAN/INN) <JP>
|
Melanocortin
|
MC1R [HSA:4157] [KO:K04199]
|
D10511 Afamelanotide (USAN/INN)
D11334 Afamelanotide acetate (USAN) <US>
D06569 Bremelanotide (USAN/INN)
D11629 Bremelanotide acetate (USAN) <US>
D12147 Dersimelagon (USAN/INN)
D12148 Dersimelagon phosphate (USAN)
D13177 Resomelagon (USAN/INN)
D13178 Resomelagon acetate (USAN)
|
MC2R [HSA:4158] [KO:K04200]
|
D00146 Corticotropin (USP/INN) <US>
D03593 Corticotropin zinc hydroxide
D06544 Corticotropin, repository (USP)
D00284 Cosyntropin (USP) <US>
D02105 Tetracosactide acetate (JAN) <JP>
D07417 Alsactide (INN)
D05827 Seractide acetate (USAN)
D09801 Giractide acetate (JAN)
D09937 Giractide (INN)
D13102 Atumelnant (USAN/INN)
D13103 Atumelnant maleate (USAN)
|
MC3R [HSA:4159] [KO:K04201]
|
D13177 Resomelagon (USAN/INN)
D13178 Resomelagon acetate (USAN)
|
MC4R [HSA:4160] [KO:K04202]
|
D11927 Setmelanotide (USAN/INN)
D11928 Setmelanotide acetate <US>
D11929 Setmelanotide hydrochloride (USAN)
D06569 Bremelanotide (USAN/INN)
D11629 Bremelanotide acetate (USAN) <US>
|
Motilin
|
MLNR [HSA:2862] [KO:K05266]
|
D02801 Alemcinal (USAN/INN)
D03216 Atilmotin (USAN/INN)
D04497 Idremcinal (USAN/INN)
D05053 Mitemcinal fumarate (USAN)
D10330 Camicinal (USAN/INN)
|
Neuropeptide Y
|
NPY5R [HSA:4889] [KO:K04207]
|
D08026 Velneperit (USAN/INN)
|
Opioid
|
OPRM1 [HSA:4988] [KO:K04215]
|
D08639 Trimebutine (INN)
D01500 Trimebutine maleate (JP18) <JP>
D06618 Methylnaltrexone bromide (JAN/USAN) <US>
D02878 Alvimopan (USAN) <US>
D10479 Naloxegol (USAN/INN)
D10375 Naloxegol oxalate (USAN) <US>
D08249 Naloxone (INN)
D01340 Naloxone hydrochloride (JP18/USP) <JP/US>
D11620 Naloxone hydrochloride dihydrate <US>
D10188 Naldemedine (USAN/INN)
D10478 Naldemedine tosylate (JAN/USAN) <JP/US>
D07861 Diphenoxylate (INN)
D03860 Diphenoxylate hydrochloride (USP)
D08144 Loperamide (INN)
D00729 Loperamide hydrochloride (JAN/USP) <JP/US>
D03809 Difenoxin (USAN/INN)
D11583 Difenoxin hydrochloride
D07113 Loperamide oxide (INN)
D10403 Eluxadoline (USAN/INN) <US>
D00320 Fentanyl (JAN/USP/INN) <JP/US>
D01399 Fentanyl citrate (JP18/USP) <JP/US>
D10811 Fentanyl hydrochloride (JAN)
D07122 Alfentanil (INN)
D00835 Alfentanil hydrochloride (USP)
D05938 Sufentanil (USAN/INN)
D00845 Sufentanil citrate (USP) <US>
D02941 Anileridine (USP/INN)
D02942 Anileridine hydrochloride (USP)
D08473 Remifentanil (INN)
D01177 Remifentanil hydrochloride (JAN/USAN) <JP/US>
D08233 Morphine (BAN)
D00842 Morphine sulfate (USP) <JP/US>
D02271 Morphine hydrochloride hydrate (JP18) <JP>
D08234 Morphine tartrate
D08047 Hydromorphone (INN)
D00839 Hydromorphone hydrochloride (JAN/USP) <JP/US>
D07285 Nicomorphine (INN)
D08273 Nicomorphine hydrochloride
D05312 Oxycodone (USAN/INN) <US>
D00847 Oxycodone hydrochloride (USP) <US>
D03783 Oxycodone terephthalate (USP)
D05462 Oxycodone hydrochloride hydrate (JP18) <JP>
D07831 Dihydrocodeine (INN)
D01481 Dihydrocodeine phosphate (JP18) <JP>
D03825 Dihydrocodeine bitartrate (USP)
D07832 Dihydrocodeine thiocyanate
D08323 Oxymorphone (INN)
D00844 Oxymorphone hydrochloride (USP) <US>
D08100 Ketobemidone (INN)
D08101 Ketobemidone hydrochloride
D08343 Pethidine (INN)
D01383 Meperidine hydrochloride (USP) <JP/US>
D07809 Dextropropoxyphene (INN)
D00482 Propoxyphene hydrochloride (USAN) <US>
D05632 Propoxyphene napsylate (USAN)
D00498 Pentazocine (JP18/USP/INN) <JP>
D02111 Pentazocine lactate (USP)
D02227 Pentazocine hydrochloride (JAN/USP) <JP>
D07132 Buprenorphine (JAN/INN) <JP/US>
D00836 Buprenorphine hydrochloride (JP18/USP) <JP/US>
D03197 Butorphanol (USAN/INN)
D00837 Butorphanol tartrate (JAN/USP) <US>
D08246 Nalbuphine (INN)
D00843 Nalbuphine hydrochloride (USAN) <US>
D08597 Tilidine (INN)
D06147 Tilidine hydrochloride (USAN)
D08623 Tramadol (INN)
D01355 Tramadol hydrochloride (JP18/USP) <JP/US>
D00838 Dezocine (USAN)
D08182 Meptazinol (INN)
D04924 Meptazinol hydrochloride (USAN)
D06007 Tapentadol (USAN/INN)
D10199 Tapentadol hydrochloride (JAN) <US>
D11214 Oliceridine (USAN/INN) <US>
D05113 Naltrexone (USAN/INN) <US>
D02095 Naltrexone hydrochloride (USP) <US>
D05111 Nalmefene (USAN/INN)
D02104 Nalmefene hydrochloride <US>
D10812 Nalmefene hydrochloride hydrate (JAN) <JP>
D08195 Methadone (BAN)
D02102 Methadone hydrochloride (JAN/USP) <JP/US>
D04716 Levomethadyl acetate (USAN)
D00840 Levomethadyl acetate hydrochloride (USAN)
D08121 Levomethadone (INN)
D08122 Levomethadone hydrochloride
D07286 Diamorphine (BAN)
D07810 Diacetylmorphine hydrochloride
D07929 Ethylmorphine (BAN)
D02205 Ethylmorphine hydrochloride hydrate (JP18)
D08045 Hydrocodone (INN)
D03725 Hydrocodone bitartrate (USP) <US>
D04461 Hydrocodone polistirex (USAN)
D08046 Hydrocodone hydrochloride
D00195 Codeine (USP)
D02101 Codeine phosphate (USP) <JP>
D03579 Codeine polistirex (USAN)
D03580 Codeine sulfate (USP) <US>
D07740 Codeine hydrochloride
D07385 Pholcodine (INN)
D07557 O-Acetyldihydrocodeine hydrochloride
D08247 Nalorphine (INN)
D08248 Nalorphine hydrochloride (USP)
D00841 Levorphanol tartrate (USP) <US>
D01435 Ethoheptazine citrate (JAN)
D02238 Levallorphan tartrate (JP18) <JP>
D03156 Brifentanil hydrochloride (USAN)
D03405 Carfentanil citrate (USAN)
D03618 Cyclazocine (USAN/INN)
D04764 Lofentanil oxalate (USAN)
D04973 Methadyl acetate (USAN)
D05048 Mirfentanil hydrochloride (USAN)
D05217 Ocfentanil hydrochloride (USAN)
D05631 Propiram fumarate (USAN)
D05667 Quadazocine mesylate (USAN)
D06189 Tonazocine mesylate (USAN)
D06208 Trefentanil hydrochloride (USAN)
D06268 Trimeperidine (INN)
D06342 Xorphanol mesylate (USAN)
D07620 Carfentanil (INN)
D07863 Diprenorphine (INN)
D07864 Diprenorphine hydrochloride
D07937 Etorphine (INN)
D08123 Levorphanol (INN)
D10162 Samidorphan (USAN)
D10163 Samidorphan l-malate (USAN)
D10349 Bevenopran (USAN/INN)
D10371 Methylsamidorphan (USAN)
D10436 Cebranopadol (USAN/INN)
D10612 Benzhydrocodone (USAN/INN)
D10648 Methylsamidorphan chloride (USAN/INN)
D10690 Axelopran sulfate (USAN)
D10692 Benzhydrocodone hydrochloride (USAN)
D10740 Axelopran (USAN/INN)
D11291 Asalhydromorphone (USAN)
D11292 Asalhydromorphone hydrochloride (USAN)
D11424 Oxycodegol (USAN/INN)
D11425 Oxycodegol phosphate (USAN)
D12660 Alphacetylmethadol (INN)
D12661 Betacetylmethadol (INN)
D12662 Allylprodine (INN)
D12666 Alphameprodine (INN)
D12667 Betameprodine (INN)
D12668 Clonitazene (INN)
D12669 Etonitazene (INN)
D12674 Alphamethadol (INN)
D12675 Betamethadol (INN)
D12676 Isomethadone (INN)
D12678 Alphaprodine (INN)
D12679 Betaprodine (INN)
D12680 Etoxeridine (INN)
D12681 Hydroxypethidine (INN)
D12682 Furethidine (INN)
D12683 Piminodine (INN)
D12685 Benzethidine (INN)
D12686 Hydromorphinol (INN)
D12687 Levophenacylmorphan (INN)
D12688 Phenomorphan (INN)
D12689 Methyldihydromorphine (INN)
D12690 Metopon (BAN)
D12691 Methyldesorphine (INN)
D12692 Norlevorphanol (INN)
D12693 Phenampromide (INN)
D12694 Diampromide (INN)
D12696 Levomethorphan (INN)
D12697 Morpheridin (INN)
D12700 Acetorphine (INN)
D13025 Properidine (INN)
|
OPRK1 [HSA:4986] [KO:K04214]
|
D08639 Trimebutine (INN)
D01500 Trimebutine maleate (JP18) <JP>
D08249 Naloxone (INN)
D01340 Naloxone hydrochloride (JP18/USP) <JP/US>
D11620 Naloxone hydrochloride dihydrate <US>
D08144 Loperamide (INN)
D00729 Loperamide hydrochloride (JAN/USP) <JP/US>
D07113 Loperamide oxide (INN)
D10403 Eluxadoline (USAN/INN) <US>
D05312 Oxycodone (USAN/INN) <US>
D00847 Oxycodone hydrochloride (USP) <US>
D03783 Oxycodone terephthalate (USP)
D05462 Oxycodone hydrochloride hydrate (JP18) <JP>
D08100 Ketobemidone (INN)
D08101 Ketobemidone hydrochloride
D00498 Pentazocine (JP18/USP/INN) <JP>
D02111 Pentazocine lactate (USP)
D02227 Pentazocine hydrochloride (JAN/USP) <JP>
D07132 Buprenorphine (JAN/INN) <JP/US>
D00836 Buprenorphine hydrochloride (JP18/USP) <JP/US>
D03197 Butorphanol (USAN/INN)
D00837 Butorphanol tartrate (JAN/USP) <US>
D08246 Nalbuphine (INN)
D00843 Nalbuphine hydrochloride (USAN) <US>
D00838 Dezocine (USAN)
D05113 Naltrexone (USAN/INN) <US>
D02095 Naltrexone hydrochloride (USP) <US>
D05111 Nalmefene (USAN/INN)
D02104 Nalmefene hydrochloride <US>
D10812 Nalmefene hydrochloride hydrate (JAN) <JP>
D08247 Nalorphine (INN)
D08248 Nalorphine hydrochloride (USP)
D06405 Nalfurafine hydrochloride (JAN/USAN) <JP>
D11111 Difelikefalin (USAN/INN)
D10890 Difelikefalin acetate (JAN) <JP/US>
D01879 Eptazocine hydrobromide (JAN)
D02238 Levallorphan tartrate (JP18) <JP>
D03618 Cyclazocine (USAN/INN)
D04649 Ketazocine (USAN/INN)
D05299 Oxilorphan (USAN/INN)
D05646 Proxorphan tartrate (USAN)
D05667 Quadazocine mesylate (USAN)
D05907 Spiradoline mesylate (USAN)
D06189 Tonazocine mesylate (USAN)
D06342 Xorphanol mesylate (USAN)
D06395 Enadoline hydrochloride (USAN)
D07863 Diprenorphine (INN)
D07864 Diprenorphine hydrochloride
D07904 Eptazocine (INN)
D07937 Etorphine (INN)
D11831 Aticaprant (USAN/INN)
D12700 Acetorphine (INN)
D12869 Navacaprant (USAN/INN)
D12870 Navacaprant hydrochloride (USAN)
D13002 Icalcaprant (USAN/INN)
|
OPRD1 [HSA:4985] [KO:K04213]
|
D08249 Naloxone (INN)
D01340 Naloxone hydrochloride (JP18/USP) <JP/US>
D11620 Naloxone hydrochloride dihydrate <US>
D08144 Loperamide (INN)
D00729 Loperamide hydrochloride (JAN/USP) <JP/US>
D07113 Loperamide oxide (INN)
D10403 Eluxadoline (USAN/INN) <US>
D05312 Oxycodone (USAN/INN) <US>
D00847 Oxycodone hydrochloride (USP) <US>
D03783 Oxycodone terephthalate (USP)
D05462 Oxycodone hydrochloride hydrate (JP18) <JP>
D08100 Ketobemidone (INN)
D08101 Ketobemidone hydrochloride
D08246 Nalbuphine (INN)
D00843 Nalbuphine hydrochloride (USAN) <US>
D05113 Naltrexone (USAN/INN) <US>
D02095 Naltrexone hydrochloride (USP) <US>
D05111 Nalmefene (USAN/INN)
D02104 Nalmefene hydrochloride <US>
D10812 Nalmefene hydrochloride hydrate (JAN) <JP>
D02238 Levallorphan tartrate (JP18) <JP>
D05007 Metkephamid acetate (USAN)
D05667 Quadazocine mesylate (USAN)
D06189 Tonazocine mesylate (USAN)
D06342 Xorphanol mesylate (USAN)
D07937 Etorphine (INN)
D12676 Isomethadone (INN)
D12700 Acetorphine (INN)
|
OPRL1 [HSA:4987] [KO:K04216]
|
D10436 Cebranopadol (USAN/INN)
|
Orexin
|
HCRTR [HSA:3061 3062] [KO:K04238 K04239]
|
D10082 Suvorexant (JAN/USAN) <JP/US>
D11022 Lemborexant (JAN/USAN/INN) <JP/US>
D11886 Daridorexant (USAN/INN)
D11887 Daridorexant hydrochloride (JAN/USAN) <JP/US>
D09964 Almorexant (INN)
D10345 Filorexant (USAN/INN)
D12611 Vornorexant hydrate (JAN) <JP>
|
HCRTR2 [HSA:3062] [KO:K04239]
|
D11269 Seltorexant (USAN/INN)
D13223 Oveporexton (USAN/INN)
|
Oxytocin
|
OXTR [HSA:5021] [KO:K04229]
|
D03008 Atosiban (USAN/INN)
D07475 Atosiban acetate
D07228 Demoxytocin (INN)
D00089 Oxytocin (JP18/USP/INN) <JP/US>
D07229 Carbetocin (USAN/INN/BAN)
D08986 Retosiban (USAN)
D09797 Cargutocin (JAN/INN)
D10117 Epelsiban (USAN)
D10118 Epelsiban besylate (USAN)
|
Relaxin
|
RXFP1 [HSA:59350] [KO:K04306]
|
D10488 Serelaxin (USAN/INN)
|
RXFP2 [HSA:122042] [KO:K04307]
|
D12783 Volenrelaxin (USAN)
|
Somatostatin
|
SSTR [HSA:6751 6752 6753 6754 6755] [KO:K04217 K04218 K04219 K04220 K04221]
|
D07431 Somatostatin (INN)
D05812 Seglitide acetate (USAN)
D11192 Veldoreotide (USAN/INN)
|
SSTR1 [HSA:6751] [KO:K04217]
|
D10147 Pasireotide (USAN)
D10497 Pasireotide diaspartate <US>
D10566 Pasireotide pamoate (JAN) <JP/US>
|
SSTR2 [HSA:6752] [KO:K04218]
|
D00442 Octreotide (USAN/INN)
D02250 Octreotide acetate (JAN) <JP>
D05230 Octreotide pamoate (USAN)
D06495 Octreotide acetate (USP) <US>
D11204 Octreotide hydrochloride (USAN)
D04666 Lanreotide acetate (JAN/USAN) <JP/US>
D06281 Vapreotide (USAN/INN)
D09988 Vapreotide acetate (USAN)
D10147 Pasireotide (USAN)
D10497 Pasireotide diaspartate <US>
D10566 Pasireotide pamoate (JAN) <JP/US>
D12477 Paltusotine (USAN/INN)
D12478 Paltusotine hydrochloride (JAN/USAN) <US>
D02108 Indium In 111 pentetreotide (USP) <JP/US>
D11651 Edotreotide gallium Ga-68 <US>
D11882 Copper Cu 64 dotatate <US>
D11033 Lutetium (177Lu) oxodotreotide (INN) <JP/US>
D11845 Tidutamab (USAN/INN)
D12431 Lutetium Lu177 edotreotide (USAN)
D12907 Actinium Ac 225 dotatate (USAN)
|
SSTR3 [HSA:6753] [KO:K04219]
|
D10147 Pasireotide (USAN)
D10497 Pasireotide diaspartate <US>
D10566 Pasireotide pamoate (JAN) <JP/US>
D02108 Indium In 111 pentetreotide (USP) <JP/US>
|
SSTR5 [HSA:6755] [KO:K04221]
|
D04666 Lanreotide acetate (JAN/USAN) <JP/US>
D06281 Vapreotide (USAN/INN)
D09988 Vapreotide acetate (USAN)
D10147 Pasireotide (USAN)
D10497 Pasireotide diaspartate <US>
D10566 Pasireotide pamoate (JAN) <JP/US>
D02108 Indium In 111 pentetreotide (USP) <JP/US>
|
Tachykinin
|
TACR1 (NK1R) [HSA:6869] [KO:K04222]
|
D02968 Aprepitant (JAN/USP/INN) <JP/US>
D10895 Fosaprepitant (INN)
D06597 Fosaprepitant dimeglumine (USAN) <JP/US>
D06574 Casopitant mesylate (USAN)
D10742 Rolapitant (USAN/INN)
D08988 Rolapitant hydrochloride (USAN) <US>
D12123 Elinzanetant (USAN/INN)
D03221 Befetupitant (USAN/INN)
D04122 Ezlopitant (USAN/INN)
D04860 Maropitant citrate (USAN)
D05152 Netupitant (USAN/INN)
D06293 Vestipitant mesylate (USAN)
D06317 Vofopitant dihydrochloride (USAN)
D09378 Serlopitant (USAN)
D09650 Orvepitant (USAN/INN)
D09651 Orvepitant maleate (USAN)
D10391 Telmapitant (USAN/INN)
D11065 Fosnetupitant (USAN/INN)
D11370 Fosnetupitant chloride hydrochloride (JAN/USAN) <JP>
D11728 Tradipitant (USAN/INN)
|
TACR3 (NK3R) [HSA:6870] [KO:K04224]
|
D11976 Fezolinetant (JAN/USAN) <US>
D12123 Elinzanetant (USAN/INN)
D05996 Talnetant hydrochloride (USAN)
D11345 Pavinetant (USAN/INN)
|
Thrombin
|
F2R (PAR1) [HSA:2149] [KO:K03914]
|
D09765 Vorapaxar (USAN/INN)
D09766 Vorapaxar sulfate (JAN/USAN)
D09866 Atopaxar (USAN)
D09867 Atopaxar hydrobromide (USAN)
|
Thyrotropin-releasing hormone
|
TRHR [HSA:7201] [KO:K04282]
|
D06120 Thyrotropin alfa (USAN/INN) <JP/US>
D00176 Protirelin (JP18/USAN/INN) <JP>
D02007 Protirelin tartrate hydrate (JP18) <JP>
D01925 Taltirelin hydrate (JP18) <JP>
D02588 Montirelin (INN)
D09845 Montirelin hydrate (JAN)
D10594 Rovatirelin hydrate (JAN)
|
Vasopressin
|
AVPR1 [HSA:552 553] [KO:K04226 K04227]
|
D00101 Vasopressin (JP18/USP) <JP/US>
D09820 Vasopressin tannate (JAN)
D02983 Argipressin tannate (USAN)
D00366 Lypressin (USAN/INN)
D06672 Terlipressin (USAN/INN)
D08571 Terlipressin acetate (JAN) <US>
D07227 Ornipressin (INN)
|
AVPR1A [HSA:552] [KO:K04226]
|
D07748 Conivaptan (INN)
D01236 Conivaptan hydrochloride (JAN/USAN)
D04137 Felypressin (USAN/INN)
D11476 Balovaptan (USAN/INN)
|
AVPR2 [HSA:554] [KO:K04228]
|
D01213 Tolvaptan (JP18/USAN/INN) <JP/US>
D11659 Tolvaptan sodium phosphate (JAN) <JP>
D07748 Conivaptan (INN)
D01236 Conivaptan hydrochloride (JAN/USAN)
D00101 Vasopressin (JP18/USP) <JP/US>
D09820 Vasopressin tannate (JAN)
D02983 Argipressin tannate (USAN)
D00291 Desmopressin (INN)
D02235 Desmopressin acetate (USP) <JP/US>
D00366 Lypressin (USAN/INN)
D06672 Terlipressin (USAN/INN)
D08571 Terlipressin acetate (JAN) <US>
D07227 Ornipressin (INN)
D01855 Mozavaptane hydrochloride (JAN)
D04752 Lixivaptan (USAN/INN)
|
Purine / pyrimidine
|
P2RY2 [HSA:5029] [KO:K04269]
|
D03864 Diquafosol tetrasodium (USAN) <JP>
D03685 Denufosol tetrasodium (USAN)
|
P2RY12 [HSA:64805] [KO:K04298]
|
D07729 Clopidogrel (USP/INN)
D00769 Clopidogrel bisulfate (USP) <JP/US>
D10823 Clopidogrel hydrochloride
D10824 Clopidogrel besilate
D08594 Ticlopidine (INN)
D01028 Ticlopidine hydrochloride (JP18/USP) <JP>
D05597 Prasugrel hydrochloride (JAN/USAN) <JP/US>
D09017 Ticagrelor (JAN/USAN/INN) <JP/US>
D03359 Cangrelor (USAN/INN)
D03361 Cangrelor tetrasodium (USAN) <US>
D08983 Regrelor disodium (USAN)
D09607 Elinogrel (USAN/INN)
D09608 Elinogrel potassium (USAN)
D12979 Sumecigrel (USAN/INN)
|
Adenosine
|
ADORA [HSA:134 135 136 140] [KO:K04265 K04266 K04267 K04268]
|
D00045 Adenosine (JAN/USP) <JP/US>
D02300 Adenosine triphosphate disodium hydrate (JAN) <JP>
D02769 Adenosine phosphate (USAN/INN)
D08646 Triphosadenine (DCF)
D08647 Triphosadenine disodium salt
|
ADORA1 [HSA:134] [KO:K04265]
|
D00528 Caffeine (USP) <JP>
D01453 Caffeine hydrate (JP18) <JP>
D07603 Caffeine citrate (USP) <US>
D00691 Dyphylline (USP) <JP>
D02017 Oxtriphylline (USP)
D01771 Proxyphylline (JAN/INN)
D00371 Theophylline (JP18) <JP/US>
D01712 Theophylline sodium acetate (JAN)
D06103 Theophylline (USP)
D06104 Theophylline sodium glycinate (USP)
D00227 Aminophylline (USP/INN)
D05429 Aminophylline hydrate (JP18) <JP>
D11630 Aminophylline dihydrate <US>
D07491 Bamifylline (INN)
D03051 Bamifylline hydrochloride (USAN)
D02964 Apaxifylline (USAN/INN)
D04006 Enprofylline (USAN/INN)
D05125 Naxifylline (USAN/INN)
D05818 Selodenoson (USAN/INN)
D06019 Tecadenoson (USAN/INN)
D08989 Rolofylline (USAN)
D09684 Tonapofylline (USAN/INN)
D10493 Trabodenoson (USAN/INN)
|
ADORA2 [HSA:135 136] [KO:K04266 K04267]
|
D01771 Proxyphylline (JAN/INN)
D04006 Enprofylline (USAN/INN)
D12369 Etrumadenant (USAN/INN)
|
ADORA2A [HSA:135] [KO:K04266]
|
D12568 Regadenoson (INN) <US>
D05711 Regadenoson (USAN) <US>
D00528 Caffeine (USP) <JP>
D01453 Caffeine hydrate (JP18) <JP>
D07603 Caffeine citrate (USP) <US>
D04641 Istradefylline (JAN/USAN/INN) <JP/US>
D02017 Oxtriphylline (USP)
D03898 Doxofylline (USAN/INN)
D03120 Binodenoson (USAN/INN)
D03212 Apadenoson (USAN)
D09003 Sonedenoson (USAN)
D09717 Preladenant (USAN/INN)
D09991 Vipadenant (USAN/INN)
D10174 Tozadenant (USAN)
D10362 Evodenoson (USAN/INN)
D11547 Ciforadenant (USAN)
D11978 Inupadenant (USAN)
D11979 Inupadenant hydrochloride (USAN)
|
ADORA2B [HSA:136] [KO:K04267]
|
D00691 Dyphylline (USP) <JP>
D00371 Theophylline (JP18) <JP/US>
D01712 Theophylline sodium acetate (JAN)
D06103 Theophylline (USP)
D06104 Theophylline sodium glycinate (USP)
D00227 Aminophylline (USP/INN)
D05429 Aminophylline hydrate (JP18) <JP>
D11630 Aminophylline dihydrate <US>
|
ADORA3 [HSA:140] [KO:K04268]
|
D10971 Piclidenoson (USAN/INN)
D11128 Namodenoson (USAN/INN)
|
Cysteinyl leukotriene
|
CYSLTR1 [HSA:10800] [KO:K04322]
|
D00411 Zafirlukast (JAN/USAN/INN) <US>
D08408 Pranlukast (INN)
D02732 Pranlukast hydrate (JP18) <JP>
D08229 Montelukast (INN)
D00529 Montelukast sodium (JP18/USP) <JP/US>
D01385 Ibudilast (JP18/INN) <JP>
D02384 Verlukast (USAN/INN)
D02739 Ablukast (USAN/INN)
D02741 Ablukast sodium (USAN)
D02846 Cinalukast (USAN/INN)
D02848 Pobilukast edamine (USAN)
D02849 Ritolukast (USAN/INN)
D02850 Sulukast (USAN/INN)
D02851 Tomelukast (USAN/INN)
D06659 Tipelukast (USAN)
|
Free fatty acid
|
FFAR1 [HSA:2864] [KO:K04325]
|
D10336 Fasiglifam (USAN/INN)
D10567 Fasiglifam hydrate (JAN)
|
Leukotriene
|
LTB4R [HSA:1241 56413] [KO:K04296 K04297]
|
D04074 Etalocib (USAN)
D05085 Moxilubant maleate (USAN)
D06140 Ticolubant (USAN/INN)
|
Lysophosphatidic acid
|
LPAR1 [HSA:1902] [KO:K04289]
|
D12642 Fipaxalparant (USAN/INN)
D12657 Admilparant (USAN)
|
Oleoylethanolamide
|
GPR119 [HSA:139760] [KO:K08424]
|
D13209 Vanoglipel (USAN)
|
Prostaglandin
|
PTGDR [HSA:5729] [KO:K04332]
|
D01128 Ramatroban (JAN/INN) <JP>
D08940 Laropiprant (INN/USAN)
D09990 Vidupiprant (USAN/INN)
D10326 Setipiprant (USAN/INN)
D10631 Fevipiprant (JAN/USAN/INN)
|
PTGER1 [HSA:5731] [KO:K04258]
|
D02722 Limaprost (INN)
D02860 Limaprost alfadex (JP18) <JP>
D00180 Alprostadil (JP18/USP/INN) <JP/US>
D02705 Alprostadil alfadex (JP18) <JP>
D02073 Gemeprost (JAN/USAN/INN) <JP>
D01869 Ornoprostil (JAN/INN)
D02723 Ecraprost (USAN/INN)
D03999 Enisoprost (USAN/INN)
|
PTGER2 [HSA:5732] [KO:K04259]
|
D00419 Misoprostol (JAN/USP/INN) <JP/US>
D01891 Enprostil (JAN/USAN/INN)
D00079 Dinoprostone (JAN/USP/INN) <JP/US>
D03269 Dinoprostone betadex (JAN)
D02725 Sulprostone (USAN/INN)
D10965 Omidenepag (USAN/INN)
D10966 Omidenepag isopropyl (JAN) <JP/US>
D02726 Meteneprost (USAN/INN)
D02975 Arbaprostil (USAN/INN)
D03187 Butaprost (USAN/INN)
D05732 Rioprostil (USAN/INN)
D06240 Trimoprostil (USAN/INN)
D09613 Evatanepag (USAN/INN)
D09614 Evatanepag sodium (USAN)
D09968 Taprenepag (USAN/INN)
D09969 Taprenepag isopropyl (USAN)
|
PTGER3 [HSA:5733] [KO:K04260]
|
D00419 Misoprostol (JAN/USP/INN) <JP/US>
D01891 Enprostil (JAN/USAN/INN)
D12617 Sepetaprost (JAN/INN) <JP>
|
PTGER4 [HSA:5734] [KO:K04261]
|
D00419 Misoprostol (JAN/USP/INN) <JP/US>
D10638 Grapiprant (USAN/INN)
D12971 Vorbipiprant (USAN/INN)
D12972 Vorbipiprant sodium (USAN)
|
PTGFR [HSA:5737] [KO:K04262]
|
D00081 Dinoprost (JP18/USAN/INN) <JP>
D01352 Dinoprost tromethamine (JAN/USP)
D02343 Carboprost (USAN/INN)
D00682 Carboprost tromethamine (USP) <US>
D03399 Carboprost methyl (USAN)
D00356 Latanoprost (JAN/USP/INN) <JP/US>
D08661 Unoprostone (INN)
D01452 Isopropyl unoprostone (JAN) <JP>
D02724 Bimatoprost (JAN/USAN/INN) <JP/US>
D12599 Bimatoprost grenod (USAN)
D01964 Travoprost (JAN/USP/INN) <JP/US>
D06274 Tafluprost (JAN/USAN/INN) <JP/US>
D10441 Latanoprostene bunod (USAN/INN) <US>
D02719 Rosaprostol (INN)
D02727 Cloprostenol sodium (USP)
D05642 Prostalene (USAN)
D07730 Cloprostenol (INN)
D07932 Etiproston (INN)
D08591 Tiaprost (INN)
D12617 Sepetaprost (JAN/INN) <JP>
|
Prostacyclin
|
PTGIR [HSA:5739] [KO:K04263]
|
D00106 Epoprostenol (USAN/INN)
D01337 Epoprostenol sodium (JAN/USAN) <JP/US>
D02721 Iloprost (USAN/INN) <US>
D08065 Iloprost tromethamine
D02720 Beraprost (USAN)
D01551 Beraprost sodium (JP18/USAN) <JP>
D06213 Treprostinil (JAN/USAN/INN) <JP/US>
D08628 Treprostinil monosodium salt <US>
D10430 Treprostinil diolamine (USAN) <US>
D12005 Treprostinil palmitil (USAN/INN)
D12629 Treprostinil phosphate (USAN)
D09994 Selexipag (JAN/USAN/INN) <JP/US>
D01385 Ibudilast (JP18/INN) <JP>
D01188 Pimilprost (JAN/INN)
D02048 Clinprost (JAN/INN)
D03522 Ciprostene calcium (USAN)
D10628 Esuberaprost (USAN/INN)
D10703 Esuberaprost sodium (USAN)
D10725 Ralinepag (USAN/INN)
D11446 Esuberaprost potassium (USAN)
|
Sphingolipid
|
S1PR [HSA:1901 9294 1903 8698 53637] [KO:K04288 K04292 K04290 K04293 K04295]
|
D10968 Ozanimod (USAN/INN)
D10967 Ozanimod hydrochloride (JAN/USAN) <JP/US>
D10904 Amiselimod hydrochloride (USAN)
D10905 Amiselimod (USAN/INN)
|
S1PR1 [HSA:1901] [KO:K04288]
|
D10001 Fingolimod (INN)
D04187 Fingolimod hydrochloride (JAN/USAN) <JP/US>
D11460 Siponimod (USAN/INN)
D11072 Siponimod fumarate (USAN) <JP/US>
D11215 Ponesimod (USAN/INN) <US>
D10930 Etrasimod (USAN)
D10931 Etrasimod arginine (USAN) <JP/US>
D11283 Cenerimod (JAN/USAN/INN)
D12376 Udifitimod (USAN)
D12377 Udifitimod hydrochloride (USAN)
D12549 Fingolimod lauryl sulfate <US>
D12771 Mocravimod (USAN/INN)
D12772 Mocravimod hydrochloride (USAN)
D12897 Tamuzimod (USAN/INN)
D13175 Vibozilimod (USAN/INN)
D13176 Vibozilimod potassium (USAN)
|
S1PR4 [HSA:8698] [KO:K04293]
|
D10930 Etrasimod (USAN)
D10931 Etrasimod arginine (USAN) <JP/US>
|
S1PR5 [HSA:53637] [KO:K04295]
|
D11460 Siponimod (USAN/INN)
D11072 Siponimod fumarate (USAN) <JP/US>
D10930 Etrasimod (USAN)
D10931 Etrasimod arginine (USAN) <JP/US>
|
Thromboxane
|
TBXA2R [HSA:6915] [KO:K04264]
|
D07140 Picotamide (BAN)
D01896 Cilostazol (JP18/USP/INN) <JP/US>
D01123 Seratrodast (JAN/USAN/INN)
D01128 Ramatroban (JAN/INN) <JP>
D03642 Daltroban (USAN/INN)
D04500 Ifetroban (USAN/INN)
D04501 Ifetroban sodium (USAN)
D05727 Ridogrel (USAN/INN)
D05970 Sulotroban (USAN/INN)
D06077 Terbogrel (USAN/INN)
D06280 Vapiprost hydrochloride (JAN/USAN)
D09774 Imitrodast sodium (JAN)
D09824 Domitroban calcium hydrate (JAN)
|
Cannabinoid
|
CNR [HSA:1268 1269] [KO:K04277 K04278]
|
D00306 Dronabinol (USP/INN) <US>
D05099 Nabilone (USAN/INN) <US>
D10915 Cannabidiol (JAN/USAN/INN) <US>
D12305 Onternabez (USAN)
|
CNR1 [HSA:1268] [KO:K04277]
|
D05731 Rimonabant (JAN/USAN/INN)
D04717 Levonantradol hydrochloride (USAN)
D05117 Nantradol hydrochloride (USAN)
D09009 Taranabant (USAN/INN)
D09349 Ibipinabant (USAN/INN)
D09362 Otenabant (USAN/INN)
D09363 Otenabant hydrochloride (USAN)
D11435 Nimacimab (USAN)
D12875 Selonabant (USAN)
|
CNR2 [HSA:1269] [KO:K04278]
|
D11312 Lenabasum (USAN/INN)
D11429 Olorinab (USAN/INN)
D12511 Vicasinabin (USAN/INN)
|
Melatonin
|
MTNR1 [HSA:4543 4544] [KO:K04285 K04286]
|
D08170 Melatonin (JAN) <JP>
D02689 Ramelteon (JAN/USAN/INN) <JP/US>
D09388 Tasimelteon (USAN/INN) <US>
D02578 Agomelatine (INN)
|
Platelet activating factor
|
PTAFR [HSA:5724] [KO:K04279]
|
D07407 Rupatadine (USAN/INN)
D08497 Rupatadine fumarate (JAN/USAN) <JP>
D01652 Apafant (JAN/USAN/INN)
D02590 Israpafant (JAN/INN)
D04724 Lexipafant (USAN/INN)
|
R-spondin
|
LGR5 [HSA:8549] [KO:K04308]
|
D12416 Petosemtamab (USAN/INN)
|
Orphan GPCR
|
GPR6 [HSA:2830] [KO:K04313]
|
D12980 Solengepras (USAN)
|
Secretin receptor family
|
Calcitonin
|
CALCR [HSA:799] [KO:K04576]
|
D05594 Pramlintide (USAN/INN)
D05595 Pramlintide acetate (USAN) <US>
D00249 Calcitonin salmon (JP18/USP/INN) <US>
D03287 Elcatonin (JP18/INN) <JP>
D02913 Amlintide (USAN/INN)
D09600 Davalintide (USAN/INN)
D09601 Davalintide acetate (USAN)
D09771 Avicatonin (JAN/INN)
D12886 Eloralintide (USAN)
|
CALCRL [HSA:10203] [KO:K04577]
|
D05594 Pramlintide (USAN/INN)
D05595 Pramlintide acetate (USAN) <US>
D10928 Erenumab (USAN/INN) <JP/US>
D10673 Ubrogepant (USAN/INN) <US>
D10662 Rimegepant (USAN/INN)
D10663 Rimegepant sulfate (USAN) <JP/US>
D11313 Atogepant (USAN) <US>
D13026 Atogepant hydrate (JAN)
D11898 Zavegepant (USAN)
D11899 Zavegepant hydrochloride (USAN) <US>
D02913 Amlintide (USAN/INN)
D09391 Telcagepant (USAN)
D09392 Telcagepant potassium (USAN)
D09600 Davalintide (USAN/INN)
D09601 Davalintide acetate (USAN)
D12886 Eloralintide (USAN)
|
Parathyroid hormone
|
PTH1R [HSA:5745] [KO:K04585]
|
D06078 Teriparatide (USP/INN) <JP/US>
D03358 Teriparatide acetate (JAN) <JP>
D06546 Teriparatide acetate (USAN) <US>
D05364 Parathyroid hormone (human) (USAN) <US>
D10885 Abaloparatide (USAN/INN) <US>
D11563 Abaloparatide acetate (JAN) <JP>
D12395 Palopegteriparatide (JAN/USAN/INN) <JP/US>
D05821 Semparatide acetate (USAN)
D12805 Eneboparatide (USAN/INN)
|
PTH2R [HSA:5746] [KO:K04586]
|
D05364 Parathyroid hormone (human) (USAN) <US>
|
Corticotropin-releasing hormone
|
CRHR [HSA:1394 1395] [KO:K04578 K04579]
|
D03905 Corticorelin (human) (JAN) <JP>
D03591 Corticorelin acetate (USAN)
D03592 Corticorelin ovine triflutate (USAN)
|
CRHR1 [HSA:1394] [KO:K04578]
|
D09610 Emicerfont (USAN/INN)
D09695 Verucerfont (USAN/INN)
D10022 Pexacerfont (USAN/INN)
D12366 Crinecerfont (USAN) <US>
D12761 Tildacerfont (USAN/INN)
|
Growth hormone-releasing hormone
|
GHRHR [HSA:2692] [KO:K04584]
|
D08509 Sermorelin (INN)
D02117 Sermorelin acetate (USAN)
D06655 Tesamorelin (USAN)
D09015 Tesamorelin acetate (USAN) <US>
D08523 Somatorelin (INN)
D03326 Somatorelin acetate (JAN)
D04491 Ibutamoren mesylate (USAN)
|
Glucagon
|
GLP1R [HSA:2740] [KO:K04581]
|
D11034 Insulin glargine and lixisenatide <JP/US>
D11567 Insulin degludec and liraglutide <JP/US>
D04121 Exenatide (JAN/USAN/INN) <US>
D06404 Liraglutide (USAN/INN) <JP/US>
D09729 Lixisenatide (JAN/USAN/INN)
D08843 Albiglutide (USAN)
D09889 Dulaglutide (USAN/INN) <JP/US>
D10025 Semaglutide (USAN/INN) <JP/US>
D11924 Beinaglutide (INN)
D11360 Tirzepatide (JAN/USAN) <JP/US>
D09723 Taspoglutide (USAN/INN)
D10970 Pegapamodutide (USAN/INN)
D11304 Cotadutide (USAN/INN)
D11418 Avexitide (USAN/INN)
D11419 Avexitide acetate (USAN)
D11607 Efinopegdutide (USAN/INN)
D11910 Danuglipron (USAN)
D11911 Danuglipron tromethamine (USAN)
D11947 Efpeglenatide (USAN/INN)
D12225 Mazdutide (USAN/INN)
D12341 Vurolenatide (USAN/INN)
D12430 Retatrutide (USAN)
D12529 Orforglipron calcium (JAN/USAN)
D12536 Orforglipron (USAN)
D12555 Lotiglipron (USAN)
D12735 Lotiglipron tromethamine (USAN)
D12861 Pemvidutide (USAN/INN)
D12898 Survodutide (USAN/INN)
D13181 Naperiglipron (USAN)
D13182 Naperiglipron erbumine (USAN)
|
GLP2R [HSA:9340] [KO:K04582]
|
D06053 Teduglutide (USAN/INN) <JP/US>
D11337 Glepaglutide (USAN)
D12903 Apraglutide (INN)
D12904 Apraglutide sodium (JAN)
|
GCGR [HSA:2642] [KO:K04583]
|
D00116 Glucagon (USP/INN) <JP/US>
D02118 Glucagon hydrochloride <US>
D11359 Dasiglucagon (USAN)
D12314 Dasiglucagon hydrochloride <US>
D11230 Crotedumab (USAN/INN)
D11304 Cotadutide (USAN/INN)
D11607 Efinopegdutide (USAN/INN)
D11614 Volagidemab (USAN/INN)
D12225 Mazdutide (USAN/INN)
D12430 Retatrutide (USAN)
D12861 Pemvidutide (USAN/INN)
D12898 Survodutide (USAN/INN)
|
Gastric inhibitory polypeptide
|
GIPR [HSA:2696] [KO:K04580]
|
D11360 Tirzepatide (JAN/USAN) <JP/US>
D12430 Retatrutide (USAN)
|
Secretin
|
SCTR [HSA:6344] [KO:K04588]
|
D02021 Secretin (JAN/USAN/INN) <US>
|
Metabotropic glutamate receptor family
|
Glutamate (metabotropic)
|
GRM2 [HSA:2912] [KO:K04605]
|
D03966 Eglumetad (USAN)
D08908 Eglumegad (INN)
D09008 Talaglumetad hydrochloride (USAN)
D09949 Pomaglumetad methionil (USAN)
D10896 Pomaglumetad methionil (INN)
|
GRM3 [HSA:2913] [KO:K04606]
|
D09008 Talaglumetad hydrochloride (USAN)
D09949 Pomaglumetad methionil (USAN)
D10896 Pomaglumetad methionil (INN)
|
GRM5 [HSA:2915] [KO:K04604]
|
D04155 Fenobam (USAN)
|
GABA (metabotropic)
|
GABBR [HSA:2550 9568] [KO:K04615]
|
D00241 Baclofen (JP18/USP/INN) <JP/US>
D00058 gamma-Aminobutyric acid (JAN) <JP>
D05621 Progabide (USAN/INN)
D08861 Arbaclofen placarbil (USAN/INN)
D09791 Arbaclofen (USAN)
D12240 Valiloxybate (USAN)
|
Chemoreception
|
TAS1R2 [HSA:80834] [KO:K04625]
|
D02381 Aspartame (NF/INN)
D08836 Acesulfame potassium (NF)
D08862 Aspartame acesulfame (NF)
|
TAS1R3 [HSA:83756] [KO:K04626]
|
D02381 Aspartame (NF/INN)
D08836 Acesulfame potassium (NF)
D08862 Aspartame acesulfame (NF)
|
Calcium-sensing
|
CASR [HSA:846] [KO:K04612]
|
D03504 Cinacalcet (USAN)
D03505 Cinacalcet hydrochloride (JAN/USAN) <JP/US>
D10676 Etelcalcetide (USAN/INN)
D10677 Etelcalcetide hydrochloride (JAN/USAN) <JP/US>
D11063 Evocalcet (JAN/INN) <JP>
D06020 Tecalcet hydrochloride (USAN)
D08991 Ronacaleret hydrochloride (USAN)
D11564 Upacicalcet sodium hydrate (JAN) <JP>
D12917 Upacicalcet sodium (USAN)
D12918 Upacicalcet (USAN/INN)
|
Orphan GPRC5
|
GPRC5D [HSA:55507] [KO:K04621]
|
D12180 Talquetamab (USAN/INN) <JP/US>
D12724 Forimtamig (USAN/INN)
|
Frizzled / Smoothened family
|
Frizzled
|
FZD7 [HSA:8324] [KO:K02432]
|
D10410 Vantictumab (USAN/INN)
|
FZD8 [HSA:8325] [KO:K02375]
|
D11758 Ipafricept (USAN/INN)
|
Smoothened
|
SMO [HSA:6608] [KO:K06226]
|
D09992 Vismodegib (USAN/INN) <US>
D10119 Sonidegib (USAN/INN)
D10729 Sonidegib phosphate (USAN) <US>
D10636 Glasdegib (USAN/INN)
D11107 Glasdegib maleate (JAN) <US>
D10324 Patidegib (USAN/INN)
D10325 Patidegib hydrochloride (USAN)
D10671 Taladegib (USAN/INN)
|
Others
|
Vomeronasal pheromone
|
V1R [HSA:57191 317701 317702 317703 317705] [KO:K04614]
|
D12524 Fasedienol (USAN/INN)
|
|
Ion channels
|
Ligand-gated ion channels
|
Acetylcholine (nicotinic)
|
CHRN [HSA:1134 1135 1136 1137 1138 8973 1139 55584 57053 1140 1141 1142 1143 1144 1145 1146] [KO:K04803 K04804 K04805 K04806 K04807 K04808 K04809 K04810 K04811 K04812 K04813 K04814 K04815 K04816 K04817 K04818]
|
D00611 Mecamylamine hydrochloride (USP) <US>
D03365 Nicotine (USP) <JP/US>
D05156 Nicotine bitartrate (USAN)
D05157 Nicotine polacrilex (USP)
D07770 Cytisinicline (USAN)
D00999 Acetylcholine chloride (JP18/USP/INN) <JP/US>
D02202 Lobeline hydrochloride (JAN)
D02364 Lobeline (INN)
D08138 Lobeline sulfate
|
CHRN (muscle type) [HSA:1134 1140 1144 1145 1146] [KO:K04803 K04812 K04816 K04817 K04818]
|
D00766 Succinylcholine chloride (USP) <US>
D02275 Suxamethonium chloride hydrate (JP18) <JP>
D00761 Metocurine iodide (USAN)
D04303 Gantacurium chloride (USAN/INN)
|
CHRN (neuronal type) [HSA:1135 1136 1137 1138 8973 1139 55584 57053 1141 1142 1143] [KO:K04804 K04805 K04806 K04807 K04808 K04809 K04810 K04811 K04813 K04814 K04815]
|
D02207 Tubocurarine chloride (USP)
D08655 Tubocurarine chloride (INN)
D07272 Dimethyltubocurarine (BAN)
D00492 Pancuronium bromide (JP18/USP/INN)
D00767 Vecuronium bromide (JAN/USP/INN) <US>
D00758 Atracurium besylate (USP) <US>
D00764 Pipecuronium bromide (JAN/USAN/INN)
D00760 Doxacurium chloride (USAN/INN)
D07273 Fazadinium bromide (INN)
D00765 Rocuronium bromide (JAN/USP/INN) <JP/US>
D00763 Mivacurium chloride (USAN/INN)
D00759 Cisatracurium besylate (USP) <US>
D02204 Hexamethonium bromide (JAN/INN)
|
CHRNA7 [HSA:1139] [KO:K04809]
|
D10613 Bradanicline (USAN/INN)
D10626 Encenicline (USAN/INN)
D10693 Bradanicline hydrochloride (USAN)
D10702 Encenicline hydrochloride (USAN)
D10789 Encenicline hydrochloride hydrate (JAN)
|
CHRNA10 [HSA:57053] [KO:K04811]
|
D00612 Trimetaphan camsilate (JAN/INN)
|
CHRNA3/CHRNB4 [HSA:1136 1143] [KO:K04805 K04815]
|
D06016 Tebanicline tosylate (USAN)
|
CHRNA4/CHRNB2 [HSA:1137 1141] [KO:K04806 K04813]
|
D08669 Varenicline (INN)
D06282 Varenicline tartrate (JAN/USAN) <JP/US>
D02839 Altinicline maleate (USAN)
D06016 Tebanicline tosylate (USAN)
D08935 Ispronicline (INN/USAN)
D08987 Rivanicline galactarate (USAN)
D09367 Pozanicline (USAN)
D09368 Pozanicline tartrate (USAN)
D09382 Sofinicline (USAN)
D09383 Sofinicline benzenesulfonate (USAN)
D10111 Dexmecamylamine (USAN)
D10112 Dexmecamylamine hydrochloride (USAN)
|
Serotonin
|
HTR3 [HSA:3359 9177 170572 200909 285242] [KO:K04819]
|
D07129 Alosetron (INN)
D02829 Alosetron hydrochloride (USAN) <US>
D03495 Cilansetron (USAN/INN)
D03496 Cilansetron hydrochloride (USAN)
D00456 Ondansetron (JAN/USP/INN) <US>
D00678 Ondansetron hydrochloride hydrate (JAN/USP) <JP/US>
D02130 Tropisetron (INN)
D02041 Tropisetron hydrochloride (JAN)
D07867 Dolasetron (INN)
D00725 Dolasetron mesylate (USP)
D07175 Palonosetron (INN)
D05343 Palonosetron hydrochloride (JAN/USP) <JP/US>
D00283 Clozapine (JAN/USP/INN) <JP/US>
D08216 Mianserin (INN)
D01358 Mianserin hydrochloride (JAN/USAN) <JP>
D00563 Mirtazapine (JAN/USP/INN) <JP/US>
D11056 Mirtazapine hydrate (JAN)
D10184 Vortioxetine (USAN)
D10185 Vortioxetine hydrobromide (JAN/USAN) <JP/US>
D12544 Vortioxetine hemihydrobromide (USAN)
D01613 Azasetron hydrochloride (JAN)
D01838 Fabesetron hydrochloride (JAN)
D02016 Ramosetron hydrochloride (JAN) <JP>
D02632 Indisetron hydrochloride (JAN)
D03060 Batanopride hydrochloride (USAN)
D03073 Bemesetron (USAN/INN)
D03662 Dazopride fumarate (USAN)
D04294 Galdansetron hydrochloride (USAN)
D04642 Itasetron (USAN/INN)
D04821 Lurosetron mesylate (USAN)
D05050 Mirisetron maleate (USAN)
D05348 Pancopride (USAN/INN)
D05685 Quipazine maleate (USAN)
D06253 Tropanserin hydrochloride (USAN)
D06353 Zacopride hydrochloride (USAN)
D06358 Zatosetron maleate (USAN)
D06396 Renzapride (INN)
D07481 Azasetron (INN)
D08466 Ramosetron (INN)
D09749 Itasetron hydrochloride hydrate (JAN)
D10170 Tedatioxetine (USAN)
D10171 Tedatioxetine hydrobromide (USAN)
|
HTR3A [HSA:3359] [KO:K04819]
|
D00274 Cisapride (USP/INN)
D02092 Cisapride (JAN)
|
HTR3B [HSA:9177] [KO:K04819]
|
D04370 Granisetron (JAN/USAN/INN) <US>
D00677 Granisetron hydrochloride (JAN/USP) <JP/US>
|
GABA (ionotropic)
|
GABR [HSA:2554 2555 2556 2557 2558 2559 2560 2561 2562 2563 2564 2565 2566 2567 2568 55879] [KO:K05175 K05181 K05184 K05185 K05186 K05189 K05192]
|
D01071 Hexobarbital (JAN/INN)
D00714 Thiopental sodium (JP18/USP/INN) <JP>
D00549 Propofol (JAN/USP/INN) <JP/US>
D04257 Fospropofol disodium (USAN)
D00700 Mephobarbital (JAN/USP)
D00506 Phenobarbital (JP18/USP/INN) <JP>
D00701 Phenobarbital sodium (JAN/USP/INN) <JP/US>
D08356 Phenobarbital diethylamine
D07298 Barbexaclone (INN)
D01382 Metharbital (JAN/INN)
D00280 Clonazepam (JP18/USP/INN) <JP/US>
D00058 gamma-Aminobutyric acid (JAN) <JP>
D00537 Topiramate (JAN/USP/INN) <JP/US>
D11150 Cenobamate (JAN/USAN/INN) <US>
D04300 Ganaxolone (USAN/INN) <US>
D00293 Diazepam (JP18/USP/INN) <JP/US>
D00267 Chlordiazepoxide (JP18/USP/INN) <JP>
D00693 Chlordiazepoxide hydrochloride (JAN/USP) <US>
D01292 Medazepam (JP18/INN) <JP>
D04882 Medazepam hydrochloride (USAN)
D00464 Oxazepam (JAN/USP/INN) <US>
D00694 Clorazepate dipotassium (JP18/USP) <JP/US>
D03562 Clorazepate monopotassium (USAN)
D00365 Lorazepam (JP18/USP/INN) <JP/US>
D02770 Adinazolam (USAN/INN)
D02771 Adinazolam mesylate (USAN)
D01245 Bromazepam (JP18/USAN/INN) <JP>
D01253 Clobazam (JAN/USAN/INN) <JP/US>
D04650 Ketazolam (USAN/INN)
D00470 Prazepam (JP18/USAN/INN)
D00225 Alprazolam (JP18/USP/INN) <JP/US>
D00338 Halazepam (USAN/INN)
D08283 Nordazepam (INN)
D01354 Fludiazepam (JP18/INN)
D01293 Ethyl loflazepate (JP18/INN) <JP>
D01514 Etizolam (JP18/INN) <JP>
D01328 Clotiazepam (JP18/INN) <JP>
D01268 Cloxazolam (JP18/INN) <JP>
D01254 Tofisopam (JP18/INN) <JP>
D01316 Mexazolam (JAN/INN) <JP>
D00376 Meprobamate (JAN/USP/INN) <US>
D00499 Pentobarbital (USP/INN)
D00500 Pentobarbital sodium (JAN/USP) <US>
D02253 Pentobarbital calcium (JP18) <JP>
D00555 Amobarbital (JP18/INN)
D02252 Amobarbital sodium (JAN/USP)
D02618 Butobarbital (BAN)
D01740 Barbital (JP18/INN)
D00698 Aprobarbital (INN)
D00430 Secobarbital (USP/INN)
D01310 Secobarbital sodium (JAN/USP)
D06887 Talbutal (INN)
D00329 Flurazepam (JAN/INN)
D00695 Flurazepam hydrochloride (USP) <US>
D01408 Flurazepam hydrochloride (JP18) <JP>
D00531 Nitrazepam (JP18/USAN/INN) <JP>
D01230 Flunitrazepam (JP18/USAN/INN) <JP>
D00311 Estazolam (JP18/USP/INN) <JP/US>
D00387 Triazolam (JP18/USP/INN) <JP/US>
D01657 Lormetazepam (JAN/USAN/INN) <JP>
D00370 Temazepam (USP/INN) <US>
D00550 Midazolam (JAN/USP/INN) <JP/US>
D00696 Midazolam hydrochloride (USAN) <US>
D05028 Midazolam maleate (USAN)
D01744 Brotizolam (JP18/USAN/INN) <JP>
D00457 Quazepam (JAN/USP/INN) <JP/US>
D07326 Loprazolam (INN)
D08145 Loprazolam mesilate
D07328 Cinolazepam (INN)
D11788 Remimazolam (USAN/INN)
D10194 Remimazolam besylate (USAN) <JP/US>
D01593 Nimetazepam (JAN/INN)
D13231 Dimdazenil (INN)
D00532 Glutethimide (JAN/INN)
D01372 Zopiclone (JP18/INN) <JP>
D08690 Zolpidem (INN)
D00706 Zolpidem tartrate (JP18/USP) <JP/US>
D02624 Eszopiclone (JAN/USP/INN) <JP/US>
D11149 Brexanolone (USAN/INN)
D11793 Zuranolone (JAN/USAN/INN) <US>
D00697 Flumazenil (JAN/USP/INN) <JP/US>
D00699 Butabarbital sodium (USP)
D00713 Thiamylal sodium (JP18) <JP>
D01278 Oxazolam (JP18/INN) <JP>
D01279 Flutoprazepam (JP18/INN)
D01286 Flutazolam (JAN/INN)
D01564 Rilmazafone hydrochloride hydrate (JP18) <JP>
D01758 Haloxazolam (JP18/INN) <JP>
D02283 Iomazenil (123I) (JAN/INN) <JP>
D02594 Abecarnil (INN)
D02616 Pagoclone (USAN/INN)
D02617 Ocinaplon (USAN/INN)
D02640 Indiplon (USAN/INN)
D02833 Alpidem (USAN/INN)
D03155 Bretazenil (USAN/INN)
D03180 Butabarbital (USP)
D03737 Dextofisopam (USAN/INN)
D04282 Gaboxadol (USAN/INN)
D04721 Levotofisopam (USAN/INN)
D05346 Panadiplon (USAN/INN)
D05378 Pazinaclone (USAN/INN)
D05980 Suritozole (USAN/INN)
D06106 Thiamylal
D07784 Delorazepam (INN)
D08481 Rilmazafone (INN)
D08507 Sarmazenil (INN)
D08840 Adipiplon (USAN)
D12146 Darigabat (USAN)
D12449 Cipepofol (USAN/INN)
|
GABRA1 [HSA:2554] [KO:K05175]
|
D04985 Methohexital (USP/INN)
D00712 Methohexital sodium (USP) <US>
D00548 Etomidate (USP/INN) <US>
D05621 Progabide (USAN/INN)
D01150 Methyprylon (JAN/INN)
D00530 Zaleplon (JAN/USP/INN) <US>
D07330 Clomethiazole (INN)
D07725 Clomethiazole edisilate
|
GABRA5 [HSA:2558] [KO:K05175]
|
D12382 Alogabat (USAN)
|
Glycine
|
GLRA1 [HSA:2741] [KO:K05193]
|
D10470 Strychnine nitrate
|
Glutamate (ionotropic), non-NMDA
|
GRIA [HSA:2890 2891 2892 2893] [KO:K05197 K05198 K05199 K05200]
|
D00537 Topiramate (JAN/USP/INN) <JP/US>
D08964 Perampanel (JAN/USAN)
D10780 Perampanel hydrate (JAN) <JP/US>
D00775 Riluzole (JAN/USP/INN) <JP/US>
D11414 Troriluzole (USAN)
D11415 Troriluzole hydrochloride (USAN)
D02696 Talampanel (INN)
D04131 Farampator (USAN/INN)
D06656 Tezampanel (USAN)
D09035 Zonampanel (INN/USAN)
D09931 Mibampator (USAN/INN)
D10107 Dasolampanel (USAN/INN)
D10108 Dasolampanel etibutil (USAN)
D10109 Dasolampanel etibutil tosylate (USAN)
D12239 Pesampator (USAN)
D13050 Osavampator (USAN/INN)
|
GRIK [HSA:2897 2898 2899 2900 2901] [KO:K05201 K05202 K05203 K05204 K05205]
|
D00537 Topiramate (JAN/USP/INN) <JP/US>
D00775 Riluzole (JAN/USP/INN) <JP/US>
D11414 Troriluzole (USAN)
D11415 Troriluzole hydrochloride (USAN)
D06656 Tezampanel (USAN)
D10107 Dasolampanel (USAN/INN)
D10108 Dasolampanel etibutil (USAN)
D10109 Dasolampanel etibutil tosylate (USAN)
|
Glutamate (ionotropic), NMDA
|
GRIN (NMDAR) [HSA:2902 2903 2904 2905 2906 116443 116444] [KO:K05208 K05209 K05210 K05211 K05212 K05213 K05214]
|
D00774 Orphenadrine citrate (USP) <US>
D00536 Felbamate (USPINN) <US>
D02599 Orphenadrine hydrochloride
D08305 Orphenadrine (INN)
D12788 Dalzanemdor (USAN/INN)
|
GRIN (NMDAR) [HSA:2902 2903 2904 2905 2906] [KO:K05208 K05209 K05210 K05211 K05212]
|
D08098 Ketamine (INN)
D00711 Ketamine hydrochloride (JP18/USP) <JP/US>
D07283 Esketamine (USAN/INN)
D10627 Esketamine hydrochloride (JAN/USAN) <US>
D07441 Amantadine (INN)
D00777 Amantadine hydrochloride (JP18/USP) <JP/US>
D07306 Budipine (INN)
D07589 Budipine hydrochloride
D08174 Memantine (INN)
D04905 Memantine hydrochloride (JAN/USP) <JP/US>
D07058 Acamprosate (INN)
D02780 Acamprosate calcium (JAN/USAN) <JP/US>
D08195 Methadone (BAN)
D02102 Methadone hydrochloride (JAN/USP) <JP/US>
D08121 Levomethadone (INN)
D08122 Levomethadone hydrochloride
D00775 Riluzole (JAN/USP/INN) <JP/US>
D11414 Troriluzole (USAN)
D11415 Troriluzole hydrochloride (USAN)
D03742 Dextromethorphan (USP)
D00848 Dextromethorphan hydrobromide (USP) <JP>
D03744 Dextromethorphan polistirex (USAN)
D02410 Selfotel (USAN/INN)
D02973 Aptiganel hydrochloride (USAN)
D03679 Delucemine hydrochloride (USAN)
D03746 Dextrorphan hydrochloride (USAN)
D03878 Dizocilpine maleate (USAN)
D04308 Gavestinel (USAN/INN)
D04728 Licostinel (USAN/INN)
D05447 Perzinfotel (USAN/INN)
D05453 Phencyclidine hydrochloride (USAN)
D05714 Remacemide hydrochloride (USAN)
D06146 Tiletamine hydrochloride (USP)
D08596 Tiletamine (INN)
D09917 Latrepirdine (USAN/INN)
D09918 Latrepirdine dihydrochloride (USAN)
D11299 Apimostinel (USAN)
D12214 Esmethadone (USAN)
D12215 Esmethadone hydrochloride (USAN)
D12553 Nevadistinel (USAN)
D12554 Risevistinel (USAN)
D12702 Tenocyclidine (INN)
|
GRIN2B (NMDAR2B) [HSA:2904] [KO:K05210]
|
D03100 Besonprodil (USAN)
D05145 Neramexane mesylate (USAN)
D06204 Traxoprodil mesylate (USAN)
D11340 Rislenemdaz (USAN)
D12787 Onfasprodil (USAN/INN)
|
Epithelial sodium channel (SCNN)
|
SCNN1 [HSA:6337 6338 6339 6340] [KO:K04824 K04825 K04826 K04827]
|
D12346 Idrevloride (USAN)
|
SCNN1 [HSA:6337 6338 6340] [KO:K04824 K04825 K04827]
|
D07447 Amiloride (INN)
D00649 Amiloride hydrochloride (USP) <US>
D00386 Triamterene (JP18/USP/INN) <JP/US>
|
ATP-gated cation channel (P2X)
|
P2RX3 [HSA:5024] [KO:K05217]
|
D11349 Gefapixant (USAN/INN)
D11693 Gefapixant citrate (JAN/USAN) <JP>
D12323 Eliapixant (USAN/INN)
D12355 Sivopixant (JAN/INN)
D12785 Camlipixant (JAN/USAN/INN)
|
P2RX7 [HSA:5027] [KO:K05220]
|
D10799 Brilliant blue G (JAN) <US>
|
Voltage-gated ion channels
|
Sodium channels
|
SCN1A [HSA:6323] [KO:K04833]
|
D08458 Quinidine (BAN)
D00642 Quinidine gluconate (USP) <US>
D00643 Quinidine polygalacturonate
D02272 Quinidine sulfate (USP) <JP/US>
D08459 Quinidine phenylethylbarbiturate
D08421 Procainamide (INN)
D00477 Procainamide hydrochloride (JP18/USP) <JP/US>
D00303 Disopyramide (JP18/USAN/INN) <JP>
D00637 Disopyramide phosphate (JAN/USP) <JP/US>
D01041 Sparteine (INN)
D02239 Sparteine sulfate (JAN/USAN)
D00199 Ajmaline (JP18)
D04774 Lorajmine hydrochloride (USAN)
D00358 Lidocaine (JP18/USP/INN) <JP/US>
D02086 Lidocaine hydrochloride (JAN/USP) <JP/US>
D08127 Lidocaine hydrochloride monohydrate <JP/US>
D08215 Mexiletine (INN)
D00639 Mexiletine hydrochloride (JP18/USP) <JP/US>
D06172 Tocainide (USAN/INN)
D02088 Tocainide hydrochloride (USP)
D02969 Aprindine (USAN/INN)
D01326 Aprindine hydrochloride (JP18/USAN) <JP>
D08435 Propafenone (INN)
D00640 Propafenone hydrochloride (JP18/USP) <JP/US>
D07962 Flecainide (INN)
D00638 Flecainide acetate (JP18/USP) <JP/US>
D07894 Encainide (INN)
D03991 Encainide hydrochloride (USAN)
D02910 Amiodarone (USAN/INN)
D00636 Amiodarone hydrochloride (JP18/USP) <JP/US>
D03492 Cifenline (USAN)
D01455 Cifenline succinate (USAN) <JP>
D00551 Tetracaine (USP/INN)
D00741 Tetracaine hydrochloride (JP18/USP) <US>
D00552 Benzocaine (USP/INN) <JP>
D00733 Dibucaine (USP)
D02220 Dibucaine hydrochloride (JP18/USP)
D08422 Procaine (INN)
D00740 Procaine hydrochloride (JP18/USP) <JP>
D01152 Oxethazaine (JP18/USAN) <JP>
D08311 Oxetacaine hydrochloride
D08407 Pramocaine (INN)
D00739 Pramoxine hydrochloride (USP)
D02456 Aminobenzoic acid (USP)
D02906 Aminobenzoate potassium (USP)
D02907 Aminobenzoate sodium (USP)
D08319 Oxybuprocaine (INN)
D01768 Benoxinate hydrochloride (USP) <JP>
D07678 Chloroprocaine (INN)
D00732 Chloroprocaine hydrochloride (USP) <US>
D07552 Bupivacaine (USAN/INN) <US>
D01450 Bupivacaine hydrochloride (USP) <JP/US>
D08181 Mepivacaine (INN)
D00738 Mepivacaine hydrochloride (JP18/USP) <JP/US>
D00553 Prilocaine (USP/INN)
D01243 Prilocaine hydrochloride (USP) <US>
D04095 Etidocaine (USAN/INN)
D00737 Etidocaine hydrochloride
D07468 Articaine (INN)
D02991 Articaine hydrochloride (JAN/USP)
D08490 Ropivacaine (INN)
D04048 Ropivacaine hydrochloride (USP) <JP/US>
D08116 Levobupivacaine (INN)
D01287 Levobupivacaine hydrochloride (JAN/USAN) <JP>
D00110 Cocaine (USP)
D02182 Cocaine hydrochloride (JP18/USP) <US>
D00512 Phenytoin (JP18/USP/INN) <JP/US>
D02103 Phenytoin sodium (USP) <JP/US>
D00375 Mephenytoin (USP/INN)
D07993 Fosphenytoin (INN)
D02096 Fosphenytoin sodium (USP) <US>
D07595 Fosphenytoin sodium hydrate (JAN) <JP>
D00252 Carbamazepine (JP18/USP/INN) <JP/US>
D00533 Oxcarbazepine (JAN/USP/INN) <US>
D05775 Rufinamide (JAN/USP/INN) <JP/US>
D09215 Eslicarbazepine (USAN/INN)
D09612 Eslicarbazepine acetate (USAN) <US>
D00354 Lamotrigine (JAN/USP/INN) <JP/US>
D00537 Topiramate (JAN/USP/INN) <JP/US>
D00538 Zonisamide (JP18/USP/INN) <JP/US>
D11150 Cenobamate (JAN/USAN/INN) <US>
D08448 Proxymetacaine (INN)
D02098 Proparacaine hydrochloride (USP) <US>
D01519 Ethyl piperidinoacetylaminobenzoate (JAN)
D01554 Pilsicainide hydrochloride hydrate (JP18) <JP>
D01785 Pirmenol hydrochloride hydrate (JAN) <JP>
D01967 p-Butylaminobenzoyldiethylaminoethyl hydrochloride (USAN)
D02762 Actisomide (USAN/INN)
D04521 Indecainide hydrochloride (USAN)
D05708 Recainam hydrochloride (USAN)
D05709 Recainam tosylate (USAN)
D06203 Transcainide (USAN/INN)
D06517 Pirmenol hydrochloride (USAN)
D08377 Pilsicainide (INN)
D08394 Pirmenol (INN)
D09833 Levosemotiadil fumarate (JAN)
D11155 Eleclazine (USAN/INN)
D12616 Bliretrigine (JAN/INN)
|
SCN2A [HSA:6326] [KO:K04834]
|
D08458 Quinidine (BAN)
D00642 Quinidine gluconate (USP) <US>
D00643 Quinidine polygalacturonate
D02272 Quinidine sulfate (USP) <JP/US>
D08459 Quinidine phenylethylbarbiturate
D08421 Procainamide (INN)
D00477 Procainamide hydrochloride (JP18/USP) <JP/US>
D00303 Disopyramide (JP18/USAN/INN) <JP>
D00637 Disopyramide phosphate (JAN/USP) <JP/US>
D01041 Sparteine (INN)
D02239 Sparteine sulfate (JAN/USAN)
D00199 Ajmaline (JP18)
D04774 Lorajmine hydrochloride (USAN)
D00358 Lidocaine (JP18/USP/INN) <JP/US>
D02086 Lidocaine hydrochloride (JAN/USP) <JP/US>
D08127 Lidocaine hydrochloride monohydrate <JP/US>
D08215 Mexiletine (INN)
D00639 Mexiletine hydrochloride (JP18/USP) <JP/US>
D06172 Tocainide (USAN/INN)
D02088 Tocainide hydrochloride (USP)
D02969 Aprindine (USAN/INN)
D01326 Aprindine hydrochloride (JP18/USAN) <JP>
D08435 Propafenone (INN)
D00640 Propafenone hydrochloride (JP18/USP) <JP/US>
D07962 Flecainide (INN)
D00638 Flecainide acetate (JP18/USP) <JP/US>
D07894 Encainide (INN)
D03991 Encainide hydrochloride (USAN)
D02910 Amiodarone (USAN/INN)
D00636 Amiodarone hydrochloride (JP18/USP) <JP/US>
D03492 Cifenline (USAN)
D01455 Cifenline succinate (USAN) <JP>
D00551 Tetracaine (USP/INN)
D00741 Tetracaine hydrochloride (JP18/USP) <US>
D00552 Benzocaine (USP/INN) <JP>
D00733 Dibucaine (USP)
D02220 Dibucaine hydrochloride (JP18/USP)
D08422 Procaine (INN)
D00740 Procaine hydrochloride (JP18/USP) <JP>
D01152 Oxethazaine (JP18/USAN) <JP>
D08311 Oxetacaine hydrochloride
D08407 Pramocaine (INN)
D00739 Pramoxine hydrochloride (USP)
D02456 Aminobenzoic acid (USP)
D02906 Aminobenzoate potassium (USP)
D02907 Aminobenzoate sodium (USP)
D08319 Oxybuprocaine (INN)
D01768 Benoxinate hydrochloride (USP) <JP>
D07678 Chloroprocaine (INN)
D00732 Chloroprocaine hydrochloride (USP) <US>
D07552 Bupivacaine (USAN/INN) <US>
D01450 Bupivacaine hydrochloride (USP) <JP/US>
D08181 Mepivacaine (INN)
D00738 Mepivacaine hydrochloride (JP18/USP) <JP/US>
D00553 Prilocaine (USP/INN)
D01243 Prilocaine hydrochloride (USP) <US>
D04095 Etidocaine (USAN/INN)
D00737 Etidocaine hydrochloride
D07468 Articaine (INN)
D02991 Articaine hydrochloride (JAN/USP)
D08490 Ropivacaine (INN)
D04048 Ropivacaine hydrochloride (USP) <JP/US>
D08116 Levobupivacaine (INN)
D01287 Levobupivacaine hydrochloride (JAN/USAN) <JP>
D00110 Cocaine (USP)
D02182 Cocaine hydrochloride (JP18/USP) <US>
D00512 Phenytoin (JP18/USP/INN) <JP/US>
D02103 Phenytoin sodium (USP) <JP/US>
D00375 Mephenytoin (USP/INN)
D07993 Fosphenytoin (INN)
D02096 Fosphenytoin sodium (USP) <US>
D07595 Fosphenytoin sodium hydrate (JAN) <JP>
D00252 Carbamazepine (JP18/USP/INN) <JP/US>
D00533 Oxcarbazepine (JAN/USP/INN) <US>
D05775 Rufinamide (JAN/USP/INN) <JP/US>
D09215 Eslicarbazepine (USAN/INN)
D09612 Eslicarbazepine acetate (USAN) <US>
D00354 Lamotrigine (JAN/USP/INN) <JP/US>
D00537 Topiramate (JAN/USP/INN) <JP/US>
D00538 Zonisamide (JP18/USP/INN) <JP/US>
D11150 Cenobamate (JAN/USAN/INN) <US>
D08448 Proxymetacaine (INN)
D02098 Proparacaine hydrochloride (USP) <US>
D01519 Ethyl piperidinoacetylaminobenzoate (JAN)
D01554 Pilsicainide hydrochloride hydrate (JP18) <JP>
D01785 Pirmenol hydrochloride hydrate (JAN) <JP>
D01967 p-Butylaminobenzoyldiethylaminoethyl hydrochloride (USAN)
D02762 Actisomide (USAN/INN)
D04521 Indecainide hydrochloride (USAN)
D05708 Recainam hydrochloride (USAN)
D05709 Recainam tosylate (USAN)
D06203 Transcainide (USAN/INN)
D06517 Pirmenol hydrochloride (USAN)
D08377 Pilsicainide (INN)
D08394 Pirmenol (INN)
D09833 Levosemotiadil fumarate (JAN)
D11155 Eleclazine (USAN/INN)
D12616 Bliretrigine (JAN/INN)
|
SCN3A [HSA:6328] [KO:K04836]
|
D08458 Quinidine (BAN)
D00642 Quinidine gluconate (USP) <US>
D00643 Quinidine polygalacturonate
D02272 Quinidine sulfate (USP) <JP/US>
D08459 Quinidine phenylethylbarbiturate
D08421 Procainamide (INN)
D00477 Procainamide hydrochloride (JP18/USP) <JP/US>
D00303 Disopyramide (JP18/USAN/INN) <JP>
D00637 Disopyramide phosphate (JAN/USP) <JP/US>
D01041 Sparteine (INN)
D02239 Sparteine sulfate (JAN/USAN)
D00199 Ajmaline (JP18)
D04774 Lorajmine hydrochloride (USAN)
D00358 Lidocaine (JP18/USP/INN) <JP/US>
D02086 Lidocaine hydrochloride (JAN/USP) <JP/US>
D08127 Lidocaine hydrochloride monohydrate <JP/US>
D08215 Mexiletine (INN)
D00639 Mexiletine hydrochloride (JP18/USP) <JP/US>
D06172 Tocainide (USAN/INN)
D02088 Tocainide hydrochloride (USP)
D02969 Aprindine (USAN/INN)
D01326 Aprindine hydrochloride (JP18/USAN) <JP>
D08435 Propafenone (INN)
D00640 Propafenone hydrochloride (JP18/USP) <JP/US>
D07962 Flecainide (INN)
D00638 Flecainide acetate (JP18/USP) <JP/US>
D07894 Encainide (INN)
D03991 Encainide hydrochloride (USAN)
D02910 Amiodarone (USAN/INN)
D00636 Amiodarone hydrochloride (JP18/USP) <JP/US>
D03492 Cifenline (USAN)
D01455 Cifenline succinate (USAN) <JP>
D00551 Tetracaine (USP/INN)
D00741 Tetracaine hydrochloride (JP18/USP) <US>
D00552 Benzocaine (USP/INN) <JP>
D00733 Dibucaine (USP)
D02220 Dibucaine hydrochloride (JP18/USP)
D08422 Procaine (INN)
D00740 Procaine hydrochloride (JP18/USP) <JP>
D01152 Oxethazaine (JP18/USAN) <JP>
D08311 Oxetacaine hydrochloride
D08407 Pramocaine (INN)
D00739 Pramoxine hydrochloride (USP)
D02456 Aminobenzoic acid (USP)
D02906 Aminobenzoate potassium (USP)
D02907 Aminobenzoate sodium (USP)
D08319 Oxybuprocaine (INN)
D01768 Benoxinate hydrochloride (USP) <JP>
D07678 Chloroprocaine (INN)
D00732 Chloroprocaine hydrochloride (USP) <US>
D07552 Bupivacaine (USAN/INN) <US>
D01450 Bupivacaine hydrochloride (USP) <JP/US>
D08181 Mepivacaine (INN)
D00738 Mepivacaine hydrochloride (JP18/USP) <JP/US>
D00553 Prilocaine (USP/INN)
D01243 Prilocaine hydrochloride (USP) <US>
D04095 Etidocaine (USAN/INN)
D00737 Etidocaine hydrochloride
D07468 Articaine (INN)
D02991 Articaine hydrochloride (JAN/USP)
D08490 Ropivacaine (INN)
D04048 Ropivacaine hydrochloride (USP) <JP/US>
D08116 Levobupivacaine (INN)
D01287 Levobupivacaine hydrochloride (JAN/USAN) <JP>
D00110 Cocaine (USP)
D02182 Cocaine hydrochloride (JP18/USP) <US>
D00512 Phenytoin (JP18/USP/INN) <JP/US>
D02103 Phenytoin sodium (USP) <JP/US>
D00375 Mephenytoin (USP/INN)
D07993 Fosphenytoin (INN)
D02096 Fosphenytoin sodium (USP) <US>
D07595 Fosphenytoin sodium hydrate (JAN) <JP>
D00252 Carbamazepine (JP18/USP/INN) <JP/US>
D00533 Oxcarbazepine (JAN/USP/INN) <US>
D05775 Rufinamide (JAN/USP/INN) <JP/US>
D09215 Eslicarbazepine (USAN/INN)
D09612 Eslicarbazepine acetate (USAN) <US>
D00354 Lamotrigine (JAN/USP/INN) <JP/US>
D00537 Topiramate (JAN/USP/INN) <JP/US>
D00538 Zonisamide (JP18/USP/INN) <JP/US>
D07299 Lacosamide (JAN/USAN/INN) <JP/US>
D11150 Cenobamate (JAN/USAN/INN) <US>
D08448 Proxymetacaine (INN)
D02098 Proparacaine hydrochloride (USP) <US>
D01519 Ethyl piperidinoacetylaminobenzoate (JAN)
D01554 Pilsicainide hydrochloride hydrate (JP18) <JP>
D01785 Pirmenol hydrochloride hydrate (JAN) <JP>
D01967 p-Butylaminobenzoyldiethylaminoethyl hydrochloride (USAN)
D02762 Actisomide (USAN/INN)
D04521 Indecainide hydrochloride (USAN)
D05708 Recainam hydrochloride (USAN)
D05709 Recainam tosylate (USAN)
D06203 Transcainide (USAN/INN)
D06517 Pirmenol hydrochloride (USAN)
D08377 Pilsicainide (INN)
D08394 Pirmenol (INN)
D09833 Levosemotiadil fumarate (JAN)
D11155 Eleclazine (USAN/INN)
D12616 Bliretrigine (JAN/INN)
|
SCN4A [HSA:6329] [KO:K04837]
|
D08458 Quinidine (BAN)
D00642 Quinidine gluconate (USP) <US>
D00643 Quinidine polygalacturonate
D02272 Quinidine sulfate (USP) <JP/US>
D08459 Quinidine phenylethylbarbiturate
D08421 Procainamide (INN)
D00477 Procainamide hydrochloride (JP18/USP) <JP/US>
D00303 Disopyramide (JP18/USAN/INN) <JP>
D00637 Disopyramide phosphate (JAN/USP) <JP/US>
D01041 Sparteine (INN)
D02239 Sparteine sulfate (JAN/USAN)
D00199 Ajmaline (JP18)
D04774 Lorajmine hydrochloride (USAN)
D00358 Lidocaine (JP18/USP/INN) <JP/US>
D02086 Lidocaine hydrochloride (JAN/USP) <JP/US>
D08127 Lidocaine hydrochloride monohydrate <JP/US>
D08215 Mexiletine (INN)
D00639 Mexiletine hydrochloride (JP18/USP) <JP/US>
D06172 Tocainide (USAN/INN)
D02088 Tocainide hydrochloride (USP)
D02969 Aprindine (USAN/INN)
D01326 Aprindine hydrochloride (JP18/USAN) <JP>
D08435 Propafenone (INN)
D00640 Propafenone hydrochloride (JP18/USP) <JP/US>
D07962 Flecainide (INN)
D00638 Flecainide acetate (JP18/USP) <JP/US>
D07894 Encainide (INN)
D03991 Encainide hydrochloride (USAN)
D02910 Amiodarone (USAN/INN)
D00636 Amiodarone hydrochloride (JP18/USP) <JP/US>
D03492 Cifenline (USAN)
D01455 Cifenline succinate (USAN) <JP>
D00551 Tetracaine (USP/INN)
D00741 Tetracaine hydrochloride (JP18/USP) <US>
D00552 Benzocaine (USP/INN) <JP>
D00733 Dibucaine (USP)
D02220 Dibucaine hydrochloride (JP18/USP)
D08422 Procaine (INN)
D00740 Procaine hydrochloride (JP18/USP) <JP>
D01152 Oxethazaine (JP18/USAN) <JP>
D08311 Oxetacaine hydrochloride
D08407 Pramocaine (INN)
D00739 Pramoxine hydrochloride (USP)
D02456 Aminobenzoic acid (USP)
D02906 Aminobenzoate potassium (USP)
D02907 Aminobenzoate sodium (USP)
D08319 Oxybuprocaine (INN)
D01768 Benoxinate hydrochloride (USP) <JP>
D07678 Chloroprocaine (INN)
D00732 Chloroprocaine hydrochloride (USP) <US>
D07552 Bupivacaine (USAN/INN) <US>
D01450 Bupivacaine hydrochloride (USP) <JP/US>
D08181 Mepivacaine (INN)
D00738 Mepivacaine hydrochloride (JP18/USP) <JP/US>
D00553 Prilocaine (USP/INN)
D01243 Prilocaine hydrochloride (USP) <US>
D04095 Etidocaine (USAN/INN)
D00737 Etidocaine hydrochloride
D07468 Articaine (INN)
D02991 Articaine hydrochloride (JAN/USP)
D08490 Ropivacaine (INN)
D04048 Ropivacaine hydrochloride (USP) <JP/US>
D08116 Levobupivacaine (INN)
D01287 Levobupivacaine hydrochloride (JAN/USAN) <JP>
D00110 Cocaine (USP)
D02182 Cocaine hydrochloride (JP18/USP) <US>
D00512 Phenytoin (JP18/USP/INN) <JP/US>
D02103 Phenytoin sodium (USP) <JP/US>
D00375 Mephenytoin (USP/INN)
D07993 Fosphenytoin (INN)
D02096 Fosphenytoin sodium (USP) <US>
D07595 Fosphenytoin sodium hydrate (JAN) <JP>
D00252 Carbamazepine (JP18/USP/INN) <JP/US>
D00533 Oxcarbazepine (JAN/USP/INN) <US>
D05775 Rufinamide (JAN/USP/INN) <JP/US>
D09215 Eslicarbazepine (USAN/INN)
D09612 Eslicarbazepine acetate (USAN) <US>
D00354 Lamotrigine (JAN/USP/INN) <JP/US>
D00537 Topiramate (JAN/USP/INN) <JP/US>
D00538 Zonisamide (JP18/USP/INN) <JP/US>
D11150 Cenobamate (JAN/USAN/INN) <US>
D08448 Proxymetacaine (INN)
D02098 Proparacaine hydrochloride (USP) <US>
D01519 Ethyl piperidinoacetylaminobenzoate (JAN)
D01554 Pilsicainide hydrochloride hydrate (JP18) <JP>
D01785 Pirmenol hydrochloride hydrate (JAN) <JP>
D01967 p-Butylaminobenzoyldiethylaminoethyl hydrochloride (USAN)
D02762 Actisomide (USAN/INN)
D04521 Indecainide hydrochloride (USAN)
D05708 Recainam hydrochloride (USAN)
D05709 Recainam tosylate (USAN)
D06203 Transcainide (USAN/INN)
D06517 Pirmenol hydrochloride (USAN)
D08377 Pilsicainide (INN)
D08394 Pirmenol (INN)
D09833 Levosemotiadil fumarate (JAN)
D11155 Eleclazine (USAN/INN)
D12616 Bliretrigine (JAN/INN)
|
SCN5A [HSA:6331] [KO:K04838]
|
D08458 Quinidine (BAN)
D00642 Quinidine gluconate (USP) <US>
D00643 Quinidine polygalacturonate
D02272 Quinidine sulfate (USP) <JP/US>
D08459 Quinidine phenylethylbarbiturate
D08421 Procainamide (INN)
D00477 Procainamide hydrochloride (JP18/USP) <JP/US>
D00303 Disopyramide (JP18/USAN/INN) <JP>
D00637 Disopyramide phosphate (JAN/USP) <JP/US>
D01041 Sparteine (INN)
D02239 Sparteine sulfate (JAN/USAN)
D00199 Ajmaline (JP18)
D04774 Lorajmine hydrochloride (USAN)
D00358 Lidocaine (JP18/USP/INN) <JP/US>
D02086 Lidocaine hydrochloride (JAN/USP) <JP/US>
D08127 Lidocaine hydrochloride monohydrate <JP/US>
D08215 Mexiletine (INN)
D00639 Mexiletine hydrochloride (JP18/USP) <JP/US>
D06172 Tocainide (USAN/INN)
D02088 Tocainide hydrochloride (USP)
D02969 Aprindine (USAN/INN)
D01326 Aprindine hydrochloride (JP18/USAN) <JP>
D08435 Propafenone (INN)
D00640 Propafenone hydrochloride (JP18/USP) <JP/US>
D07962 Flecainide (INN)
D00638 Flecainide acetate (JP18/USP) <JP/US>
D07894 Encainide (INN)
D03991 Encainide hydrochloride (USAN)
D02910 Amiodarone (USAN/INN)
D00636 Amiodarone hydrochloride (JP18/USP) <JP/US>
D05077 Moricizine (USAN)
D02087 Moricizine hydrochloride (USP)
D03492 Cifenline (USAN)
D01455 Cifenline succinate (USAN) <JP>
D06665 Vernakalant hydrochloride (USAN)
D00551 Tetracaine (USP/INN)
D00741 Tetracaine hydrochloride (JP18/USP) <US>
D00552 Benzocaine (USP/INN) <JP>
D00733 Dibucaine (USP)
D02220 Dibucaine hydrochloride (JP18/USP)
D08422 Procaine (INN)
D00740 Procaine hydrochloride (JP18/USP) <JP>
D01152 Oxethazaine (JP18/USAN) <JP>
D08311 Oxetacaine hydrochloride
D08407 Pramocaine (INN)
D00739 Pramoxine hydrochloride (USP)
D02456 Aminobenzoic acid (USP)
D02906 Aminobenzoate potassium (USP)
D02907 Aminobenzoate sodium (USP)
D08319 Oxybuprocaine (INN)
D01768 Benoxinate hydrochloride (USP) <JP>
D07678 Chloroprocaine (INN)
D00732 Chloroprocaine hydrochloride (USP) <US>
D07552 Bupivacaine (USAN/INN) <US>
D01450 Bupivacaine hydrochloride (USP) <JP/US>
D08181 Mepivacaine (INN)
D00738 Mepivacaine hydrochloride (JP18/USP) <JP/US>
D00553 Prilocaine (USP/INN)
D01243 Prilocaine hydrochloride (USP) <US>
D04095 Etidocaine (USAN/INN)
D00737 Etidocaine hydrochloride
D07468 Articaine (INN)
D02991 Articaine hydrochloride (JAN/USP)
D08490 Ropivacaine (INN)
D04048 Ropivacaine hydrochloride (USP) <JP/US>
D08116 Levobupivacaine (INN)
D01287 Levobupivacaine hydrochloride (JAN/USAN) <JP>
D00110 Cocaine (USP)
D02182 Cocaine hydrochloride (JP18/USP) <US>
D00512 Phenytoin (JP18/USP/INN) <JP/US>
D02103 Phenytoin sodium (USP) <JP/US>
D00375 Mephenytoin (USP/INN)
D07993 Fosphenytoin (INN)
D02096 Fosphenytoin sodium (USP) <US>
D07595 Fosphenytoin sodium hydrate (JAN) <JP>
D00252 Carbamazepine (JP18/USP/INN) <JP/US>
D00533 Oxcarbazepine (JAN/USP/INN) <US>
D05775 Rufinamide (JAN/USP/INN) <JP/US>
D09215 Eslicarbazepine (USAN/INN)
D09612 Eslicarbazepine acetate (USAN) <US>
D00354 Lamotrigine (JAN/USP/INN) <JP/US>
D00537 Topiramate (JAN/USP/INN) <JP/US>
D00538 Zonisamide (JP18/USP/INN) <JP/US>
D11150 Cenobamate (JAN/USAN/INN) <US>
D08448 Proxymetacaine (INN)
D02098 Proparacaine hydrochloride (USP) <US>
D01519 Ethyl piperidinoacetylaminobenzoate (JAN)
D01554 Pilsicainide hydrochloride hydrate (JP18) <JP>
D01785 Pirmenol hydrochloride hydrate (JAN) <JP>
D01967 p-Butylaminobenzoyldiethylaminoethyl hydrochloride (USAN)
D02762 Actisomide (USAN/INN)
D04521 Indecainide hydrochloride (USAN)
D05708 Recainam hydrochloride (USAN)
D05709 Recainam tosylate (USAN)
D06203 Transcainide (USAN/INN)
D06517 Pirmenol hydrochloride (USAN)
D08377 Pilsicainide (INN)
D08394 Pirmenol (INN)
D09833 Levosemotiadil fumarate (JAN)
D11155 Eleclazine (USAN/INN)
D12616 Bliretrigine (JAN/INN)
|
SCN8A [HSA:6334] [KO:K04840]
|
D08458 Quinidine (BAN)
D00642 Quinidine gluconate (USP) <US>
D00643 Quinidine polygalacturonate
D02272 Quinidine sulfate (USP) <JP/US>
D08459 Quinidine phenylethylbarbiturate
D08421 Procainamide (INN)
D00477 Procainamide hydrochloride (JP18/USP) <JP/US>
D00303 Disopyramide (JP18/USAN/INN) <JP>
D00637 Disopyramide phosphate (JAN/USP) <JP/US>
D01041 Sparteine (INN)
D02239 Sparteine sulfate (JAN/USAN)
D00199 Ajmaline (JP18)
D04774 Lorajmine hydrochloride (USAN)
D00358 Lidocaine (JP18/USP/INN) <JP/US>
D02086 Lidocaine hydrochloride (JAN/USP) <JP/US>
D08127 Lidocaine hydrochloride monohydrate <JP/US>
D08215 Mexiletine (INN)
D00639 Mexiletine hydrochloride (JP18/USP) <JP/US>
D06172 Tocainide (USAN/INN)
D02088 Tocainide hydrochloride (USP)
D02969 Aprindine (USAN/INN)
D01326 Aprindine hydrochloride (JP18/USAN) <JP>
D08435 Propafenone (INN)
D00640 Propafenone hydrochloride (JP18/USP) <JP/US>
D07962 Flecainide (INN)
D00638 Flecainide acetate (JP18/USP) <JP/US>
D07894 Encainide (INN)
D03991 Encainide hydrochloride (USAN)
D02910 Amiodarone (USAN/INN)
D00636 Amiodarone hydrochloride (JP18/USP) <JP/US>
D03492 Cifenline (USAN)
D01455 Cifenline succinate (USAN) <JP>
D00551 Tetracaine (USP/INN)
D00741 Tetracaine hydrochloride (JP18/USP) <US>
D00552 Benzocaine (USP/INN) <JP>
D00733 Dibucaine (USP)
D02220 Dibucaine hydrochloride (JP18/USP)
D08422 Procaine (INN)
D00740 Procaine hydrochloride (JP18/USP) <JP>
D01152 Oxethazaine (JP18/USAN) <JP>
D08311 Oxetacaine hydrochloride
D08407 Pramocaine (INN)
D00739 Pramoxine hydrochloride (USP)
D02456 Aminobenzoic acid (USP)
D02906 Aminobenzoate potassium (USP)
D02907 Aminobenzoate sodium (USP)
D08319 Oxybuprocaine (INN)
D01768 Benoxinate hydrochloride (USP) <JP>
D07678 Chloroprocaine (INN)
D00732 Chloroprocaine hydrochloride (USP) <US>
D07552 Bupivacaine (USAN/INN) <US>
D01450 Bupivacaine hydrochloride (USP) <JP/US>
D08181 Mepivacaine (INN)
D00738 Mepivacaine hydrochloride (JP18/USP) <JP/US>
D00553 Prilocaine (USP/INN)
D01243 Prilocaine hydrochloride (USP) <US>
D04095 Etidocaine (USAN/INN)
D00737 Etidocaine hydrochloride
D07468 Articaine (INN)
D02991 Articaine hydrochloride (JAN/USP)
D08490 Ropivacaine (INN)
D04048 Ropivacaine hydrochloride (USP) <JP/US>
D08116 Levobupivacaine (INN)
D01287 Levobupivacaine hydrochloride (JAN/USAN) <JP>
D00110 Cocaine (USP)
D02182 Cocaine hydrochloride (JP18/USP) <US>
D00512 Phenytoin (JP18/USP/INN) <JP/US>
D02103 Phenytoin sodium (USP) <JP/US>
D00375 Mephenytoin (USP/INN)
D07993 Fosphenytoin (INN)
D02096 Fosphenytoin sodium (USP) <US>
D07595 Fosphenytoin sodium hydrate (JAN) <JP>
D00252 Carbamazepine (JP18/USP/INN) <JP/US>
D00533 Oxcarbazepine (JAN/USP/INN) <US>
D05775 Rufinamide (JAN/USP/INN) <JP/US>
D09215 Eslicarbazepine (USAN/INN)
D09612 Eslicarbazepine acetate (USAN) <US>
D00354 Lamotrigine (JAN/USP/INN) <JP/US>
D00537 Topiramate (JAN/USP/INN) <JP/US>
D00538 Zonisamide (JP18/USP/INN) <JP/US>
D11150 Cenobamate (JAN/USAN/INN) <US>
D08448 Proxymetacaine (INN)
D02098 Proparacaine hydrochloride (USP) <US>
D01519 Ethyl piperidinoacetylaminobenzoate (JAN)
D01554 Pilsicainide hydrochloride hydrate (JP18) <JP>
D01785 Pirmenol hydrochloride hydrate (JAN) <JP>
D01967 p-Butylaminobenzoyldiethylaminoethyl hydrochloride (USAN)
D02762 Actisomide (USAN/INN)
D04521 Indecainide hydrochloride (USAN)
D05708 Recainam hydrochloride (USAN)
D05709 Recainam tosylate (USAN)
D06203 Transcainide (USAN/INN)
D06517 Pirmenol hydrochloride (USAN)
D08377 Pilsicainide (INN)
D08394 Pirmenol (INN)
D09833 Levosemotiadil fumarate (JAN)
D11155 Eleclazine (USAN/INN)
D12616 Bliretrigine (JAN/INN)
D12896 Zandatrigine (USAN/INN)
|
SCN9A [HSA:6335] [KO:K04841]
|
D08458 Quinidine (BAN)
D00642 Quinidine gluconate (USP) <US>
D00643 Quinidine polygalacturonate
D02272 Quinidine sulfate (USP) <JP/US>
D08459 Quinidine phenylethylbarbiturate
D08421 Procainamide (INN)
D00477 Procainamide hydrochloride (JP18/USP) <JP/US>
D00303 Disopyramide (JP18/USAN/INN) <JP>
D00637 Disopyramide phosphate (JAN/USP) <JP/US>
D01041 Sparteine (INN)
D02239 Sparteine sulfate (JAN/USAN)
D00199 Ajmaline (JP18)
D04774 Lorajmine hydrochloride (USAN)
D00358 Lidocaine (JP18/USP/INN) <JP/US>
D02086 Lidocaine hydrochloride (JAN/USP) <JP/US>
D08127 Lidocaine hydrochloride monohydrate <JP/US>
D08215 Mexiletine (INN)
D00639 Mexiletine hydrochloride (JP18/USP) <JP/US>
D06172 Tocainide (USAN/INN)
D02088 Tocainide hydrochloride (USP)
D02969 Aprindine (USAN/INN)
D01326 Aprindine hydrochloride (JP18/USAN) <JP>
D08435 Propafenone (INN)
D00640 Propafenone hydrochloride (JP18/USP) <JP/US>
D07962 Flecainide (INN)
D00638 Flecainide acetate (JP18/USP) <JP/US>
D07894 Encainide (INN)
D03991 Encainide hydrochloride (USAN)
D02910 Amiodarone (USAN/INN)
D00636 Amiodarone hydrochloride (JP18/USP) <JP/US>
D03492 Cifenline (USAN)
D01455 Cifenline succinate (USAN) <JP>
D00551 Tetracaine (USP/INN)
D00741 Tetracaine hydrochloride (JP18/USP) <US>
D00552 Benzocaine (USP/INN) <JP>
D00733 Dibucaine (USP)
D02220 Dibucaine hydrochloride (JP18/USP)
D08422 Procaine (INN)
D00740 Procaine hydrochloride (JP18/USP) <JP>
D01152 Oxethazaine (JP18/USAN) <JP>
D08311 Oxetacaine hydrochloride
D08407 Pramocaine (INN)
D00739 Pramoxine hydrochloride (USP)
D02456 Aminobenzoic acid (USP)
D02906 Aminobenzoate potassium (USP)
D02907 Aminobenzoate sodium (USP)
D08319 Oxybuprocaine (INN)
D01768 Benoxinate hydrochloride (USP) <JP>
D07678 Chloroprocaine (INN)
D00732 Chloroprocaine hydrochloride (USP) <US>
D07552 Bupivacaine (USAN/INN) <US>
D01450 Bupivacaine hydrochloride (USP) <JP/US>
D08181 Mepivacaine (INN)
D00738 Mepivacaine hydrochloride (JP18/USP) <JP/US>
D00553 Prilocaine (USP/INN)
D01243 Prilocaine hydrochloride (USP) <US>
D04095 Etidocaine (USAN/INN)
D00737 Etidocaine hydrochloride
D07468 Articaine (INN)
D02991 Articaine hydrochloride (JAN/USP)
D08490 Ropivacaine (INN)
D04048 Ropivacaine hydrochloride (USP) <JP/US>
D08116 Levobupivacaine (INN)
D01287 Levobupivacaine hydrochloride (JAN/USAN) <JP>
D00110 Cocaine (USP)
D02182 Cocaine hydrochloride (JP18/USP) <US>
D00512 Phenytoin (JP18/USP/INN) <JP/US>
D02103 Phenytoin sodium (USP) <JP/US>
D00375 Mephenytoin (USP/INN)
D07993 Fosphenytoin (INN)
D02096 Fosphenytoin sodium (USP) <US>
D07595 Fosphenytoin sodium hydrate (JAN) <JP>
D00252 Carbamazepine (JP18/USP/INN) <JP/US>
D00533 Oxcarbazepine (JAN/USP/INN) <US>
D05775 Rufinamide (JAN/USP/INN) <JP/US>
D09215 Eslicarbazepine (USAN/INN)
D09612 Eslicarbazepine acetate (USAN) <US>
D00354 Lamotrigine (JAN/USP/INN) <JP/US>
D00537 Topiramate (JAN/USP/INN) <JP/US>
D00538 Zonisamide (JP18/USP/INN) <JP/US>
D07299 Lacosamide (JAN/USAN/INN) <JP/US>
D11150 Cenobamate (JAN/USAN/INN) <US>
D08448 Proxymetacaine (INN)
D02098 Proparacaine hydrochloride (USP) <US>
D01519 Ethyl piperidinoacetylaminobenzoate (JAN)
D01554 Pilsicainide hydrochloride hydrate (JP18) <JP>
D01785 Pirmenol hydrochloride hydrate (JAN) <JP>
D01967 p-Butylaminobenzoyldiethylaminoethyl hydrochloride (USAN)
D02762 Actisomide (USAN/INN)
D04521 Indecainide hydrochloride (USAN)
D05708 Recainam hydrochloride (USAN)
D05709 Recainam tosylate (USAN)
D06203 Transcainide (USAN/INN)
D06517 Pirmenol hydrochloride (USAN)
D08377 Pilsicainide (INN)
D08394 Pirmenol (INN)
D09833 Levosemotiadil fumarate (JAN)
D11155 Eleclazine (USAN/INN)
D11156 Funapide (USAN/INN)
D11179 Vixotrigine (USAN/INN)
D11180 Vixotrigine hydrochloride (USAN)
D12616 Bliretrigine (JAN/INN)
|
SCN10A [HSA:6336] [KO:K04842]
|
D08458 Quinidine (BAN)
D00642 Quinidine gluconate (USP) <US>
D00643 Quinidine polygalacturonate
D02272 Quinidine sulfate (USP) <JP/US>
D08459 Quinidine phenylethylbarbiturate
D08421 Procainamide (INN)
D00477 Procainamide hydrochloride (JP18/USP) <JP/US>
D00303 Disopyramide (JP18/USAN/INN) <JP>
D00637 Disopyramide phosphate (JAN/USP) <JP/US>
D01041 Sparteine (INN)
D02239 Sparteine sulfate (JAN/USAN)
D00199 Ajmaline (JP18)
D04774 Lorajmine hydrochloride (USAN)
D00358 Lidocaine (JP18/USP/INN) <JP/US>
D02086 Lidocaine hydrochloride (JAN/USP) <JP/US>
D08127 Lidocaine hydrochloride monohydrate <JP/US>
D08215 Mexiletine (INN)
D00639 Mexiletine hydrochloride (JP18/USP) <JP/US>
D06172 Tocainide (USAN/INN)
D02088 Tocainide hydrochloride (USP)
D02969 Aprindine (USAN/INN)
D01326 Aprindine hydrochloride (JP18/USAN) <JP>
D08435 Propafenone (INN)
D00640 Propafenone hydrochloride (JP18/USP) <JP/US>
D07962 Flecainide (INN)
D00638 Flecainide acetate (JP18/USP) <JP/US>
D07894 Encainide (INN)
D03991 Encainide hydrochloride (USAN)
D02910 Amiodarone (USAN/INN)
D00636 Amiodarone hydrochloride (JP18/USP) <JP/US>
D03492 Cifenline (USAN)
D01455 Cifenline succinate (USAN) <JP>
D00551 Tetracaine (USP/INN)
D00741 Tetracaine hydrochloride (JP18/USP) <US>
D00552 Benzocaine (USP/INN) <JP>
D00733 Dibucaine (USP)
D02220 Dibucaine hydrochloride (JP18/USP)
D08422 Procaine (INN)
D00740 Procaine hydrochloride (JP18/USP) <JP>
D01152 Oxethazaine (JP18/USAN) <JP>
D08311 Oxetacaine hydrochloride
D08407 Pramocaine (INN)
D00739 Pramoxine hydrochloride (USP)
D02456 Aminobenzoic acid (USP)
D02906 Aminobenzoate potassium (USP)
D02907 Aminobenzoate sodium (USP)
D08319 Oxybuprocaine (INN)
D01768 Benoxinate hydrochloride (USP) <JP>
D07678 Chloroprocaine (INN)
D00732 Chloroprocaine hydrochloride (USP) <US>
D07552 Bupivacaine (USAN/INN) <US>
D01450 Bupivacaine hydrochloride (USP) <JP/US>
D08181 Mepivacaine (INN)
D00738 Mepivacaine hydrochloride (JP18/USP) <JP/US>
D00553 Prilocaine (USP/INN)
D01243 Prilocaine hydrochloride (USP) <US>
D04095 Etidocaine (USAN/INN)
D00737 Etidocaine hydrochloride
D07468 Articaine (INN)
D02991 Articaine hydrochloride (JAN/USP)
D08490 Ropivacaine (INN)
D04048 Ropivacaine hydrochloride (USP) <JP/US>
D08116 Levobupivacaine (INN)
D01287 Levobupivacaine hydrochloride (JAN/USAN) <JP>
D00110 Cocaine (USP)
D02182 Cocaine hydrochloride (JP18/USP) <US>
D00512 Phenytoin (JP18/USP/INN) <JP/US>
D02103 Phenytoin sodium (USP) <JP/US>
D00375 Mephenytoin (USP/INN)
D07993 Fosphenytoin (INN)
D02096 Fosphenytoin sodium (USP) <US>
D07595 Fosphenytoin sodium hydrate (JAN) <JP>
D00252 Carbamazepine (JP18/USP/INN) <JP/US>
D00533 Oxcarbazepine (JAN/USP/INN) <US>
D05775 Rufinamide (JAN/USP/INN) <JP/US>
D09215 Eslicarbazepine (USAN/INN)
D09612 Eslicarbazepine acetate (USAN) <US>
D00354 Lamotrigine (JAN/USP/INN) <JP/US>
D00537 Topiramate (JAN/USP/INN) <JP/US>
D00538 Zonisamide (JP18/USP/INN) <JP/US>
D07299 Lacosamide (JAN/USAN/INN) <JP/US>
D11150 Cenobamate (JAN/USAN/INN) <US>
D08448 Proxymetacaine (INN)
D02098 Proparacaine hydrochloride (USP) <US>
D01519 Ethyl piperidinoacetylaminobenzoate (JAN)
D01554 Pilsicainide hydrochloride hydrate (JP18) <JP>
D01785 Pirmenol hydrochloride hydrate (JAN) <JP>
D01967 p-Butylaminobenzoyldiethylaminoethyl hydrochloride (USAN)
D02762 Actisomide (USAN/INN)
D04521 Indecainide hydrochloride (USAN)
D05708 Recainam hydrochloride (USAN)
D05709 Recainam tosylate (USAN)
D06203 Transcainide (USAN/INN)
D06517 Pirmenol hydrochloride (USAN)
D08377 Pilsicainide (INN)
D08394 Pirmenol (INN)
D09833 Levosemotiadil fumarate (JAN)
D11155 Eleclazine (USAN/INN)
D12616 Bliretrigine (JAN/INN)
D12860 Suzetrigine (USAN/INN) <US>
|
SCN11A [HSA:11280] [KO:K04843]
|
D08458 Quinidine (BAN)
D00642 Quinidine gluconate (USP) <US>
D00643 Quinidine polygalacturonate
D02272 Quinidine sulfate (USP) <JP/US>
D08459 Quinidine phenylethylbarbiturate
D08421 Procainamide (INN)
D00477 Procainamide hydrochloride (JP18/USP) <JP/US>
D00303 Disopyramide (JP18/USAN/INN) <JP>
D00637 Disopyramide phosphate (JAN/USP) <JP/US>
D01041 Sparteine (INN)
D02239 Sparteine sulfate (JAN/USAN)
D00199 Ajmaline (JP18)
D04774 Lorajmine hydrochloride (USAN)
D00358 Lidocaine (JP18/USP/INN) <JP/US>
D02086 Lidocaine hydrochloride (JAN/USP) <JP/US>
D08127 Lidocaine hydrochloride monohydrate <JP/US>
D08215 Mexiletine (INN)
D00639 Mexiletine hydrochloride (JP18/USP) <JP/US>
D06172 Tocainide (USAN/INN)
D02088 Tocainide hydrochloride (USP)
D02969 Aprindine (USAN/INN)
D01326 Aprindine hydrochloride (JP18/USAN) <JP>
D08435 Propafenone (INN)
D00640 Propafenone hydrochloride (JP18/USP) <JP/US>
D07962 Flecainide (INN)
D00638 Flecainide acetate (JP18/USP) <JP/US>
D07894 Encainide (INN)
D03991 Encainide hydrochloride (USAN)
D02910 Amiodarone (USAN/INN)
D00636 Amiodarone hydrochloride (JP18/USP) <JP/US>
D03492 Cifenline (USAN)
D01455 Cifenline succinate (USAN) <JP>
D00551 Tetracaine (USP/INN)
D00741 Tetracaine hydrochloride (JP18/USP) <US>
D00552 Benzocaine (USP/INN) <JP>
D00733 Dibucaine (USP)
D02220 Dibucaine hydrochloride (JP18/USP)
D08422 Procaine (INN)
D00740 Procaine hydrochloride (JP18/USP) <JP>
D01152 Oxethazaine (JP18/USAN) <JP>
D08311 Oxetacaine hydrochloride
D08407 Pramocaine (INN)
D00739 Pramoxine hydrochloride (USP)
D02456 Aminobenzoic acid (USP)
D02906 Aminobenzoate potassium (USP)
D02907 Aminobenzoate sodium (USP)
D08319 Oxybuprocaine (INN)
D01768 Benoxinate hydrochloride (USP) <JP>
D07678 Chloroprocaine (INN)
D00732 Chloroprocaine hydrochloride (USP) <US>
D07552 Bupivacaine (USAN/INN) <US>
D01450 Bupivacaine hydrochloride (USP) <JP/US>
D08181 Mepivacaine (INN)
D00738 Mepivacaine hydrochloride (JP18/USP) <JP/US>
D00553 Prilocaine (USP/INN)
D01243 Prilocaine hydrochloride (USP) <US>
D07468 Articaine (INN)
D02991 Articaine hydrochloride (JAN/USP)
D08490 Ropivacaine (INN)
D04048 Ropivacaine hydrochloride (USP) <JP/US>
D08116 Levobupivacaine (INN)
D01287 Levobupivacaine hydrochloride (JAN/USAN) <JP>
D00110 Cocaine (USP)
D02182 Cocaine hydrochloride (JP18/USP) <US>
D00512 Phenytoin (JP18/USP/INN) <JP/US>
D02103 Phenytoin sodium (USP) <JP/US>
D00375 Mephenytoin (USP/INN)
D07993 Fosphenytoin (INN)
D02096 Fosphenytoin sodium (USP) <US>
D07595 Fosphenytoin sodium hydrate (JAN) <JP>
D00252 Carbamazepine (JP18/USP/INN) <JP/US>
D00533 Oxcarbazepine (JAN/USP/INN) <US>
D05775 Rufinamide (JAN/USP/INN) <JP/US>
D09215 Eslicarbazepine (USAN/INN)
D09612 Eslicarbazepine acetate (USAN) <US>
D00354 Lamotrigine (JAN/USP/INN) <JP/US>
D00537 Topiramate (JAN/USP/INN) <JP/US>
D00538 Zonisamide (JP18/USP/INN) <JP/US>
D11150 Cenobamate (JAN/USAN/INN) <US>
D08448 Proxymetacaine (INN)
D02098 Proparacaine hydrochloride (USP) <US>
D01519 Ethyl piperidinoacetylaminobenzoate (JAN)
D01554 Pilsicainide hydrochloride hydrate (JP18) <JP>
D01785 Pirmenol hydrochloride hydrate (JAN) <JP>
D01967 p-Butylaminobenzoyldiethylaminoethyl hydrochloride (USAN)
D02762 Actisomide (USAN/INN)
D04521 Indecainide hydrochloride (USAN)
D05708 Recainam hydrochloride (USAN)
D05709 Recainam tosylate (USAN)
D06203 Transcainide (USAN/INN)
D06517 Pirmenol hydrochloride (USAN)
D08377 Pilsicainide (INN)
D08394 Pirmenol (INN)
D09833 Levosemotiadil fumarate (JAN)
D11155 Eleclazine (USAN/INN)
D12616 Bliretrigine (JAN/INN)
|
Calcium channels
|
CACNA1-T [HSA:8911 8912 8913] [KO:K04856 K04855 K04854]
|
D08217 Mibefradil (INN)
D05024 Mibefradil dihydrochloride (USAN)
D07520 Bepridil (INN)
D00631 Bepridil hydrochloride (USAN) <JP>
D00539 Ethosuximide (JP18/USP/INN) <JP/US>
D00404 Methsuximide (USP) <US>
D00399 Valproic acid (USP) <US>
D00304 Divalproex sodium (USP) <US>
D00710 Valproate sodium (USAN) <JP/US>
D08667 Calcium valproate
D00538 Zonisamide (JP18/USP/INN) <JP/US>
D02630 Penfluridol (USAN/INN)
D07971 Flunarizine (INN)
D01303 Flunarizine hydrochloride (JAN/USAN)
D02633 Lomerizine hydrochloride (JAN) <JP>
D12061 Suvecaltamide (USAN)
D12062 Suvecaltamide hydrocloride (USAN)
D12819 Ulixacaltamide (USAN/INN)
D12820 Ulixacaltamide hydrochloride (USAN)
|
CACNA1-L [HSA:775 776 778 779] [KO:K04850 K04851 K04853 K04857]
|
D02537 Dronedarone (INN)
D03914 Dronedarone hydrochloride (USP) <US>
D07845 Diltiazem (INN)
D00616 Diltiazem hydrochloride (JP18/USP) <JP/US>
D03830 Diltiazem malate (USAN)
D01369 Bevantolol hydrochloride (JAN/USAN) <JP>
D07450 Amlodipine (USP/INN)
D00615 Amlodipine besylate (USP) <JP/US>
D02914 Amlodipine maleate (USAN)
D11881 Amlodipine benzoate <US>
D00319 Felodipine (JP18/USP/INN) <JP/US>
D00349 Isradipine (USP/INN) <US>
D08270 Nicardipine (INN)
D00617 Nicardipine hydrochloride (JP18/USAN) <JP/US>
D00437 Nifedipine (JP18/USP/INN) <JP/US>
D00438 Nimodipine (USP/INN) <US>
D00618 Nisoldipine (JAN/USAN/INN) <US>
D00629 Nitrendipine (JP18/USAN/INN) <JP>
D04657 Lacidipine (USAN/INN)
D01908 Nilvadipine (JP18/USAN/INN) <JP>
D08155 Manidipine (INN)
D01553 Manidipine hydrochloride (JP18) <JP>
D07494 Barnidipine (INN)
D01104 Barnidipine hydrochloride (JAN) <JP>
D08111 Lercanidipine (INN)
D01849 Lercanidipine hydrochloride (JAN/USAN)
D01173 Cilnidipine (JP18/INN) <JP>
D07509 Benidipine (INN)
D02045 Benidipine hydrochloride (JP18) <JP>
D08892 Clevidipine (USAN/INN) <US>
D08941 Levamlodipine malate (USAN)
D11723 Levamlodipine maleate (USAN) <US>
D08217 Mibefradil (INN)
D05024 Mibefradil dihydrochloride (USAN)
D02356 Verapamil (USAN/INN)
D00619 Verapamil hydrochloride (JP18/USP) <JP/US>
D08009 Gallopamil (INN)
D01969 Gallopamil hydrochloride (JAN)
D10932 Etripamil (USAN/INN)
D07185 Fendiline (INN)
D07943 Fendiline hydrochloride
D07520 Bepridil (INN)
D00631 Bepridil hydrochloride (USAN) <JP>
D08340 Perhexiline (INN)
D05442 Perhexiline maleate (USAN)
D08441 Propiverine (INN)
D01007 Propiverine hydrochloride (JP18) <JP>
D00495 Paramethadione (INN)
D00537 Topiramate (JAN/USP/INN) <JP/US>
D01145 Azelnidipine (JP18/INN) <JP>
D01151 Lemildipine (JAN/INN)
D01171 Monatepil maleate (JAN/USAN)
D01562 Aranidipine (JAN/INN)
D01604 Efonidipine hydrochloride ethanolate (JAN) <JP>
D01933 Vatanidipine hydrochloride (JAN)
D03067 Belfosdil (USAN/INN)
D03536 Clentiazem maleate (JAN/USAN)
D03655 Darodipine (USAN/INN)
D04193 Flordipine (USAN/INN)
D04260 Fostedil (USAN/INN)
D06129 Tiapamil hydrochloride (USAN)
D07886 Efonidipine (INN)
D09789 Kirenidipine hydrochloride (JAN)
D09833 Levosemotiadil fumarate (JAN)
D11102 Tamolarizine hydrochloride (JAN)
|
CACNA1B [HSA:774] [KO:K04849]
|
D01173 Cilnidipine (JP18/INN) <JP>
D06363 Ziconotide (USAN/INN)
D08686 Ziconotide acetate <US>
|
CACNA1S [HSA:779] [KO:K04857]
|
D07094 Pinaverium bromide (INN)
|
CACNA2D [HSA:781 9254 55799 93589] [KO:K04858 K04859 K04860 K04861]
|
D00332 Gabapentin (JAN/USP/INN) <JP/US>
D09539 Gabapentin enacarbil (JAN/USAN/INN) <JP/US>
D02716 Pregabalin (JAN/USAN/INN) <JP/US>
|
CACNA2D1 [HSA:781] [KO:K04858]
|
D11203 Mirogabalin (USAN/INN)
D10790 Mirogabalin besylate (USAN) <JP>
|
CACNA2D2 [HSA:9254] [KO:K04859]
|
D11203 Mirogabalin (USAN/INN)
D10790 Mirogabalin besylate (USAN) <JP>
|
CACNA1G [HSA:8913] [KO:K04854]
|
D12867 Ismidenon (USAN)
D12910 Apinocaltamide (USAN/INN)
|
CACNA1H [HSA:8912] [KO:K04855]
|
D12910 Apinocaltamide (USAN/INN)
|
CACNA1I [HSA:8911] [KO:K04856]
|
D12910 Apinocaltamide (USAN/INN)
|
Potassium channels
|
KCNA [HSA:3736 3737 3738 3739 3741 3742 3743 3744] [KO:K04874 K04875 K04876 K04877 K04878 K04879 K04880 K04881]
|
D10228 Amifampridine (USAN/INN)
D10689 Amifampridine phosphate (JAN/USAN) <JP/US>
D04127 Dalfampridine (USAN) <US>
|
KCNA1 [HSA:3736] [KO:K04874]
|
D06652 Tedisamil (USAN)
D06653 Tedisamil sesquifumarate (USAN)
|
KCNA5 [HSA:3741] [KO:K04878]
|
D06665 Vernakalant hydrochloride (USAN)
D07520 Bepridil (INN)
D00631 Bepridil hydrochloride (USAN) <JP>
|
KCNB [HSA:3745 9312] [KO:K04885 K04886]
|
D10228 Amifampridine (USAN/INN)
D10689 Amifampridine phosphate (JAN/USAN) <JP/US>
D04127 Dalfampridine (USAN) <US>
|
KCNC [HSA:3746 3747 3748 3749] [KO:K04887 K04888 K04889 K04890]
|
D10228 Amifampridine (USAN/INN)
D10689 Amifampridine phosphate (JAN/USAN) <JP/US>
D04127 Dalfampridine (USAN) <US>
|
KCND [HSA:3750 3751 3752] [KO:K04891 K04892 K04893]
|
D10228 Amifampridine (USAN/INN)
D10689 Amifampridine phosphate (JAN/USAN) <JP/US>
D04127 Dalfampridine (USAN) <US>
D00730 Butamben (USP)
D03547 Clofilium phosphate (USAN/INN)
|
KCND3 [HSA:3752] [KO:K04893]
|
D02910 Amiodarone (USAN/INN)
D00636 Amiodarone hydrochloride (JP18/USP) <JP/US>
D02537 Dronedarone (INN)
D03914 Dronedarone hydrochloride (USP) <US>
D06665 Vernakalant hydrochloride (USAN)
D07520 Bepridil (INN)
D00631 Bepridil hydrochloride (USAN) <JP>
D01856 Nifekalant hydrochloride (JAN) <JP>
|
KCNH1 [HSA:3756] [KO:K04904]
|
D03547 Clofilium phosphate (USAN/INN)
|
KCNH2 [HSA:3757] [KO:K04905]
|
D02910 Amiodarone (USAN/INN)
D00636 Amiodarone hydrochloride (JP18/USP) <JP/US>
D00647 Dofetilide (JAN/USP/INN) <US>
D08060 Ibutilide (INN)
D00648 Ibutilide fumarate (USP) <US>
D02537 Dronedarone (INN)
D03914 Dronedarone hydrochloride (USP) <US>
D08525 Sotalol (INN)
D01026 Sotalol hydrochloride (JAN/USP) <JP/US>
D07520 Bepridil (INN)
D00631 Bepridil hydrochloride (USAN) <JP>
D00110 Cocaine (USP)
D02182 Cocaine hydrochloride (JP18/USP) <US>
D00521 Terfenadine (JAN/USAN/INN)
D01856 Nifekalant hydrochloride (JAN) <JP>
D03037 Azimilide dihydrochloride (USAN)
D03547 Clofilium phosphate (USAN/INN)
D03732 Dexsotalol hydrochloride (USAN)
D04955 Sematilide hydrochloride (USAN)
D06206 Trecetilide fumarate (USAN)
D09757 Terikalant (INN)
D09758 Ambasilide (INN)
D09759 Trecetilide (INN)
|
KCNQ [HSA:3784 3785 3786 9132 56479] [KO:K04926 K04927 K04928 K04929 K04930]
|
D09569 Ezogabine (USAN)
D04192 Flindokalner (USAN/INN)
|
KCNQ1 [HSA:3784] [KO:K04926]
|
D02910 Amiodarone (USAN/INN)
D00636 Amiodarone hydrochloride (JP18/USP) <JP/US>
D02537 Dronedarone (INN)
D03914 Dronedarone hydrochloride (USP) <US>
D07520 Bepridil (INN)
D00631 Bepridil hydrochloride (USAN) <JP>
D03037 Azimilide dihydrochloride (USAN)
D09757 Terikalant (INN)
D09758 Ambasilide (INN)
|
KCNQ2 [HSA:3785] [KO:K04927]
|
D12890 Azetukalner (USAN/INN)
D13061 Opakalim (USAN)
|
KCNQ3 [HSA:3786] [KO:K04928]
|
D12890 Azetukalner (USAN/INN)
D13061 Opakalim (USAN)
|
KCNMB1 [HSA:3779] [KO:K04937]
|
D04192 Flindokalner (USAN/INN)
|
KCNN4 [HSA:3783] [KO:K04945]
|
D06640 Senicapoc (USAN)
|
KCNT2 (SLICK) [HSA:343450] [KO:K04947]
|
D03547 Clofilium phosphate (USAN/INN)
|
Inward rectifier channels (Kir)
|
KCNJ1 [HSA:3758] [KO:K04995]
|
D01603 Bethanidine sulfate (JAN/USAN)
|
KCNJ3 [HSA:3760] [KO:K04997]
|
D02910 Amiodarone (USAN/INN)
D00636 Amiodarone hydrochloride (JP18/USP) <JP/US>
D02537 Dronedarone (INN)
D03914 Dronedarone hydrochloride (USP) <US>
D07520 Bepridil (INN)
D00631 Bepridil hydrochloride (USAN) <JP>
|
KCNJ5 [HSA:3762] [KO:K04999]
|
D02910 Amiodarone (USAN/INN)
D00636 Amiodarone hydrochloride (JP18/USP) <JP/US>
D02537 Dronedarone (INN)
D03914 Dronedarone hydrochloride (USP) <US>
D07520 Bepridil (INN)
D00631 Bepridil hydrochloride (USAN) <JP>
|
KCNJ8 [HSA:3764] [KO:K05001]
|
D02910 Amiodarone (USAN/INN)
D00636 Amiodarone hydrochloride (JP18/USP) <JP/US>
D07520 Bepridil (INN)
D00631 Bepridil hydrochloride (USAN) <JP>
|
KCNJ11 [HSA:3767] [KO:K05004]
|
D02910 Amiodarone (USAN/INN)
D00636 Amiodarone hydrochloride (JP18/USP) <JP/US>
D03914 Dronedarone hydrochloride (USP) <US>
D07520 Bepridil (INN)
D00631 Bepridil hydrochloride (USAN) <JP>
|
KCNJ12 [HSA:3768] [KO:K05005]
|
D02910 Amiodarone (USAN/INN)
D00636 Amiodarone hydrochloride (JP18/USP) <JP/US>
D07520 Bepridil (INN)
D00631 Bepridil hydrochloride (USAN) <JP>
D01856 Nifekalant hydrochloride (JAN) <JP>
D09757 Terikalant (INN)
|
Ryanodine receptors (RYR)
|
RYR [HSA:6261 6262 6263] [KO:K04961 K04962 K04963]
|
D10304 Aladorian (USAN/INN)
D10305 Aladorian sodium (USAN)
D13172 Surlorian (USAN/INN)
D13173 Surlorian fumarate (USAN)
|
Transient receptor potential channels
|
TRPA1 [HSA:8989] [KO:K04984]
|
D00064 l-Menthol (JP18) <JP>
D04849 dl-Menthol (JP18)
D04918 Menthol (USP)
|
TRPC5 [HSA:7224] [KO:K04968]
|
D01705 Clemizole hydrochloride (JAN/USAN)
D02013 Clemizole undecylate (JAN)
D13060 Clemizole (USAN/INN)
|
TRPM8 [HSA:79054] [KO:K04983]
|
D00064 l-Menthol (JP18) <JP>
D04849 dl-Menthol (JP18)
D04918 Menthol (USP)
D13125 Acoltremon (USAN/INN) <US>
|
TRPV1 [HSA:7442] [KO:K05222]
|
D00250 Capsaicin (JAN/USP) <US>
D06388 Zucapsaicin (USAN/INN)
D05249 Olvanil (USAN)
D08282 Nonivamide (INN)
D10370 Mavatrep (USAN)
D12841 Motugivatrep (JAN/INN)
|
Other ion channels
|
Chloride channel
|
CLCN2 [HSA:1181] [KO:K05011]
|
D04790 Lubiprostone (JAN/USAN/INN) <JP/US>
|
CLCA [HSA:1179 9635 22802] [KO:K05027 K05028 K05030]
|
D03605 Crofelemer (USAN) <US>
D08275 Niflumic acid (INN)
|
Calcium channel
|
ORAI1 [HSA:84876] [KO:K16056]
|
D13009 Zegocractin (USAN/INN)
|
Hyperpolarization-activated ion channel
|
HCN [HSA:348980 610 57657 10021] [KO:K04954 K04955 K04956 K04957]
|
D07165 Ivabradine (USAN/INN)
D08095 Ivabradine hydrochloride (JAN/USAN) <JP/US>
|
|
Nuclear receptors
|
Thyroid hormone like receptors
|
Thyroid hormone receptor (THR)
|
NR1A (THR) [HSA:7067 7068] [KO:K05547 K08362]
|
D03750 Dextrothyroxine sodium (USAN)
D07214 Tiratricol (USAN/INN)
D11113 Levothyroxine sodium (INN) <US>
D01010 Levothyroxine sodium (USP) <JP/US>
D01011 Liothyronine sodium (JP18/USP) <JP/US>
D01012 Dried thyroid (JP18)
D06482 Thyroid (USP)
D08125 Levothyroxine (BAN)
D08128 Liothyronine (INN)
D08129 Liothyronine hydrochloride
|
NR1A2 (THRB) [HSA:7068] [KO:K08362]
|
D11602 Resmetirom (USAN/INN) <US>
D09381 Sobetirome (USAN)
|
Retinoic acid receptor (RAR)
|
NR1B (RAR) [HSA:5914 5915 5916] [KO:K08527 K08528 K08529]
|
D06543 Vitamin A (USP) <JP>
D00164 Retinol palmitate (JP18) <JP/US>
D01621 Retinol acetate (JP18)
D08477 Retinol propionate
D01132 Tazarotene (JAN/USAN/INN) <US>
D00316 Etretinate (JAN/USAN/INN) <JP>
D02754 Acitretin (USP/INN) <US>
D00094 Tretinoin (JAN/USP/INN) <JP/US>
D01516 Tretinoin tocoferil (JAN) <JP>
D00348 Isotretinoin (JAN/USP) <US>
D04636 Isotretinoin anisatil (USAN)
D02815 Alitretinoin (USAN) <US>
D04162 Fenretinide (USAN/INN)
|
NR1B1 (RARA) [HSA:5914] [KO:K08527]
|
D01418 Tamibarotene (JAN/USAN/INN) <JP>
|
NR1B2 (RARB) [HSA:5915] [KO:K08528]
|
D01112 Adapalene (JAN/USP/INN) <JP/US>
|
NR1B3 (RARG) [HSA:5916] [KO:K08529]
|
D01112 Adapalene (JAN/USP/INN) <JP/US>
D11225 Trifarotene (USAN/INN) <US>
D09365 Palovarotene (JAN/USAN/INN) <US>
|
PML-RARA [HSA:5371 5914] [KO:K10054 K08527]
|
D00094 Tretinoin (JAN/USP/INN) <JP/US>
D02106 Arsenic trioxide (JP18/USAN) <JP/US>
|
Peroxisome proliferator-activated receptor (PPAR)
|
NR1C (PPAR) [HSA:5465 5467 5468] [KO:K07294 K04504 K08530]
|
D06647 Sodelglitazar (USAN)
D09350 Indeglitazar (USAN)
D12614 Trisdecanoin (JAN/INN)
D13044 Saroglitazar (USAN/INN)
D13045 Saroglitazar magnesium (USAN)
|
NR1C1 (PPARA) [HSA:5465] [KO:K07294]
|
D11208 Elafibranor (USAN) <US>
D12484 Carfloglitazar (INN)
D00279 Clofibrate (JP18/USP/INN) <JP>
D01208 Aluminum clofibrate (JAN/INN)
D07724 Magnesium clofibrate (INN)
D01366 Bezafibrate (JP18/USAN/INN) <JP>
D00334 Gemfibrozil (JAN/USP/INN) <US>
D00565 Fenofibrate (JP18/USP/INN) <JP/US>
D03521 Ciprofibrate (USAN/INN)
D07187 Etofibrate (INN)
D08890 Choline fenofibrate (USAN/INN) <US>
D10711 Pemafibrate (JAN) <JP>
D01274 Tesaglitazar (JAN/USAN/INN)
D05091 Muraglitazar (USAN/INN)
D05397 Peliglitazar (USAN)
D06102 Theofibrate (USAN)
D08845 Aleglitazar (USAN)
D08949 Naveglitazar (USAN/INN)
D11579 Fenofibric acid
|
NR1C3 (PPARG) [HSA:5468] [KO:K08530]
|
D11256 Seladelpar (USAN/INN)
D11257 Seladelpar lysine (USAN) <US>
D00395 Troglitazone (JAN/USAN/INN)
D08491 Rosiglitazone (INN)
D00596 Rosiglitazone maleate (JAN/USP)
D08378 Pioglitazone (INN)
D00945 Pioglitazone hydrochloride (JP18/USP) <JP/US>
D11923 Lobeglitazone (INN)
D12484 Carfloglitazar (INN)
D11603 Leriglitazone (USAN/INN)
D11604 Leriglitazone hydrochloride (USAN)
D01274 Tesaglitazar (JAN/USAN/INN)
D01971 Reglitazar (JAN/INN)
D03493 Ciglitazone (USAN/INN)
D03653 Darglitazone sodium (USAN)
D03941 Edaglitazone sodium (USAN)
D03996 Englitazone sodium (USAN)
D04132 Farglitazar (USAN/INN)
D04411 Halofenate (USAN/INN)
D05030 Mifobate (USAN/INN)
D05091 Muraglitazar (USAN/INN)
D05150 Netoglitazone (USAN/INN)
D05397 Peliglitazar (USAN)
D05739 Rivoglitazone (USAN/INN)
D08845 Aleglitazar (USAN)
D09579 Arhalofenate (USAN/INN)
D12242 Bocidelpar (USAN)
D12243 Bocidelpar sulfate (USAN)
D12644 Mavodelpar (USAN/INN)
D12645 Mavodelpar sodium (USAN)
|
RAR-related orphan receptor
|
NR1F3 (RORC) [HSA:6097] [KO:K08534]
|
D12274 Cedirogant (USAN/INN)
|
Liver X receptor like receptor
|
NR1H2 (LXRB) [HSA:7376] [KO:K08535]
|
D12298 Abequolixron (USAN/INN)
D12299 Abequolixron zinc (USAN)
|
NR1H3 (LXRA) [HSA:10062] [KO:K08536]
|
D12298 Abequolixron (USAN/INN)
D12299 Abequolixron zinc (USAN)
|
NR1H4 (FXR) [HSA:9971] [KO:K08537]
|
D00163 Chenodiol (USAN) <JP/US>
D00734 Ursodiol (USP) <JP/US>
D10699 Cholic acid (JAN/USAN) <JP/US>
D09360 Obeticholic acid (JAN/USAN/INN)
D13241 Norucholic acid (INN)
D08277 Turofexorate isopropyl (USAN/INN)
D11548 Tropifexor (USAN)
|
Vitamin D3 like receptor
|
NR1I1 (VDR) [HSA:7421] [KO:K08539]
|
D00187 Ergocalciferol (JP18/USP) <US>
D00299 Dihydrotachysterol (JAN/USP/INN)
D01518 Alfacalcidol (JAN/INN) <JP>
D00129 Calcitriol (JAN/USP/INN) <JP/US>
D00188 Cholecalciferol (JP18/USP)
D00122 Calcifediol (USP/INN) <US>
D01125 Calcipotriene (USP) <JP/US>
D10198 Calcipotriol hydrate (JAN) <US>
D08554 Tacalcitol (INN)
D01472 Tacalcitol hydrate (JP18) <JP>
D00930 Paricalcitol (JAN/USP/INN) <US>
D01009 Doxercalciferol (USAN/INN) <US>
D00628 Secalciferol (JAN/USAN/INN)
D01098 Maxacalcitol (JAN/USAN/INN) <JP>
D01662 Falecalcitriol (JAN/INN) <JP>
D03930 Ecalcidene (USAN/INN)
D07578 Eldecalcitol (JAN/INN) <JP>
D08868 Becocalcidiol (USAN/INN)
D10565 Pefcalcitol (JAN/USAN/INN)
|
Hepatocyte nuclear factor 4 like receptors
|
Retinoid X receptor (RXR)
|
NR2B (RXR) [HSA:6256 6257 6258] [KO:K08524 K08525 K08526]
|
D00316 Etretinate (JAN/USAN/INN) <JP>
D02754 Acitretin (USP/INN) <US>
D02815 Alitretinoin (USAN) <US>
D03106 Bexarotene (JAN/USAN/INN) <JP/US>
|
NR2B2 (RXRB) [HSA:6257] [KO:K08525]
|
D01132 Tazarotene (JAN/USAN/INN) <US>
D01112 Adapalene (JAN/USP/INN) <JP/US>
|
NR2B3 (RXRG) [HSA:6258] [KO:K08526]
|
D01112 Adapalene (JAN/USP/INN) <JP/US>
|
Estrogen like receptors
|
Estrogen receptor
|
NR3A (ESR) [HSA:2099 2100] [KO:K08550 K08551]
|
D08409 Prasterone (USAN/INN) <US>
D01616 Sodium prasterone sulfate hydrate (JP18)
D00105 Estradiol (JAN/USP/INN) <JP/US>
D01413 Estradiol valerate (JAN/USP/INN) <JP/US>
D01617 Estradiol dipropionate (JAN)
D01953 Estradiol benzoate (JP18/USP)
D04061 Estradiol acetate (USAN) <US>
D04063 Estradiol cypionate (USP) <US>
D04064 Estradiol enanthate (USAN)
D04065 Estradiol undecylate (USAN/INN)
D07918 Estradiol hemihydrate <US>
D07919 Estradiol 17 beta-hemisuccinate
D00185 Estriol (JP18/USP) <JP>
D01986 Estriol tripropionate (JAN)
D01989 Estriol diacetate benzoate (JAN)
D07920 Estriol succinate
D07921 Estriol sodium succinate (BAN)
D00269 Chlorotrianisene (INN)
D00067 Estrone (JAN/USP/INN)
D00312 Estrone sodium sulfate
D00948 Estropipate (USP)
D07221 Promestriene (INN)
D11513 Estetrol (USAN)
D11514 Estetrol (JAN/USAN)
D00898 Dienestrol (USP/INN)
D00577 Diethylstilbestrol (USP/INN)
D00946 Diethylstilbestrol diphosphate (USP)
D07826 Hexestrol diphosphate sodium
D07726 Clomifene (INN)
D00962 Clomiphene citrate (USP) <JP/US>
D08465 Raloxifene (INN)
D02217 Raloxifene hydrochloride (JAN/USP) <JP/US>
D10606 Raloxifene hydrochloride hydrate (JAN) <JP>
D03062 Bazedoxifene acetate (JAN/USAN) <JP>
D04672 Lasofoxifene tartrate (JAN/USAN)
D08301 Ormeloxifene (INN)
D08559 Tamoxifen (INN)
D00966 Tamoxifen citrate (JP18/USP) <JP/US>
D08620 Toremifene (INN)
D00967 Toremifene citrate (JAN/USAN) <JP/US>
D01161 Fulvestrant (JAN/USP/INN) <JP/US>
D11829 Fluoroestradiol F18 <US>
D00575 Mestranol (JP18/USP/INN)
D01265 Epitiostanol (JAN/INN)
D01602 Mepitiostane (JP18/INN)
D01641 Hexestrol (JAN/INN)
D01853 Miproxifene phosphate (JAN)
D02018 Hexestrol diacetate (JAN)
D02758 Acolbifene hydrochloride (USAN)
D02993 Arzoxifene hydrochloride (USAN)
D03551 Clometherone (USAN/INN)
D03911 Droloxifene (USAN/INN)
D03912 Droloxifene citrate (USAN)
D04041 Equilin (USP)
D04071 Estrogens, esterified (USP) <US>
D04496 Idoxifene (USAN/INN)
D05106 Nafoxidine hydrochloride (USAN)
D05192 Nitromifene citrate (USAN)
D06245 Trioxifene mesylate (USAN)
D06551 Afimoxifene (USAN/INN)
D07121 Alfatradiol (INN)
D07783 Delmadinone (INN)
D08910 Enclomiphene (USAN)
D09834 Levormeloxifene fumarate (JAN)
D10008 Fispemifene (USAN/INN)
D10876 Enclomiphene citrate (USAN)
D11264 Brilanestrant (USAN/INN)
|
NR3A1 (ESR1) [HSA:2099] [KO:K08550]
|
D04104 Etonogestrel (USAN/INN) <US>
D02367 Desogestrel (USAN/INN)
D00554 Ethinyl estradiol (USP) <JP>
D07928 Ethinylestradiol propanesulfonate
D01639 Tibolone (JAN/USAN/INN)
D07939 Etynodiol (INN)
D01294 Ethynodiol diacetate (JAN/USP)
D00289 Danazol (JP18/USP/INN) <JP/US>
D08958 Ospemifene (INN/USAN/BAN) <US>
D07434 Polyestradiol phosphate (INN)
D11671 Elacestrant (USAN/INN)
D12049 Camizestrant (JAN/USAN)
D00576 Quinestrol (USAN/INN)
D11961 Giredestrant (USAN/INN)
D12145 Amcenestrant (JAN/USAN/INN)
D12216 Imlunestrant (USAN)
D12217 Imlunestrant tosylate (USAN)
D12628 Vepdegestrant (JAN/USAN/INN)
D12827 Palazestrant (USAN/INN)
D12943 Giredestrant tartrate (JAN)
|
NR3A1* (ESR1) [HSA_VAR:2099v2] [HSA:2099] [KO:K08550]
|
D11672 Elacestrant hydrochloride (USAN) <US>
|
NR3A2 (ESR2) [HSA:2100] [KO:K08551]
|
D06631 Prinaberel (USAN/INN)
D09899 Erteberel (USAN/INN)
|
3-Ketosteroid receptor
|
NR3C1 (GR) [HSA:2908] [KO:K05771]
|
D00385 Triamcinolone (JP18/USP/INN) <JP>
D00983 Triamcinolone acetonide (JP18/USP) <JP/US>
D00984 Triamcinolone diacetate (JAN/USP)
D00985 Triamcinolone hexacetonide (USP/INN)
D06216 Triamcinolone acetonide sodium phosphate (USAN)
D00292 Dexamethasone (JP18/USP/INN) <JP/US>
D00975 Dexamethasone sodium phosphate (JAN/USP) <JP/US>
D01510 Dexamethasone metasulfobenzoate sodium (JAN) <JP>
D01615 Dexamethasone palmitate (JAN) <JP>
D01632 Dexamethasone dipropionate (USAN) <JP>
D01948 Dexamethasone valerate (JAN) <JP>
D02174 Dexamethasone acetate (JAN/USP)
D02591 Dexamethasone acefurate (USAN/INN)
D02592 Dexamethasone beloxil (USAN)
D07073 Dexamethasone cipecilate (JAN/INN) <JP>
D07796 Dexamethasone 21-acetate
D07797 Dexamethasone isonicotinate
D07798 Dexamethasone sodium hemisulfate
D07799 Dexamethasone 21-tebutate
D07800 Dexamethasone 21-valerate
D07801 Dexamethasone phenylpropionate
D07802 Dexamethasone phosphate
D00088 Hydrocortisone (JP18/USP/INN) <JP/US>
D00165 Hydrocortisone acetate (JP18/USP) <US>
D00976 Hydrocortisone cypionate
D00977 Hydrocortisone sodium phosphate (JP18/USP) <JP>
D00978 Hydrocortisone sodium succinate (JP18/USP) <JP/US>
D01442 Hydrocortisone succinate (JP18)
D01619 Hydrocortisone butyrate (JP18/USP) <JP/US>
D01886 Hydrocortisone probutate (USAN) <JP>
D02288 Hydrocortisone valerate (USP) <US>
D04467 Hydrocortisone hemisuccinate (USP)
D06876 Hydrocortisone aceponate (INN)
D09796 Hydrocortisone caproate (JAN)
D00472 Prednisolone (JP18/USP/INN) <JP/US>
D00980 Prednisolone acetate (JP18/USP/INN) <JP/US>
D00981 Prednisolone sodium phosphate (JP18/USP) <JP/US>
D00982 Prednisolone tebutate (JAN/USP)
D01239 Prednisolone sodium succinate (JP18/USP) <JP>
D01998 Prednisolone farnesylate (JAN)
D02156 Prednisolone hemisuccinate (USP)
D03301 Prednisolone valerate acetate (JAN) <JP>
D08412 Prednisolone pivalate
D08413 Prednisolone sodium metazoate (USAN)
D08414 Prednisolone 21-(sodium tetrahydrophthalate)
D08415 Prednisolone steaglate (BAN)
D00473 Prednisone (USP) <US>
D08416 Prednisone acetate
D00244 Betamethasone (JP18/USP/INN) <JP>
D00972 Betamethasone sodium phosphate (JP18/USP) <JP>
D01357 Betamethasone valerate (JP18/USP) <JP/US>
D01402 Betamethasone acetate (JAN/USP)
D01637 Betamethasone dipropionate (JP18/USP) <JP/US>
D02032 Betamethasone butyrate propionate (JAN) <JP>
D02286 Betamethasone benzoate (USP)
D08610 Tixocortol (INN)
D06171 Tixocortol pivalate (USAN)
D00246 Budesonide (JP18/USP/INN) <JP/US>
D07495 Beclometasone (INN)
D00689 Beclomethasone dipropionate (USP) <JP/US>
D11572 Beclomethasone dipropionate monohydrate
D01367 Fluorometholone (JP18/USP/INN) <JP/US>
D04221 Fluorometholone acetate (USP) <US>
D04218 Fluocortolone (USAN/INN)
D04219 Fluocortolone caproate (USAN)
D07973 Fluocortolone 21-pivalate
D01825 Fluocinolone acetonide (JP18/USP/INN) <JP/US>
D00325 Fluocinonide (JP18/USP/INN) <JP/US>
D00407 Methylprednisolone (JP18/USP/INN) <JP/US>
D00751 Methylprednisolone sodium succinate (JAN/USP) <JP/US>
D00979 Methylprednisolone acetate (JAN/USP) <JP/US>
D05000 Methylprednisolone hemisuccinate (USP)
D05001 Methylprednisolone sodium phosphate (USAN)
D05002 Methylprednisolone suleptanate (USAN/INN)
D07203 Methylprednisolone aceponate (INN)
D07717 Clobetasone (INN)
D01273 Clobetasone butyrate (JAN/USAN) <JP>
D04208 Flumethasone (USAN)
D01464 Flumethasone pivalate (USP)
D07972 Fluocortin (INN)
D04217 Fluocortin butyl (USAN)
D07201 Fluprednidene (INN)
D07980 Fluprednidene acetate
D03696 Desonide (USP/INN) <US>
D07116 Alclometasone (INN)
D01820 Alclometasone dipropionate (JAN/USP) <JP/US>
D07719 Clocortolone (INN)
D02287 Clocortolone pivalate (USP) <US>
D03541 Clocortolone acetate (USAN)
D04201 Flucloronide (USAN)
D03697 Desoximetasone (USP/INN) <US>
D03812 Diflucortolone (USAN)
D01764 Diflucortolone valerate (JP18) <JP>
D03813 Diflucortolone pivalate (USAN)
D00328 Flurandrenolide (USP) <US>
D07827 Diflorasone (INN)
D01327 Diflorasone diacetate (JP18/USP) <JP/US>
D01387 Amcinonide (JAN/USP/INN) <JP/US>
D07202 Halometasone (INN)
D08227 Mometasone (INN)
D00690 Mometasone furoate (JAN/USP) <JP/US>
D03325 Mometasone furoate hydrate (JAN) <JP/US>
D07981 Fluticasone (INN)
D01708 Fluticasone propionate (JAN/USP) <JP/US>
D06315 Fluticasone furoate (JAN/USAN/INN) <JP/US>
D05601 Prednicarbate (USP/INN)
D01266 Difluprednate (JAN/USAN/INN) <JP/US>
D08660 Ulobetasol (INN)
D04409 Halobetasol propionate (USP) <US>
D07715 Clobetasol (INN)
D01272 Clobetasol propionate (JP18/USP) <JP/US>
D01308 Halcinonide (JAN/USP/INN) <US>
D00585 Mifepristone (JAN/USAN/INN) <US>
D07464 Paramethasone (INN)
D01229 Paramethasone acetate (JAN/USAN)
D07749 Cortisone (INN)
D00973 Cortisone acetate (JP18/USP) <JP/US>
D07230 Prednylidene (INN)
D05729 Rimexolone (USP/INN)
D03671 Deflazacort (USAN/INN) <US>
D03561 Cloprednol (USAN/INN)
D06673 Meprednisone (USP/INN)
D03594 Cortivazol (USAN)
D11000 Vamorolone (USAN/INN) <US>
D00324 Flunisolide (JAN/USP) <US>
D04214 Flunisolide acetate (USAN)
D01703 Ciclesonide (JAN/USAN/INN) <JP/US>
D02289 Medrysone (USAN)
D04244 Formocortal (USAN/INN)
D08147 Loteprednol (INN)
D01689 Loteprednol etabonate (JAN/USAN) <US>
D01434 Deprodone propionate (JAN) <JP>
D01743 Halopredone acetate (JAN/USAN)
D03691 Descinolone acetonide (USAN)
D04227 Fluprednisolone (USAN/INN)
D04228 Fluprednisolone valerate (USAN)
D05194 Nivazol (USAN)
D05603 Prednival (USAN)
D05719 Resocortol butyrate (USAN)
D06135 Ticabesone propionate (USAN)
D06161 Tipredane (USAN)
D06201 Tralonide (USAN/INN)
D07814 Dichlorisone (INN)
D07815 Dichlorisone acetate
D07975 Flupamesone
D08036 Halopredone (INN)
D08429 Proligestone (INN)
D08476 Resocortol (INN)
D10136 Mapracorat (USAN)
D10617 Dagrocorat (USAN/INN)
D10634 Fosdagrocorat (USAN/INN)
D11336 Relacorilant (USAN)
D11665 Exicorilant (USAN/INN)
D11667 Miricorilant (USAN/INN)
D11937 Velsecorat (USAN/INN)
D12638 Dazucorilant (USAN/INN)
|
NR3C2 (MR) [HSA:4306] [KO:K08555]
|
D00443 Spironolactone (JP18/USP/INN) <JP/US>
D01943 Canrenoate potassium (USAN) <JP>
D03363 Canrenone (USAN)
D01115 Eplerenone (JP18/USAN/INN) <JP/US>
D10633 Finerenone (JAN/USAN/INN) <JP/US>
D00386 Triamterene (JP18/USP/INN) <JP/US>
D03917 Drospirenone (JAN/USP/INN) <JP/US>
D10528 Aldosterone (INN)
D07967 Fludrocortisone (INN)
D00986 Fludrocortisone acetate (JP18/USP) <JP/US>
D07792 Desoxycortone (INN)
D03698 Desoxycorticosterone acetate (USP)
D03699 Desoxycorticosterone pivalate (USP)
D03792 Dicirenone (USAN)
D05020 Mexrenoate potassium (USAN)
D05640 Prorenoate potassium (USAN/INN)
D05912 Spiroxasone (USAN/INN)
D10892 Esaxerenone (JAN/INN) <JP>
D11667 Miricorilant (USAN/INN)
D13184 Balcinrenone (JAN/INN)
|
NR3C3 (PGR) [HSA:5241] [KO:K08556]
|
D01414 Ethylestrenol (USAN/INN)
D00182 Norethindrone (USP) <JP/US>
D00953 Norethindrone acetate (USP) <US>
D08285 Norethisterone enantate
D01580 Lynestrenol (JAN/USAN)
D00950 Levonorgestrel (JAN/USP/INN) <JP/US>
D05679 Quingestanol acetate (USAN)
D08167 Megestrol (INN)
D00952 Megestrol acetate (USP) <US>
D08166 Medroxyprogesterone (INN)
D00951 Medroxyprogesterone acetate (JP18/USP) <JP/US>
D07220 Norgestrienone (INN)
D04104 Etonogestrel (USAN/INN) <US>
D02367 Desogestrel (USAN/INN)
D03917 Drospirenone (JAN/USP/INN) <JP/US>
D09567 Ulipristal (USAN/INN)
D09687 Ulipristal acetate (JAN/USAN) <US>
D01159 Gestonorone caproate (JAN/USAN) <JP>
D08052 Hydroxyprogesterone (INN)
D00949 Hydroxyprogesterone caproate (JAN/USP/INN) <JP/US>
D08053 Hydroxyprogesterone 17alfa-acetate
D00066 Progesterone (JP18/USP/INN) <JP/US>
D01217 Dydrogesterone (JP18/USP/INN) <JP>
D04885 Medrogestone (USAN/INN)
D07222 Nomegestrol (USAN/INN)
D08281 Nomegestrol acetate (USAN)
D07223 Demegestone (INN)
D07670 Chlormadinone (INN)
D01299 Chlormadinone acetate (JP18/USAN) <JP>
D08431 Promegestone (INN)
D03799 Dienogest (JAN/USAN/INN) <JP>
D01374 Allylestrenol (JAN/INN)
D07939 Etynodiol (INN)
D01294 Ethynodiol diacetate (JAN/USP)
D00289 Danazol (JP18/USP/INN) <JP/US>
D00585 Mifepristone (JAN/USAN/INN) <US>
D00954 Norgestrel (JP18/USP/INN)
D02840 Altrenogest (USAN/INN)
D02881 Amadinone acetate (USAN)
D02996 Asoprisnil (USAN/INN)
D04315 Gestaclone (USAN/INN)
D04316 Gestodene (USAN/INN)
D05003 Methynodiol diacetate (USAN)
D05009 Metogest (USAN/INN)
D05205 Norelgestromin (USP/INN)
D05207 Norethynodrel (USAN)
D05209 Norgestimate (USP/INN)
D05308 Oxogestone phenpropionate (USAN)
D05680 Quingestrone (USAN/INN)
D06003 Tanaproget (USAN/INN)
D06145 Tigestol (USAN/INN)
D06197 Tosagestin (USAN/INN)
D06235 Trimegestone (USAN/INN)
D07096 Aglepristone (INN)
D07968 Flugestone (INN)
D08429 Proligestone (INN)
D09571 Onapristone (INN)
D09972 Telapristone acetate (USAN)
D10016 Lonaprisan (USAN/INN)
D10986 Segesterone acetate (USAN)
D10987 Segesterone (USAN/INN)
D11181 Vilaprisan (JAN/USAN/INN)
|
NR3C4 (AR) [HSA:367] [KO:K08557]
|
D07456 Androstanolone (INN)
D00444 Stanozolol (JAN/USP/INN)
D00389 Metandienone (INN)
D08193 Metenolone (INN)
D01301 Methenolone enanthate (USAN)
D01375 Methenolone acetate (USAN) <JP>
D00490 Oxymetholone (JP18/USP/INN)
D05674 Quinbolone (USAN/INN)
D08409 Prasterone (USAN/INN) <US>
D01616 Sodium prasterone sulfate hydrate (JP18)
D00462 Oxandrolone (JAN/USP/INN)
D07127 Norethandrolone (INN)
D08250 Nandrolone (INN)
D00955 Nandrolone decanoate (JAN/USP)
D00956 Nandrolone phenpropionate (USP)
D01476 Nandrolone cyclohexylpropionate (JAN)
D01737 Nandrolone furylpropionate (JAN)
D05116 Nandrolone cyclotate (USAN)
D08251 Nandrolone laurate
D01149 Oxabolone cipionate (JAN/INN)
D11451 Clascoterone (USAN) <US>
D00327 Fluoxymesterone (JAN/USP/INN)
D00408 Methyltestosterone (JP18/USP/INN) <US>
D00075 Testosterone (JAN/USP) <US>
D00957 Testosterone cypionate (USP) <US>
D00958 Testosterone enanthate (JP18/USP) <JP/US>
D00959 Testosterone propionate (JP18/USP)
D06085 Testosterone ketolaurate (USAN/INN)
D06086 Testosterone phenylacetate (USAN)
D06087 Testosterone undecanoate (USAN) <US>
D08573 Testosterone decanoate
D08574 Testosterone phenylpropionate
D04947 Mesterolone (USAN/INN)
D07670 Chlormadinone (INN)
D01299 Chlormadinone acetate (JP18/USAN) <JP>
D07766 Cyproterone (INN)
D01368 Cyproterone acetate (JAN/USAN)
D00289 Danazol (JP18/USP/INN) <JP/US>
D00586 Flutamide (JP18/USP/INN) <JP/US>
D00965 Nilutamide (USAN/INN) <US>
D00961 Bicalutamide (JP18/USP/INN) <JP/US>
D10218 Enzalutamide (JAN/USAN) <JP/US>
D11040 Apalutamide (JAN/INN) <JP/US>
D11045 Darolutamide (JAN/USAN/INN) <JP/US>
D01329 Oxendolone (JAN/USAN/INN)
D01533 Mestanolone (JAN/INN)
D01534 Dromostanolone propionate (USAN)
D03079 Benorterone (USAN/INN)
D03144 Bolasterone (USAN/INN)
D03145 Boldenone undecylenate (USAN)
D03338 Calusterone (USAN/INN)
D03515 Cioteronel (USAN/INN)
D03551 Clometherone (USAN/INN)
D03675 Delmadinone acetate (USAN)
D05025 Mibolerone (USP/INN)
D05174 Nisterime acetate (USAN)
D05837 Silandrone (USAN/INN)
D06191 Topterone (USAN/INN)
D06211 Trenbolone acetate (USP)
D06357 Zanoterone (USAN/INN)
D07536 Boldenone (INN)
D07783 Delmadinone (INN)
D08196 Methandriol (INN)
D08197 Methandriol dipropionate
D08627 Trenbolone (INN)
D10221 Enobosarm (USAN)
D11105 Osaterone acetate (JAN)
D11184 Ralaniten (USAN/INN)
D11185 Ralaniten acetate (USAN)
D12303 Deutenzalutamide (USAN)
D12316 Bavdegalutamide (USAN)
D12643 Masofaniten (USAN/INN)
D12866 Gridegalutamide (USAN)
D13046 Vosilasarm (USAN/INN)
D13059 Luxdegalutamide (USAN/INN)
D13211 Orevandrodeg (USAN)
D13217 Dezandrodeg (USAN)
|
|
Protein kinases
|
Serine/threonine kinases
|
AGC group
|
PRKCA [HSA:5578] [KO:K02677]
|
D05029 Midostaurin (JAN/USAN/INN) <US>
D02970 Aprinocarsen sodium (USAN)
D11191 Tigilanol tiglate (USAN/INN)
|
PRKCB [HSA:5579] [KO:K19662]
|
D05029 Midostaurin (JAN/USAN/INN) <US>
D04014 Enzastaurin hydrochloride (JAN/USAN)
D05784 Safingol (USAN/INN)
D05785 Safingol hydrochloride (USAN)
D11191 Tigilanol tiglate (USAN/INN)
D11935 Enzastaurin (USAN/INN)
|
PRKCG [HSA:5582] [KO:K19663]
|
D05029 Midostaurin (JAN/USAN/INN) <US>
D11191 Tigilanol tiglate (USAN/INN)
|
PRKCD [HSA:5580] [KO:K06068]
|
D05784 Safingol (USAN/INN)
D05785 Safingol hydrochloride (USAN)
D09671 Sotrastaurin (USAN/INN)
D09718 Sotrastaurin acetate (USAN)
D10456 Delcasertib (USAN/INN)
D10457 Delcasertib acetate (USAN)
|
PRKCE [HSA:5581] [KO:K18050]
|
D05784 Safingol (USAN/INN)
D05785 Safingol hydrochloride (USAN)
D09671 Sotrastaurin (USAN/INN)
D09718 Sotrastaurin acetate (USAN)
|
PRKCH [HSA:5583] [KO:K18051]
|
D09671 Sotrastaurin (USAN/INN)
D09718 Sotrastaurin acetate (USAN)
|
PRKCQ [HSA:5588] [KO:K18052]
|
D09671 Sotrastaurin (USAN/INN)
D09718 Sotrastaurin acetate (USAN)
|
AURK [HSA:6790 9212 6795] [KO:K11481 K11479 K11480]
|
D08279 Tozasertib (USAN)
D08344 Tozasertib lactate (USAN)
D10423 Ilorasertib (USAN/INN)
|
AURKA [HSA:6790] [KO:K11481]
|
D10085 Alisertib (USAN)
D10086 Alisertib sodium (USAN)
D12545 Tinengotinib (USAN/INN)
|
AURKB [HSA:9212] [KO:K11479]
|
D12545 Tinengotinib (USAN/INN)
|
AKT (PKB) [HSA:207 208 10000] [KO:K04456]
|
D11371 Capivasertib (JAN/USAN) <JP/US>
D06221 Triciribine phosphate (USAN)
D10381 Afuresertib (USAN/INN)
D10382 Afuresertib hydrochloride (USAN)
D10641 Ipatasertib (USAN/INN)
D10674 Uprosertib (USAN/INN)
D11074 Ipatasertib hydrochloride (JAN)
D11409 Miransertib (USAN/INN)
D11508 Miransertib mesylate (USAN)
|
DMPK [HSA:1760] [KO:K08788]
|
D10907 Baliforsen (USAN/INN)
|
ROCK [HSA:6093 9475] [KO:K04514 K17388]
|
D07941 Fasudil (INN)
D01840 Fasudil hydrochloride (JAN)
D03115 Fasudil hydrochloride hydrate (JAN) <JP>
D11030 Netarsudil (USAN/INN)
D11031 Netarsudil mesylate (USAN) <US>
D13014 Ripasudil (USAN/INN)
D10463 Ripasudil hydrochloride hydrate (JAN/USAN) <JP>
D10737 Verosudil (USAN/INN)
D10738 Verosudil hydrochloride (USAN)
|
ROCK2 [HSA:9475] [KO:K17388]
|
D11815 Belumosudil (USAN)
D11816 Belumosudil mesylate (USAN) <JP/US>
|
CAMK group
|
CHEK1 [HSA:1111] [KO:K02216]
|
D10397 Rabusertib (USAN/INN)
D11206 Prexasertib (USAN/INN)
|
AMPK (PRKAA) [HSA:5562 5563] [KO:K07198]
|
D08351 Phenformin (BAN)
D08352 Phenformin hydrochloride
D04966 Metformin (USAN/INN)
D00944 Metformin hydrochloride (JP18/USP) <JP/US>
D00595 Buformin (USAN/INN)
D02206 Buformin hydrochloride (JP18)
|
MAPKAPK2 [HSA:9261] [KO:K04443]
|
D12237 Zunsemetinib (USAN)
D12560 Gamcemetinib (USAN)
|
MKNK [HSA:8569 2872] [KO:K04372]
|
D11452 Tomivosertib (USAN/INN)
D11481 Tomivosertib hydrochloride (USAN)
D11763 Merestinib (USAN/INN)
|
PIM1 [HSA:5292] [KO:K04702]
|
D13179 Nuvisertib (USAN/INN)
D13180 Nuvisertib hydrochloride (USAN)
|
CK1 group
|
CSNK1E [HSA:1454] [KO:K08960]
|
D11322 Umbralisib (USAN/INN)
D11323 Umbralisib tosylate (USAN)
|
CMGC group
|
CDK1 [HSA:983] [KO:K02087]
|
D02880 Alvocidib hydrochloride (USAN)
D09604 Dinaciclib (USAN/INN)
D09868 Alvocidib (USAN/INN)
D11599 Zotiraciclib (USAN)
D11600 Zotiraciclib citrate (USAN)
|
CDK2 [HSA:1017] [KO:K02206]
|
D02880 Alvocidib hydrochloride (USAN)
D09604 Dinaciclib (USAN/INN)
D09868 Alvocidib (USAN/INN)
D11599 Zotiraciclib (USAN)
D11600 Zotiraciclib citrate (USAN)
D12601 Tegtociclib (USAN)
D12946 Certociclib (USAN)
|
CDK4/6 [HSA:1019 1021] [KO:K02089 K02091]
|
D10372 Palbociclib (JAN/USAN) <JP/US>
D10652 Palbociclib isethionate (USAN)
D10883 Ribociclib (USAN/INN)
D10979 Ribociclib succinate (USAN) <US>
D10688 Abemaciclib (JAN/USAN/INN) <JP/US>
D11130 Trilaciclib (USAN/INN)
D11987 Trilaciclib dihydrochloride <US>
D11455 Lerociclib (USAN)
D12834 Atirmociclib (USAN)
|
CDK4 [HSA:1019] [KO:K02089]
|
D02880 Alvocidib hydrochloride (USAN)
D09868 Alvocidib (USAN/INN)
|
CDK6 [HSA:1021] [KO:K02091]
|
D02880 Alvocidib hydrochloride (USAN)
D09868 Alvocidib (USAN/INN)
|
CDK7 [HSA:1022] [KO:K02202]
|
D02880 Alvocidib hydrochloride (USAN)
D09868 Alvocidib (USAN/INN)
D11599 Zotiraciclib (USAN)
D11600 Zotiraciclib citrate (USAN)
|
CDK9 [HSA:1025] [KO:K02211]
|
D09604 Dinaciclib (USAN/INN)
D11599 Zotiraciclib (USAN)
D11600 Zotiraciclib citrate (USAN)
D12525 Enitociclib (USAN/INN)
D12868 Istisociclib (USAN)
D13188 Tambiciclib (USAN/INN)
|
CDK5 [HSA:1020] [KO:K02090]
|
D09604 Dinaciclib (USAN/INN)
|
ERK [HSA:5594 5595] [KO:K04371]
|
D11038 Ulixertinib (INN)
D11285 Ravoxertinib (USAN/INN)
D12059 Temuterkib (USAN)
D12060 Temuterkib mesylate (USAN)
D12865 Beroterkib (USAN)
D12921 Tizaterkib (USAN/INN)
D12922 Tizaterkib adipate (USAN)
D12932 Bezisterim (USAN/INN)
|
JNK [HSA:5599 5601 5602] [KO:K04440]
|
D10168 Tanzisertib (USAN)
|
P38 [HSA:1432 5600 5603 6300] [KO:K04441]
|
D03736 Doramapimod (USAN/INN)
D09602 Dilmapimod (USAN/INN)
D09603 Dilmapimod tosylate (USAN)
D09639 Losmapimod (USAN/INN)
D10658 Ralimetinib (USAN/INN)
D10659 Ralimetinib mesylate (USAN)
D10959 Neflamapimod (USAN/INN)
|
P38alpha (MAPK14) [HSA:1432] [KO:K04441]
|
D08963 Pamapimod (INN/USAN)
D09386 Talmapimod (USAN/INN)
|
CLK2 [HSA:1196] [KO:K08823]
|
D11588 Lorecivivint (USAN/INN)
|
GSK3 [HSA:2931 2932] [KO:K08822 K03083]
|
D12196 Laduviglusib (USAN)
|
GSK3B [HSA:2932] [KO:K03083]
|
D12304 Elraglusib (USAN)
|
DYRK1A [HSA:1859] [KO:K08825]
|
D11588 Lorecivivint (USAN/INN)
|
STE group
|
MAP2K (MEK) [HSA:5604 5605] [KO:K04368 K04369]
|
D10175 Trametinib (USAN)
D10176 Trametinib dimethyl sulfoxide (JAN/USAN) <JP/US>
D10405 Cobimetinib (USAN/INN)
D10615 Cobimetinib fumarate (USAN) <US>
D10604 Binimetinib (JAN/USAN/INN) <JP/US>
D09666 Selumetinib (USAN/INN)
D10024 Selumetinib sulfate (JAN/USAN) <JP/US>
D11675 Mirdametinib (USAN) <US>
D13236 Tunlametinib (INN)
D10426 Pimasertib (USAN/INN)
D10486 Pimasertib hydrochloride (USAN)
D12473 Zapnometinib (USAN/INN)
D12515 Avutometinib (USAN/INN)
D12534 Avutometinib potassium (USAN)
D13039 Nedometinib (USAN/INN)
D13097 Polfurmetinib (USAN)
|
MAP2K1 (MEK1) [HSA:5604] [KO:K04368]
|
MAP2K2 (MEK2) [HSA:5605] [KO:K04369]
|
MAP3K5 (ASK1) [HSA:4217] [KO:K04426]
|
D10988 Selonsertib (JAN/USAN/INN)
|
TNIK [HSA:23043] [KO:K08840]
|
D13106 Rentosertib (USAN)
D13107 Rentosertib acetate (USAN)
|
TKL group
|
BRAF [HSA:673] [KO:K04365]
|
D10064 Dabrafenib (USAN)
D08524 Sorafenib (USAN/INN)
D06272 Sorafenib tosylate (USAN) <JP/US>
D10138 Regorafenib (USAN/INN)
D10137 Regorafenib hydrate (JAN) <JP/US>
D11410 Lifirafenib (USAN/INN)
D11411 Lifirafenib maleate (USAN)
D12831 Naporafenib (USAN/INN)
D12947 Claturafenib (USAN)
D13132 Flezurafenib (USAN/INN)
D13174 Mosperafenib (USAN/INN)
D13204 Plixorafenib (USAN/INN)
|
BRAF* [HSA_VAR:673v1] [HSA:673] [KO:K04365]
|
D09996 Vemurafenib (JAN/USAN/INN) <JP/US>
D10104 Dabrafenib mesylate (USAN) <JP/US>
D11053 Encorafenib (JAN/USAN/INN) <JP/US>
|
BRAF* [HSA_VAR:673v1 673v2] [HSA:673] [KO:K04365]
|
D12291 Tovorafenib (USAN/INN) <US>
|
RAF1 [HSA:5894] [KO:K04366]
|
D12291 Tovorafenib (USAN/INN) <US>
D08524 Sorafenib (USAN/INN)
D06272 Sorafenib tosylate (USAN) <JP/US>
D10138 Regorafenib (USAN/INN)
D10137 Regorafenib hydrate (JAN) <JP/US>
D12515 Avutometinib (USAN/INN)
D12534 Avutometinib potassium (USAN)
D12831 Naporafenib (USAN/INN)
D13132 Flezurafenib (USAN/INN)
|
IRAK4 [HSA:51135] [KO:K04733]
|
D12167 Zimlovisertib (USAN)
D12411 Emavusertib (USAN/INN)
D12412 Emavusertib hydrochloride (USAN)
D12532 Emavusertib mesylate (USAN)
D12533 Emavusertib maleate (USAN)
D12538 Emavusertib phosphate (USAN)
D12539 emavusertib tosylate (USAN)
|
RIPK1 [HSA:8737] [KO:K02861]
|
D12352 Eclitasertib (USAN/INN)
D12821 Flizasertib (USAN/INN)
D12846 Ocadusertib (USAN)
D12940 Oditrasertib (USAN/INN)
|
Other
|
NPR [HSA:4881 4882] [KO:K12323 K12324]
|
D04051 Erythrityl tetranitrate (USAN)
D02935 Anaritide acetate (USAN)
|
NPR1 [HSA:4881] [KO:K12323]
|
D05147 Nesiritide (USAN/INN)
D05148 Nesiritide citrate (USAN)
D03328 Carperitide (USAN/INN) <JP>
D10063 Cenderitide (USAN)
|
NPR2 [HSA:4882] [KO:K12324]
|
D11190 Vosoritide (USAN/INN) <JP/US>
|
CDC7 [HSA:8317] [KO:K02214]
|
D12176 Simurosertib (USAN/INN)
|
IKBKB [HSA:3551] [KO:K07209]
|
D04050 Ertiprotafib (USAN/INN)
|
AAK1 [HSA:22848] [KO:K08853]
|
D13080 Pilavapadin (USAN/INN)
D13081 Pilavapadin phosphate (USAN)
|
NEK7 [HSA:140609] [KO:K20876]
|
D13076 Ofirnoflast (USAN/INN)
|
PLK1 [HSA:5347] [KO:K06631]
|
D10154 Rigosertib (USAN)
D10155 Rigosertib sodium (JAN/USAN)
D10182 Volasertib (USAN)
D10183 Volasertib trihydrochloride (USAN)
D11458 Onvansertib (USAN)
D11459 Onvansertib fumarate (USAN)
|
MTOR [HSA:2475] [KO:K07203]
|
D06068 Temsirolimus (JAN/USAN/INN) <JP/US>
D02714 Everolimus (JAN/USAN/INN) <JP/US>
D08900 Ridaforolimus (JAN/USAN/INN)
D00753 Sirolimus (JAN/USAN/INN) <JP/US>
D06669 Zotarolimus (USAN/INN)
D10076 Olcorolimus (USAN)
D10543 Apitolisib (USAN/INN)
D10552 Dactolisib (USAN/INN)
D10616 Dactolisib tosylate (USAN)
D10635 Gedatolisib (USAN/INN)
D10718 Omipalisib (USAN/INN)
D11440 Bimiralisib (USAN/INN)
D11501 Samotolisib (USAN)
D11663 Onatasertib (USAN)
D11727 Voxtalisib (USAN/INN)
D11869 Paxalisib (USAN/INN)
|
PDK [HSA:5164 5165 5166] [KO:K00898]
|
D05857 Sodium dichloroacetate (USAN)
|
ATM [HSA:472] [KO:K04728]
|
D13010 Lartesertib (USAN/INN)
|
ATR [HSA:545] [KO:K06640]
|
D11148 Berzosertib (USAN/INN)
D11787 Ceralasertib (JAN/USAN/INN)
D12321 Camonsertib (USAN)
D12882 Tuvusertib (USAN/INN)
|
PKMYT1 [HSA:9088] [KO:K06633]
|
D12736 Lunresertib (USAN)
|
WEE1 [HSA:7465] [KO:K06632]
|
D11361 Adavosertib (USAN)
|
BRD2 [HSA:6046] [KO:K08871]
|
D12266 Pelabresib (USAN/INN)
D10911 Birabresib (USAN/INN)
D11131 Apabetalone (USAN/INN)
D12006 Trotabresib (USAN)
D13101 Repibresib (USAN)
|
BRD3 [HSA:8019] [KO:K11721]
|
D12266 Pelabresib (USAN/INN)
D10911 Birabresib (USAN/INN)
D11131 Apabetalone (USAN/INN)
D12006 Trotabresib (USAN)
D13101 Repibresib (USAN)
|
BRD4 [HSA:23476] [KO:K11722]
|
D12266 Pelabresib (USAN/INN)
D10911 Birabresib (USAN/INN)
D11131 Apabetalone (USAN/INN)
D11326 Molibresib (USAN)
D11347 Molibresib besylate (USAN)
D11479 Mivebresib (USAN/INN)
D12006 Trotabresib (USAN)
D12710 Ezobresib (USAN)
D13101 Repibresib (USAN)
|
BRDT [HSA:676] [KO:K11724]
|
D12266 Pelabresib (USAN/INN)
D11131 Apabetalone (USAN/INN)
D12006 Trotabresib (USAN)
D13101 Repibresib (USAN)
|
ULK1 [HSA:8408] [KO:K21357]
|
D13122 Inlexisertib (USAN/INN)
|
ULK2 [HSA:9706] [KO:K08269]
|
D13122 Inlexisertib (USAN/INN)
|
Receptor serine/threonine kinases (RSTK)
|
TGFBR1 family
|
ACVR1 (ALK2) [HSA:90] [KO:K04675]
|
D10889 Momelotinib hydrochloride hydrate (JAN) <JP/US>
D12547 Zilurgisertib (USAN/INN)
D12548 Zilurgisertib fumarate (USAN)
D12711 Fidrisertib (USAN/INN)
|
ACVRL1 [HSA:94] [KO:K13594]
|
D10106 Dalantercept (USAN)
D11709 Ascrinvacumab (USAN/INN)
|
TGFBR1 [HSA:7046] [KO:K04674]
|
D10437 Galunisertib (USAN/INN)
|
TGFBR2 family
|
ACVR2A [HSA:92] [KO:K04670]
|
D09670 Sotatercept (USAN/INN) <JP/US>
D10620 Bimagrumab (JAN/USAN/INN)
D12891 Elritercept (USAN/INN)
|
ACVR2B [HSA:93] [KO:K13596]
|
D11701 Luspatercept (USAN/INN) <JP/US>
D10620 Bimagrumab (JAN/USAN/INN)
D12999 Cibotercept (USAN/INN)
|
BMPR2 [HSA:659] [KO:K04671]
|
D03779 Dibotermin alfa (USAN/INN)
|
TGFBR2 [HSA:7048] [KO:K04388]
|
D11893 Bintrafusp alfa (USAN/INN)
D12768 Ficerafusp alfa (USAN)
|
Receptor tyrosine kinases (RTK)
|
EGFR family
|
EGFR [HSA:1956] [KO:K04361]
|
D07907 Erlotinib (INN)
D09724 Afatinib (USAN/INN)
D10858 Rociletinib (USAN/INN)
D10859 Olmutinib (USAN/INN)
D11115 Olmutinib hydrochloride (USAN)
D09883 Dacomitinib (INN)
D11251 Icotinib
D12001 Mobocertinib (USAN/INN)
D08108 Lapatinib (INN)
D04024 Lapatinib ditosylate (USAN) <JP/US>
D08950 Neratinib (USAN/INN)
D10898 Neratinib maleate <US>
D13235 Mifanertinib (INN)
D13098 Sevabertinib (USAN)
D13116 Sevabertinib hydrate (JAN) <US>
D06407 Vandetanib (JAN/USAN/INN) <JP/US>
D03455 Cetuximab (USAN/INN) <JP/US>
D05350 Panitumumab (USAN/INN) <JP/US>
D10018 Necitumumab (USAN/INN) <JP/US>
D04862 Masoprocol (USAN/INN)
D03350 Canertinib dihydrochloride (USAN)
D05399 Pelitinib (USAN/INN)
D09660 Rindopepimut (USAN)
D09689 Varlitinib (USAN/INN)
D09690 Varlitinib tosylate (USAN)
D10031 Zalutumumab (USAN/INN)
D10439 Imgatuzumab (USAN/INN)
D10886 Naquotinib mesylate (USAN)
D10958 Naquotinib (USAN/INN)
D11125 Modotuximab (USAN/INN)
D11368 Mavelertinib (USAN/INN)
D11410 Lifirafenib (USAN/INN)
D11411 Lifirafenib maleate (USAN)
D11430 Nazartinib (USAN/INN)
D11434 Nazartinib mesylate (USAN)
D11750 Duligotuzumab (USAN)
D11772 Tesevatinib (USAN/INN)
D11773 Tesevatinib tosylate (USAN)
D11803 Cetuximab sarotalocan (USAN/INN)
D11805 Cetuximab sarotalocan sodium (genetical recombination) (JAN) <JP>
D11872 Serclutamab (USAN/INN)
D11874 Serclutamab talirine (USAN/INN)
D12229 Poziotinib (USAN/INN)
D12230 Poziotinib hydrochloride (USAN)
D12416 Petosemtamab (USAN/INN)
D12457 Tuxobertinib (USAN/INN)
D12709 Marlotamig (USAN)
D12768 Ficerafusp alfa (USAN)
D12809 Bafisontamab (USAN/INN)
D13052 Izalontamab (USAN/INN)
D13053 Izalontamab brengitecan (USAN/INN)
D13066 Tilatamig (USAN/INN)
D13067 Tilatamig samrotecan (USAN/INN)
D13156 Pamvatamig (USAN/INN)
|
EGFR* [HSA_VAR:1956v2] [HSA:1956] [KO:K04361]
|
D01977 Gefitinib (JP18/USAN/INN) <JP/US>
D04023 Erlotinib hydrochloride (JAN/USAN) <JP/US>
D09733 Afatinib dimaleate (USAN) <JP/US>
D10766 Osimertinib mesylate (USAN) <JP/US>
D10514 Dacomitinib (USAN) <JP/US>
D11980 Lazertinib (USAN/INN)
D12245 Lazertinib mesylate (USAN) <JP/US>
D11969 Mobocertinib succinate (JAN)
D12258 Aumolertinib (USAN/INN)
D12259 Aumolertinib mesylate (USAN)
D12956 Firmonertinib (USAN/INN)
D12957 Firmonertinib mesylate (USAN)
D11894 Amivantamab (USAN/INN) <JP/US>
D13229 Amivantamab (genetical recombination) and vorhyaluronidase alfa (genetical recombination)
D12506 Sunvozertinib (USAN/INN)
D12730 Tigozertinib (USAN)
D12859 Pebezertinib (USAN)
D13062 Zipalertinib (JAN/USAN/INN)
|
ERBB2 (HER2, CD340) [HSA:2064] [KO:K05083]
|
D09724 Afatinib (USAN/INN)
D09733 Afatinib dimaleate (USAN) <JP/US>
D09883 Dacomitinib (INN)
D10514 Dacomitinib (USAN) <JP/US>
D08108 Lapatinib (INN)
D08950 Neratinib (USAN/INN)
D12879 Zongertinib (JAN/USAN/INN) <JP/US>
D11375 Trastuzumab duocarmazine (USAN/INN)
D12011 Zanidatamab (USAN/INN) <US>
D03350 Canertinib dihydrochloride (USAN)
D04025 Mubritinib (USAN/INN)
D06610 Lapuleucel-T (USAN)
D09689 Varlitinib (USAN/INN)
D09690 Varlitinib tosylate (USAN)
D10344 Nelipepimut-S (USAN)
D11772 Tesevatinib (USAN/INN)
D11773 Tesevatinib tosylate (USAN)
D11991 Zenocutuzumab (USAN/INN) <US>
D12229 Poziotinib (USAN/INN)
D12230 Poziotinib hydrochloride (USAN)
D12236 Runimotamab (USAN/INN)
D12457 Tuxobertinib (USAN/INN)
D12583 Anvatabart opadotin (USAN/INN)
D12584 Anvatabart pactil (USAN/INN)
D12978 Trastuzumab pamirtecan (USAN)
D12988 Disitamab (USAN/INN)
D12989 Disitamab vedotin (USAN/INN)
|
ERBB2* (HER2, CD340) [HSA_VAR:2064v1] [HSA:2064] [KO:K05083]
|
D04024 Lapatinib ditosylate (USAN) <JP/US>
D11141 Tucatinib (USAN/INN) <US>
D12442 Tucatinib ethanolate (JAN)
D03257 Trastuzumab (USAN/INN) <JP/US>
D11529 Trastuzumab deruxtecan (USAN/INN) <JP/US>
D10446 Margetuximab (USAN/INN) <US>
|
ERBB2* (HER2, CD340) [HSA_VAR:2064v1 2064v2] [HSA:2064] [KO:K05083]
|
D13116 Sevabertinib hydrate (JAN) <US>
|
ERBB2* (HER2, CD340) [HSA_VAR:2064v1 2064v3] [HSA:2064] [KO:K05083]
|
D10898 Neratinib maleate <US>
D05446 Pertuzumab (USAN/INN) <JP/US>
D09980 Trastuzumab emtansine (USAN/INN) <JP/US>
|
ERBB3 (HER3) [HSA:2065] [KO:K05084]
|
D11141 Tucatinib (USAN/INN) <US>
D12442 Tucatinib ethanolate (JAN)
D12184 Patritumab deruxtecan (USAN/INN)
D03350 Canertinib dihydrochloride (USAN)
D10943 Istiratumab (USAN/INN)
D11239 Lumretuzumab (USAN/INN)
D11750 Duligotuzumab (USAN)
D11777 Seribantumab (USAN/INN)
D11991 Zenocutuzumab (USAN/INN) <US>
D12185 Patritumab (USAN/INN)
D13052 Izalontamab (USAN/INN)
D13053 Izalontamab brengitecan (USAN/INN)
|
ERBB4 (HER4) [HSA:2066] [KO:K05085]
|
D09724 Afatinib (USAN/INN)
D09733 Afatinib dimaleate (USAN) <JP/US>
D09883 Dacomitinib (INN)
D10514 Dacomitinib (USAN) <JP/US>
D08950 Neratinib (USAN/INN)
D10898 Neratinib maleate <US>
D03350 Canertinib dihydrochloride (USAN)
D09689 Varlitinib (USAN/INN)
D09690 Varlitinib tosylate (USAN)
|
INSR family
|
INSR (CD220) [HSA:3643] [KO:K04527]
|
D03230 Insulin human (USP/INN) <JP/US>
D04548 Insulin, neutral (USAN)
D04477 Insulin lispro (USP/INN) <JP/US>
D04475 Insulin aspart (USP/INN) <JP/US>
D04540 Insulin glulisine (USAN/INN) <JP/US>
D03250 Insulin glargine (USAN/INN) <JP/US>
D04539 Insulin detemir (USAN/INN) <JP/US>
D09727 Insulin degludec (USAN/INN) <JP/US>
D12358 Insulin icodec (USAN/INN) <JP>
D11034 Insulin glargine and lixisenatide <JP/US>
D11567 Insulin degludec and liraglutide <JP/US>
D13242 Verenafusp alfa (INN)
D00085 Insulin (JAN/USP)
D04541 Insulin human, isophane (USP)
D04542 Insulin human zinc (USP)
D04543 Insulin human zinc, extended (USP)
D04544 Insulin I 125 (USAN)
D04545 Insulin I 131 (USAN)
D04546 Insulin, dalanated (USAN)
D04547 Insulin, isophane (USP) <JP>
D04549 Insulin zinc, extended (USP)
D04550 Insulin zinc, prompt (USP)
D04551 Insulin zinc (USP)
D05622 Proinsulin human (USAN)
D08080 Insulin injection, biphasic isophane (BAN) <JP>
D10473 Insulin peglispro (USAN/INN)
D12912 Ersodetug (USAN/INN)
D13028 Insulin efsitora alfa (INN)
|
IGF1R (CD221) [HSA:3480] [KO:K05087]
|
D03297 Mecasermin (USAN/INN) <JP/US>
D04870 Mecasermin rinfabate (USAN/INN)
D08620 Toremifene (INN)
D09680 Teprotumumab (USAN/INN) <JP/US>
D04491 Ibutamoren mesylate (USAN)
D09328 Cixutumumab (USAN)
D09345 Figitumumab (USAN)
D09746 Dalotuzumab (USAN)
D09908 Ganitumab (USAN/INN)
D09925 Linsitinib (USAN/INN)
D10056 Robatumumab (USAN/INN)
D10943 Istiratumab (USAN/INN)
D12952 Veligrotug (USAN/INN)
|
ROS1 [HSA:6098] [KO:K05088]
|
D11012 Lorlatinib (JAN/USAN/INN) <JP/US>
D12363 Taletrectinib (USAN/INN)
D12364 Taletrectinib adipate (JAN/USAN) <JP/US>
D12899 Zidesamtinib (USAN/INN)
|
ROS1* [HSA_VAR:6098v1] [HSA:6098] [KO:K05088]
|
D09731 Crizotinib (JAN/USAN/INN) <JP/US>
D10926 Entrectinib (JAN/USAN/INN) <JP/US>
D11454 Repotrectinib (JAN/USAN) <JP/US>
|
PDGFR family
|
PDGFR [HSA:5156 5159] [KO:K04363 K05089]
|
D08953 Nilotinib (USAN/INN) <US>
D06413 Nilotinib hydrochloride hydrate (JAN) <JP/US>
D12444 Nilotinib hydrochloride dihydrate (JAN) <JP>
D12854 Nilotinib laurylsulfate (USAN)
D13008 Nilotinib D-tartrate (USAN) <US>
D08552 Sunitinib (INN)
D06402 Sunitinib malate (JAN/USAN) <JP/US>
D05380 Pazopanib hydrochloride (JAN/USAN) <JP/US>
D10481 Nintedanib (USAN/INN)
D10396 Nintedanib esylate (USAN) <JP/US>
D05029 Midostaurin (JAN/USAN/INN) <US>
D11140 Sitravatinib (USAN/INN)
D11541 Sitravatinib malate (USAN)
D06678 Motesanib (USAN)
D08503 Toceranib (USAN)
D08544 Toceranib phosphate (USAN)
D09635 Linifanib (USAN/INN)
D10102 Crenolanib (USAN)
D10103 Crenolanib besylate (USAN)
D10423 Ilorasertib (USAN/INN)
D12002 Seralutinib (USAN/INN)
D12526 Catequentinib (USAN/INN)
D12537 Catequentinib hydrochloride (USAN)
|
PDGFRA [HSA:5156] [KO:K04363]
|
D11353 Ripretinib (USAN) <US>
D09939 Olaratumab (USAN/INN)
D08947 Motesanib diphosphate (USAN)
D10411 Tovetumab (USAN/INN)
D13058 Migaldendranib (USAN/INN)
|
PDGFRA* [HSA_VAR:5156v2] [HSA:5156] [KO:K04363]
|
D11279 Avapritinib (USAN/INN) <US>
|
FIP1L1-PDGFRA [HSA:5156] [KO:K04363]
|
D08066 Imatinib (INN)
D01441 Imatinib mesylate (USAN) <JP/US>
|
PDGFRB [HSA:5159] [KO:K05089]
|
D03065 Becaplermin (USAN/INN)
D03658 Dasatinib (JAN/INN) <JP>
D06414 Dasatinib (USAN) <JP/US>
D12609 Dasatinib laurylsulfate (USAN)
D10190 Tivozanib hydrochloride (USAN) <US>
D08524 Sorafenib (USAN/INN)
D06272 Sorafenib tosylate (USAN) <JP/US>
D10138 Regorafenib (USAN/INN)
D10137 Regorafenib hydrate (JAN) <JP/US>
D06005 Tandutinib (USAN/INN)
D06285 Vatalanib (USAN/INN)
D08907 Dovitinib lactate (USAN)
D08947 Motesanib diphosphate (USAN)
D13058 Migaldendranib (USAN/INN)
|
KIT (CD117) [HSA:3815] [KO:K05091]
|
D08066 Imatinib (INN)
D01441 Imatinib mesylate (USAN) <JP/US>
D03658 Dasatinib (JAN/INN) <JP>
D06414 Dasatinib (USAN) <JP/US>
D12609 Dasatinib laurylsulfate (USAN)
D08953 Nilotinib (USAN/INN) <US>
D06413 Nilotinib hydrochloride hydrate (JAN) <JP/US>
D12444 Nilotinib hydrochloride dihydrate (JAN) <JP>
D12854 Nilotinib laurylsulfate (USAN)
D13008 Nilotinib D-tartrate (USAN) <US>
D10190 Tivozanib hydrochloride (USAN) <US>
D08552 Sunitinib (INN)
D06402 Sunitinib malate (JAN/USAN) <JP/US>
D08524 Sorafenib (USAN/INN)
D06272 Sorafenib tosylate (USAN) <JP/US>
D05380 Pazopanib hydrochloride (JAN/USAN) <JP/US>
D10138 Regorafenib (USAN/INN)
D10137 Regorafenib hydrate (JAN) <JP/US>
D10229 Masitinib (INN)
D05029 Midostaurin (JAN/USAN/INN) <US>
D11270 Pexidartinib (USAN/INN)
D11271 Pexidartinib hydrochloride (JAN/USAN) <US>
D11353 Ripretinib (USAN) <US>
D02937 Ancestim (USAN/INN)
D05819 Semaxanib (USAN/INN)
D06005 Tandutinib (USAN/INN)
D06285 Vatalanib (USAN/INN)
D06678 Motesanib (USAN)
D08503 Toceranib (USAN)
D08544 Toceranib phosphate (USAN)
D08907 Dovitinib lactate (USAN)
D08947 Motesanib diphosphate (USAN)
D09864 Amuvatinib (USAN/INN)
D09865 Amuvatinib hydrochloride (USAN)
D12175 Olverembatinib (USAN/INN)
D12409 Barzolvolimab (USAN/INN)
D12450 Elenestinib (USAN)
D12526 Catequentinib (USAN/INN)
D12537 Catequentinib hydrochloride (USAN)
D12540 Briquilimab (USAN/INN)
D13058 Migaldendranib (USAN/INN)
|
KIT* (CD117) [HSA_VAR:3815v1] [HSA:3815] [KO:K05091]
|
D11279 Avapritinib (USAN/INN) <US>
D12476 Tuspetinib (USAN/INN)
D12600 Bezuclastinib (USAN/INN)
|
FLT3 (CD135) [HSA:2322] [KO:K05092]
|
D11768 Pacritinib (USAN/INN) <US>
D08552 Sunitinib (INN)
D06402 Sunitinib malate (JAN/USAN) <JP/US>
D08524 Sorafenib (USAN/INN)
D06272 Sorafenib tosylate (USAN) <JP/US>
D09955 Quizartinib (USAN/INN)
D10709 Gilteritinib (USAN/INN)
D04696 Lestaurtinib (USAN/INN)
D05819 Semaxanib (USAN/INN)
D06005 Tandutinib (USAN/INN)
D08279 Tozasertib (USAN)
D08344 Tozasertib lactate (USAN)
D08907 Dovitinib lactate (USAN)
D10102 Crenolanib (USAN)
D10103 Crenolanib besylate (USAN)
D11599 Zotiraciclib (USAN)
D11600 Zotiraciclib citrate (USAN)
D12476 Tuspetinib (USAN/INN)
D12641 Emirodatamab (USAN/INN)
|
FLT3* (CD135) [HSA_VAR:2322v1 2322v2] [HSA:2322] [KO:K05092]
|
D05029 Midostaurin (JAN/USAN/INN) <US>
D10800 Gilteritinib fumarate (JAN/USAN) <JP/US>
|
FLT3* (CD135) [HSA_VAR:2322v2] [HSA:2322] [KO:K05092]
|
D09956 Quizartinib dihydrochloride (USAN) <JP/US>
D11270 Pexidartinib (USAN/INN)
D11271 Pexidartinib hydrochloride (JAN/USAN) <US>
|
FGFR family
|
FGFR [HSA:2260 2263 2261 2264] [KO:K04362 K05093 K05094 K05095]
|
D09919 Lenvatinib (USAN/INN)
D09920 Lenvatinib mesylate (USAN) <JP/US>
D05716 Repifermin (USAN/INN)
D11461 Derazantinib hydrochloride (USAN)
D12526 Catequentinib (USAN/INN)
D12537 Catequentinib hydrochloride (USAN)
|
FGFR1 (CD331) [HSA:2260] [KO:K04362]
|
D11417 Pemigatinib (JAN/USAN/INN) <JP/US>
D11589 Infigratinib (USAN/INN)
D11611 Infigratinib phosphate (USAN)
D10138 Regorafenib (USAN/INN)
D10137 Regorafenib hydrate (JAN) <JP/US>
D10481 Nintedanib (USAN/INN)
D10396 Nintedanib esylate (USAN) <JP/US>
D11885 Surufatinib (USAN/INN)
D08878 Brivanib alaninate (JAN/USAN/INN)
D09589 Brivanib (USAN)
D11762 Lucitanib (USAN/INN)
D12404 Tasurgratinib (INN)
D12405 Tasurgratinib succinate (JAN) <JP>
D12490 Fazpilodemab (USAN/INN)
D12545 Tinengotinib (USAN/INN)
|
FGFR2 (CD332) [HSA:2263] [KO:K05093]
|
D11589 Infigratinib (USAN/INN)
D10481 Nintedanib (USAN/INN)
D10396 Nintedanib esylate (USAN) <JP/US>
D13029 Bemarituzumab (INN)
D05338 Palifermin (USAN/INN) <US>
D11762 Lucitanib (USAN/INN)
D12404 Tasurgratinib (INN)
D12455 Lirafugratinib (USAN)
D12456 Lirafugratinib hydrochloride (USAN)
D12545 Tinengotinib (USAN/INN)
|
FGFR2* (CD332) [HSA_VAR:2263v2] [HSA:2263] [KO:K05093]
|
D10927 Erdafitinib (JAN/USAN/INN) <JP/US>
D11417 Pemigatinib (JAN/USAN/INN) <JP/US>
D11725 Futibatinib (JAN/USAN/INN) <JP/US>
D12405 Tasurgratinib succinate (JAN) <JP>
|
FGFR2* (CD332) [HSA_VAR:2263v2 2263v1] [HSA:2263] [KO:K05093]
|
D11611 Infigratinib phosphate (USAN)
|
FGFR3 (CD333) [HSA:2261] [KO:K05094]
|
D11417 Pemigatinib (JAN/USAN/INN) <JP/US>
D11589 Infigratinib (USAN/INN)
D11611 Infigratinib phosphate (USAN)
D10481 Nintedanib (USAN/INN)
D10396 Nintedanib esylate (USAN) <JP/US>
D08907 Dovitinib lactate (USAN)
D11445 Vofatamab (USAN)
D12284 Recifercept (USAN/INN)
D12404 Tasurgratinib (INN)
D12405 Tasurgratinib succinate (JAN) <JP>
D12545 Tinengotinib (USAN/INN)
D13203 Vepugratinib (USAN)
|
FGFR3* (CD333) [HSA_VAR:2261v2] [HSA:2261] [KO:K05094]
|
D10927 Erdafitinib (JAN/USAN/INN) <JP/US>
|
FGFR4 [HSA:2264] [KO:K05095]
|
D11737 Fisogatinib (USAN/INN)
|
VEGFR family
|
VEGFR1 (FLT1) [HSA:2321] [KO:K05096]
|
D03218 Axitinib (JAN/USAN) <JP/US>
D08881 Cediranib (USAN/INN)
D08883 Cediranib maleate (JAN/USAN)
D09683 Tivozanib (USAN/INN)
D10190 Tivozanib hydrochloride (USAN) <US>
D11977 Fruquintinib (JAN/USAN) <JP/US>
D08552 Sunitinib (INN)
D06402 Sunitinib malate (JAN/USAN) <JP/US>
D05380 Pazopanib hydrochloride (JAN/USAN) <JP/US>
D10138 Regorafenib (USAN/INN)
D10137 Regorafenib hydrate (JAN) <JP/US>
D09919 Lenvatinib (USAN/INN)
D09920 Lenvatinib mesylate (USAN) <JP/US>
D10481 Nintedanib (USAN/INN)
D10396 Nintedanib esylate (USAN) <JP/US>
D11713 Selpercatinib (JAN/USAN/INN) <JP/US>
D11885 Surufatinib (USAN/INN)
D11140 Sitravatinib (USAN/INN)
D11541 Sitravatinib malate (USAN)
D06285 Vatalanib (USAN/INN)
D06678 Motesanib (USAN)
D08907 Dovitinib lactate (USAN)
D08947 Motesanib diphosphate (USAN)
D09635 Linifanib (USAN/INN)
D09926 Icrucumab (USAN/INN)
D10423 Ilorasertib (USAN/INN)
D11762 Lucitanib (USAN/INN)
D12526 Catequentinib (USAN/INN)
D12537 Catequentinib hydrochloride (USAN)
D12545 Tinengotinib (USAN/INN)
D13058 Migaldendranib (USAN/INN)
|
VEGFR2 (KDR) [HSA:3791] [KO:K05098]
|
D03218 Axitinib (JAN/USAN) <JP/US>
D08881 Cediranib (USAN/INN)
D08883 Cediranib maleate (JAN/USAN)
D09683 Tivozanib (USAN/INN)
D10190 Tivozanib hydrochloride (USAN) <US>
D11977 Fruquintinib (JAN/USAN) <JP/US>
D11288 Rivoceranib (USAN/INN)
D11289 Rivoceranib mesylate (USAN)
D08552 Sunitinib (INN)
D06402 Sunitinib malate (JAN/USAN) <JP/US>
D08524 Sorafenib (USAN/INN)
D06272 Sorafenib tosylate (USAN) <JP/US>
D05380 Pazopanib hydrochloride (JAN/USAN) <JP/US>
D06407 Vandetanib (JAN/USAN/INN) <JP/US>
D10138 Regorafenib (USAN/INN)
D10137 Regorafenib hydrate (JAN) <JP/US>
D10062 Cabozantinib (USAN)
D10095 Cabozantinib s-malate (USAN) <JP/US>
D09919 Lenvatinib (USAN/INN)
D09920 Lenvatinib mesylate (USAN) <JP/US>
D10481 Nintedanib (USAN/INN)
D10396 Nintedanib esylate (USAN) <JP/US>
D05029 Midostaurin (JAN/USAN/INN) <US>
D11885 Surufatinib (USAN/INN)
D11140 Sitravatinib (USAN/INN)
D11541 Sitravatinib malate (USAN)
D09371 Ramucirumab (USAN) <JP/US>
D05819 Semaxanib (USAN/INN)
D06285 Vatalanib (USAN/INN)
D06678 Motesanib (USAN)
D08503 Toceranib (USAN)
D08544 Toceranib phosphate (USAN)
D08878 Brivanib alaninate (JAN/USAN/INN)
D08907 Dovitinib lactate (USAN)
D08947 Motesanib diphosphate (USAN)
D09589 Brivanib (USAN)
D09618 Foretinib (USAN/INN)
D09635 Linifanib (USAN/INN)
D09945 Pegdinetanib (USAN/INN)
D10224 Golvatinib (USAN)
D10465 Golvatinib tartrate (USAN)
D10862 Altiratinib (USAN)
D11762 Lucitanib (USAN/INN)
D11772 Tesevatinib (USAN/INN)
D11773 Tesevatinib tosylate (USAN)
D12526 Catequentinib (USAN/INN)
D12537 Catequentinib hydrochloride (USAN)
D12545 Tinengotinib (USAN/INN)
D12650 Zanzalintinib (USAN/INN)
D12651 Zanzalintinib fumarate (USAN)
D13058 Migaldendranib (USAN/INN)
|
VEGFR3 (FLT4) [HSA:2324] [KO:K05097]
|
D03218 Axitinib (JAN/USAN) <JP/US>
D08881 Cediranib (USAN/INN)
D08883 Cediranib maleate (JAN/USAN)
D09683 Tivozanib (USAN/INN)
D10190 Tivozanib hydrochloride (USAN) <US>
D11977 Fruquintinib (JAN/USAN) <JP/US>
D08552 Sunitinib (INN)
D06402 Sunitinib malate (JAN/USAN) <JP/US>
D08524 Sorafenib (USAN/INN)
D06272 Sorafenib tosylate (USAN) <JP/US>
D05380 Pazopanib hydrochloride (JAN/USAN) <JP/US>
D10138 Regorafenib (USAN/INN)
D10137 Regorafenib hydrate (JAN) <JP/US>
D09919 Lenvatinib (USAN/INN)
D09920 Lenvatinib mesylate (USAN) <JP/US>
D10481 Nintedanib (USAN/INN)
D10396 Nintedanib esylate (USAN) <JP/US>
D11713 Selpercatinib (JAN/USAN/INN) <JP/US>
D11885 Surufatinib (USAN/INN)
D11140 Sitravatinib (USAN/INN)
D11541 Sitravatinib malate (USAN)
D06285 Vatalanib (USAN/INN)
D06678 Motesanib (USAN)
D08907 Dovitinib lactate (USAN)
D08947 Motesanib diphosphate (USAN)
D09635 Linifanib (USAN/INN)
D11762 Lucitanib (USAN/INN)
D11772 Tesevatinib (USAN/INN)
D11773 Tesevatinib tosylate (USAN)
D12526 Catequentinib (USAN/INN)
D12537 Catequentinib hydrochloride (USAN)
D12545 Tinengotinib (USAN/INN)
D12635 Sozinibercept (USAN/INN)
|
MET family
|
MET [HSA:4233] [KO:K05099]
|
D10696 Capmatinib (USAN/INN)
D11717 Tepotinib (USAN/INN)
D11139 Savolitinib (JAN/USAN/INN)
D10062 Cabozantinib (USAN)
D10095 Cabozantinib s-malate (USAN) <JP/US>
D11140 Sitravatinib (USAN/INN)
D11541 Sitravatinib malate (USAN)
D11894 Amivantamab (USAN/INN) <JP/US>
D13229 Amivantamab (genetical recombination) and vorhyaluronidase alfa (genetical recombination)
D09618 Foretinib (USAN/INN)
D09864 Amuvatinib (USAN/INN)
D09865 Amuvatinib hydrochloride (USAN)
D09941 Onartuzumab (USAN/INN)
D10173 Tivantinib (JAN/USAN/INN)
D10224 Golvatinib (USAN)
D10465 Golvatinib tartrate (USAN)
D10862 Altiratinib (USAN)
D11136 Glesatinib (USAN/INN)
D11307 Telisotuzumab (USAN)
D11763 Merestinib (USAN/INN)
D12287 Terevalefim (USAN/INN)
D12392 Fosgonimeton (USAN/INN)
D12393 Fosgonimeton sodium (USAN)
D12424 Davutamig (USAN)
D12557 Elzovantinib (USAN/INN)
D12650 Zanzalintinib (USAN/INN)
D12651 Zanzalintinib fumarate (USAN)
D12809 Bafisontamab (USAN/INN)
D13066 Tilatamig (USAN/INN)
D13067 Tilatamig samrotecan (USAN/INN)
D13156 Pamvatamig (USAN/INN)
|
MET* [HSA_VAR:4233v2] [HSA:4233] [KO:K05099]
|
D11344 Telisotuzumab vedotin (USAN) <US>
|
MET* [HSA_VAR:4233v4] [HSA:4233] [KO:K05099]
|
D10891 Capmatinib hydrochloride (USAN) <JP/US>
D11073 Tepotinib hydrochloride (USAN) <JP/US>
D12053 Vebreltinib (USAN)
D12705 Gumarontinib hydrate (JAN) <JP>
|
RON [HSA:4486] [KO:K05100]
|
D10074 Narnatumab (USAN)
D11763 Merestinib (USAN/INN)
|
TRK family
|
NTRK [HSA:4914 4915 4916] [KO:K03176 K04360 K05101]
|
D11137 Larotrectinib (USAN/INN)
D11138 Larotrectinib sulfate (JAN/USAN) <JP/US>
D12363 Taletrectinib (USAN/INN)
D12364 Taletrectinib adipate (JAN/USAN) <JP/US>
D12432 Zurletrectinib (USAN)
D12646 Paltimatrectinib (USAN/INN)
|
NTRK1 (TRKA) [HSA:4914] [KO:K03176]
|
D11454 Repotrectinib (JAN/USAN) <JP/US>
D11484 Pegcantratinib (USAN/INN)
|
NTRK1* (TRKA) [HSA_VAR:4914v1] [HSA:4914] [KO:K03176]
|
D10926 Entrectinib (JAN/USAN/INN) <JP/US>
|
NTRK2 (TRKB) [HSA:4915] [KO:K04360]
|
D10926 Entrectinib (JAN/USAN/INN) <JP/US>
D11454 Repotrectinib (JAN/USAN) <JP/US>
|
NTRK3 (TRKC) [HSA:4916] [KO:K05101]
|
D10926 Entrectinib (JAN/USAN/INN) <JP/US>
D11454 Repotrectinib (JAN/USAN) <JP/US>
|
EPH family
|
EPHA1 [HSA:2041] [KO:K05102]
|
D11140 Sitravatinib (USAN/INN)
D11541 Sitravatinib malate (USAN)
|
EPHA2 [HSA:1969] [KO:K05103]
|
D03658 Dasatinib (JAN/INN) <JP>
D06414 Dasatinib (USAN) <JP/US>
D12609 Dasatinib laurylsulfate (USAN)
D11140 Sitravatinib (USAN/INN)
D11541 Sitravatinib malate (USAN)
|
EPHB1 [HSA:2047] [KO:K05110]
|
D11140 Sitravatinib (USAN/INN)
D11541 Sitravatinib malate (USAN)
|
EPHB2 [HSA:2048] [KO:K05111]
|
D11140 Sitravatinib (USAN/INN)
D11541 Sitravatinib malate (USAN)
|
EPHB4 [HSA:2050] [KO:K05113]
|
D11140 Sitravatinib (USAN/INN)
D11541 Sitravatinib malate (USAN)
D11772 Tesevatinib (USAN/INN)
D11773 Tesevatinib tosylate (USAN)
|
AXL family
|
AXL [HSA:558] [KO:K05115]
|
D10062 Cabozantinib (USAN)
D10095 Cabozantinib s-malate (USAN) <JP/US>
D11140 Sitravatinib (USAN/INN)
D11541 Sitravatinib malate (USAN)
D09864 Amuvatinib (USAN/INN)
D09865 Amuvatinib hydrochloride (USAN)
D11438 Bemcentinib (USAN/INN)
D11732 Dubermatinib (USAN/INN)
D11733 Dubermatinib tartrate (USAN)
D11763 Merestinib (USAN/INN)
D12219 Mecbotamab (USAN)
D12220 Mecbotamab vedotin
D12271 Batiraxcept (USAN)
D12279 Mipasetamab (USAN/INN)
D12280 Mipasetamab uzoptirine (USAN/INN)
D12650 Zanzalintinib (USAN/INN)
D12651 Zanzalintinib fumarate (USAN)
|
TYRO3 [HSA:7301] [KO:K05116]
|
D12650 Zanzalintinib (USAN/INN)
D12651 Zanzalintinib fumarate (USAN)
|
MERTK [HSA:10461] [KO:K05117]
|
D12650 Zanzalintinib (USAN/INN)
D12651 Zanzalintinib fumarate (USAN)
|
ALK family
|
ALK (CD246) [HSA:238] [KO:K05119]
|
D10542 Alectinib (USAN/INN)
D11012 Lorlatinib (JAN/USAN/INN) <JP/US>
D10926 Entrectinib (JAN/USAN/INN) <JP/US>
D11346 Ensartinib (USAN)
D13079 Neladalkib (USAN/INN)
|
EML4-ALK [HSA_VAR:238v1] [HSA:238] [KO:K05119]
|
D09731 Crizotinib (JAN/USAN/INN) <JP/US>
D10551 Ceritinib (JAN/USAN/INN) <JP/US>
D10450 Alectinib hydrochloride (JAN) <JP/US>
D10866 Brigatinib (JAN/USAN) <JP/US>
D11012 Lorlatinib (JAN/USAN/INN) <JP/US>
D11356 Ensartinib hydrochloride (USAN) <US>
|
ALK* (CD246) [HSA_VAR:238v2] [HSA:238] [KO:K05119]
|
D11356 Ensartinib hydrochloride (USAN) <US>
|
TIE family
|
TEK (TIE2, CD202) [HSA:7010] [KO:K05121]
|
D10138 Regorafenib (USAN/INN)
D10137 Regorafenib hydrate (JAN) <JP/US>
D10334 Rebastinib (USAN)
D10399 Rebastinib Tosylate (USAN)
D10862 Altiratinib (USAN)
D11540 Razuprotafib (USAN)
|
ROR family
|
ROR2 [HSA:4920] [KO:K05123]
|
D12209 Ozuriftamab (USAN)
D12210 Ozuriftmab vedotin (USAN)
|
RET family
|
RET [HSA:5979] [KO:K05126]
|
D08552 Sunitinib (INN)
D06402 Sunitinib malate (JAN/USAN) <JP/US>
D08524 Sorafenib (USAN/INN)
D06272 Sorafenib tosylate (USAN) <JP/US>
D06407 Vandetanib (JAN/USAN/INN) <JP/US>
D10138 Regorafenib (USAN/INN)
D10137 Regorafenib hydrate (JAN) <JP/US>
D09919 Lenvatinib (USAN/INN)
D09920 Lenvatinib mesylate (USAN) <JP/US>
D06678 Motesanib (USAN)
D08947 Motesanib diphosphate (USAN)
D12330 Zeteletinib (USAN)
D12331 Zeteletinib adipate (USAN)
D12559 Enbezotinib (USAN/INN)
|
RET* [HSA_VAR:5979v1] [HSA:5979] [KO:K05126]
|
D11712 Pralsetinib (USAN/INN) <US>
D12354 Pralsetinib hydrate (JAN)
|
RET* [HSA_VAR:5979v1 5979v2] [HSA:5979] [KO:K05126]
|
D11713 Selpercatinib (JAN/USAN/INN) <JP/US>
|
CCK family
|
PTK7 [HSA:5754] [KO:K05127]
|
D11118 Cofetuzumab pelidotin (USAN)
D11119 Cofetuzumab (USAN/INN)
|
Non-receptor tyrosine kinases
|
SRC family
|
SRC [HSA:6714] [KO:K05704]
|
D11691 Tirbanibulin (JAN/USAN/INN) <US>
D11692 Tirbanibulin mesylate (USAN)
D03658 Dasatinib (JAN/INN) <JP>
D06414 Dasatinib (USAN) <JP/US>
D12609 Dasatinib laurylsulfate (USAN)
D03252 Bosutinib (USAN)
D09728 Bosutinib hydrate (JAN) <JP/US>
D09664 Saracatinib (USAN/INN)
D09665 Saracatinib difumarate (USAN)
D10423 Ilorasertib (USAN/INN)
|
FYN [HSA:2534] [KO:K05703]
|
D03658 Dasatinib (JAN/INN) <JP>
D06414 Dasatinib (USAN) <JP/US>
D12609 Dasatinib laurylsulfate (USAN)
|
LYN [HSA:4067] [KO:K05854]
|
D06182 Tolimidone (USAN)
D10202 Bafetinib (USAN)
|
LCK [HSA:3932] [KO:K05856]
|
D03658 Dasatinib (JAN/INN) <JP>
D06414 Dasatinib (USAN) <JP/US>
D12609 Dasatinib laurylsulfate (USAN)
|
YES1 [HSA:7525] [KO:K05705]
|
D03658 Dasatinib (JAN/INN) <JP>
D06414 Dasatinib (USAN) <JP/US>
D12609 Dasatinib laurylsulfate (USAN)
|
ABL family
|
ABL1 [HSA:25] [KO:K06619]
|
D03252 Bosutinib (USAN)
D09664 Saracatinib (USAN/INN)
D09665 Saracatinib difumarate (USAN)
D12828 Risvodetinib (USAN/INN)
D12829 Risvodetinib succinate (USAN)
|
BCR-ABL [HSA_VAR:25v1] [HSA:25] [KO:K06619]
|
D08066 Imatinib (INN)
D01441 Imatinib mesylate (USAN) <JP/US>
D03658 Dasatinib (JAN/INN) <JP>
D06414 Dasatinib (USAN) <JP/US>
D12609 Dasatinib laurylsulfate (USAN)
D08953 Nilotinib (USAN/INN) <US>
D06413 Nilotinib hydrochloride hydrate (JAN) <JP/US>
D12444 Nilotinib hydrochloride dihydrate (JAN) <JP>
D12854 Nilotinib laurylsulfate (USAN)
D13008 Nilotinib D-tartrate (USAN) <US>
D09728 Bosutinib hydrate (JAN) <JP/US>
D09950 Ponatinib (USAN/INN)
D09951 Ponatinib hydrochloride (JAN/USAN) <JP/US>
D11403 Asciminib (USAN/INN)
D11404 Asciminib hydrochloride (JAN/USAN) <JP/US>
D08279 Tozasertib (USAN)
D08344 Tozasertib lactate (USAN)
D10202 Bafetinib (USAN)
D10334 Rebastinib (USAN)
D10399 Rebastinib Tosylate (USAN)
D11786 Vodobatinib (USAN)
D12175 Olverembatinib (USAN/INN)
|
SYK family
|
SYK [HSA:6850] [KO:K05855]
|
D09347 Fostamatinib (USAN)
D09348 Fostamatinib disodium (USAN) <JP/US>
D11209 Entospletinib (USAN/INN)
D11676 Gusacitinib (USAN/INN)
D11677 Gusacitinib hydrochloride (USAN)
D11789 Mivavotinib (USAN/INN)
D11790 Mivavotinib citrate (USAN)
D12476 Tuspetinib (USAN/INN)
D12953 Sovleplenib (USAN/INN)
D12954 Sovleplenib acetate (USAN)
|
JAK family
|
JAK [HSA:3716 3717 3718] [KO:K11217 K04447 K11218]
|
D12476 Tuspetinib (USAN/INN)
|
JAK1 [HSA:3716] [KO:K11217]
|
D11400 Abrocitinib (JAN/USAN) <JP/US>
D09959 Ruxolitinib (USAN/INN)
D09960 Ruxolitinib phosphate (JAN/USAN) <JP/US>
D11046 Delgocitinib (JAN/USAN/INN) <JP/US>
D10315 Momelotinib (USAN/INN)
D10358 Momelotinib dihydrochloride (USAN)
D10889 Momelotinib hydrochloride hydrate (JAN) <JP/US>
D09970 Tofacitinib (USAN)
D09783 Tofacitinib citrate (JAN/USAN) <JP/US>
D10308 Baricitinib (JAN/USAN/INN) <JP/US>
D10994 Upadacitinib (USAN/INN)
D10995 Upadacitinib tartrate (USAN)
D11048 Upadacitinib hydrate (JAN) <JP/US>
D10871 Filgotinib (USAN/INN)
D10872 Filgotinib hydrochloride (USAN)
D11106 Filgotinib maleate (JAN/USAN) <JP>
D10944 Itacitinib (USAN/INN)
D10945 Itacitinib adipate (JAN/USAN)
D10653 Peficitinib (USAN/INN)
D10721 Peficitinib hydrobromide (JAN/USAN) <JP>
D11866 Deuruxolitinib (USAN)
D11867 Deuruxolitinib phosphate (USAN) <US>
D10141 Oclacitinib (USAN)
D10142 Oclacitinib maleate (USAN)
D10728 Solcitinib (USAN/INN)
D11537 Brepocitinib (USAN)
D11538 Brepocitinib tosylate (USAN)
D11676 Gusacitinib (USAN/INN)
D11677 Gusacitinib hydrochloride (USAN)
D12118 Nezulcitinib (USAN)
D12211 Ivarmacitinib (USAN)
D12212 Ivarmacitinib sulfate (USAN)
D12502 Golidocitinib (USAN/INN)
D12545 Tinengotinib (USAN/INN)
D12575 Povorcitinib (USAN/INN)
D12576 Povorcitinib phosphate (JAN/USAN)
D12786 Lepzacitinib (USAN)
D12993 Frevecitinib (USAN/INN)
D13040 Londamocitinib (USAN/INN)
D13041 Londamocitinib xinafoate (USAN)
|
JAK2 [HSA:3717] [KO:K04447]
|
D09959 Ruxolitinib (USAN/INN)
D09960 Ruxolitinib phosphate (JAN/USAN) <JP/US>
D11046 Delgocitinib (JAN/USAN/INN) <JP/US>
D10630 Fedratinib (USAN/INN)
D11296 Fedratinib hydrochloride (USAN) <JP/US>
D11768 Pacritinib (USAN/INN) <US>
D10315 Momelotinib (USAN/INN)
D10358 Momelotinib dihydrochloride (USAN)
D10889 Momelotinib hydrochloride hydrate (JAN) <JP/US>
D09970 Tofacitinib (USAN)
D09783 Tofacitinib citrate (JAN/USAN) <JP/US>
D10308 Baricitinib (JAN/USAN/INN) <JP/US>
D11106 Filgotinib maleate (JAN/USAN) <JP>
D10653 Peficitinib (USAN/INN)
D10721 Peficitinib hydrobromide (JAN/USAN) <JP>
D11866 Deuruxolitinib (USAN)
D11867 Deuruxolitinib phosphate (USAN) <US>
D10365 Gandotinib (USAN/INN)
D11599 Zotiraciclib (USAN)
D11600 Zotiraciclib citrate (USAN)
D11676 Gusacitinib (USAN/INN)
D11677 Gusacitinib hydrochloride (USAN)
D12118 Nezulcitinib (USAN)
D12545 Tinengotinib (USAN/INN)
D12993 Frevecitinib (USAN/INN)
|
JAK2* [HSA_VAR:3717v1] [HSA:3717] [KO:K04447]
|
D10889 Momelotinib hydrochloride hydrate (JAN) <JP/US>
|
JAK3 [HSA:3718] [KO:K11218]
|
D11046 Delgocitinib (JAN/USAN/INN) <JP/US>
D09970 Tofacitinib (USAN)
D09783 Tofacitinib citrate (JAN/USAN) <JP/US>
D11106 Filgotinib maleate (JAN/USAN) <JP>
D10653 Peficitinib (USAN/INN)
D10721 Peficitinib hydrobromide (JAN/USAN) <JP>
D11970 Ritlecitinib tosylate (USAN) <JP/US>
D10585 Decernotinib (USAN/INN)
D11676 Gusacitinib (USAN/INN)
D11677 Gusacitinib hydrochloride (USAN)
D12118 Nezulcitinib (USAN)
D12786 Lepzacitinib (USAN)
D12993 Frevecitinib (USAN/INN)
|
TYK2 [HSA:7297] [KO:K11219]
|
D11046 Delgocitinib (JAN/USAN/INN) <JP/US>
D09970 Tofacitinib (USAN)
D09783 Tofacitinib citrate (JAN/USAN) <JP/US>
D11106 Filgotinib maleate (JAN/USAN) <JP>
D11817 Deucravacitinib (JAN/USAN) <JP/US>
D11867 Deuruxolitinib phosphate (USAN) <US>
D11537 Brepocitinib (USAN)
D11538 Brepocitinib tosylate (USAN)
D12056 Ropsacitinib (USAN)
D12118 Nezulcitinib (USAN)
D12725 Lomedeucitinib (USAN)
D12941 Zasocitinib (JAN/USAN/INN)
D13123 Envudeucitinib (USAN/INN)
D13124 Envudeucitinib hydrochloride (USAN)
|
FAK family
|
PTK2B [HSA:2185] [KO:K05871]
|
D10618 Defactinib (USAN/INN)
D10619 Defactinib hydrochloride (USAN)
|
TEC family
|
BTK [HSA:695] [KO:K07370]
|
D10223 Ibrutinib (JAN/USAN) <JP/US>
D10893 Acalabrutinib (JAN/USAN/INN) <JP>
D11720 Acalabrutinib maleate (USAN)
D12704 Acalabrutinib maleate hydrate (JAN) <JP/US>
D11422 Zanubrutinib (JAN/USAN/INN) <JP/US>
D12160 Orelabrutinib (USAN/INN)
D12050 Pirtobrutinib (JAN/USAN) <JP/US>
D12594 Tirabrutinib (USAN/INN)
D11070 Tirabrutinib hydrochloride (JAN/USAN) <JP>
D12285 Remibrutinib (JAN/USAN/INN) <US>
D12213 Tolebrutinib (JAN/USAN/INN)
D10730 Spebrutinib (USAN/INN)
D10731 Spebrutinib besylate (USAN)
D11428 Vecabrutinib (USAN/INN)
D11457 Fenebrutinib (USAN/INN)
D11478 Branebrutinib (USAN)
D11502 Vecabrutinib succinate (USAN)
D11873 Rilzabrutinib (JAN/USAN/INN) <US>
D12052 Luxeptinib (USAN)
D12158 Elsubrutinib (USAN/INN)
D12383 Edralbrutinib (USAN/INN)
D12467 Evobrutinib (USAN/INN)
D12489 Atuzabrutinib (USAN/INN)
D12504 Nemtabrutinib (USAN/INN)
D12858 Zelebrudomide (USAN)
D13115 Bexobrutideg (USAN)
D13142 Docirbrutinib (USAN/INN)
D13143 Docirbrutinib mesylate (USAN)
|
ITK [HSA:3702] [KO:K07363]
|
D12762 Soquelitinib (USAN)
|
|
Peptidases and inhibitors
|
Aspartic peptidases
|
Pepsin family
|
BACE [HSA:23621 25825] [KO:K04521 K07747]
|
D10739 Verubecestat (JAN/USAN/INN)
D11509 Elenbecestat (JAN/USAN)
|
BACE1 [HSA:23621] [KO:K04521]
|
D10946 Lanabecestat (USAN/INN)
D10947 Lanabecestat camsylate (USAN)
D11456 Atabecestat (USAN/INN)
D11690 Umibecestat (USAN/INN)
|
REN [HSA:5972] [KO:K01380]
|
D09038 Remikiren (INN)
D03208 Aliskiren (USAN/INN)
D06412 Aliskiren fumarate (JAN/USAN) <JP/US>
D03738 Enalkiren (USAN/INN)
D03741 Ditekiren (USAN)
D03743 Terlakiren (USAN/INN)
D03745 Zankiren hydrochloride (USAN)
|
Presenilin family
|
PSEN1/PSENEN/NCSTN/APH1A [HSA:5663 55851 23385 51107] [KO:K04505 K06170 K06171 K06172]
|
D10960 Nirogacestat (USAN/INN)
D11453 Nirogacestat hydrobromide (USAN) <US>
D08869 Begacestat (USAN/INN)
D09010 Tarenflurbil (USAN/INN)
D09377 Semagacestat (USAN/INN)
D09869 Avagacestat (USAN)
D11151 Crenigacestat (USAN/INN)
D12235 Osugacestat (USAN/INN)
D13031 Varegacestat (USAN/INN)
D13199 Nivegacetor (USAN/INN)
|
Cysteine peptidases
|
Papain family
|
CTSC (DPP1) [HSA:1075] [KO:K01275]
|
D12120 Brensocatib (USAN/INN)
D12746 Brensocatib hydrate (JAN) <US>
|
CTSK [HSA:1513] [KO:K01371]
|
D06634 Relacatib (USAN/INN)
D08955 Odanacatib (JAN/USAN)
|
CTSL [HSA:1514] [KO:K01365]
|
D12777 Olgotrelvir (USAN)
D12778 Olgotrelvir sodium (USAN)
|
CTSS [HSA:1520] [KO:K01368]
|
D11376 Petesicatib (USAN)
|
Caspase family
|
CASP1 [HSA:834] [KO:K01370]
|
D08978 Pralnacasan (USAN/INN)
D09938 Nivocasan (USAN)
D10004 Emricasan (USAN/INN)
D10416 Belnacasan (USAN/INN)
|
CASP9 [HSA:842] [KO:K04399]
|
D11195 Rimiducid (USAN/INN)
|
Metallo peptidases
|
Family M1
|
ANPEP (CD13) [HSA:290] [KO:K11140]
|
D00087 Ubenimex (JP18/INN) <JP>
D10026 Tosedostat (USAN/INN)
|
Family M2
|
ACE (CD143) [HSA:1636] [KO:K01283]
|
D00251 Captopril (JP18/USP/INN) <JP/US>
D07892 Enalapril (INN)
D00621 Enalapril maleate (JP18/USP) <JP/US>
D08131 Lisinopril (INN)
D00362 Lisinopril (USP) <JP/US>
D03753 Perindopril (USAN/INN)
D00624 Perindopril erbumine (JAN/USP) <JP/US>
D11580 Perindopril arginine
D00421 Ramipril (USP/INN) <US>
D03752 Quinapril (INN)
D00459 Quinapril hydrochloride (JP18/USP) <US>
D07499 Benazepril (INN)
D00620 Benazepril hydrochloride (JAN/USP) <US>
D07699 Cilazapril (INN)
D01069 Cilazapril (USAN)
D07992 Fosinopril (INN)
D00622 Fosinopril sodium (USP) <US>
D00383 Trandolapril (JAN/USP/INN) <JP/US>
D08529 Spirapril (INN)
D03765 Spirapril hydrochloride (USAN)
D07781 Delapril (INN)
D01667 Delapril hydrochloride (JAN/USAN) <JP>
D08225 Moexipril (INN)
D00623 Moexipril hydrochloride (USP) <US>
D08566 Temocapril (INN)
D01119 Temocapril hydrochloride (JP18/USAN) <JP>
D08688 Zofenopril (INN)
D03767 Zofenopril calcium (USAN)
D08068 Imidapril (INN)
D01549 Imidapril hydrochloride (JP18) <JP>
D01900 Alacepril (JP18/INN) <JP>
D03077 Benazeprilat (USAN/INN)
D03440 Ceronapril (USAN/INN)
D03756 Indolapril hydrochloride (USAN)
D03758 Libenzapril (USAN/INN)
D03760 Pentopril (USAN/INN)
D03763 Pivopril (USAN/INN)
D03769 Enalaprilat (USP) <US>
D03772 Fosinoprilat (USAN/INN)
D03773 Quinaprilat (USAN/INN)
D03775 Spiraprilat (USAN/INN)
D03776 Zofenoprilat arginine (USAN)
D04312 Gemopatrilat (USAN/INN)
D06076 Teprotide (USAN/INN)
|
Family M10
|
MMP1 [HSA:4312] [KO:K01388]
|
D03517 Cipemastat (USAN/INN)
D03795 Marimastat (USAN/INN)
D03800 Rebimastat (USAN/INN)
D03802 Tanomastat (USAN/INN)
D11020 Diclofenac etalhyaluronate sodium (JAN) <JP>
|
MMP2 [HSA:4313] [KO:K01398]
|
D03061 Batimastat (USAN/INN)
D03793 Ilomastat (USAN/INN)
D03795 Marimastat (USAN/INN)
D03797 Prinomastat (USAN/INN)
D03800 Rebimastat (USAN/INN)
D03802 Tanomastat (USAN/INN)
|
MMP3 [HSA:4314] [KO:K01394]
|
D03795 Marimastat (USAN/INN)
D03797 Prinomastat (USAN/INN)
|
MMP7 [HSA:4316] [KO:K01397]
|
D03795 Marimastat (USAN/INN)
|
MMP8 [HSA:4317] [KO:K01402]
|
D03517 Cipemastat (USAN/INN)
D03800 Rebimastat (USAN/INN)
|
MMP9 [HSA:4318] [KO:K01403]
|
D03061 Batimastat (USAN/INN)
D03517 Cipemastat (USAN/INN)
D03793 Ilomastat (USAN/INN)
D03795 Marimastat (USAN/INN)
D03797 Prinomastat (USAN/INN)
D03800 Rebimastat (USAN/INN)
D03802 Tanomastat (USAN/INN)
D11262 Andecaliximab (USAN/INN)
|
MMP12 [HSA:4321] [KO:K01413]
|
D03795 Marimastat (USAN/INN)
D12909 Aderamastat (USAN/INN)
|
MMP13 [HSA:4322] [KO:K07994]
|
D03517 Cipemastat (USAN/INN)
D03797 Prinomastat (USAN/INN)
D08859 Apratastat (USAN/INN)
|
MMP14 [HSA:4323] [KO:K07763]
|
D03797 Prinomastat (USAN/INN)
D03800 Rebimastat (USAN/INN)
|
Family M12
|
ADAM10 [HSA:102] [KO:K06704]
|
D09320 Aderbasib (USAN/INN)
|
ADAM17 [HSA:6868] [KO:K06059]
|
D08859 Apratastat (USAN/INN)
D09320 Aderbasib (USAN/INN)
|
ADAMTS5 [HSA:11096] [KO:K08620]
|
D11995 Aldumastat (USAN)
|
ADAMTS13 [HSA:11093] [KO:K08627]
|
D12835 Apadamtase alfa and cinaxadamtase alfa <JP/US>
D12569 Apadamtase alfa (INN)
D12570 Cinaxadamtase alfa (INN)
|
Family M13
|
MME (CD10) [HSA:4311] [KO:K01389]
|
D08464 Racecadotril (INN)
D10226 Sacubitril valsartan sodium hydrate (JAN) <JP/US>
D01070 Candoxatril (JAN/USAN/INN)
D01970 Omapatrilat (JAN/USAN/INN)
D03349 Candoxatrilat (USAN/INN)
D03929 Ecadotril (USAN/INN)
D10225 Sacubitril (JAN/USAN/INN)
|
Family M19
|
DPEP1 [HSA:1800] [KO:K01273]
|
D02194 Cilastatin sodium (JP18/USP)
D07698 Cilastatin (INN)
|
Family M28
|
FOLH1 (PSMA) [HSA:2346] [KO:K14592]
|
D10683 Technetium Tc99m trofolastat chloride (USAN/INN)
D04525 Indium In 111 capromab pendetide (USP)
D12257 Gallium Ga 68 gozetotide (USAN) <JP/US>
D12132 Piflufolastat F-18 (USAN) <US>
D12606 Flotufolastat F18 gallium (USAN) <US>
D13230 Vidoflufolastat F 18 (USAN)
D12335 Lutetium Lu 177 vipivotide tetraxetan (USAN) <JP/US>
D03372 Capromab pendetide (USAN)
D10070 Iofolastat I 123 (USAN)
D12121 Acapatamab (USAN)
D12566 Nezastomig (USAN)
D13129 Abefolastat tesaroxetan (USAN/INN)
|
TFRC (CD71) [HSA:7037] [KO:K06503]
|
D11812 Pabinafusp alfa (genetical recombination) (JAN) <JP>
D12509 Trontinemab (USAN/INN)
D12806 Tividenofusp alfa (USAN/INN)
D13112 Zeleciment (USAN/INN)
D13225 Delpacibart (USAN/INN)
|
Serine peptidases
|
Chymotrypsin family
|
CTRB [HSA:1504 440387] [KO:K01310]
|
D05183 Ulinastatin (JP18) <JP>
|
PRSS [HSA:5644 5645 5646] [KO:K01312]
|
D05183 Ulinastatin (JP18) <JP>
|
ELANE [HSA:1991] [KO:K01327]
|
D05183 Ulinastatin (JP18) <JP>
D01918 Sivelestat sodium (USAN) <JP>
D03686 Depelestat (USAN/INN)
D03788 Sivelestat (USAN/INN)
|
CELA1 [HSA:1990] [KO:K01326]
|
D11770 Vonapanitase (USAN/INN)
|
KLK [HSA:3816 3817] [KO:K01325]
|
D01672 Gabexate mesilate (JP18) <JP>
D08004 Gabexate (INN)
|
KLK1 [HSA:3816] [KO:K01325]
|
D12830 Rinvecalinase alfa (USAN/INN)
|
KLK2 [HSA:3817] [KO:K01325]
|
D13137 Alpitatug (USAN/INN)
D13159 Pasritamig (USAN/INN)
|
KLKB1 [HSA:3818] [KO:K01324]
|
D03931 Ecallantide (USAN/INN) <US>
D10845 Conestat alfa (INN) <US>
D11094 Lanadelumab (USAN) <JP/US>
D11673 Berotralstat (USAN/INN)
D11674 Berotralstat hydrochloride (JAN/USAN) <JP/US>
D12396 Sebetralstat (JAN/USAN/INN) <US>
D13154 Donidalorsen sodium (USAN) <US>
D01672 Gabexate mesilate (JP18) <JP>
D08004 Gabexate (INN)
D12573 Feniralstat (USAN/INN)
D12574 Feniralstat hydrochloride (USAN)
D12770 Navenibart (USAN)
|
MASP1 (MASP-3) [HSA:5648] [KO:K03992]
|
D12920 Zaltenibart (USAN/INN)
|
MASP2 [HSA:10747] [KO:K03993]
|
D11531 Narsoplimab (USAN)
|
C1R [HSA:715] [KO:K01330]
|
D10845 Conestat alfa (INN) <US>
|
C1S [HSA:716] [KO:K01331]
|
D10845 Conestat alfa (INN) <US>
D11530 Sutimlimab (USAN/INN) <JP/US>
D12895 Riliprubart (USAN/INN)
|
C2 [HSA:717] [KO:K01332]
|
D12992 Empasiprubart (USAN/INN)
|
CFB [HSA:629] [KO:K01335]
|
D12251 Iptacopan (USAN/INN)
D12252 Iptacopan hydrochloride (USAN) <JP/US>
D12857 Ruxoprubart (USAN)
|
CFD [HSA:1675] [KO:K01334]
|
D11641 Danicopan (JAN/USAN/INN) <JP/US>
D10440 Lampalizumab (USAN/INN)
D12481 Vemircopan (USAN/INN)
|
F2a [CPD:C00752] [HSA:2147] [KO:K01313]
|
D03692 Desirudin (USAN/INN)
D06880 Lepirudin (INN)
D00181 Argatroban (USP) <JP/US>
D07143 Melagatran (INN)
D01981 Ximelagatran (JAN/USAN/INN)
D03136 Bivalirudin (USAN/INN)
D11280 Bivalirudin trifluoroacetate (USAN) <US>
D07144 Dabigatran etexilate (USAN/INN)
D07082 Dabigatran etexilate mesylate (USAN) <JP/US>
D03722 Efegatran sulfate (USAN)
D03728 Napsagatran (USAN)
D06410 Thrombomodulin alfa (USAN/INN) <JP>
D09707 Dabigatran (USAN/INN)
|
F3 (CD142, TF) [HSA:2152] [KO:K03901]
|
D11814 Tisotumab vedotin (USAN/INN) <JP/US>
D06142 Tifacogin (USAN/INN)
D11813 Tisotumab (USAN)
|
F7a [CPD:C03378] [HSA:2155] [KO:K01320]
|
D12421 Freeze-dried activated human blood coagulation factor VII concentrate containing factor X <JP>
D00172 Eptacog alfa (INN) <JP/US>
D10139 Vatreptacog alfa (activated) (genetical recombination) (JAN)
D06142 Tifacogin (USAN/INN)
|
F9 [HSA:2158] [KO:K01321]
|
D12500 Etranacogene dezaparvovec (USAN/INN) <US>
D12541 Gruticibart (USAN)
|
F9a [CPD:C03259] [HSA:2158] [KO:K01321]
|
D10821 Emicizumab (USAN/INN) <JP/US>
D10150 Pegnivacogin sodium (USAN)
D10484 Pegnivacogin (USAN/INN)
D12797 Denecimig (USAN/INN)
|
F9* [HSA_VAR:2158v1] [HSA:2158] [KO:K01321]
|
D08797 Freeze-dried human blood-coagulation factor IX <JP/US>
D08794 Human blood-coagulation factor IX complex, dried <JP>
D05201 Nonacog alfa (USAN/INN) <JP>
D10401 Trenonacog alfa (USAN/INN)
D10522 Eftrenonacog alfa (INN) <JP>
D10538 Nonacog gamma (INN)
D10757 Nonacog beta pegol (INN) <JP>
D10770 Albutrepenonacog alfa (INN) <JP>
D12908 Fidanacogene elaparvovec (USAN/INN)
|
F10 [HSA:2159] [KO:K01314]
|
D12421 Freeze-dried activated human blood coagulation factor VII concentrate containing factor X <JP>
D10821 Emicizumab (USAN/INN) <JP/US>
D12797 Denecimig (USAN/INN)
|
F10a [CPD:C01065] [HSA:2159] [KO:K01314]
|
D07086 Rivaroxaban (JAN/USAN/INN) <JP/US>
D03213 Apixaban (JAN/USAN/INN) <JP/US>
D09710 Edoxaban (USAN/INN)
D09546 Edoxaban tosilate hydrate (JAN) <JP/US>
D11568 Edoxaban tosylate (USAN)
D08873 Betrixaban (USAN)
D01844 Fondaparinux sodium (JAN/USP/INN) <JP/US>
D11029 Andexanet alfa (USAN/INN) <JP/US>
D04029 Razaxaban hydrochloride (USAN)
D04183 Fidexaban (USAN/INN)
D08913 Eribaxaban (USAN)
D09817 Darexaban maleate (JAN)
D09923 Letaxaban (USAN/INN)
D10471 Idraparinux sodium (USAN)
|
F11a [CPD:C03262] [HSA:2160] [KO:K01323]
|
D11802 Milvexian (USAN)
D12563 Frunexian (USAN)
D12564 Frunexian hydrochloride (USAN)
D12838 Asundexian (JAN/INN)
|
F12a [CPD:C03379] [HSA:2161] [KO:K01328]
|
D12613 Garadacimab (INN) <JP/US>
|
PLAT [HSA:5327] [KO:K01343]
|
D00160 Aminocaproic acid (USP/INN) <US>
|
PLG [HSA:5340] [KO:K01315]
|
D12149 Plasminogen
|
Plasmin [CPD:C00471] [HSA:5340] [KO:K01315]
|
D00160 Aminocaproic acid (USP/INN) <US>
D01136 Tranexamic acid (JP18/USP/INN) <JP/US>
D07568 Aminomethylbenzoic acid
|
LPA [HSA:4018] [KO:K09644]
|
D12460 Muvalaplin (USAN)
|
HTRA1 [HSA:5654] [KO:K08784]
|
D12379 Galegenimab (USAN/INN)
|
Subtilisin family
|
PCSK9 [HSA:255738] [KO:K13050]
|
D10557 Evolocumab (USAN/INN) <JP/US>
D10335 Alirocumab (USAN) <US>
D11931 Inclisiran (USAN/INN)
D12293 Inclisiran sodium (JAN) <JP/US>
D13095 Lerodalcibep (USAN/INN)
D10621 Bococizumab (USAN/INN)
D11398 Frovocimab (USAN/INN)
|
Prolyl oligopeptidase family
|
DPP4 (CD26) [HSA:1803] [KO:K01278]
|
D08516 Sitagliptin (USAN/INN) <US>
D06645 Sitagliptin phosphate (USAN) <JP/US>
D12294 Sitagliptin phosphate (JAN)
D13055 Sitagliptin hydrochloride <US>
D07080 Vildagliptin (JAN/USAN/INN) <JP>
D08996 Saxagliptin (USAN/INN)
D09753 Saxagliptin hydrate (JAN) <JP/US>
D10262 Saxagliptin hydrochloride <US>
D06553 Alogliptin benzoate (JAN/USAN) <JP/US>
D09566 Linagliptin (JAN/USAN/INN) <JP/US>
D12703 Linagliptin hydrate (JAN)
D10502 Gemigliptin (INN)
D11023 Evogliptin (INN)
D08616 Teneligliptin (INN)
D09756 Teneligliptin hydrobromide hydrate (JAN) <JP>
D11968 Teneligliptin hydrobromide (JAN)
D06578 Denagliptin tosylate (USAN)
D08631 Carmegliptin (USAN/INN)
D09326 Carmegliptin dihydrochloride (USAN)
D09333 Dutogliptin (USAN)
D09334 Dutogliptin tartrate (USAN)
D09625 Gosogliptin (USAN/INN)
D09780 Anagliptin (JAN/INN) <JP>
D10178 Trelagliptin (USAN)
D10179 Trelagliptin succinate (JAN/USAN) <JP>
D10317 Omarigliptin (JAN/USAN/INN) <JP>
|
DPP8 [HSA:54878] [KO:K08655]
|
D05989 Talabostat (USAN/INN)
D05990 Talabostat mesylate (USAN)
|
DPP9 [HSA:91039] [KO:K08656]
|
D05989 Talabostat (USAN/INN)
D05990 Talabostat mesylate (USAN)
|
ClpP endopeptidase family
|
CLPP [HSA:8192] [KO:K01358]
|
D12733 Dordaviprone (USAN/INN)
D12734 Dordaviprone hydrochloride (JAN/USAN) <US>
|
Family S53
|
TPP1* [HSA_VAR:1200v1] [HSA:1200] [KO:K01279]
|
D10813 Cerliponase alfa (USAN/INN) <JP/US>
|
Threonine peptidases
|
Proteasome family
|
PSMB2 [HSA:5690] [KO:K02734]
|
D09640 Marizomib (USAN/INN)
|
PSMB5 [HSA:5693] [KO:K02737]
|
D03150 Bortezomib (JAN/USAN/INN) <JP/US>
D12311 Bortezomib hydrate (JAN) <JP/US>
D08880 Carfilzomib (JAN/USAN/INN) <JP/US>
D10130 Ixazomib (USAN)
D10131 Ixazomib citrate (JAN/USAN) <JP/US>
D09640 Marizomib (USAN/INN)
D10110 Delanzomib (USAN)
D10318 Oprozomib (USAN/INN)
|
PSMB1 [HSA:5689] [KO:K02732]
|
D09640 Marizomib (USAN/INN)
D10110 Delanzomib (USAN)
|
PSMB8 [HSA:5696] [KO:K02740]
|
D12512 Zetomipzomib (USAN/INN)
D12513 Zetomipzomib maleate (USAN)
|
PSMB9 [HSA:5698] [KO:K02741]
|
D12512 Zetomipzomib (USAN/INN)
D12513 Zetomipzomib maleate (USAN)
|
Peptidase inhibitors
|
Kunitz/BPTI family
|
TFPI [HSA:7035] [KO:K03909]
|
D11847 Concizumab (USAN) <JP/US>
D11261 Marstacimab (USAN) <JP/US>
|
Serpin family
|
SERPINA1 [HSA:5265] [KO:K03984]
|
D11965 alpha 1-Antitrypsin <JP>
|
AGT [HSA:183] [KO:K09821]
|
D12840 Zilebesiran sodium (JAN/USAN)
|
SERPINC1 (AT3) [HSA:462] [KO:K03911]
|
D07510 Adomiparin (USAN)
D02112 Heparin sodium (JP18/USP/INN) <JP/US>
D04427 Heparin calcium (JP18) <JP>
D03353 Dalteparin sodium (JAN/USP/INN) <JP/US>
D03674 Enoxaparin sodium (JAN/USP/INN) <JP/US>
D04977 Parnaparin sodium (JP18) <JP>
D03337 Reviparin sodium (JAN)
D03644 Danaparoid sodium (JAN/USAN)
D06398 Tinzaparin sodium (USAN)
D08547 Sulodexide (INN)
D01844 Fondaparinux sodium (JAN/USP/INN) <JP/US>
D11810 Fitusiran sodium (JAN) <US>
D02956 Anticoagulant heparin (USP)
D02980 Adomiparin sodium (USAN)
D03673 Deligoparin sodium (USAN/INN)
D10418 Delparantag pentahydrochloride (USAN)
|
SERPIND1 [HSA:3053] [KO:K03912]
|
D08547 Sulodexide (INN)
D02980 Adomiparin sodium (USAN)
|
SERPINE1 (PAI1) [HSA:5054] [KO:K03982]
|
D03766 Diaplasinin (USAN)
D06160 Tiplasinin (USAN)
D08656 Aleplasinin (USAN/INN)
|
Cystatin family
|
KNG1 [HSA:3827] [KO:K03898]
|
D03330 Kallidinogenase (JP18/INN) <JP>
|
alpha2M family
|
C3 (C3b) [HSA:718] [KO:K03990]
|
D11613 Pegcetacoplan (JAN/USAN/INN) <JP/US>
|
C5 [HSA:727] [KO:K03994]
|
D03940 Eculizumab (USAN/INN) <JP/US>
D11054 Ravulizumab (USAN/INN) <JP/US>
D12357 Zilucoplan (USAN/INN)
D12356 Zilucoplan sodium (JAN) <JP/US>
D11696 Crovalimab (USAN/INN) <JP/US>
D11477 Pozelimab (USAN) <US>
D11748 Avacincaptad pegol sodium (JAN/USAN) <JP/US>
D10023 Pexelizumab (USAN/INN)
D11473 Nomacopan (USAN/INN)
D12208 Gefurulimab (USAN)
|
C5 (C5a) [HSA:727] [KO:K03994]
|
D11838 Vilobelimab (USAN) <US>
D11331 Olendalizumab (USAN)
|
IAP family
|
BIRC5 [HSA:332] [KO:K08731]
|
D09909 Gataparsen (USAN/INN)
D09910 Gataparsen sodium (USAN)
D10164 Sepantronium bromide (JAN/USAN)
|
|
Signaling molecules and receptors
|
Cytokines
|
Interleukins
|
IL1 [HSA:3552 3553] [KO:K04383 K04519]
|
D06635 Rilonacept (USAN/INN) <US>
D01583 Pirfenidone (JAN/USAN/INN) <JP/US>
D12370 Lutikizumab (INN)
|
IL1A [HSA:3552] [KO:K04383]
|
D11253 Bermekimab (USAN)
D12350 Vilamakitug (USAN)
D12851 Lunlekitug (USAN)
|
IL1B [HSA:3553] [KO:K04519]
|
D09315 Canakinumab (USAN/INN) <JP/US>
D09911 Gevokizumab (USAN/INN)
|
IL2 [HSA:3558] [KO:K05429]
|
D12625 Pegenzileukin (USAN/INN)
D12791 Eciskafusp alfa (USAN/INN)
D12850 Imneskibart (USAN)
|
IL4 [HSA:3565] [KO:K05430]
|
D03117 Binetrakin (USAN/INN)
D05377 Pascolizumab (USAN/INN)
D12962 Tilrekimig (USAN)
D12985 Ompekimig (USAN)
|
IL5 [HSA:3567] [KO:K05428]
|
D08985 Reslizumab (USAN) <US>
D04923 Mepolizumab (USAN/INN) <JP/US>
D12169 Depemokimab (USAN)
|
IL6 [HSA:3569] [KO:K05405]
|
D09669 Siltuximab (USAN/INN) <US>
D10080 Sirukumab (USAN)
D12487 Olokizumab (INN)
D01583 Pirfenidone (JAN/USAN/INN) <JP/US>
D08976 Pomalidomide (JAN/USAN/INN) <JP/US>
D12807 Ziltivekimab (USAN/INN)
D12929 Vamikibart (USAN/INN)
D13049 Pacibekitug (USAN/INN)
|
IL8 [HSA:3576] [KO:K10030]
|
D12656 Adakitug (USAN)
|
IL9 [HSA:3578] [KO:K05432]
|
D09897 Enokizumab (USAN/INN)
|
IL10 [HSA:3586] [KO:K05443]
|
D01583 Pirfenidone (JAN/USAN/INN) <JP/US>
|
IL12 [HSA:3592 3593] [KO:K05406 K05425]
|
D09214 Ustekinumab (USAN/INN) <JP/US>
D09588 Briakinumab (USAN/INN)
D04748 Lisofylline (USAN/INN)
D06556 Apilimod mesylate (USAN)
|
IL13 [HSA:3596] [KO:K05435]
|
D09979 Tralokinumab (USAN/INN) <JP/US>
D09633 Lebrikizumab (USAN/INN) <JP/US>
D11843 Cendakimab (USAN/INN)
D08857 Anrukinzumab (USAN)
D11598 Romilkimab (USAN/INN)
D12962 Tilrekimig (USAN)
D12985 Ompekimig (USAN)
D13054 Lunsekimig (USAN/INN)
D13155 Donzakimig (USAN/INN)
|
IL15 [HSA:3600] [KO:K05433]
|
D12306 Ordesekimab (USAN)
|
IL17A [HSA:3605] [KO:K05489]
|
D09967 Secukinumab (USAN/INN) <JP/US>
D10071 Ixekizumab (USAN) <JP/US>
D11550 Bimekizumab (USAN/INN) <JP/US>
D10902 Afasevikumab (USAN/INN)
D11127 Tibulizumab (USAN/INN)
D12278 Izokibep (USAN/INN)
D13089 Simepdekinra (USAN)
D13160 Galvokimig (USAN/INN)
D13227 Sonelokimab (USAN/INN)
|
IL17F [HSA:112744] [KO:K05494]
|
D11550 Bimekizumab (USAN/INN) <JP/US>
D10902 Afasevikumab (USAN/INN)
D13160 Galvokimig (USAN/INN)
D13227 Sonelokimab (USAN/INN)
|
IL18 [HSA:3606] [KO:K05482]
|
D04487 Iboctadekin (USAN/INN)
D13196 Aletekitug (USAN/INN)
|
IL20 [HSA:50604] [KO:K22667]
|
D11756 Fletikumab (USAN/INN)
|
IL22 [HSA:50616] [KO:K05445]
|
D09615 Fezakinumab (USAN/INN)
D11953 Efmarodocokin alfa (USAN/INN)
D13155 Donzakimig (USAN/INN)
|
IL23A [HSA:51561] [KO:K05426]
|
D09214 Ustekinumab (USAN/INN) <JP/US>
D09588 Briakinumab (USAN/INN)
D10438 Guselkumab (USAN/INN) <JP/US>
D10400 Tildrakizumab (USAN) <JP/US>
D11052 Risankizumab (USAN/INN) <JP/US>
D11123 Mirikizumab (USAN/INN) <JP/US>
D06556 Apilimod mesylate (USAN)
D10912 Brazikumab (USAN/INN)
|
IL27 [HSA:246778] [KO:K22629]
|
D12784 Casdozokitug (USAN/INN)
|
IL33 [HSA:90865] [KO:K12967]
|
D11449 Etokimab (USAN)
D11999 Itepekimab (USAN/INN)
D12375 Tozorakimab (USAN/INN)
D12985 Ompekimig (USAN)
|
Interferons
|
IFNA [HSA:3439 3440 3441 3442 3443 3444 3445 3446 3447 3448 3449 3451 3452] [KO:K05414]
|
D09662 Rontalizumab (USAN/INN)
D09668 Sifalimumab (USAN/INN)
|
IFNA2 [HSA:3440] [KO:K05414]
|
D12531 Nadofaragene firadenovec (USAN/INN) <US>
|
IFNB [HSA:3456] [KO:K05415]
|
D12464 Dazukibart (USAN)
|
IFNG [HSA:3458] [KO:K04687]
|
D11120 Emapalumab (USAN/INN) <US>
D04242 Fontolizumab (USAN/INN)
|
CSF and other factors
|
CSF2 [HSA:1437] [KO:K05427]
|
D11121 Gimsilumab (USAN/INN)
D11236 Lenzilumab (USAN/INN)
D11343 Otilimab (USAN)
|
PRL [HSA:5617] [KO:K05439]
|
D03165 Bromocriptine (USAN/INN)
D00780 Bromocriptine mesylate (USP) <JP/US>
D00987 Cabergoline (JP18/USP/INN) <JP/US>
D01348 Terguride (JAN/INN)
|
TSLP [HSA:85480] [KO:K05436]
|
D11771 Tezepelumab (USAN/INN) <JP/US>
D12962 Tilrekimig (USAN)
D13054 Lunsekimig (USAN/INN)
|
LIF [HSA:3976] [KO:K05419]
|
D12810 Falbikitug (USAN/INN)
|
CNTF [HSA:1270] [KO:K05420]
|
D13084 Revakinagene taroretcel (USAN/INN) <US>
|
Chemokines
|
CCL2 [HSA:6347] [KO:K14624]
|
D01583 Pirfenidone (JAN/USAN/INN) <JP/US>
D03116 Bindarit (USAN/INN)
D09877 Carlumab (USAN)
D12654 Emapticap pegol (INN)
|
CCL11 [HSA:6356] [KO:K16597]
|
D11741 Lazucirnon (USAN)
D11742 Lazucirnon hydrochloride (USAN)
|
CCL24 [HSA:6369] [KO:K21097]
|
D13213 Nebokitug (USAN/INN)
|
CXCL10 [HSA:3627] [KO:K12671]
|
D10404 Eldelumab (USAN/INN)
|
CXCL12 [HSA:6387] [KO:K10031]
|
D12655 Olaptesed pegol (INN)
|
CX3CL1 [HSA:6376] [KO:K05508]
|
D11498 Quetmolimab (USAN)
|
Tumor necrosis factors
|
TNF (TNFA, TNFSF2) [HSA:7124] [KO:K03156]
|
D00742 Etanercept (USAN/INN) <JP/US>
D02598 Infliximab (USAN/INN) <JP/US>
D07436 Afelimomab (INN)
D02597 Adalimumab (USAN/INN) <JP/US>
D03441 Certolizumab pegol (USAN/INN) <JP/US>
D04358 Golimumab (USAN/INN) <JP/US>
D11703 Opinercept (INN)
D00754 Thalidomide (JAN/USP/INN) <JP/US>
D04687 Lenalidomide (JAN/USAN/INN) <JP/US>
D09813 Lenalidomide hydrate (JAN) <JP>
D01583 Pirfenidone (JAN/USAN/INN) <JP/US>
D08976 Pomalidomide (JAN/USAN/INN) <JP/US>
D04690 Lenercept (USAN/INN)
D05146 Nerelimomab (USAN/INN)
D05263 Onercept (USAN/INN)
D05393 Pegsunercept (USAN)
D09944 Ozoralizumab (USAN) <JP>
D10320 Placulumab (USAN/INN)
D12420 Licaminlimab (USAN/INN)
D12790 Adalimumab fosimdesonide (USAN/INN)
D13138 Brivekimig (USAN/INN)
|
LTA (TNFB, TNFSF1) [HSA:4049] [KO:K05468]
|
D00742 Etanercept (USAN/INN) <JP/US>
D04690 Lenercept (USAN/INN)
D10187 Pateclizumab (USAN)
|
LTB (TNFC, TNFSF3) [HSA:4050] [KO:K03157]
|
D04690 Lenercept (USAN/INN)
D08866 Baminercept (USAN/INN)
|
TNFSF4 (CD252, OX40L) [HSA:7292] [KO:K05469]
|
D09943 Oxelumab (USAN/INN)
D12550 Amlitelimab (USAN/INN)
D13138 Brivekimig (USAN/INN)
|
TNFSF5 (CD154) [HSA:959] [KO:K03161]
|
D05777 Ruplizumab (USAN/INN)
D06193 Toralizumab (USAN/INN)
D11122 Letolizumab (USAN/INN)
D12620 Frexalimab (USAN/INN)
|
TNFSF7 (CD70) [HSA:970] [KO:K05470]
|
D10341 Vorsetuzumab mafodotin (USAN/INN)
D10342 Vorsetuzumab (USAN/INN)
|
TNFSF11 (RANKL, CD254) [HSA:8600] [KO:K05473]
|
D03684 Denosumab (USAN) <JP/US>
|
TNFSF13 (APRIL, CD256) [HSA:8741] [KO:K05475]
|
D12374 Sibeprenlimab (USAN/INN) <US>
D09704 Atacicept (USAN/INN)
D12800 Zigakibart (USAN/INN)
|
TNFSF13B (BAFF, CD257) [HSA:10673] [KO:K05476]
|
D03068 Belimumab (USAN) <JP/US>
D02979 Ardenermin (USAN)
D08877 Briobacept (USAN)
D09704 Atacicept (USAN/INN)
D10083 Tabalumab (USAN)
D11127 Tibulizumab (USAN/INN)
D11907 Rozibafusp alfa (USAN/INN)
|
TNFSF14 [HSA:8740] [KO:K05477]
|
D12648 Quisovalimab (USAN/INN)
|
TNFSF15 [HSA:9966] [KO:K05478]
|
D12760 Tulisokibart (USAN/INN)
D12950 Duvakitug (USAN/INN)
D13220 Afimkibart (USAN/INN)
|
Transforming growth factors (RSTK-binding)
|
TGFB [HSA:7040 7042 7043] [KO:K13375 K13376 K13377]
|
D09620 Fresolimumab (USAN/INN)
|
TGFB1 [HSA:7040] [KO:K13375]
|
D12793 Livmoniplimab (USAN/INN)
D12801 Linavonkibart (USAN/INN)
|
TGFB2 [HSA:7042] [KO:K13376]
|
D06563 Belagenpumatucel-L (USAN)
D10203 Trabedersen (INN/BAN)
|
MSTN [HSA:2660] [KO:K05497]
|
D11797 Apitegromab (USAN)
D05917 Stamulumab (USAN)
D10347 Ramatercept (USAN/INN)
D11047 Domagrozumab (USAN/INN)
D11235 Landogrozumab (USAN/INN)
D11242 Trevogrumab (USAN/INN)
D11265 Taldefgrobep alfa (USAN/INN)
|
GDF15 [HSA:9518] [KO:K05504]
|
D11909 Ponsegromab (USAN)
D12852 Rilogrotug (USAN)
D13004 Visugromab (USAN/INN)
|
Growth factors (RTK-binding)
|
PGF [HSA:5228] [KO:K16859]
|
D09574 Aflibercept (USAN/INN) <JP/US>
D10819 Aflibercept beta (genetical recombination) (JAN) <JP>
|
VEGFA [HSA:7422] [KO:K05448]
|
D06409 Bevacizumab (USAN) <JP/US>
D09574 Aflibercept (USAN/INN) <JP/US>
D05386 Pegaptanib sodium (JAN/USAN)
D05697 Ranibizumab (USAN/INN) <JP/US>
D11083 Brolucizumab (USAN/INN) <JP/US>
D11517 Abicipar pegol (USAN/INN)
D11516 Faricimab (USAN/INN) <JP/US>
D08874 Bevasiranib sodium (USAN)
D10819 Aflibercept beta (genetical recombination) (JAN) <JP>
D11126 Navicixizumab (USAN/INN)
D11244 Vanucizumab (USAN/INN)
D11642 Dilpacimab (USAN/INN)
D11890 Emvododstat (USAN)
D12507 Tarcocimab (INN)
D12508 Tarcocimab tedromer (INN)
D12808 Ivonescimab (USAN/INN)
|
VEGFB [HSA:7423] [KO:K16858]
|
D09574 Aflibercept (USAN/INN) <JP/US>
D10819 Aflibercept beta (genetical recombination) (JAN) <JP>
|
IGF1 [HSA:3479] [KO:K05459]
|
D04862 Masoprocol (USAN/INN)
D00967 Toremifene citrate (JAN/USAN) <JP/US>
|
IGF2 [HSA:3481] [KO:K13769]
|
D10352 Dusigitumab (USAN/INN)
|
NGF [HSA:4803] [KO:K02582]
|
D09387 Tanezumab (USAN/INN)
D09907 Fulranumab (USAN/INN)
|
HGF [HSA:3082] [KO:K05460]
|
D09659 Rilotumumab (USAN/INN)
D10123 Ficlatuzumab (USAN)
D12398 Oremepermin alfa (USAN/INN)
|
TGFA [HSA:7039] [KO:K08774]
|
D12343 Fepixnebart (USAN)
|
EREG [HSA:2069] [KO:K09784]
|
D12343 Fepixnebart (USAN)
D13226 Turigrobart (USAN)
|
ANGPT1 [HSA:284] [KO:K05465]
|
D10177 Trebananib (USAN)
|
ANGPT2 [HSA:285] [KO:K05466]
|
D11516 Faricimab (USAN/INN) <JP/US>
D10177 Trebananib (USAN)
D10395 Nesvacumab (USAN/INN)
D11244 Vanucizumab (USAN/INN)
D11904 Zansecimab (USAN)
|
ANGPTL3 [HSA:27329] [KO:K22288]
|
D11753 Evinacumab (USAN/INN) <JP/US>
|
FGF19 [HSA:9965] [KO:K22603]
|
D11734 Aldafermin (USAN/INN)
|
FGF21 [HSA:26291] [KO:K22429]
|
D11512 Pegbelfermin (USAN)
D11868 Efruxifermin (USAN)
D12327 Pegozafermin (USAN)
|
FGF23 [HSA:8074] [KO:K22428]
|
D10913 Burosumab (USAN/INN) <JP/US>
|
Neuropeptides
|
Neuropeptides (GPCR-binding)
|
NPY [HSA:4852] [KO:K05232]
|
D12769 Nisotirostide (USAN)
|
GNRH1 (LHRH) [HSA:2796] [KO:K05252]
|
D03701 Detirelix acetate (USAN)
|
CALCA (CGRP) [HSA:796] [KO:K12332]
|
D10936 Galcanezumab (USAN/INN) <JP/US>
D11055 Fremanezumab (USAN/INN) <JP/US>
D11303 Eptinezumab (USAN) <US>
|
ADCYAP [HSA:116] [KO:K05262]
|
D12459 Vipalanebart (USAN)
|
Other signaling molecules
|
Hepcidin
|
HAMP [HSA:57817] [KO:K23106]
|
D12064 Rusfertide (USAN)
|
Cytokine receptors
|
Interleukin receptors
|
IL2RA (CD25) [HSA:3559] [KO:K05068]
|
D03682 Denileukin diftitox (USAN/INN) <JP/US>
D00748 Aldesleukin (USAN/INN) <US>
D09190 Anti-human thymocyte immunoglobulin, rabbit (JAN) <JP/US>
D03639 Daclizumab (USAN/INN)
D03058 Basiliximab (USAN/INN) <JP/US>
D02743 Celmoleukin (genetical recombination) (JP18)
D02749 Teceleukin (USAN) <JP>
D11324 Camidanlumab (USAN)
D11325 Camidanlumab tesirine (USAN)
D12328 Rezpegaldesleukin (USAN)
D12371 Nemvaleukin alfa (USAN/INN)
D12386 Melredableukin alfa (USAN/INN)
D12928 Vopikitug (USAN/INN)
D13048 Onvapegleukin alfa (USAN/INN)
D13094 Efpixileukin alfa (USAN)
|
IL2RB (CD122) [HSA:3560] [KO:K05069]
|
D00748 Aldesleukin (USAN/INN) <US>
D02743 Celmoleukin (genetical recombination) (JP18)
D02749 Teceleukin (USAN) <JP>
D11669 Bempegaldesleukin (USAN/INN)
D12328 Rezpegaldesleukin (USAN)
|
IL2RG (CD132) [HSA:3561] [KO:K05070]
|
D00748 Aldesleukin (USAN/INN) <US>
D02743 Celmoleukin (genetical recombination) (JP18)
D02749 Teceleukin (USAN) <JP>
D12328 Rezpegaldesleukin (USAN)
|
IL4R (CD124) [HSA:3566] [KO:K05071]
|
D10354 Dupilumab (USAN/INN) <JP/US>
|
IL7R (CD127) [HSA:3575] [KO:K05072]
|
D12479 Lusvertikimab (USAN/INN)
D12739 Bempikibart (USAN/INN)
|
IL15RA (CD215) [HSA:3601] [KO:K05074]
|
D12888 Nogapendekin alfa inbakicept <US>
D11747 Inbakicept (USAN/INN)
D11821 Nogapendekin alfa (USAN/INN)
D12623 Nanrilkefusp alfa (USAN/INN)
|
IL21R (CD360) [HSA:50615] [KO:K05075]
|
D09332 Denenicokin (USAN/INN)
|
CRLF2 (TSLPR) [HSA:64109] [KO:K05078]
|
D12973 Verekitug (USAN/INN)
D13085 Solrikitug (USAN/INN)
|
IL3RA (CD123) [HSA:3563] [KO:K04737]
|
D11358 Tagraxofusp (USAN/INN) <US>
D03645 Daniplestim (USAN/INN)
D04695 Leridistim (USAN/INN)
D05036 Milodistim (USAN/INN)
D05090 Muplestim (USAN/INN)
D11306 Flotetuzumab (USAN/INN)
D11841 Vibecotamab (USAN/INN)
D12307 Pivekimab (USAN)
D12308 Pivekimab sunirine (USAN)
D13057 Bexatamig (USAN/INN)
|
IL5RA (CD125) [HSA:3568] [KO:K05067]
|
D09874 Benralizumab (USAN/INN) <JP/US>
|
IL6R (CD126) [HSA:3570] [KO:K05055]
|
D02596 Tocilizumab (USAN/INN) <JP/US>
D10161 Sarilumab (USAN) <JP/US>
D11079 Satralizumab (USAN/INN) <JP/US>
D12748 Levilimab (INN)
|
IL11RA [HSA:3590] [KO:K05056]
|
D05266 Oprelvekin (USAN/INN)
|
IL12RB [HSA:3594 3595] [KO:K05063 K05064]
|
D13096 Tolododekin alfa (USAN)
|
IL23R [HSA:149233] [KO:K05065]
|
D13093 Icotrokinra hydrochloride (JAN/USAN)
D13108 Icotrokinra (USAN/INN)
|
IL31RA [HSA:133396] [KO:K22630]
|
D11080 Nemolizumab (USAN/INN) <JP/US>
|
OSMR [HSA:9180] [KO:K05057]
|
D11800 Vixarelimab (USAN)
|
IL10R [HSA:3587 3588] [KO:K05134 K05135]
|
D04505 Ilodecakin (USAN/INN)
D11200 Pegilodecakin (USAN/INN)
|
IL22RA1 [HSA:58985] [KO:K05138]
|
D12824 Temtokibart (USAN/INN)
|
IL1R (CD121) [HSA:3554 7850] [KO:K04386 K04387]
|
D02934 Anakinra (USAN/INN) <US>
D11759 Isunakinra (USAN/INN)
|
IL1RL1 [HSA:9173] [KO:K05171]
|
D11796 Melrilimab (USAN)
D11832 Astegolimab (USAN/INN)
|
IL1RL2 (IL-36R) [HSA:8808] [KO:K05172]
|
D12066 Spesolimab (USAN/INN) <JP/US>
D11892 Imsidolimab (USAN)
|
IL17RA (CD217) [HSA:23765] [KO:K05164]
|
D10061 Brodalumab (USAN) <JP/US>
|
Interferon receptors
|
IFNAR1 [HSA:3454] [KO:K05130]
|
D03305 Interferon alfa (NAMALWA) (JP18) <JP>
D03304 Interferon beta (JAN)
D00745 Interferon alfa-2a (USAN/INN)
D02745 Interferon alfa-2b (USAN)
D04552 Interferon alfa-n1 (USAN)
D04554 Interferon beta-1a (USAN) <JP/US>
D00746 Interferon beta-1b (USAN/INN) <JP/US>
D02744 Interferon alfacon-1 (USAN/INN)
D02748 Peginterferon alfa-2b (USAN/INN)
D02747 Peginterferon alfa-2a (USAN/INN) <JP/US>
D08844 Albinterferon alfa-2b (USAN)
D10483 Peginterferon beta-1a (USAN/INN) <US>
D11027 Ropeginterferon alfa-2b (INN) <JP/US>
D11082 Anifrolumab (USAN) <JP/US>
D04553 Interferon alfa-n3 (USAN)
|
IFNAR2 [HSA:3455] [KO:K05131]
|
D03305 Interferon alfa (NAMALWA) (JP18) <JP>
D03304 Interferon beta (JAN)
D00745 Interferon alfa-2a (USAN/INN)
D02745 Interferon alfa-2b (USAN)
D04552 Interferon alfa-n1 (USAN)
D04554 Interferon beta-1a (USAN) <JP/US>
D00746 Interferon beta-1b (USAN/INN) <JP/US>
D02744 Interferon alfacon-1 (USAN/INN)
D02748 Peginterferon alfa-2b (USAN/INN)
D02747 Peginterferon alfa-2a (USAN/INN) <JP/US>
D08844 Albinterferon alfa-2b (USAN)
D10483 Peginterferon beta-1a (USAN/INN) <US>
D11027 Ropeginterferon alfa-2b (INN) <JP/US>
D11082 Anifrolumab (USAN) <JP/US>
D04553 Interferon alfa-n3 (USAN)
|
IFNGR1 (CD119) [HSA:3459] [KO:K05132]
|
D00747 Interferon gamma-1b (USAN/INN) <US>
D03357 Interferon gamma-1a (genetical recombination) (JAN) <JP>
D08805 Interferon gamma-n1 (JAN)
|
IFNGR2 [HSA:3460] [KO:K05133]
|
D00747 Interferon gamma-1b (USAN/INN) <US>
D03357 Interferon gamma-1a (genetical recombination) (JAN) <JP>
D08805 Interferon gamma-n1 (JAN)
|
IFNLR1 [HSA:163702] [KO:K05140]
|
D10078 Peginterferon lambda-1a (USAN)
|
CSF and other factor receptors
|
CSF1R (FMS, CD115) [HSA:1436] [KO:K05090]
|
D08552 Sunitinib (INN)
D06402 Sunitinib malate (JAN/USAN) <JP/US>
D11270 Pexidartinib (USAN/INN)
D11271 Pexidartinib hydrochloride (JAN/USAN) <US>
D11885 Surufatinib (USAN/INN)
D12238 Vimseltinib (USAN/INN)
D13166 Vimseltinib dihydrate <US>
D11952 Axatilimab (USAN/INN) <US>
D02664 Mirimostim (JAN/INN)
D09635 Linifanib (USAN/INN)
D11234 Emactuzumab (USAN/INN)
D11378 Edicotinib (USAN)
D11379 Edicotinib hydrochloride (USAN)
D12545 Tinengotinib (USAN/INN)
D12938 Pimicotinib (USAN/INN)
D12939 Pimicotinib hydrochloride (USAN)
D13058 Migaldendranib (USAN/INN)
|
CSF2RA (GMCSFR, CD116) [HSA:1438] [KO:K05066]
|
D05066 Molgramostim (USAN/INN)
D05803 Sargramostim (USP/INN) <JP/US>
D05712 Regramostim (USAN/INN)
D09930 Mavrilimumab (USAN/INN)
D10015 Litgenprostucel-L (USAN)
|
CSF3R (GCSFR, CD114) [HSA:1441] [KO:K05061]
|
D03235 Filgrastim (USP/INN) <JP/US>
D03247 Lenograstim (USAN/INN) <JP>
D06889 Pegfilgrastim (USAN/INN) <JP/US>
D10242 Lipegfilgrastim (USAN)
D10310 Balugrastim (USAN/INN)
D11026 Pegteograstim (INN)
D11986 Efbemalenograstim alfa (USAN/INN) <US>
D11188 Eflapegrastim (USAN/INN) <US>
D03245 Nartograstim (genetical recombination) (JAN)
D04695 Leridistim (USAN/INN)
D05036 Milodistim (USAN/INN)
D05389 Pegnartograstim (USAN/INN)
D12731 Anumigilimab (USAN/INN)
|
EPOR [HSA:2057] [KO:K05079]
|
D03231 Epoetin alfa (USAN/INN) <JP/US>
D03232 Epoetin beta (USAN/INN) <JP>
D04032 Epoetin delta (USAN)
D10000 Epoetin epsilon (INN)
D10846 Epoetin theta (INN)
D10847 Epoetin zeta (INN)
D03651 Darbepoetin alfa (USAN/INN) <JP/US>
D09998 Epoetin beta pegol (genetical recombination) (JAN) <JP/US>
D09946 Peginesatide (USAN/INN)
D09947 Peginesatide acetate (JAN/USAN)
D13016 Efepoetin alfa (INN)
|
LEPR (CD295) [HSA:3953] [KO:K05062]
|
D05014 Metreleptin (USAN/INN) <JP/US>
|
GHR [HSA:2690] [KO:K05080]
|
D02691 Somatropin (USP/INN) <JP/US>
D05884 Somatrem (USAN)
D03297 Mecasermin (USAN/INN) <JP/US>
D04870 Mecasermin rinfabate (USAN/INN)
D11194 Somapacitan (USAN/INN) <JP/US>
D10990 Somatrogon (USAN/INN) <JP/US>
D11486 Lonapegsomatropin (USAN/INN) <US>
D05394 Pegvisomant (USAN/INN) <JP/US>
D11161 Atesidorsen (USAN/INN)
D11162 Atesidorsen sodium (USAN)
D11193 Somavaratan (USAN/INN)
|
MPL (TPOR, CD110) [HSA:4352] [KO:K05082]
|
D08990 Romiplostim (USAN/INN) <JP/US>
D03978 Eltrombopag olamine (JAN/USAN) <JP/US>
D12815 Eltrombopag choline <US>
D10476 Lusutrombopag (JAN/USAN/INN) <JP/US>
D10306 Avatrombopag (USAN/INN)
D10307 Avatrombopag maleate (JAN/USAN) <JP/US>
D09024 Totrombopag choline (USAN)
|
CNTFR [HSA:1271] [KO:K05059]
|
D03647 Dapiclermin (USAN/INN)
|
Chemokine receptors
|
CCR2 (CD192) [HSA:729230] [KO:K04177]
|
D09878 Cenicriviroc (USAN/INN)
D09879 Cenicriviroc mesylate (USAN)
D10972 Plozalizumab (USAN/INN)
D11997 Ilacirnon (USAN)
D11998 Ilacirnon sodium (USAN)
|
CCR4 (CD194) [HSA:1233] [KO:K04179]
|
D09761 Mogamulizumab (USAN) <JP/US>
D12884 Tivumecirnon (USAN/INN)
D12885 Tivumecirnon besylate (USAN)
|
CCR5 (CD195) [HSA:1234] [KO:K04180]
|
D06670 Maraviroc (JAN/INN) <JP/US>
D03210 Ancriviroc (USAN/INN)
D06297 Vicriviroc maleate (USAN)
D06557 Aplaviroc hydrochloride (USAN)
D09878 Cenicriviroc (USAN/INN)
D09879 Cenicriviroc mesylate (USAN)
D11399 Leronlimab (USAN/INN)
|
CCR8 [HSA:1237] [KO:K04183]
|
D12849 Imzokitug (USAN)
D13088 Tagmokitug (USAN)
D13130 Azirkitug (USAN/INN)
D13224 Lanerkitug (USAN/INN)
|
CCR9 (CD199) [HSA:10803] [KO:K04184]
|
D10378 Vercirnon (USAN/INN)
D10379 Vercirnon sodium (USAN)
|
CXCR1 (IL8RA, CD181) [HSA:3577] [KO:K04175]
|
D08984 Reparixin (USAN/INN)
D10075 Navarixin (USAN)
D12556 Eltrekibart (USAN)
|
CXCR2 (IL8RB, CD182) [HSA:3579] [KO:K05050]
|
D08984 Reparixin (USAN/INN)
D10075 Navarixin (USAN)
D10332 Elubrixin (USAN)
D10387 Danirixin (USAN/INN)
D10420 Elubrixin tosylate (USAN)
|
CXCR4 (CD184) [HSA:7852] [KO:K04189]
|
D08971 Plerixafor (JAN/USAN/INN) <JP/US>
D12281 Motixafortide (USAN/INN)
D12282 Motixafortide acetate (USAN) <US>
D11510 Mavorixafor (USAN) <US>
D12128 Balixafortide (USAN/INN)
|
CXCR7 (ACKR3) [HSA:57007] [KO:K04304]
|
D13139 Canverixin (USAN)
|
CMKLR1 (ChemR23) [HSA:1240] [KO:K04245]
|
D13113 Urcosimod (USAN)
|
Tumor necrosis factor receptors
|
TNFRSF1 (CD120) [HSA:7132 7133] [KO:K03158 K05141]
|
D08562 Tasonermin (INN)
|
TNFRSF4 (CD134, OX40) [HSA:7293] [KO:K05142]
|
D11268 Vonlerolizumab (USAN/INN)
D11301 Tavolimab (USAN/INN)
D12543 Rocatinlimab (USAN/INN)
D13100 Ordastobart (USAN)
|
TNFRSF5 (CD40) [HSA:958] [KO:K03160]
|
D06071 Teneliximab (USAN/INN)
D08896 Dacetuzumab (USAN)
D08942 Lucatumumab (USAN)
D11357 Bleselumab (USAN/INN)
D11491 Selicrelumab (USAN/INN)
D11597 Ravagalimab (USAN/INN)
D11610 Iscalimab (USAN/INN)
D12178 Sotigalimab (USAN)
D13033 Abiprubart (USAN/INN)
|
TNFRSF7 (CD27) [HSA:939] [KO:K05144]
|
D12256 Boserolimab (USAN)
|
TNFRSF8 (CD30) [HSA:943] [KO:K05145]
|
D09587 Brentuximab vedotin (USAN/INN) <JP/US>
D04612 Iratumumab (USAN)
|
TNFRSF9 (CD137) [HSA:3604] [KO:K05146]
|
D09984 Urelumab (USAN/INN)
|
TNFRSF10A (TRAILR1, CD261) [HSA:8797] [KO:K04722]
|
D04858 Mapatumumab (USAN/INN)
|
TNFRSF10B (TRAILR2, CD262) [HSA:8795] [KO:K04722]
|
D06611 Lexatumumab (USAN/INN)
D09329 Conatumumab (USAN/INN)
D09888 Drozitumab (USAN/INN)
D12458 Ozekibart (USAN)
|
TNFRSF12A (TWEAKR, CD266) [HSA:51330] [KO:K05149]
|
D09896 Enavatuzumab (USAN/INN)
|
TNFRSF13B (CD267, TACI) [HSA:23495] [KO:K05150]
|
D12803 Povetacicept (USAN/INN)
|
TNFRSF13C (BAFF-R, CD268) [HSA:115650] [KO:K05151]
|
D12151 Ianalumab (USAN/INN)
|
TNFRSF18 [HSA:8784] [KO:K05154]
|
D12165 Ragifilimab (USAN/INN)
|
NGFR (TNFRSF16, CD271) [HSA:4804] [KO:K02583]
|
D11028 Cenegermin (INN) <US>
|
TNFRSF17 (BCMA, CD269) [HSA:608] [KO:K05153]
|
D11595 Belantamab mafodotin (USAN) <JP>
D12177 Teclistamab (USAN/INN) <JP/US>
D12222 Linvoseltamab (USAN) <US>
D12315 Ciltacabtagene autoleucel (USAN/INN) <US>
D11556 Idecabtagene vicleucel (USAN) <US>
D11594 Belantamab (USAN/INN)
D11992 Pavurutamab (USAN)
D12010 Pacanalotamab (USAN)
D12913 Ingitamig (USAN)
D12990 Etentamig (USAN/INN)
D13214 Cizutamig (USAN/INN)
|
Pattern recognition receptors
|
Toll-like receptors
|
TLR2 (CD282) [HSA:7097] [KO:K10159]
|
D11503 Tomaralimab (USAN)
|
TLR3 (CD283) [HSA:7098] [KO:K05401]
|
D09661 Rintatolimod (USAN/INN)
|
TLR4 (CD284) [HSA:7099] [KO:K10160]
|
D06619 Mifamurtide (USAN)
D04043 Eritoran tetrasodium (USAN)
D09573 Eritoran sodium (JAN)
D11668 Mosedipimod (USAN/INN)
D12624 Paridiprubart (USAN/INN)
|
TLR5 [HSA:7100] [KO:K10168]
|
D10368 Entolimod (USAN/INN)
|
TLR7 [HSA:51284] [KO:K05404]
|
D02500 Imiquimod (JAN/USP/INN) <JP/US>
D01666 Bropirimine (JAN/USAN/INN)
D04619 Isatoribine (USAN)
D04787 Loxoribine (USAN/INN)
D11003 Vesatolimod (USAN/INN)
D12261 Enpatoran (USAN/INN)
D12453 Guretolimod (USAN/INN)
D12521 Ruzotolimod (USAN/INN)
D13051 Resiquimod sulfate (USAN)
|
TLR8 (CD288) [HSA:51311] [KO:K10170]
|
D10716 Motolimod (USAN/INN)
D11871 Selgantolimod (USAN/INN)
D12261 Enpatoran (USAN/INN)
D13051 Resiquimod sulfate (USAN)
|
TLR9 (CD289) [HSA:54106] [KO:K10161]
|
D08841 Agatolimod (USAN)
D08842 Agatolimod sodium (USAN)
D11504 Tilsotolimod (USAN/INN)
D11505 Tilsotolimod sodium (USAN)
D12275 Cobitolimod (USAN/INN)
D12276 Cobitolimod sodium (USAN)
D12855 Nelitolimod (USAN)
D12856 Nelitolimod sodium (USAN)
D12936 Vidutolimod (USAN/INN)
|
C-type lectin receptors
|
CLEC4C (BDCA2, CD303) [HSA:170482] [KO:K06723]
|
D12232 Litifilimab (USAN)
|
KLRC1 (NKG2A) [HSA:3821] [KO:K06541]
|
D12893 Zimistobart
D13238 Monalizumab (USAN/INN)
|
MRC1 (CD206) [HSA:4360] [KO:K06560]
|
D11543 Technetium Tc99m tilmanocept (USAN) <US>
|
NOD-like receptors
|
NOD2 [HSA:64127] [KO:K10165]
|
D06619 Mifamurtide (USAN)
D11385 Inarigivir soproxil (USAN)
|
NLRP3 [HSA:114548] [KO:K12800]
|
D12422 Selnoflast (USAN/INN)
D12423 Selnoflast potassium (USAN)
D12720 Nibrozetone (USAN)
D13195 Usnoflast (USAN/INN)
|
|
Cell surface molecules and ligands
|
Cell adhesion molecules: Ig superfamiy
|
CD2 family
|
CD2 [HSA:914] [KO:K06449]
|
D09190 Anti-human thymocyte immunoglobulin, rabbit (JAN) <JP/US>
D05847 Siplizumab (USAN/INN)
|
CD58 (LFA3) [HSA:965] [KO:K06492]
|
D02800 Alefacept (USAN/INN)
|
SLAMF7 (CD319) [HSA:57823] [KO:K06733]
|
D09337 Elotuzumab (USAN) <JP/US>
|
SIGLEC family
|
CD22 (SIGLEC2) [HSA:933] [KO:K06467]
|
D08933 Inotuzumab ozogamicin (USAN/INN) <JP/US>
D09932 Moxetumomab pasudotox (USAN/INN)
D03066 Bectumomab (USAN/INN)
D04036 Epratuzumab (USAN/INN)
D06348 Yttrium Y 90 epratuzumab (USAN)
D06349 Yttrium Y 90 epratuzumab tetraxetan (USAN)
|
CD33 (SIGLEC3) [HSA:945] [KO:K06473]
|
D03259 Gemtuzumab ozogamicin (USAN) <JP/US>
D11294 Vadastuximab (USAN/INN)
D11295 Vadastuximab talirine (USAN)
D12141 Emerfetamab (USAN)
D12152 Eluvixtamab (USAN)
D12721 Avitotamig (USAN)
|
SIGLEC8 [HSA:27181] [KO:K06748]
|
D11906 Lirentelimab (USAN)
|
MHC
|
MHC1 [HSA:3105 3106 3107 3133 3134 3135] [KO:K06751]
|
D04318 Glatiramer acetate (JAN/USAN) <JP/US>
|
MHC2 [HSA:3108 3109 3111 3112 3113 3115 3117 3118 3119 3122 3123 3125 3126 3127] [KO:K06752]
|
D04318 Glatiramer acetate (JAN/USAN) <JP/US>
|
HLA-DRB [HSA:3123 3125 3126 3127] [KO:K06752]
|
D02967 Apolizumab (USAN/INN)
|
CAMs
|
ICAM1 (CD54) [HSA:3383] [KO:K06490]
|
D02811 Alicaforsen sodium (USAN)
D04000 Enlimomab (USAN/INN)
|
NCAM1 (CD56) [HSA:4684] [KO:K06491]
|
D09927 Lorvotuzumab mertansine (USAN/INN)
|
CEACAM [HSA:1048 1084 1087 1088 1089 4680 634 90273] [KO:K06499]
|
D04524 Indium In 111 altumomab pentetate (USAN)
D06028 Technetium Tc 99m arcitumomab (USP)
D02977 Arcitumomab (USAN/INN)
D06350 Yttrium Y 90 labetuzumab (USAN)
D06351 Yttrium Y 90 labetuzumab tetraxetan (USAN)
D08936 Labetuzumab (INN/USAN)
D10917 Cergutuzumab amunaleukin (USAN/INN)
D11110 Cergutuzumab (USAN)
|
EPCAM (CD326) [HSA:4072] [KO:K06737]
|
D03958 Edrecolomab (USAN/INN)
D09207 Catumaxomab (INN)
D09027 Tucotuzumab celmoleukin (USAN/INN)
|
VCAM1 [HSA:7412] [KO:K06527]
|
D06570 Camobucol (USAN/INN)
D06582 Elsibucol (USAN/INN)
D06648 Succinobucol (USAN)
|
Cell adhesion molecules: other families
|
Integrins
|
ITGA4 (CD49D) [HSA:3676] [KO:K06483]
|
D06886 Natalizumab (USAN/INN) <JP/US>
D06590 Firategrast (USAN)
|
ITGAL (CD11A) [HSA:3683] [KO:K05718]
|
D09190 Anti-human thymocyte immunoglobulin, rabbit (JAN) <JP/US>
D03959 Efalizumab (USAN/INN)
D10374 Lifitegrast (USAN/INN) <US>
D10392 Lifitegrast sodium (USAN)
D08993 Rovelizumab (USAN/INN)
|
ITGAM (CD11B) [HSA:3684] [KO:K06461]
|
D08993 Rovelizumab (USAN/INN)
D11919 Fuzapladib sodium hydrate (JAN)
|
ITGAV (CD51) [HSA:3685] [KO:K06487]
|
D09631 Intetumumab (USAN/INN)
|
ITGB2 (CD18) [HSA:3689] [KO:K06464]
|
D08993 Rovelizumab (USAN/INN)
D11919 Fuzapladib sodium hydrate (JAN)
|
ITGB6 [HSA:3694] [KO:K06589]
|
D12722 Bexotegrast (USAN/INN)
D13006 Sigvotatug (USAN/INN)
D13007 Sigvotatug vedotin (USAN/INN)
|
ITGB7 [HSA:3695] [KO:K06590]
|
D09901 Etrolizumab (USAN/INN)
|
ITGA2B/ITGB3 [HSA:3674 3690] [KO:K06476 K06493]
|
D02778 Abciximab (USAN/INN)
D06888 Eptifibatide (INN) <US>
D08607 Tirofiban (INN)
D01029 Tirofiban hydrochloride (USAN) <US>
D03971 Elarofiban (USAN)
D04659 Lamifiban (USAN/INN)
D04660 Lamifiban hydrochloride (USAN)
D04785 Lotrafiban hydrochloride (USAN)
D05267 Orbofiban acetate (USAN)
D05772 Roxifiban acetate (USAN)
D05834 Sibrafiban (USAN/INN)
D06335 Xemilofiban hydrochloride (USAN)
D06649 Tadocizumab (USAN)
D12051 Zalunfiban (USAN)
D12163 Zalunfiban acetate (USAN)
|
ITGA4/ITGB1 [HSA:3676 3688] [KO:K06483 K05719]
|
D09799 Carotegrast methyl (JAN) <JP>
D10028 Valategrast hydrochloride (USAN)
|
ITGA4/ITGB7 [HSA:3676 3695] [KO:K06483 K06590]
|
D08083 Vedolizumab (USAN) <JP/US>
D09799 Carotegrast methyl (JAN) <JP>
D10028 Valategrast hydrochloride (USAN)
D10540 Abrilumab (USAN/INN)
D13087 Trosunilimab (USAN/INN)
|
ITGA5/ITGB1 [HSA:3678 3688] [KO:K06484 K05719]
|
D06319 Volociximab (USAN)
D12722 Bexotegrast (USAN/INN)
|
ITGAV/ITGB3 [HSA:3685 3690] [KO:K06487 K06493]
|
D09342 Etaracizumab (USAN/INN)
D09929 Maraciclatide (USAN/INN)
|
ITGAV-ITGB3/ITGB5 [HSA:3685 3690 3693] [KO:K06487 K06493 K06588]
|
D03497 Cilengitide (USAN/INN)
D09903 Fluciclatide F 18 (USAN/INN)
|
ITGB2/ITGAL [HSA:3689 3683] [KO:K06464 K05718]
|
D04045 Erlizumab (USAN/INN)
|
Cadherins
|
CDH6 [HSA:1004] [KO:K06798]
|
D13068 Raludotatug (USAN/INN)
D13069 Raludotatug deruxtecan (USAN/INN)
|
Selectins
|
SEL [HSA:6401 6402 6403] [KO:K06494 K06495 K06496]
|
D03114 Bimosiamose disodium (USAN)
|
SELE (CD62E) [HSA:6401] [KO:K06494]
|
D10487 Rivipansel (USAN/INN)
D11310 Uproleselan sodium (USAN)
D11332 Uproleselan (USAN/INN)
|
SELP (CD62P) [HSA:6403] [KO:K06496]
|
D11480 Crizanlizumab (USAN/INN) <US>
D06194 Torapsel (USAN/INN)
D10356 Inclacumab (USAN/INN)
|
Collectins
|
SFTPD [HSA:6441] [KO:K10068]
|
D12333 Zelpultide alfa (USAN/INN)
|
CAM ligands
|
CTGF [HSA:1490] [KO:K06827]
|
D10969 Pamrevlumab (USAN/INN)
|
Other cell surface molecules
|
Immune checkpoints
|
CTLA4 (CD152) [HSA:1493] [KO:K06538]
|
D04603 Ipilimumab (USAN/INN) <JP/US>
D06657 Tremelimumab (USAN/INN) <JP/US>
D11823 Zalifrelimab (USAN/INN)
D12186 Vudalimab (USAN)
D12190 Cadonilimab (USAN/INN)
D12233 Quavonlimab (USAN/INN)
D12317 Bavunalimab (USAN/INN)
D12347 Volrustomig (USAN)
D12448 Botensilimab (USAN/INN)
D13005 Vilastobart (USAN/INN)
D13064 Gotistobart (USAN/INN)
|
PDCD1 (PD1, CD279) [HSA:5133] [KO:K06744]
|
D10316 Nivolumab (USAN/INN) <JP/US>
D10574 Pembrolizumab (USAN) <JP/US>
D13168 Pembrolizumab and berahyaluronidase alfa <US>
D11108 Cemiplimab (USAN) <JP/US>
D11366 Dostarlimab (USAN) <US>
D11487 Tislelizumab (USAN/INN) <JP/US>
D11827 Retifanlimab (USAN) <US>
D12751 Serplulimab (USAN/INN)
D12202 Toripalimab (USAN/INN) <US>
D13234 Camrelizumab (INN)
D12839 Sasanlimab (USAN/INN)
D10390 Pidilizumab (USAN/INN)
D11488 Cetrelimab (USAN/INN)
D11605 Spartalizumab (USAN/INN)
D11643 Budigalimab (USAN/INN)
D11820 Balstilimab (USAN/INN)
D11948 Pacmilimab (USAN/INN)
D12063 Zimberelimab (USAN)
D12119 Sintilimab (USAN/INN)
D12186 Vudalimab (USAN)
D12190 Cadonilimab (USAN/INN)
D12195 Izuralimab (USAN)
D12198 Penpulimab (USAN) <US>
D12223 Rosnilimab (USAN)
D12231 Peresolimab (USAN)
D12332 Zeluvalimab (USAN/INN)
D12347 Volrustomig (USAN)
D12764 Rilvegostomig (USAN/INN)
D12791 Eciskafusp alfa (USAN/INN)
D12808 Ivonescimab (USAN/INN)
D12961 Tobemstomig (USAN/INN)
|
PDL1 (CD274) [HSA:29126] [KO:K06745]
|
D10808 Durvalumab (USAN/INN) <JP/US>
D10817 Avelumab (USAN/INN) <JP/US>
D10773 Atezolizumab (USAN/INN) <JP/US>
D12750 Sugemalimab (INN)
D13233 Envafolimab (INN)
D11532 Lodapolimab (USAN)
D11747 Inbakicept (USAN/INN)
D11893 Bintrafusp alfa (USAN/INN)
D11946 Cosibelimab (USAN/INN) <US>
D12143 Pimivalimab (USAN)
D12344 Socazolimab (USAN)
D12349 Danburstotug (USAN)
D12561 Enristomig (USAN)
|
LAG3 (CD223) [HSA:3902] [KO:K06565]
|
D11350 Relatlimab (USAN)
D12156 Ieramilimab (USAN/INN)
D12317 Bavunalimab (USAN/INN)
D12469 Favezelimab (USAN/INN)
D12480 Tuparstobart (USAN/INN)
D12961 Tobemstomig (USAN/INN)
|
TIGIT [HSA:201633] [KO:K16350]
|
D11482 Tiragolumab (USAN/INN)
D11593 Etigilimab (USAN/INN)
D11795 Vibostolimab (USAN/INN)
D12283 Ociperlimab (USAN/INN)
D12348 Belrestotug (USAN)
D12367 Domvanalimab (USAN/INN)
D12764 Rilvegostomig (USAN/INN)
D13000 Dargistotug (USAN/INN)
|
B7H4 (VTCN1) [HSA:79679] [KO:K06747]
|
D12926 Puxitatug (USAN/INN)
D12927 Puxitatug samrotecan (USAN/INN)
|
CD molecules
|
CD3 [HSA:915 916 917] [KO:K06450 K06451 K06452]
|
D09013 Teplizumab (USAN/INN) <US>
D09207 Catumaxomab (INN)
D09325 Blinatumomab (USAN/INN) <JP/US>
D12296 Tebentafusp (USAN/INN) <US>
D09190 Anti-human thymocyte immunoglobulin, rabbit (JAN) <JP/US>
D05092 Muromonab-CD3 (JAN/USAN/INN)
D06314 Visilizumab (USAN/INN)
D08959 Otelixizumab (USAN)
D11306 Flotetuzumab (USAN/INN)
|
CD3E [HSA:916] [KO:K06451]
|
D12177 Teclistamab (USAN/INN) <JP/US>
D11463 Mosunetuzumab (USAN/INN) <JP/US>
D12368 Epcoritamab (USAN/INN) <JP/US>
D11833 Glofitamab (USAN/INN) <US>
D12180 Talquetamab (USAN/INN) <JP/US>
D12058 Elranatamab (USAN) <JP/US>
D12234 Tarlatamab (USAN) <JP/US>
D11534 Odronextamab (USAN)
D11372 Duvortuxizumab (USAN)
D11489 Cibisatamab (USAN/INN)
D11686 Plamotamab (USAN/INN)
D11841 Vibecotamab (USAN/INN)
D11845 Tidutamab (USAN/INN)
D11984 Cevostamab (USAN/INN)
D11992 Pavurutamab (USAN)
D12007 Ubamatamab (USAN)
D12121 Acapatamab (USAN)
D12236 Runimotamab (USAN/INN)
D12567 Imvotamab (USAN/INN)
D12641 Emirodatamab (USAN/INN)
D12721 Avitotamig (USAN)
D12724 Forimtamig (USAN/INN)
D12990 Etentamig (USAN/INN)
D13159 Pasritamig (USAN/INN)
D13214 Cizutamig (USAN/INN)
|
CD4 [HSA:920] [KO:K06454]
|
D09575 Ibalizumab (USAN/INN) <US>
D12833 Lifileucel (USAN/INN) <US>
D09190 Anti-human thymocyte immunoglobulin, rabbit (JAN) <JP/US>
D03420 Cedelizumab (USAN/INN)
D05610 Priliximab (USAN/INN)
D06356 Zanolimumab (USAN/INN)
|
CD5 [HSA:921] [KO:K06455]
|
D09190 Anti-human thymocyte immunoglobulin, rabbit (JAN) <JP/US>
D06381 Zolimomab aritox (USAN)
|
CD6 (TP120) [HSA:923] [KO:K06456]
|
D12426 Itolizumab (USAN/INN)
|
CD7 [HSA:924] [KO:K06457]
|
D09190 Anti-human thymocyte immunoglobulin, rabbit (JAN) <JP/US>
|
CD8 [HSA:925 926] [KO:K06458 K06459]
|
D10993 Tucidinostat (JAN/USAN/INN) <JP>
D12833 Lifileucel (USAN/INN) <US>
D09190 Anti-human thymocyte immunoglobulin, rabbit (JAN) <JP/US>
|
CD19 [HSA:930] [KO:K06465]
|
D09325 Blinatumomab (USAN/INN) <JP/US>
D11601 Tafasitamab (USAN/INN) <US>
D11338 Loncastuximab tesirine (USAN) <US>
D11144 Axicabtagene ciloleucel (USAN) <US>
D11386 Tisagenlecleucel-T (USAN) <US>
D11880 Brexucabtagene autoleucel (USAN) <US>
D11990 Lisocabtagene maraleucel (USAN/INN) <US>
D13022 Obecabtagene autoleucel (USAN/INN) <US>
D11757 Inebilizumab (USAN/INN) <JP/US>
D11231 Denintuzumab (USAN/INN)
D11232 Denintuzumab mafodotin (USAN/INN)
D11333 Loncastuximab (USAN)
D11372 Duvortuxizumab (USAN)
D11496 Obexelimab (USAN/INN)
|
CD20 [HSA:931] [KO:K06466]
|
D02994 Rituximab (USAN/INN) <JP/US>
D09314 Ofatumumab (USAN/INN) <JP/US>
D09321 Obinutuzumab (USAN/INN) <JP/US>
D11463 Mosunetuzumab (USAN/INN) <JP/US>
D12368 Epcoritamab (USAN/INN) <JP/US>
D11833 Glofitamab (USAN/INN) <US>
D11534 Odronextamab (USAN)
D05218 Ocrelizumab (USAN) <US>
D11243 Ublituximab (USAN/INN) <US>
D12747 Divozilimab (INN)
D08622 Tositumomab 131 iodine
D04489 Ibritumomab tiuxetan (USAN/INN) <US>
D08621 Tositumomab (INN)
D09031 Veltuzumab (USAN)
D10482 Ocaratuzumab (USAN/INN)
D11686 Plamotamab (USAN/INN)
D12567 Imvotamab (USAN/INN)
|
CD23 [HSA:2208] [KO:K06468]
|
D06463 Lumiliximab (USAN/INN)
|
CD28 [HSA:940] [KO:K06470]
|
D11281 Reltecimod (USAN/INN)
D11348 Reltecimod sodium (USAN)
D12300 Acazicolcept (USAN/INN)
D12566 Nezastomig (USAN)
D12709 Marlotamig (USAN)
|
CD34 [HSA:947] [KO:K06474]
|
D12877 Atidarsagene autotemcel (USAN/INN) <US>
D13157 Dorocubicel (USAN/INN)
D11930 Betibeglogene autotemcel (USAN/INN) <US>
D12749 Exagamglogene autotemcel (USAN/INN) <US>
D12765 Lovotibeglogene autotemcel (USAN/INN) <US>
D12592 Omidubicel (USAN) <US>
|
CD37 [HSA:951] [KO:K06475]
|
D12124 Lilotomab (USAN/INN)
D12125 Lutetium (177Lu) lilotomab satetraxetan (USAN/INN)
|
CD47 [HSA:961] [KO:K06266]
|
D11846 Magrolimab (USAN/INN)
D12193 Evorpacept (USAN)
D12385 Lemzoparlimab (USAN/INN)
D13158 Spevatamig (USAN/INN)
D13161 Peluntamig (USAN/INN)
|
CD52 [HSA:1043] [KO:K06488]
|
D02802 Alemtuzumab (USAN/INN) <JP/US>
|
CEACAM5 (CD66e) [HSA:1048] [KO:K06499]
|
D11489 Cibisatamab (USAN/INN)
D12309 Tusamitamab (USAN/INN)
D12310 Tusamitamab ravtansine (USAN/INN)
D13201 Precemtabart (USAN/INN)
D13202 Precemtabart tocentecan (USAN/INN)
|
CD74 [HSA:972] [KO:K06505]
|
D08944 Milatuzumab (USAN)
|
CD79B [HSA:974] [KO:K06507]
|
D10761 Polatuzumab vedotin (USAN) <JP/US>
|
CD80 [HSA:941] [KO:K05412]
|
D03203 Abatacept (USAN/INN) <JP/US>
D03222 Belatacept (USAN/INN) <US>
D04295 Galiximab (USAN/INN)
D12463 Davoceticept (USAN/INN)
|
LILRA4 [HSA:23547] [KO:K06512]
|
D11778 Daxdilimab (USAN)
|
LILRB2 [HSA:10288] [KO:K06512]
|
D12775 Polzastobart (USAN/INN)
|
CD86 [HSA:942] [KO:K05413]
|
D03203 Abatacept (USAN/INN) <JP/US>
D03222 Belatacept (USAN/INN) <US>
|
CD96 [HSA:10225] [KO:K06517]
|
D12914 Nelistotug (USAN/INN)
|
SEMA4 (CD100) [HSA:10507] [KO:K06521]
|
D11469 Pepinemab (USAN)
|
ENG (CD105) [HSA:2022] [KO:K06526]
|
D11260 Carotuximab (USAN/INN)
|
KIR2DL (CD158) [HSA:3802 3803 3804] [KO:K07981]
|
D10444 Lirilumab (USAN/INN)
|
ALCAM (CD166) [HSA:214] [KO:K06547]
|
D11959 Praluzatamab (USAN/INN)
|
SIRPA (CD172A) [HSA:140885] [KO:K06551]
|
D12342 Anzurstobart (USAN)
D12826 Maplirpacept (USAN/INN)
|
CD200 [HSA:4345] [KO:K06556]
|
D09961 Samalizumab (USAN/INN)
|
LY75 (CD205) [HSA:4065] [KO:K06559]
|
D12915 Oberotatug (USAN/INN)
D12916 Oberotatug ravtansine (USAN/INN)
|
MUC1 (CD227) [HSA:4582] [KO:K06568]
|
D06028 Technetium Tc 99m arcitumomab (USP)
D02977 Arcitumomab (USAN/INN)
D09700 Yttrium Y 90 clivatuzumab tetraxetan (USAN)
D09895 Emepepimut-S (USAN)
|
RHD (CD240D) [HSA:6007] [KO:K06579]
|
D09663 Rozrolimupab (USAN)
|
CD244 [HSA:51744] [KO:K06582]
|
D10993 Tucidinostat (JAN/USAN/INN) <JP>
|
BTLA (CD272) [HSA:151888] [KO:K06707]
|
D12546 Venanprubart (USAN)
|
ICOSLG (CD275) [HSA:23308] [KO:K06710]
|
D11907 Rozibafusp alfa (USAN/INN)
|
CD276 [HSA:80381] [KO:K06746]
|
D12753 Ifinatamab deruxtecan (USAN/INN)
D11515 Omburtamab (USAN/INN)
D11752 Enoblituzumab (USAN/INN)
D12154 Mirzotamab (USAN/INN)
D12517 Vobramitamab (USAN/INN)
D12518 Voramitamab duocarmazine (USAN/INN)
D13070 Ifinatamab (USAN/INN)
|
ICOS (CD278) [HSA:29851] [KO:K06713]
|
D11433 Vopratelimab (USAN/INN)
D11996 Feladilimab (USAN/INN)
D12195 Izuralimab (USAN)
D12300 Acazicolcept (USAN/INN)
|
NRP1 (CD304) [HSA:8829] [KO:K06724]
|
D10494 Vesencumab (USAN/INN)
|
KLRK1 (CD314, NKG2D) [HSA:22914] [KO:K06728]
|
D12179 Tesnatilimab (USAN/INN)
D12913 Ingitamig (USAN)
|
NCR1 (CD335) [HSA:9437] [KO:K06741]
|
D13057 Bexatamig (USAN/INN)
|
HAVCR2 (CD366) [HSA:84868] [KO:K20414]
|
D12164 Sabatolimab (USAN/INN)
D11377 Cobolimab (USAN)
D12429 Surzebiclimab (USAN/INN)
D12798 Verzistobart (USAN/INN)
|
Other
|
MUC16 (CA125) [HSA:94025] [KO:K16145]
|
D05269 Oregovomab (USAN/INN)
D11240 Sofituzumab (USAN)
D11241 Sofituzumab vedotin (USAN/INN)
D12007 Ubamatamab (USAN)
|
TACSTD2 (TROP2) [HSA:4070] [KO:K17288]
|
D10985 Sacituzumab govitecan (USAN/INN) <JP/US>
D12359 Datopotamab deruxtecan (USAN/INN) <JP/US>
D12360 Datopotamab (USAN/INN)
|
VSIR (VISTA) [HSA:64115] [KO:K23268]
|
D11474 Onvatilimab (USAN/INN)
D13219 Solnerstotug (USAN/INN)
|
CLDN1 [HSA:9076] [KO:K06087]
|
D12997 Lixudebart (USAN/INN)
|
CLDN18 [HSA:51208] [KO:K06087]
|
D11527 Zolbetuximab (USAN/INN) <JP/US>
D12781 Osemitamab (USAN/INN)
D13158 Spevatamig (USAN/INN)
D13163 Sonesitatug (USAN/INN)
D13164 Sonesitatug vedotin (USAN/INN)
|
PVRL4 (NECTIN4) [HSA:81607] [KO:K06593]
|
D11525 Enfortumab vedotin (USAN) <JP/US>
D11524 Enfortumab (USAN)
|
CD200R [HSA:131450] [KO:K21668]
|
D12603 Ucenprubart (USAN)
|
KLRG1 [HSA:10219] [KO:K10076]
|
D12825 Ulviprubart (USAN/INN)
|
BTN1A1 [HSA:696] [KO:K06712]
|
D13065 Nelmastobart (USAN/INN)
|
|
Transporters
|
ABC transporters
|
ABCB (MDR/TAP) subfamily
|
ABCB1 (CD243) [HSA:5243] [KO:K05658]
|
D03128 Biricodar dicitrate (USAN)
D03968 Elacridar hydrochloride (USAN)
D06008 Tariquidar (USAN/INN)
D06084 Tesmilifene hydrochloride (USAN)
D06277 Valspodar (USAN/INN)
D06387 Zosuquidar trihydrochloride (USAN)
D11782 Encequidar (USAN/INN)
D11783 Encequidar mesylate (USAN)
|
ABCC subfamily
|
ABCC8 (SUR1) [HSA:6833] [KO:K05032]
|
D02427 Glibornuride (USAN/INN)
D02425 Carbutamide (INN)
D00335 Glipizide (USP/INN) <US>
D02430 Gliquidone (INN)
D01599 Gliclazide (JP18/INN) <JP>
D07117 Metahexamide (INN)
D07118 Glisoxepide (INN)
D00593 Glimepiride (JP18/USP/INN) <JP/US>
D00219 Acetohexamide (JP18/USP/INN)
D01799 Glyclopyramide (JAN/INN)
|
ABCC8(SUR1)/KCNJ11(KIR6.2) [HSA:6833 3767] [KO:K05032 K05004]
|
D00336 Glyburide (USP) <JP/US>
D00271 Chlorpropamide (JP18/USP/INN)
D00380 Tolbutamide (JAN/USP/INN)
D06177 Tolbutamide sodium, sterile
D00379 Tolazamide (JAN/USP/INN)
D01356 Glymidine sodium (JAN/USAN/INN)
D00594 Repaglinide (JAN/USP/INN) <JP/US>
D01111 Nateglinide (JP18/USP/INN) <JP/US>
D01854 Mitiglinide calcium hydrate (JP18) <JP>
D01810 Nicorandil (JP18/USAN/INN) <JP>
D00294 Diazoxide (JAN/USP/INN) <JP/US>
D00418 Minoxidil (JAN/USP/INN) <US>
D05482 Pinacidil (USAN)
D02385 Levcromakalim (USAN/INN)
D04739 Linogliride (USAN/INN)
D04740 Linogliride fumarate (USAN)
D05114 Naminidil (USAN/INN)
D12987 Diazoxide choline (USAN) <US>
|
ABCC9(SUR2)/KCNJ11(KIR6.2) [HSA:10060 3767] [KO:K05033 K05004]
|
D01810 Nicorandil (JP18/USAN/INN) <JP>
D05482 Pinacidil (USAN)
D02385 Levcromakalim (USAN/INN)
D05114 Naminidil (USAN/INN)
|
CFTR (ABCC7) [HSA:1080] [KO:K05031]
|
D03605 Crofelemer (USAN) <US>
D09916 Ivacaftor (USAN/INN) <US>
D10134 Lumacaftor (USAN/INN)
D11041 Tezacaftor (USAN/INN)
D11402 Olacaftor (USAN/INN)
D11423 Deutivacaftor (USAN/INN)
D11507 Elexacaftor (USAN)
D11535 Bamocaftor (USAN)
D11536 Bamocaftor potassium (USAN)
D11682 Nesolicaftor (USAN)
D11683 Posenacaftor (USAN)
D11724 Galicaftor (USAN/INN)
D12140 Navocaftor (USAN/INN)
D12454 Icenticaftor (USAN/INN)
D12718 Vanzacaftor (USAN/INN)
D12719 Vanzacaftor calcium (USAN)
|
CFTR* [HSA_VAR:1080v1] [HSA:1080] [KO:K05031]
|
D10685 Lumacaftor and ivacaftor <US>
D11042 Tezacaftor and ivacaftor <US>
D11700 Elexacaftor, ivacaftor and tezacaftor <US>
D13024 Vanzacaftor, tezacaftor and deutivacaftor <US>
|
ABCD (ALD) subfamily
|
ABCD1 (ALDP) [HSA:215] [KO:K05675]
|
D12150 Elivaldogene autotemcel (USAN/INN) <US>
|
Solute carrier family
|
SLC5
|
SLC5A1 (SGLT1) [HSA:6523] [KO:K14158]
|
D10669 Sotagliflozin (USAN/INN) <US>
|
SLC5A2 (SGLT2) [HSA:6524] [KO:K14382]
|
D08897 Dapagliflozin (JAN/USAN/INN) <JP>
D09763 Dapagliflozin propanediol (USAN) <JP/US>
D09592 Canagliflozin (USAN/INN) <JP/US>
D10459 Empagliflozin (JAN/USAN/INN) <JP/US>
D10313 Ertugliflozin (USAN/INN)
D11043 Ertugliflozin pidolate <US>
D10196 Ipragliflozin (INN)
D10200 Ipragliflozin L-proline (JAN) <JP>
D10669 Sotagliflozin (USAN/INN) <US>
D10195 Luseogliflozin hydrate (JAN) <JP>
D10865 Bexagliflozin (USAN) <US>
D13015 Enavogliflozin (INN)
D06641 Sergliflozin etabonate (USAN)
D09978 Tofogliflozin (USAN) <JP>
D10055 Remogliflozin etabonate (USAN/INN)
|
SLC6
|
SLC6A1 (GAT1) [HSA:6529] [KO:K05034]
|
D00332 Gabapentin (JAN/USP/INN) <JP/US>
D09539 Gabapentin enacarbil (JAN/USAN/INN) <JP/US>
D08588 Tiagabine (INN)
D02097 Tiagabine hydrochloride (USP) <US>
|
SLC6A2 (NAT1) [HSA:6530] [KO:K05035]
|
D05458 Phentermine (USAN/INN)
D05459 Phentermine hydrochloride (USP) <US>
D07444 Amfepramone (INN)
D03801 Diethylpropion hydrochloride (USP) <US>
D00367 Mazindol (JAN/USP/INN) <JP>
D08513 Sibutramine (INN)
D02571 Sibutramine hydrochloride (USP)
D01304 Amezinium metilsulfate (JAN) <JP>
D08030 Guanethidine (INN)
D02237 Guanethidine sulfate (USAN)
D04382 Guanethidine monosulfate (USP)
D07875 Doxepin (INN)
D00814 Doxepin hydrochloride (USP) <US>
D00110 Cocaine (USP)
D02182 Cocaine hydrochloride (JP18/USP) <US>
D06007 Tapentadol (USAN/INN)
D10199 Tapentadol hydrochloride (JAN) <US>
D07791 Desipramine (INN)
D00812 Desipramine hydrochloride (JAN/USP) <US>
D08070 Imipramine (INN)
D00815 Imipramine hydrochloride (JP18/USP) <JP/US>
D08071 Imipramine pamoate (USP) <US>
D07727 Clomipramine (INN)
D00811 Clomipramine hydrochloride (JP18/USP) <JP/US>
D00394 Trimipramine (USAN/INN)
D02408 Trimipramine maleate (JAN/USP) <JP/US>
D08140 Lofepramine (INN)
D01285 Lofepramine hydrochloride (JAN/USAN)
D07448 Amitriptyline (INN)
D00809 Amitriptyline hydrochloride (JP18/USP) <JP/US>
D08288 Nortriptyline (INN)
D00816 Nortriptyline hydrochloride (JP18/USP/INN) <JP/US>
D08447 Protriptyline (INN)
D00484 Protriptyline hydrochloride (USP) <US>
D07872 Dosulepin (INN)
D01546 Dothiepin hydrochloride (USAN) <JP>
D00228 Amoxapine (JP18/USP/INN) <JP/US>
D02566 Maprotiline (USAN)
D00818 Maprotiline hydrochloride (JP18/USP) <JP>
D05200 Nomifensine maleate (USAN)
D08673 Viloxazine (INN)
D02572 Viloxazine hydrochloride (USAN) <US>
D07591 Bupropion (INN)
D00817 Bupropion hydrochloride (JAN/USP) <US>
D07938 Bupropion hydrobromide (USAN) <US>
D08670 Venlafaxine (INN)
D00821 Venlafaxine hydrochloride (JAN/USP) <JP/US>
D12403 Venlafaxine besylate monohydrate <US>
D08222 Milnacipran (INN)
D01107 Milnacipran hydrochloride (JAN/USAN) <JP/US>
D08472 Reboxetine (INN)
D02573 Reboxetine mesylate (USAN)
D07880 Duloxetine (INN)
D01179 Duloxetine hydrochloride (JAN/USP) <JP/US>
D07793 Desvenlafaxine (INN) <US>
D02570 Desvenlafaxine succinate (USAN) <US>
D11619 Desvenlafaxine succinate anhydrous
D10072 Levomilnacipran (USAN/INN)
D10133 Levomilnacipran hydrochloride (USAN) <US>
D07445 Amfetamine (INN) <US>
D02074 Amphetamine sulfate (USP) <US>
D11622 Amphetamine aspartate monohydrate
D03740 Dextroamphetamine (USAN) <US>
D02078 Dextroamphetamine sulfate (USP) <US>
D08187 Metamfetamine (INN)
D02242 Methamphetamine hydrochloride (JP18/USP) <JP/US>
D04999 Methylphenidate (USAN/INN) <US>
D01296 Methylphenidate hydrochloride (JAN/USP) <JP/US>
D07473 Atomoxetine (USP/INN)
D02574 Atomoxetine hydrochloride (JAN/USP) <JP/US>
D07806 Dexmethylphenidate (INN)
D03721 Dexmethylphenidate hydrochloride (USAN) <US>
D08130 Lisdexamfetamine (INN)
D04747 Lisdexamfetamine dimesylate (USAN) <JP/US>
D11315 Solriamfetol (USAN)
D11328 Solriamfetol hydrochloride (USAN) <US>
D02080 Phendimetrazine tartrate (USP) <US>
D02170 Indeloxazine hydrochloride (JAN/USAN)
D02704 Tampramine fumarate (USAN)
D03491 Cidoxepin hydrochloride (USAN)
D04473 Hydroxyamphetamine hydrobromide (USP)
D04781 Lortalamine (USAN/INN)
D05119 Napamezole hydrochloride (USAN)
D05120 Napitane mesylate (USAN)
D05173 Nisoxetine (USAN/INN)
D05284 Oxaprotiline hydrochloride (USAN)
D05454 Phenmetrazine hydrochloride (USP)
D05663 Pyrovalerone hydrochloride (USAN)
D05692 Radafaxine hydrochloride (USAN)
D05997 Talopram hydrochloride (USAN)
D06004 Tandamine hydrochloride (USAN)
D07334 Imipraminoxide (INN)
D07449 Amitriptylinoxide (INN)
D07514 Benzfetamine (INN)
D07515 Benzfetamine hydrochloride <US>
D08072 Imipraminoxide hydrochloride
D08077 Indeloxazine (INN)
D08347 Phendimetrazine (INN)
D08348 Phendimetrazine hydrochloride
D09340 Esreboxetine (USAN/INN)
D09341 Esreboxetine succinate (USAN)
D09890 Edivoxetine (USAN/INN)
D09891 Edivoxetine hydrochloride (USAN)
D10088 Amitifadine (USAN)
D10089 Amitifadine hydrochloride (USAN)
D10443 Liafensine (USAN/INN)
D10697 Centanafadine (USAN/INN)
D10698 Centanafadine hydrochloride (USAN)
D10700 Dasotraline (USAN/INN)
D10870 Dasotraline hydrochloride (USAN)
D11172 Midomafetamine (USAN/INN)
D11623 Dextroamphetamine saccharate
D11688 Ampreloxetine (USAN/INN)
D11689 Ampreloxetine hydrochloride (USAN)
D11940 Toludesvenlafaxine (USAN/INN)
D11941 Toludesvenlafaxine hydrochloride (USAN)
D12715 Tenamfetamine (INN)
D12937 Midomafetamine hydrochloride (USAN)
|
SLC6A3 (DAT1) [HSA:6531] [KO:K05036]
|
D05458 Phentermine (USAN/INN)
D05459 Phentermine hydrochloride (USP) <US>
D07444 Amfepramone (INN)
D03801 Diethylpropion hydrochloride (USP) <US>
D00367 Mazindol (JAN/USP/INN) <JP>
D08513 Sibutramine (INN)
D02571 Sibutramine hydrochloride (USP)
D00110 Cocaine (USP)
D02182 Cocaine hydrochloride (JP18/USP) <US>
D07591 Bupropion (INN)
D00817 Bupropion hydrochloride (JAN/USP) <US>
D07938 Bupropion hydrobromide (USAN) <US>
D07445 Amfetamine (INN) <US>
D02074 Amphetamine sulfate (USP) <US>
D11622 Amphetamine aspartate monohydrate
D03740 Dextroamphetamine (USAN) <US>
D02078 Dextroamphetamine sulfate (USP) <US>
D08187 Metamfetamine (INN)
D02242 Methamphetamine hydrochloride (JP18/USP) <JP/US>
D04999 Methylphenidate (USAN/INN) <US>
D01296 Methylphenidate hydrochloride (JAN/USP) <JP/US>
D07806 Dexmethylphenidate (INN)
D03721 Dexmethylphenidate hydrochloride (USAN) <US>
D08130 Lisdexamfetamine (INN)
D04747 Lisdexamfetamine dimesylate (USAN) <JP/US>
D03215 Armodafinil (USAN/INN) <US>
D11315 Solriamfetol (USAN)
D11328 Solriamfetol hydrochloride (USAN) <US>
D10014 Ioflupane I 123 (USAN) <JP/US>
D02897 Amfonelic acid (USAN)
D03153 Brasofensine maleate (USAN)
D05119 Napamezole hydrochloride (USAN)
D05454 Phenmetrazine hydrochloride (USP)
D05663 Pyrovalerone hydrochloride (USAN)
D05692 Radafaxine hydrochloride (USAN)
D07514 Benzfetamine (INN)
D07515 Benzfetamine hydrochloride <US>
D10088 Amitifadine (USAN)
D10089 Amitifadine hydrochloride (USAN)
D10697 Centanafadine (USAN/INN)
D10698 Centanafadine hydrochloride (USAN)
D10700 Dasotraline (USAN/INN)
D10870 Dasotraline hydrochloride (USAN)
D11172 Midomafetamine (USAN/INN)
D11623 Dextroamphetamine saccharate
D12715 Tenamfetamine (INN)
D12716 Mesocarb (INN)
D12937 Midomafetamine hydrochloride (USAN)
|
SLC6A4 (HTT) [HSA:6532] [KO:K05037]
|
D05458 Phentermine (USAN/INN)
D05459 Phentermine hydrochloride (USP) <US>
D07945 Fenfluramine (INN)
D04148 Fenfluramine hydrochloride (JAN/USAN) <JP/US>
D07805 Dexfenfluramine (INN)
D03713 Dexfenfluramine hydrochloride (USAN)
D00367 Mazindol (JAN/USP/INN) <JP>
D08513 Sibutramine (INN)
D02571 Sibutramine hydrochloride (USP)
D07875 Doxepin (INN)
D00814 Doxepin hydrochloride (USP) <US>
D03649 Dapoxetine hydrochloride (USAN)
D00110 Cocaine (USP)
D02182 Cocaine hydrochloride (JP18/USP) <US>
D07791 Desipramine (INN)
D00812 Desipramine hydrochloride (JAN/USP) <US>
D08070 Imipramine (INN)
D00815 Imipramine hydrochloride (JP18/USP) <JP/US>
D08071 Imipramine pamoate (USP) <US>
D07727 Clomipramine (INN)
D00811 Clomipramine hydrochloride (JP18/USP) <JP/US>
D00394 Trimipramine (USAN/INN)
D02408 Trimipramine maleate (JAN/USP) <JP/US>
D08140 Lofepramine (INN)
D01285 Lofepramine hydrochloride (JAN/USAN)
D07448 Amitriptyline (INN)
D00809 Amitriptyline hydrochloride (JP18/USP) <JP/US>
D08288 Nortriptyline (INN)
D00816 Nortriptyline hydrochloride (JP18/USP/INN) <JP/US>
D08447 Protriptyline (INN)
D00484 Protriptyline hydrochloride (USP) <US>
D07872 Dosulepin (INN)
D01546 Dothiepin hydrochloride (USAN) <JP>
D00228 Amoxapine (JP18/USP/INN) <JP/US>
D00326 Fluoxetine (USAN/INN)
D00823 Fluoxetine hydrochloride (JAN/USP) <US>
D07704 Citalopram (USP/INN)
D00822 Citalopram hydrobromide (USP) <US>
D07705 Citalopram hydrochloride
D02362 Paroxetine (USP/INN)
D02260 Paroxetine hydrochloride hemihydrate (USP) <JP/US>
D05374 Paroxetine hydrochloride (USP) <US>
D05375 Paroxetine mesylate (USAN) <US>
D02360 Sertraline (INN)
D00825 Sertraline hydrochloride (JAN/USP) <JP/US>
D02787 Alaproclate (USAN/INN)
D07984 Fluvoxamine (INN)
D00824 Fluvoxamine maleate (JP18/USP) <JP/US>
D07913 Escitalopram (INN)
D02567 Escitalopram oxalate (JAN/USP) <JP/US>
D08626 Trazodone (INN)
D00820 Trazodone hydrochloride (JAN/USP) <JP/US>
D08670 Venlafaxine (INN)
D00821 Venlafaxine hydrochloride (JAN/USP) <JP/US>
D12403 Venlafaxine besylate monohydrate <US>
D08222 Milnacipran (INN)
D01107 Milnacipran hydrochloride (JAN/USAN) <JP/US>
D07880 Duloxetine (INN)
D01179 Duloxetine hydrochloride (JAN/USP) <JP/US>
D07793 Desvenlafaxine (INN) <US>
D02570 Desvenlafaxine succinate (USAN) <US>
D11619 Desvenlafaxine succinate anhydrous
D09698 Vilazodone (USAN/INN)
D09699 Vilazodone hydrochloride (USAN) <US>
D10184 Vortioxetine (USAN)
D10185 Vortioxetine hydrobromide (JAN/USAN) <JP/US>
D12544 Vortioxetine hemihydrobromide (USAN)
D10072 Levomilnacipran (USAN/INN)
D10133 Levomilnacipran hydrochloride (USAN) <US>
D08187 Metamfetamine (INN)
D02242 Methamphetamine hydrochloride (JP18/USP) <JP/US>
D07806 Dexmethylphenidate (INN)
D03721 Dexmethylphenidate hydrochloride (USAN) <US>
D02170 Indeloxazine hydrochloride (JAN/USAN)
D03491 Cidoxepin hydrochloride (USAN)
D04788 Lubazodone hydrochloride (USAN)
D05491 Pirandamine hydrochloride (USAN)
D07334 Imipraminoxide (INN)
D07449 Amitriptylinoxide (INN)
D08072 Imipraminoxide hydrochloride
D08077 Indeloxazine (INN)
D10088 Amitifadine (USAN)
D10089 Amitifadine hydrochloride (USAN)
D10443 Liafensine (USAN/INN)
D10697 Centanafadine (USAN/INN)
D10698 Centanafadine hydrochloride (USAN)
D11172 Midomafetamine (USAN/INN)
D11688 Ampreloxetine (USAN/INN)
D11689 Ampreloxetine hydrochloride (USAN)
D11940 Toludesvenlafaxine (USAN/INN)
D11941 Toludesvenlafaxine hydrochloride (USAN)
D12715 Tenamfetamine (INN)
D12937 Midomafetamine hydrochloride (USAN)
|
SLC6A8 [HSA:6535] [KO:K05041]
|
D12779 Ompenaclid (USAN/INN)
D12780 Ompenaclid succinate (USAN)
|
SLC6A9 (GLYT1) [HSA:6536] [KO:K05038]
|
D10186 Bitopertin (JAN/USAN/INN)
D12527 Iclepertin (JAN/USAN/INN)
|
SLC6A19 [HSA:340024] [KO:K05334]
|
D13149 Repinatrabit (USAN/INN)
|
SLC7
|
SLC7A5 (LAT1) [HSA:8140] [KO:K13780]
|
D12443 Nanvuranlat hydrochloride hydrate (JAN)
|
SLC9
|
SLC9A1 (NHE1) [HSA:6548] [KO:K05742]
|
D03406 Cariporide mesylate (USAN)
D09036 Zoniporide mesylate (INN/USAN)
|
SLC9A3 (NHE3) [HSA:6550] [KO:K12040]
|
D11652 Tenapanor (USAN/INN)
D11653 Tenapanor hydrochloride (JAN/USAN) <JP/US>
|
SLC10
|
SLC10A [HSA:6554 6555 8273 347051 201780 345274 84068] [KO:K14341 K14342 K14343 K14344 K14346 K14347]
|
D10951 Maralixibat (USAN)
|
SLC10A2 (ASBT, IBAT) [HSA:6555] [KO:K14342]
|
D10952 Maralixibat chloride (JAN/USAN/INN) <JP/US>
D11716 Odevixibat (USAN)
D13092 Odevixibat hydrate (JAN) <JP/US>
D11539 Linerixibat (JAN/USAN)
D10796 Elobixibat (USAN/INN)
D10795 Elobixibat hydrate (JAN) <JP>
|
SLC12
|
SLC12A1 (NKCC2) [HSA:6557] [KO:K14425]
|
D00654 Hydroflumethiazide (JAN/USP/INN)
D00658 Trichlormethiazide (JP18/USP/INN) <JP>
D00656 Methyclothiazide (JAN/USP/INN)
D00461 Quinethazone (JAN/INN)
D00272 Chlorthalidone (USP) <US>
D00331 Furosemide (JP18/USP/INN) <JP/US>
D07999 Sodium furosemide
D08001 Furosemide diolamine
D00247 Bumetanide (JP18/USP/INN) <US>
D01634 Piretanide (JAN/USAN/INN)
D00382 Torsemide (USP) <JP/US>
D08619 Torasemide sodium
D00313 Ethacrynic acid (USP) <US>
D04079 Ethacrynate sodium (USP) <US>
D02386 Ticrynafen (USAN)
D05093 Muzolimine (USAN/INN)
D04111 Etozolin (USAN/INN)
D01323 Azosemide (JP18/USAN/INN) <JP>
D02453 Flumethiazide (INN)
D09772 Alilusem potassium (JAN)
|
SLC12A2 (NKCC1) [HSA:6558] [KO:K10951]
|
D00331 Furosemide (JP18/USP/INN) <JP/US>
D07999 Sodium furosemide
D08001 Furosemide diolamine
D00247 Bumetanide (JP18/USP/INN) <US>
D01634 Piretanide (JAN/USAN/INN)
D00382 Torsemide (USP) <JP/US>
D08619 Torasemide sodium
D00313 Ethacrynic acid (USP) <US>
D04079 Ethacrynate sodium (USP) <US>
D02386 Ticrynafen (USAN)
D05093 Muzolimine (USAN/INN)
D04111 Etozolin (USAN/INN)
D01323 Azosemide (JP18/USAN/INN) <JP>
D09772 Alilusem potassium (JAN)
|
SLC12A3 (TSC) [HSA:6559] [KO:K14426]
|
D00650 Bendroflumethiazide (JAN/USP/INN)
D00654 Hydroflumethiazide (JAN/USP/INN)
D00340 Hydrochlorothiazide (JP18/USP/INN) <JP/US>
D00519 Chlorothiazide (JAN/USP/INN) <US>
D03471 Chlorothiazide sodium (USP) <US>
D00657 Polythiazide (JAN/USAN/INN)
D00658 Trichlormethiazide (JP18/USP/INN) <JP>
D00656 Methyclothiazide (JAN/USP/INN)
D00461 Quinethazone (JAN/INN)
D00272 Chlorthalidone (USP) <US>
D01877 Mefruside (JP18/USAN/INN) <JP>
D00431 Metolazone (JAN/USP/INN) <US>
D01605 Meticrane (JP18/INN)
D00345 Indapamide (JP18/USP) <JP/US>
D06401 Indapamide hydrate
D00651 Benzthiazide (JAN/INN)
D01241 Penflutizide (JAN/INN)
D01246 Benzylhydrochlorothiazide (JAN)
D01895 Tripamide (JAN/USAN/INN)
D02453 Flumethiazide (INN)
|
SLC12A4 [HSA:6560] [KO:K14427]
|
D00247 Bumetanide (JP18/USP/INN) <US>
|
SLC18
|
SLC18A1 (VMAT1) [HSA:6570] [KO:K08155]
|
D00197 Reserpine (JP18/USP/INN)
D08187 Metamfetamine (INN)
D02242 Methamphetamine hydrochloride (JP18/USP) <JP/US>
D10170 Tedatioxetine (USAN)
D10171 Tedatioxetine hydrobromide (USAN)
|
SLC18A2 (VMAT2) [HSA:6571] [KO:K08155]
|
D07097 Isometheptene mucate (USP)
D00197 Reserpine (JP18/USP/INN)
D07445 Amfetamine (INN) <US>
D02074 Amphetamine sulfate (USP) <US>
D11622 Amphetamine aspartate monohydrate
D03740 Dextroamphetamine (USAN) <US>
D02078 Dextroamphetamine sulfate (USP) <US>
D08187 Metamfetamine (INN)
D02242 Methamphetamine hydrochloride (JP18/USP) <JP/US>
D08575 Tetrabenazine (JAN/INN) <JP/US>
D10675 Valbenazine (USAN/INN)
D10999 Valbenazine tosylate (USAN) <JP/US>
D10701 Deutetrabenazine (USAN/INN) <US>
D07514 Benzfetamine (INN)
D07515 Benzfetamine hydrochloride <US>
D10170 Tedatioxetine (USAN)
D10171 Tedatioxetine hydrobromide (USAN)
D11172 Midomafetamine (USAN/INN)
D11623 Dextroamphetamine saccharate
D12937 Midomafetamine hydrochloride (USAN)
|
SLC22
|
SLC22A11 (OAT4) [HSA:55867] [KO:K08207]
|
D09921 Lesinurad (USAN/INN)
D09922 Lesinurad sodium (USAN)
|
SLC22A12 (URAT1) [HSA:116085] [KO:K08208]
|
D01056 Benzbromarone (JP18/USAN/INN) <JP>
D09921 Lesinurad (USAN/INN)
D09922 Lesinurad sodium (USAN)
D11071 Dotinurad (JAN/INN) <JP>
D11129 Verinurad (USAN/INN)
D13063 Pozdeutinurad (USAN/INN)
|
SLC29
|
SLC29A1 (ENT1) [HSA:2030] [KO:K15014]
|
D07843 Dilazep (INN)
D02631 Dilazep dihydrochloride hydrate (JP18) <JP>
D03906 Draflazine (USAN/INN)
|
SLC29A2 (ENT2) [HSA:3177] [KO:K15014]
|
D11828 Clervonafusp alfa (USAN/INN)
|
SLC34
|
SLC34A2 [HSA:10568] [KO:K14683]
|
D11237 Lifastuzumab (USAN)
D11238 Lifastuzumab vedotin (USAN/INN)
|
SLC40
|
SLC40A1 (FPN1, IREG1) [HSA:30061] [KO:K14685]
|
D12289 Vamifeport (USAN/INN)
D12290 Vamifeport trihydrochloride (USAN)
|
Major facilitator superfamily
|
VNT family
|
SV2 [HSA:9900 9899 22987] [KO:K06258]
|
D11842 Padsevonil (JAN/USAN)
|
SV2A [HSA:9900] [KO:K06258]
|
D00709 Levetiracetam (JAN/USP/INN) <JP/US>
D08879 Brivaracetam (JAN/USAN/INN) <JP/US>
D01914 Piracetam (JAN/USAN/INN) <JP>
D05817 Seletracetam (USAN/INN)
D13077 Plosaracetam (USAN/INN)
|
Other transporters
|
Channels and pores (TC:1)
|
CETP [HSA:1071] [KO:K16835]
|
D05255 Omega-3-acid ethyl esters (USP) <JP/US>
D06195 Torcetrapib (USAN/INN)
D08855 Anacetrapib (JAN/USAN)
D09708 Dalcetrapib (USAN/INN)
D10121 Evacetrapib (USAN)
D12900 Obicetrapib (USAN/INN)
D12901 Obicetrapib calcium (USAN)
|
XPO1 [HSA:7514] [KO:K14290]
|
D11222 Selinexor (USAN/INN) <US>
D11223 Verdinexor (USAN/INN)
D11499 Eltanexor (USAN/INN)
|
Auxiliary transport proteins (TC:8.A)
|
SIGMAR1 [HSA:10280] [KO:K20719]
|
D07945 Fenfluramine (INN)
D04148 Fenfluramine hydrochloride (JAN/USAN) <JP/US>
D07316 Captodiame (BAN)
D08297 Opipramol (INN)
D01477 Opipramol hydrochloride (JAN/USAN)
D11383 Blarcamesine (USAN/INN)
D11549 Blarcamesine hydrochloride (USAN)
D03742 Dextromethorphan (USP)
D00848 Dextromethorphan hydrobromide (USP) <JP>
D03744 Dextromethorphan polistirex (USAN)
D02684 Rimcazole hydrochloride (USAN)
D02688 Tiospirone hydrochloride (USAN)
D04502 Igmesine hydrochloride (USAN)
|
KLB [HSA:152831] [KO:K22404]
|
D12490 Fazpilodemab (USAN/INN)
|
Others
|
TTR [HSA:7276] [KO:K20731]
|
D11972 Acoramidis (USAN)
D11973 Acoramidis hydrochloride (JAN/USAN) <JP/US>
D09673 Tafamidis (JAN/USAN/INN) <JP>
D09674 Tafamidis meglumine (JAN/USAN) <JP/US>
D11116 Patisiran (USAN/INN)
D10794 Patisiran sodium (JAN) <JP/US>
D10940 Inotersen (USAN/INN)
D10941 Inotersen sodium (USAN) <US>
D11917 Vutrisiran (USAN/INN)
D11916 Vutrisiran sodium (JAN) <JP/US>
D12754 Eplontersen sodium (JAN/USAN) <US>
D13140 Coramitug (USAN/INN)
|
FOLR [HSA:2348 2350 2352] [KO:K13649]
|
D10434 Vintafolide (USAN/INN)
D12249 Pafolacianine (USAN/INN)
D12250 Pafolacianine sodium (USAN) <US>
|
FOLR1 [HSA:2348] [KO:K13649]
|
D10954 Mirvetuximab soravtansine (USAN/INN) <US>
D09343 Farletuzumab (USAN)
D10953 Mirvetuximab (USAN/INN)
D12183 Farletuzumab ecteribulin (USAN)
D12880 Pasifolate exatecan (USAN)
D13208 Torvutatug (USAN/INN)
|
NPC1L1 [HSA:29881] [KO:K14461]
|
D01966 Ezetimibe (JAN/USP/INN) <JP/US>
|
|
Enzymes
|
Oxidoreductases (EC1)
|
Dehydrogenases [EC:1.1.1.-]
|
ADH [HSA:124 125 126] [KO:K13951]
|
D00707 Fomepizole (JAN/USAN/INN) <JP/US>
|
AKR1B1 [HSA:231] [KO:K00011]
|
D02323 Tolrestat (USAN/INN)
D12384 Govorestat (USAN/INN)
D01688 Epalrestat (JP18/INN) <JP>
D01715 Risarestat (INN)
D01842 Fidarestat (JAN/INN)
D02328 Zopolrestat (USAN/INN)
D02835 Alrestatin sodium (USAN)
D03803 Lidorestat (USAN)
D03805 Minalrestat (USAN/INN)
D03806 Ponalrestat (USAN/INN)
D03807 Zenarestat (USAN/INN)
D05893 Sorbinil (USAN/INN)
D06403 Ranirestat (JAN/INN)
D12390 Caficrestat (USAN/INN)
|
LDHA [HSA:3939] [KO:K00016]
|
D12723 Nedosiran sodium (USAN) <US>
|
HMGCR [HSA:3156] [KO:K00021]
|
D00434 Simvastatin (JP18/USP/INN) <JP/US>
D00359 Lovastatin (USP/INN) <US>
D08410 Pravastatin (INN)
D00893 Pravastatin sodium (JP18/USP) <JP/US>
D07983 Fluvastatin (INN)
D00892 Fluvastatin sodium (JAN/USP) <JP/US>
D07474 Atorvastatin (INN)
D00887 Atorvastatin calcium anhydorous
D02258 Atorvastatin calcium (USP) <JP/US>
D11095 Atorvastatin calcium propylene glycol solvate <US>
D07661 Cerivastatin (INN)
D00889 Cerivastatin sodium (JAN/USAN)
D08492 Rosuvastatin (INN)
D01915 Rosuvastatin calcium (JP18/USP) <JP/US>
D01862 Pitavastatin calcium (JAN) <US>
D10568 Pitavastatin calcium hydrate (JP18) <JP/US>
D11092 Pitavastatin magnesium <US>
D03601 Crilvastatin (USAN/INN)
D03643 Dalvastatin (USAN/INN)
D03816 Tenivastatin calcium (USAN)
|
IDH [HSA:3417 3418] [KO:K00031]
|
D11834 Vorasidenib (USAN/INN)
D11835 Vorasidenib citrate (USAN) <JP/US>
|
IDH1 [HSA:3417] [KO:K00031]
|
D12708 Crelosidenib (USAN)
D12717 Crelosidenib gentisate (USAN)
|
IDH1* [HSA_VAR:3417v1] [HSA:3417] [KO:K00031]
|
D11090 Ivosidenib (JAN/USAN/INN) <JP/US>
D12483 Olutasidenib (USAN/INN) <US>
|
IDH2 [HSA:3418] [KO:K00031]
|
D10901 Enasidenib (USAN/INN)
|
IDH2* [HSA_VAR:3418v1] [HSA:3418] [KO:K00031]
|
D11044 Enasidenib mesylate (USAN) <US>
|
HSD3B [HSA:3283 3284] [KO:K00070]
|
D01180 Trilostane (JAN/USAN) <JP>
D04035 Epostane (USAN/INN)
|
HSD11B1 [HSA:3290] [KO:K15680]
|
D07615 Carbenoxolone (INN)
D01899 Carbenoxolone sodium (JAN/USAN)
D00156 Glycyrrhetinic acid (JAN) <JP>
D02028 Diammonium glycyrrhizinate (JAN)
D02264 Dipotassium glycyrrhizinate (JAN)
D04987 Monoammonium glycyrrhizinate (JAN)
D12948 Clofutriben (USAN/INN)
D13200 Emestedastat (USAN/INN)
|
HSD17B1 [HSA:3292] [KO:K00044]
|
D13078 Linustedastat (USAN/INN)
|
IMPDH [HSA:3614 3615] [KO:K00088]
|
D06130 Tiazofurin (USAN)
D05096 Mycophenolic acid (USAN/INN)
D00752 Mycophenolate mofetil (JAN/USP) <JP/US>
D05094 Mycophenolate mofetil hydrochloride (USAN) <US>
D05095 Mycophenolate sodium (USP) <US>
D01392 Mizoribine (JP18/INN) <JP>
D04936 Merimepodib (USAN/INN)
|
Oxidases [EC:1.1.3.-]
|
HAO1 [HSA:54363] [KO:K11517]
|
D11925 Lumasiran (USAN/INN)
D11926 Lumasiran sodium <US>
|
Dehydrogenases [EC:1.2.1.-]
|
ALDH [HSA:217 219 224] [KO:K00128]
|
D00131 Disulfiram (JP18/USP/INN) <JP/US>
D00123 Cyanamide (JP18) <JP>
|
GAPDH [HSA:2597] [KO:K00134]
|
D12792 Misetionamide (USAN/INN)
|
SSADH [HSA:7915] [KO:K00139]
|
D00399 Valproic acid (USP) <US>
D00304 Divalproex sodium (USP) <US>
D00710 Valproate sodium (USAN) <JP/US>
D08667 Calcium valproate
|
Dehydrogenases [EC:1.3.-.-]
|
DPYD [HSA:1806] [KO:K00207]
|
D01846 Gimeracil (JAN/INN)
D03998 Eniluracil (USAN/INN)
|
SRD5A1 [HSA:6715] [KO:K12343]
|
D03820 Dutasteride (JAN/USP/INN) <JP/US>
D01134 Epristeride (JAN/USAN/INN)
D03107 Bexlosteride (USAN/INN)
D04498 Idronoxil (USAN/INN)
D04646 Izonsteride (USAN/INN)
D07121 Alfatradiol (INN)
|
SRD5A2 [HSA:6716] [KO:K12344]
|
D00321 Finasteride (JAN/USP/INN) <JP/US>
D03820 Dutasteride (JAN/USP/INN) <JP/US>
D04066 Estramustine (USAN/INN)
D02398 Estramustine phosphate sodium (USAN)
D06397 Estramustine phosphate sodium hydrate (JAN) <JP>
D01134 Epristeride (JAN/USAN/INN)
D04498 Idronoxil (USAN/INN)
D04646 Izonsteride (USAN/INN)
D07121 Alfatradiol (INN)
|
SRD5A3 [HSA:79644] [KO:K12345]
|
D04498 Idronoxil (USAN/INN)
|
DHODH [HSA:1723] [KO:K00254]
|
D00749 Leflunomide (JAN/USP/INN) <JP/US>
D10172 Teriflunomide (USAN) <US>
D03154 Brequinar sodium (USAN)
D11890 Emvododstat (USAN)
D13127 Vidofludimus (USAN/INN)
D13128 Vidofludimus calcium (USAN)
|
Amine oxidases [EC:1.4.3.-]
|
DAO [HSA:1610] [KO:K00273]
|
D11981 Luvadaxistat (USAN/INN)
|
MAO [HSA:4128 4129] [KO:K00274]
|
D05458 Phentermine (USAN/INN)
D05459 Phentermine hydrochloride (USP) <US>
D08453 Pargyline (INN)
D02564 Pargyline hydrochloride (USAN)
D02580 Isocarboxazid (INN)
D07337 Nialamide (INN)
D08349 Phenelzine (BAN)
D00505 Phenelzine sulfate (USP) <US>
D08625 Tranylcypromine (INN)
D00826 Tranylcypromine sulfate (USP) <US>
D02579 Iproniazid (INN)
D08085 Iproniazid phosphate
D07338 Iproclozide (INN)
D01888 Safrazine hydrochloride (JAN)
D03239 Ladostigil tartrate (USAN)
D03409 Caroxazone (USAN/INN)
D04092 Etryptamine acetate (USAN)
|
MAOA [HSA:4128] [KO:K00274]
|
D02561 Moclobemide (USAN/INN)
D02559 Toloxatone (INN)
D05039 Minaprine (USAN/INN)
D05040 Minaprine hydrochloride (USAN)
D02560 Brofaromine (INN)
D02563 Befloxatone (INN)
D02581 Cimoxatone (INN)
D03248 Clorgiline (INN)
D08392 Pirlindole (INN)
D08393 Pirlindole hydrochloride
|
MAOB [HSA:4129] [KO:K00274]
|
D03731 Selegiline (USAN/INN) <US>
D00785 Selegiline hydrochloride (JAN/USP) <JP/US>
D08469 Rasagiline (USAN/INN)
D02562 Rasagiline mesylate (USAN) <JP/US>
D10829 Rasagiline tartrate
D10158 Safinamide (USAN/INN)
D10191 Safinamide mesylate (USAN) <JP/US>
D01097 Lazabemide hydrochloride (JAN/USAN)
D03733 Mofegiline hydrochloride (USAN)
D04681 Lazabemide (USAN/INN)
D05033 Milacemide hydrochloride (USAN)
D11224 Sembragiline (USAN/INN)
|
LOX [HSA:4015] [KO:K00277]
|
D13190 Amsulostat (USAN/INN)
D13191 Amsulostat hydrochloride (USAN)
|
AOC3 [HSA:8639] [KO:K00276]
|
D08044 Hydralazine (INN)
D04458 Hydralazine polistirex (USAN)
|
AOC1 (DAO) [HSA:26] [KO:K11182]
|
D05479 Pimagedine hydrochloride (USAN)
|
Dihydrofolate reductase [EC:1.5.1.3]
|
DHFR [HSA:1719 200895] [KO:K00287]
|
D00142 Methotrexate (JP18/USP/INN) <JP/US>
D02115 Methotrexate sodium <US>
D07472 Pemetrexed (INN) <US>
D03828 Pemetrexed disodium (USAN) <US>
D06503 Pemetrexed sodium hydrate (JAN) <JP/US>
D10596 Pemetrexed sodium hemipentahydrate (JAN) <JP/US>
D11352 Pemetrexed tromethamine (USAN)
D13147 Pemetrexed dipotassium heptahydrate <US>
D05589 Pralatrexate (JAN/USAN/INN) <JP/US>
D06238 Trimetrexate (USAN/INN)
D06239 Trimetrexate glucuronate (USAN)
D03942 Edatrexate (USAN/INN)
D05500 Piritrexim isethionate (USAN)
D05999 Talotrexin ammonium (USAN)
|
NAD(P)H dehydrogenase [EC:1.6.5.2]
|
NQO1 [HSA:1728] [KO:K00355]
|
D08682 Warfarin (INN)
D00564 Warfarin sodium (USP) <US>
D01280 Warfarin potassium (JP18) <JP>
D07064 Acenocoumarol (INN)
|
Peroxidase [EC:1.11.1.-]
|
TPO [HSA:7173] [KO:K00431]
|
D07231 Methylthiouracil (INN)
D00562 Propylthiouracil (JP18/USP/INN) <JP/US>
D07519 Benzylthiouracil
D07616 Carbimazole (INN)
D00401 Methimazole (USP) <JP/US>
|
Peroxygenase [EC:1.11.2.-]
|
MPO [HSA:4353] [KO:K10789]
|
D11684 Verdiperstat (USAN/INN)
D12647 Mitiperstat (USAN/INN)
|
Dioxygenases [EC:1.13.11.-]
|
HPD [HSA:3242] [KO:K00457]
|
D05177 Nitisinone (JAN/USAN/INN) <JP/US>
|
ALOX15 [HSA:246] [KO:K00460]
|
D12510 Utreloxastat (JAN/USAN/INN)
|
ALOX5 [HSA:240] [KO:K00461]
|
D07516 Benzydamine (INN)
D01410 Benzydamine hydrochloride (JAN/USAN)
D07517 Benzydamine salicylate
D03080 Benoxaprofen (USAN/INN)
D01773 Oxatomide (JAN/USAN/INN) <JP>
D00414 Zileuton (USP/INN) <US>
D03010 Atreleuton (USAN/INN)
D03652 Darbufelone mesylate (USAN)
D03882 Docebenone (USAN/INN)
D03990 Enazadrem phosphate (USAN)
D04151 Fenleuton (USAN/INN)
D04770 Lonapalene (USAN)
D05498 Piriprost (USAN/INN)
D05499 Piriprost potassium (USAN)
D06017 Tebufelone (USAN/INN)
D06075 Tepoxalin (USAN/INN)
D09667 Setileuton (USAN/INN)
D09850 Linazolast (JAN)
|
IDO [HSA:3620 169355] [KO:K00463]
|
D10640 Indoximod (USAN/INN)
|
IDO1 [HSA:3620] [KO:K00463]
|
D11049 Epacadostat (JAN/USAN/INN)
D11255 Navoximod (USAN/INN)
D11412 Linrodostat (USAN/INN)
D11413 Linrodostat mesylate (USAN)
|
Prolyl 4-hydroxylase [EC:1.14.11.2]
|
P4HA [HSA:5033 8974 283208] [KO:K00472]
|
D04793 Lufironil (USAN/INN)
|
HIF hydroxylase [EC:1.14.11.29]
|
EGLN (HPH) [HSA:54583 112398 112399] [KO:K09592]
|
D10593 Roxadustat (JAN/USAN/INN) <JP>
D10874 Daprodustat (JAN/USAN/INN) <JP/US>
D11078 Vadadustat (JAN/USAN/INN) <JP/US>
D12122 Molidustat (USAN/INN)
D11273 Molidustat sodium (JAN/USAN) <JP>
D11523 Enarodustat (JAN) <JP>
|
Nitic oxide synthase [EC:1.14.13.39]
|
NOS [HSA:4842 4843 4846] [KO:K13240 K13241 K13242]
|
D05479 Pimagedine hydrochloride (USAN)
D09018 Tilarginine acetate (USAN)
|
NOS2 [HSA:4843] [KO:K13241]
|
D10386 Cindunistat (USAN/INN)
D10419 Cindunistat hydrochloride maleate (USAN)
|
Cytochrome P450 [EC:1.14.14.-]
|
CYP3A [HSA:1551 1576 1577 64816] [KO:K17691 K17689 K17690 K17692]
|
D09881 Cobicistat (JAN/USAN/INN) <US>
|
CYP19A1 (ARO) [HSA:1588] [KO:K07434]
|
D00574 Aminoglutethimide (USP/INN)
D07260 Formestane (INN)
D00960 Anastrozole (JP18/USP/INN) <JP/US>
D00964 Letrozole (JAN/USP/INN) <JP/US>
D03786 Vorozole (USAN/INN)
D00963 Exemestane (JAN/USP/INN) <JP/US>
D00153 Testolactone (USP/INN)
D02451 Fadrozole hydrochloride (USAN)
D03749 Plomestane (USAN/INN)
D03778 Fadrozole hydrochloride hydrate (JAN)
D03781 Liarozole fumarate (USAN)
D03784 Liarozole hydrochloride (USAN)
D05746 Rogletimide (USAN/INN)
D07940 Fadrozole (INN)
|
CYP17A1 [HSA:1586] [KO:K00512]
|
D10950 Levoketoconazole (USAN/INN) <US>
D00420 Mitotane (JAN/USP/INN) <JP/US>
D09701 Abiraterone acetate (JAN/USP) <JP/US>
D10125 Galeterone (USAN)
D10146 Orteronel (JAN/USAN)
|
CYP46A1 [HSA:10858] [KO:K07440]
|
D11590 Soticlestat (JAN/USAN/INN)
|
CYP51A1 [HSA:1595] [KO:K05917]
|
D03025 Azalanstat dihydrochloride (USAN)
|
CYP11B1 [HSA:1584] [KO:K00497]
|
D10950 Levoketoconazole (USAN/INN) <US>
D00410 Metyrapone (JP18/USP/INN) <JP/US>
D05019 Metyrapone tartrate (USAN)
|
CYP11B2 [HSA:1585] [KO:K07433]
|
D12789 Baxdrostat (JAN/USAN/INN)
D11061 Osilodrostat (USAN/INN)
D11062 Osilodrostat phosphate (JAN/USAN) <JP/US>
D12773 Lorundrostat (USAN/INN)
D12774 Lorundrostat hydrobromide (USAN)
D13192 Vicadrostat (USAN/INN)
|
CYP11A1 [HSA:1583] [KO:K00498]
|
D10950 Levoketoconazole (USAN/INN) <US>
D13110 Opevesostat (USAN/INN)
D13111 Opevesostat tosylate (USAN)
|
CYP26 [HSA:1592 56603 340665] [KO:K07437 K12664 K12665]
|
D09385 Talarozole (USAN/INN)
|
Other monooxygenases [EC:1.14.16.- 1.14.17.- 1.14.18.-]
|
PAH* [HSA_VAR:5053v1] [HSA:5053] [KO:K00500]
|
D11077 Pegvaliase (INN) <JP/US>
|
TH [HSA:7054] [KO:K00501]
|
D00762 Metyrosine (USP) <JP/US>
|
TPH [HSA:7166 121278] [KO:K00502]
|
D09973 Telotristat (USAN/INN)
D09974 Telotristat ethyl (USAN)
D09975 Telotristat etiprate (USAN) <US>
|
TPH1 [HSA:7166] [KO:K00502]
|
D11317 Rodatristat (USAN)
D11318 Rodatristat ethyl (USAN)
|
DBH [HSA:1621] [KO:K00503]
|
D03787 Nepicastat hydrochloride (USAN)
|
TYR [HSA:7299] [KO:K00505]
|
D00073 Hydroquinone (USP)
|
HMOX [HSA:3162 3163] [KO:K00510 K21418]
|
D05922 Stannsoporfin (USAN/INN)
|
Prostaglandin synthase [EC:1.14.99.1]
|
PTGS1 (COX1) [HSA:5742] [KO:K00509]
|
D07516 Benzydamine (INN)
D01410 Benzydamine hydrochloride (JAN/USAN)
D07517 Benzydamine salicylate
D00109 Aspirin (JP18/USP) <JP>
D05181 Aspirin aluminum (JP18)
D07579 Aspirin calcium salt
D07580 Aspirin DL-lysine (JAN)
D07581 Aspirin magnesium salt
D07582 Aspirin sodium
D12595 Aspirin trelamine (USAN)
D12596 Aspirin trelamine hydrochloride (USAN)
D07141 Indobufen (INN)
D07421 Aloxiprin (INN)
D07142 Triflusal (INN)
D00141 Indomethacin (USP) <JP/US>
D01565 Indometacin farnesil (JAN) <JP>
D02110 Indomethacin sodium (USP) <JP>
D00126 Ibuprofen (JP18/USP/INN) <JP/US>
D01122 Ibuprofen piconol (JP18/USAN) <JP>
D04490 Ibuprofen aluminum (USAN)
D06606 Ibuprofen lysine (USAN) <JP/US>
D08058 Ibuprofen arginine salt
D08059 Ibuprofen sodium
D09760 Ibuprofen sodium (USAN)
D12597 Ibuprofen trelamine (USAN)
D12598 Ibuprofen trelamine hydrochloride (USAN)
D08501 Trolamine salicylate (USP)
D07816 Diclofenac (USAN/INN)
D00903 Diclofenac potassium (USP) <US>
D00904 Diclofenac sodium (JP18/USP) <JP/US>
D07817 Diclofenac diethylamine
D07818 Diclofenac epolamine <US>
D07819 Diclofenac calcium
D00118 Naproxen (JP18/USP/INN) <JP/US>
D00970 Naproxen sodium (USP) <US>
D10017 Naproxen etemesil (USAN)
D00510 Phenylbutazone (JP18/USP/INN)
D08363 Phenylbutazone calcium
D08364 Phenylbutazone sodium
D08324 Oxyphenbutazone (INN)
D05319 Oxyphenbutazone hydrate
D00120 Sulindac (JP18/USP/INN) <US>
D02355 Tolmetin (USAN/INN)
D00158 Tolmetin sodium (JAN/USP) <US>
D01582 Acemetacin (JP18/INN) <JP>
D08427 Proglumetacin (INN)
D01765 Proglumetacin maleate (JAN)
D08104 Ketorolac (INN)
D00813 Ketorolac tromethamine (USP) <US>
D01545 Aceclofenac (JAN/INN)
D01271 Bufexamac (JAN/INN)
D00127 Piroxicam (JP18/USP/INN) <US>
D05511 Piroxicam betadex (USAN)
D05512 Piroxicam cinnamate (USAN)
D05513 Piroxicam olamine (USAN)
D01767 Tenoxicam (JAN/USAN/INN)
D07267 Droxicam (INN)
D01866 Lornoxicam (JP18/USAN/INN) <JP>
D00132 Ketoprofen (JP18/USP/INN) <JP/US>
D08102 Ketoprofen lysine
D08103 Ketoprofen sodium
D02350 Fenoprofen (USAN/INN)
D00968 Fenoprofen calcium (JAN/USP) <US>
D01344 Fenbufen (JP18/USAN/INN)
D00330 Flurbiprofen (JP18/USP/INN) <JP/US>
D01475 Flurbiprofen axetil (JAN) <JP>
D02290 Flurbiprofen sodium (USP) <US>
D10254 Esflurbiprofen (JAN)
D01325 Tiaprofenic acid (JAN/INN)
D00463 Oxaprozin (JP18/USP/INN) <JP/US>
D07268 Ibuproxam (INN)
D03715 Dexibuprofen (USAN/INN)
D03718 Dexibuprofen lysine (USAN)
D01513 Alminoprofen (JP18/INN)
D07269 Dexketoprofen (INN)
D09568 Naproxcinod (USAN/INN)
D08149 Loxoprofen (INN)
D01709 Loxoprofen sodium hydrate (JP18) <JP>
D00151 Mefenamic acid (JP18/USP/INN) <JP/US>
D01183 Tolfenamic acid (JAN/INN)
D01581 Flufenamic acid (JAN/USAN/INN)
D01823 Ufenamate (JAN/INN) <JP>
D03254 Flufenamate aluminum (JAN)
D02341 Meclofenamic acid (USAN/INN)
D00169 Meclofenamate sodium (USP) <US>
D08162 Meclofenamate sodium
D00425 Nabumetone (JP18/USP/INN) <JP/US>
D06072 Tenidap (USAN/INN)
D06073 Tenidap sodium (USAN)
D04102 Etofenamate (USAN/INN)
D01675 Felbinac (JP18/USAN/INN) <JP>
D01841 Felbinac ethyl (JAN)
D08374 Piketoprofen (INN)
D08375 Piketoprofen hydrochloride
D00810 Choline salicylate (JAN/USAN/INN)
D00566 Sodium salicylate (JP18/USP) <JP>
D01811 Salicylamide (JAN/USP/INN)
D00428 Salsalate (USP/INN)
D00217 Acetaminophen (JP18/USP) <JP/US>
D07294 Propacetamol (INN)
D08434 Propacetamol hydrochloride
D01578 Pranoprofen (JP18/INN) <JP>
D05143 Nepafenac (JAN/USAN/INN) <JP/US>
D07541 Bromfenac (INN)
D03163 Bromfenac sodium (USAN) <JP/US>
D00827 Magnesium salicylate (USP)
D01090 Pamicogrel (JAN/INN)
D01397 Ampiroxicam (JP18/INN)
D01527 Epidihydrocholesterin (JAN)
D01547 Zaltoprofen (JP18/INN) <JP>
D01557 Glycol salicylate (JAN)
D01718 Mofezolac (JAN/INN)
D01788 Amfenac sodium (USAN)
D03410 Carprofen (USP/INN)
D05275 Orpanoxin (USAN/INN)
D05451 Phenbutazone sodium glycerate (USAN)
D05598 Pravadoline maleate (USAN)
D05791 Salicylate meglumine (USAN)
D06017 Tebufelone (USAN/INN)
D06364 Zidometacin (USAN/INN)
D07443 Amfenac (INN)
D07453 Amtolmetin guacil (INN)
|
PTGS2 (COX2) [HSA:5743] [KO:K11987]
|
D07516 Benzydamine (INN)
D01410 Benzydamine hydrochloride (JAN/USAN)
D07517 Benzydamine salicylate
D00109 Aspirin (JP18/USP) <JP>
D05181 Aspirin aluminum (JP18)
D07579 Aspirin calcium salt
D07580 Aspirin DL-lysine (JAN)
D07581 Aspirin magnesium salt
D07582 Aspirin sodium
D12595 Aspirin trelamine (USAN)
D12596 Aspirin trelamine hydrochloride (USAN)
D07141 Indobufen (INN)
D07421 Aloxiprin (INN)
D00141 Indomethacin (USP) <JP/US>
D01565 Indometacin farnesil (JAN) <JP>
D02110 Indomethacin sodium (USP) <JP>
D00126 Ibuprofen (JP18/USP/INN) <JP/US>
D01122 Ibuprofen piconol (JP18/USAN) <JP>
D04490 Ibuprofen aluminum (USAN)
D06606 Ibuprofen lysine (USAN) <JP/US>
D08058 Ibuprofen arginine salt
D08059 Ibuprofen sodium
D09760 Ibuprofen sodium (USAN)
D12597 Ibuprofen trelamine (USAN)
D12598 Ibuprofen trelamine hydrochloride (USAN)
D08501 Trolamine salicylate (USP)
D07816 Diclofenac (USAN/INN)
D00903 Diclofenac potassium (USP) <US>
D00904 Diclofenac sodium (JP18/USP) <JP/US>
D07817 Diclofenac diethylamine
D07818 Diclofenac epolamine <US>
D07819 Diclofenac calcium
D00118 Naproxen (JP18/USP/INN) <JP/US>
D00970 Naproxen sodium (USP) <US>
D10017 Naproxen etemesil (USAN)
D00567 Celecoxib (JP18/USP/INN) <JP/US>
D00510 Phenylbutazone (JP18/USP/INN)
D08363 Phenylbutazone calcium
D08364 Phenylbutazone sodium
D08324 Oxyphenbutazone (INN)
D05319 Oxyphenbutazone hydrate
D00120 Sulindac (JP18/USP/INN) <US>
D02355 Tolmetin (USAN/INN)
D00158 Tolmetin sodium (JAN/USP) <US>
D01252 Alclofenac (JAN/USP/INN)
D00315 Etodolac (JP18/USP/INN) <JP/US>
D01582 Acemetacin (JP18/INN) <JP>
D08427 Proglumetacin (INN)
D01765 Proglumetacin maleate (JAN)
D08104 Ketorolac (INN)
D00813 Ketorolac tromethamine (USP) <US>
D01545 Aceclofenac (JAN/INN)
D01271 Bufexamac (JAN/INN)
D00127 Piroxicam (JP18/USP/INN) <US>
D05511 Piroxicam betadex (USAN)
D05512 Piroxicam cinnamate (USAN)
D05513 Piroxicam olamine (USAN)
D01767 Tenoxicam (JAN/USAN/INN)
D07267 Droxicam (INN)
D01866 Lornoxicam (JP18/USAN/INN) <JP>
D00969 Meloxicam (JAN/USP/INN) <JP/US>
D00132 Ketoprofen (JP18/USP/INN) <JP/US>
D08102 Ketoprofen lysine
D08103 Ketoprofen sodium
D02350 Fenoprofen (USAN/INN)
D00968 Fenoprofen calcium (JAN/USP) <US>
D01344 Fenbufen (JP18/USAN/INN)
D00330 Flurbiprofen (JP18/USP/INN) <JP/US>
D01475 Flurbiprofen axetil (JAN) <JP>
D02290 Flurbiprofen sodium (USP) <US>
D10254 Esflurbiprofen (JAN)
D01325 Tiaprofenic acid (JAN/INN)
D00463 Oxaprozin (JP18/USP/INN) <JP/US>
D07268 Ibuproxam (INN)
D03715 Dexibuprofen (USAN/INN)
D03718 Dexibuprofen lysine (USAN)
D01513 Alminoprofen (JP18/INN)
D07269 Dexketoprofen (INN)
D09568 Naproxcinod (USAN/INN)
D08149 Loxoprofen (INN)
D01709 Loxoprofen sodium hydrate (JP18) <JP>
D00151 Mefenamic acid (JP18/USP/INN) <JP/US>
D01183 Tolfenamic acid (JAN/INN)
D01581 Flufenamic acid (JAN/USAN/INN)
D01823 Ufenamate (JAN/INN) <JP>
D03254 Flufenamate aluminum (JAN)
D02341 Meclofenamic acid (USAN/INN)
D00169 Meclofenamate sodium (USP) <US>
D08162 Meclofenamate sodium
D00568 Rofecoxib (JAN/USAN/INN)
D02709 Valdecoxib (USAN/INN)
D03716 Parecoxib (USAN/INN)
D03717 Parecoxib sodium (USAN)
D03710 Etoricoxib (USAN/INN)
D03714 Lumiracoxib (USAN/INN)
D10656 Polmacoxib (USAN/INN)
D00425 Nabumetone (JP18/USP/INN) <JP/US>
D08275 Niflumic acid (INN)
D01049 Nimesulide (JAN/INN)
D06072 Tenidap (USAN/INN)
D06073 Tenidap sodium (USAN)
D04102 Etofenamate (USAN/INN)
D01675 Felbinac (JP18/USAN/INN) <JP>
D01841 Felbinac ethyl (JAN)
D08374 Piketoprofen (INN)
D08375 Piketoprofen hydrochloride
D00810 Choline salicylate (JAN/USAN/INN)
D00566 Sodium salicylate (JP18/USP) <JP>
D01811 Salicylamide (JAN/USP/INN)
D00428 Salsalate (USP/INN)
D00130 Diflunisal (JAN/USP/INN) <US>
D00217 Acetaminophen (JP18/USP) <JP/US>
D07294 Propacetamol (INN)
D08434 Propacetamol hydrochloride
D01578 Pranoprofen (JP18/INN) <JP>
D05143 Nepafenac (JAN/USAN/INN) <JP/US>
D07541 Bromfenac (INN)
D03163 Bromfenac sodium (USAN) <JP/US>
D00827 Magnesium salicylate (USP)
D01090 Pamicogrel (JAN/INN)
D01397 Ampiroxicam (JP18/INN)
D01547 Zaltoprofen (JP18/INN) <JP>
D01557 Glycol salicylate (JAN)
D01788 Amfenac sodium (USAN)
D01974 Tilmacoxib (JAN/USAN/INN)
D03410 Carprofen (USP/INN)
D03652 Darbufelone mesylate (USAN)
D03689 Deracoxib (USAN)
D03712 Firocoxib (USAN/INN)
D04863 Mavacoxib (USAN)
D05275 Orpanoxin (USAN/INN)
D05451 Phenbutazone sodium glycerate (USAN)
D05598 Pravadoline maleate (USAN)
D05791 Salicylate meglumine (USAN)
D06017 Tebufelone (USAN/INN)
D06364 Zidometacin (USAN/INN)
D07443 Amfenac (INN)
D07453 Amtolmetin guacil (INN)
D07888 Eltenac (INN)
D08657 Apricoxib (USAN/INN)
D11020 Diclofenac etalhyaluronate sodium (JAN) <JP>
|
Histone demethylase [EC:1.14.99.66]
|
KDM1A (LSD1) [HSA:23028] [KO:K11450]
|
D12263 Bomedemstat (USAN/INN)
D12264 Bomedemstat tosylate (USAN)
D12577 Seclidemstat (USAN/INN)
D12578 Seclidemstat mesylate (USAN)
|
Superoxide dismutase [EC:1.15.1.1]
|
SOD1* [HSA_VAR:6647v1] [HSA:6647] [KO:K04565]
|
D11811 Tofersen (JAN/USAN/INN) <JP/US>
|
Xanthine dehydrogenase/oxidase [EC:1.17.1.4 1.17.3.2]
|
XDH [HSA:7498] [KO:K00106]
|
D00224 Allopurinol (JP18/USP/INN) <JP/US>
D07564 Allopurinol sodium <US>
D07278 Tisopurine (INN)
D01206 Febuxostat (JP18/USAN/INN) <JP/US>
D11081 Febuxostat hydrate (JAN) <JP/US>
D02365 Oxypurinol (USAN)
D02896 Amflutizole (USAN/INN)
D09786 Topiroxostat (JAN/INN) <JP>
|
Ribonucleoside-diphosphate reductase [EC:1.17.4.1]
|
RRM1 [HSA:6240] [KO:K10807]
|
D01370 Cladribine (JAN/USP/INN) <JP/US>
D07966 Fludarabine (INN)
D01907 Fludarabine phosphate (JAN/USP) <JP/US>
D03546 Clofarabine (JAN/USAN/INN) <JP/US>
D02368 Gemcitabine (USAN/INN)
D01155 Gemcitabine hydrochloride (JAN/USP) <JP/US>
D10222 Gemcitabine elaidate (USAN/INN)
D03378 Caracemide (USAN)
D06100 Tezacitabine (USAN)
D12387 Fosgemcitabine palabenamide (USAN/INN)
|
RRM2 [HSA:6241] [KO:K10808]
|
D00341 Hydroxyurea (USP) <JP/US>
|
Vitamin-K-epoxide reductase [EC:1.17.4.4]
|
VKORC1 [HSA:79001] [KO:K05357]
|
D03798 Dicumarol (USAN)
D08354 Phenindione (INN)
D08682 Warfarin (INN)
D00564 Warfarin sodium (USP) <US>
D01280 Warfarin potassium (JP18) <JP>
D05457 Phenprocoumon (USAN/INN)
D07064 Acenocoumarol (INN)
D07131 Ethyl biscoumacetate (INN)
D07135 Clorindione (INN)
D07136 Diphenadione (INN)
D07137 Tioclomarol (INN)
D07969 Fluindione (INN)
D07134 Flocoumafen (JAN)
D09676 Tecarfarin (USAN/INN)
D09677 Tecarfarin sodium (USAN)
|
Thyroxine 5'-deiodinase [EC:1.21.99.4]
|
DIO1 [HSA:1733] [KO:K01562]
|
D00562 Propylthiouracil (JP18/USP/INN) <JP/US>
|
DIO2 [HSA:1734] [KO:K17904]
|
D00562 Propylthiouracil (JP18/USP/INN) <JP/US>
|
Transferases (EC2)
|
Methyltransferases [EC:2.1.1.-]
|
COMT [HSA:1312] [KO:K00545]
|
D00152 Phloroglucinol (JAN)
D08369 Polyphloroglucinol phosphate
D00786 Tolcapone (JAN/USP/INN) <US>
D00781 Entacapone (JP18/USP/INN) <JP/US>
D10825 Opicapone (JAN/USAN/INN) <JP/US>
D01259 Flopropione (JP18/INN) <JP>
D03241 Nitecapone (INN)
|
DNMT [HSA:1786 1788 1789] [KO:K00558 K17398 K17399]
|
D03021 Azacitidine (JAN/USAN/INN) <JP/US>
D03665 Decitabine (USAN/INN) <US>
|
DNMT1 [HSA:1786] [KO:K00558]
|
D11740 Roducitabine (USAN)
|
EZH [HSA:2145 2146] [KO:K17451 K11430]
|
D11551 Valemetostat (INN)
D11662 Valemetostat tosilate (JAN) <JP>
|
EZH2 [HSA:2146] [KO:K11430]
|
D11444 Tazemetostat (USAN/INN)
D12602 Tulmimetostat (USAN/INN)
D12845 Mevrometostat (USAN)
|
EZH2* [HSA_VAR:2146v1] [HSA:2146] [KO:K11430]
|
D11485 Tazemetostat hydrobromide (JAN/USAN) <JP/US>
|
TYMS [HSA:7298] [KO:K00560]
|
D01064 Raltitrexed (JAN/USAN/INN)
D07472 Pemetrexed (INN) <US>
D03828 Pemetrexed disodium (USAN) <US>
D06503 Pemetrexed sodium hydrate (JAN) <JP/US>
D10596 Pemetrexed sodium hemipentahydrate (JAN) <JP/US>
D11352 Pemetrexed tromethamine (USAN)
D13147 Pemetrexed dipotassium heptahydrate <US>
D00584 Fluorouracil (JP18/USP/INN) <JP/US>
D07974 Fluorouracil sodium salt
D01244 Tegafur (JP18/USAN/INN)
D01784 Carmofur (JP18/INN)
D01223 Capecitabine (JAN/USP/INN) <JP/US>
D04197 Floxuridine (USP/INN) <US>
D01309 Doxifluridine (JP18/INN) <JP>
D04964 Metesind glucuronate (USAN)
D10803 Plevitrexed (INN)
D11447 Arfolitixorin (USAN/INN)
D12388 Fosifloxuridine nafalbenamide
D12528 Arfolitixorin sulfate (JAN)
|
Acyltransferases [EC:2.3.1.-]
|
DGAT1 [HSA:8694] [KO:K11155]
|
D10657 Pradigastat sodium (USAN)
D10664 Pradigastat (USAN)
|
CPT [HSA:1374 1375 126129 1376] [KO:K08765 K19523 K19524 K08766]
|
D08340 Perhexiline (INN)
D05442 Perhexiline maleate (USAN)
|
CPT1 [HSA:1374 1375 126129] [KO:K08765 K19523 K19524]
|
D05292 Oxfenicine (USAN/INN)
|
SOAT [HSA:6646 8435] [KO:K00637]
|
D01202 Melinamide (JAN)
D03012 Avasimibe (USAN/INN)
D03447 Cetaben sodium (USAN)
D03734 Eldacimibe (USAN/INN)
D03735 Lecimibide (USAN)
|
ALAS [HSA:211 212] [KO:K00643]
|
D10003 Hemin (JAN) <JP/US>
|
ALAS1 [HSA:211] [KO:K00643]
|
D11702 Givosiran (USAN/INN)
D11708 Givosiran sodium (JAN) <JP/US>
|
LCAT [HSA:3931] [KO:K00650]
|
D04268 Elastase ES <JP>
|
KAT6A [HSA:7994] [KO:K11305]
|
D12983 Prifetrastat (USAN)
|
KAT6B [HSA:23522] [KO:K11306]
|
D12983 Prifetrastat (USAN)
|
CREBBP/EP300 [HSA:1387 2033] [KO:K04498]
|
D12394 Inobrodib (USAN)
D12924 Pocenbrodib (USAN/INN)
D12925 Pocenbrodib hydrochloride (USAN)
|
FASN [HSA:2194] [KO:K00665]
|
D12391 Denifanstat (USAN/INN)
|
SIRT6 [HSA:51548] [KO:K11416]
|
D13109 Forvisirvat (USAN)
|
gamma-Glutamyltransferase [EC:2.3.2.2]
|
GGT [HSA:2678 2687 124975 2686] [KO:K18592 K00681]
|
D02755 Acivicin (USAN/INN)
|
E3 ubiquitin-protein ligase [EC:2.3.2.27]
|
MDM2 [HSA:4193] [KO:K06643]
|
D11219 Idasanutlin (USAN/INN)
D12378 Navtemadlin (USAN/INN)
D12399 Sulanemadlin (USAN/INN)
D12417 Siremadlin (USAN/INN)
D12418 Siremadlin succinate (USAN)
D12621 Milademetan (USAN/INN)
D12622 Milademetan tosylate (USAN)
D12842 Brigimadlin (JAN/USAN/INN)
|
MDM4 [HSA:4194] [KO:K10127]
|
D12399 Sulanemadlin (USAN/INN)
|
ATP citrate synthase [EC:2.3.3.8]
|
ACLY (ACL) [HSA:47] [KO:K01648]
|
D10691 Bempedoic acid (JAN/USAN/INN) <JP/US>
|
Hexosyltransferases [EC:2.4.1.-]
|
PYG [HSA:5834 5836 5837] [KO:K00688]
|
D04537 Ingliforib (USAN/INN)
|
UGCG [HSA:7357] [KO:K00720]
|
D05032 Miglustat (JAN/USAN/INN) <JP/US>
D09893 Eliglustat (USAN/INN)
D09894 Eliglustat tartrate (JAN/USAN) <JP/US>
D11439 Lucerastat (JAN/USAN/INN)
D11633 Venglustat (USAN/INN)
|
A3GALT2 [HSA:127550] [KO:K20736]
|
D10429 Tergenpumatucel-L (USAN)
|
Pentosyltransferases [EC:2.4.2.-]
|
PNP [HSA:4860] [KO:K03783]
|
D04245 Forodesine hydrochloride (JAN/USAN) <JP>
D05396 Peldesine (USAN)
D06596 Forodesine (USAN/INN)
D10431 Ulodesine (USAN/INN)
D10432 Ulodesine succinate (USAN)
|
HPRT1 [HSA:3251] [KO:K00760]
|
D04931 Mercaptopurine (INN)
D00161 Mercaptopurine (USP) <JP/US>
D08603 Tioguanine (INN)
D06109 Thioguanine (USP) <US>
|
NAMPT [HSA:10135] [KO:K03462]
|
D09678 Teglarinad chloride (USAN/INN)
|
PARP [HSA:142 10038 10039 143] [KO:K24070 K28005 K10798]
|
D09692 Veliparib (JAN/USAN/INN)
|
PARP1 [HSA:142] [KO:K24070]
|
D09730 Olaparib (JAN/USAN/INN) <JP/US>
D10140 Niraparib (USAN)
D11895 Niraparib tosylate (USAN) <JP/US>
D10079 Rucaparib (USAN/INN)
D10157 Rucaparib phosphate (USAN)
D10982 Rucaparib camsylate (USAN) <US>
D10732 Talazoparib (USAN/INN)
D10733 Talazoparib tosylate (USAN) <JP/US>
D11426 Pamiparib (USAN/INN)
D13232 Senaparib (INN)
D09913 Iniparib (USAN/INN)
D12981 Saruparib (USAN/INN)
|
PARP2 [HSA:10038] [KO:K28005]
|
D09730 Olaparib (JAN/USAN/INN) <JP/US>
D10140 Niraparib (USAN)
D11895 Niraparib tosylate (USAN) <JP/US>
D10079 Rucaparib (USAN/INN)
D10157 Rucaparib phosphate (USAN)
D10982 Rucaparib camsylate (USAN) <US>
D10732 Talazoparib (USAN/INN)
D10733 Talazoparib tosylate (USAN) <JP/US>
D11426 Pamiparib (USAN/INN)
D13232 Senaparib (INN)
|
PARP3 [HSA:10039] [KO:K10798]
|
D10079 Rucaparib (USAN/INN)
D10157 Rucaparib phosphate (USAN)
D10982 Rucaparib camsylate (USAN) <US>
D11426 Pamiparib (USAN/INN)
|
TIPARP (PARP7) [HSA:25976] [KO:K15259]
|
D12408 Atamparib (USAN/INN)
|
Alkyl/Aryl transferases [EC:2.5.1.-]
|
FDPS [HSA:2224] [KO:K00787]
|
D07281 Pamidronic acid (INN)
D00941 Pamidronate disodium (USP) <JP/US>
D07119 Alendronic acid (INN)
D00939 Alendronate sodium (USP) <JP/US>
D08056 Ibandronic acid (INN)
D04486 Ibandronate sodium (USAN) <JP/US>
D08484 Risedronic acid (INN)
D00942 Risedronate sodium (USP) <US>
D03234 Sodium risedronate hydrate (JP18) <JP/US>
D11570 Risedronate sodium monohydrate <US>
D08689 Zoledronic acid (INN)
D01968 Zoledronic acid (USAN) <JP/US>
D06378 Zoledronate disodium (USAN)
D06379 Zoledronate trisodium (USAN)
D10515 Zoledronic acid hemipentahydrate (JAN)
D07123 Incadronate disodium hydrate (JAN)
D08073 Incadronic acid (INN)
D09198 Minodronic acid hydrate (JAN) <JP>
|
GSTP1 [HSA:2950] [KO:K23790]
|
D08917 Ezatiostat hydrochloride (USAN)
|
FDFT1 [HSA:2222] [KO:K00801]
|
D06609 Lapaquistat acetate (JAN/USAN)
|
FNT [HSA:2339 2342] [KO:K05955 K05954]
|
D04768 Lonafarnib (JAN/USAN/INN) <JP/US>
D03720 Tipifarnib (USAN/INN)
|
Aminotransferase [EC:2.6.1.-]
|
ABAT [HSA:18] [KO:K13524]
|
D00399 Valproic acid (USP) <US>
D00304 Divalproex sodium (USP) <US>
D00710 Valproate sodium (USAN) <JP/US>
D08667 Calcium valproate
D00535 Vigabatrin (JAN/USP/INN) <JP/US>
|
Phosphotransferase [EC:2.7.1.-]
|
HK [HSA:3098 3099 3101 80201] [KO:K00844]
|
D07257 Lonidamine (INN)
|
GCK [HSA:2645] [KO:K12407]
|
D11342 Dorzagliatin (USAN)
D08970 Piragliatin (USAN)
D12320 Cadisegliatin (USAN)
|
TK2 [HSA:7084] [KO:K00857]
|
D12465 Doxecitine (USAN/INN)
D12466 Doxribtimine (USAN/INN)
|
PKLR [HSA:5313] [KO:K12406]
|
D11408 Mitapivat sulfate (USAN) <US>
D12362 Etavopivat (USAN/INN)
D13032 Tebapivat (USAN/INN)
|
PIK3C3 [HSA:5289] [KO:K00914]
|
D05784 Safingol (USAN/INN)
D05785 Safingol hydrochloride (USAN)
D11319 Fimepinostat (USAN/INN)
|
PIK3CA [HSA:5290] [KO:K00922]
|
D10867 Copanlisib (USAN/INN)
D10797 Copanlisib hydrochloride (USAN)
D10798 Copanlisib hydrochloride hydrate (JAN)
D11942 Inavolisib (USAN/INN) <US>
D11869 Paxalisib (USAN/INN)
D12836 Risovalisib (INN)
D12837 Risovalisib mesilate hydrate (JAN)
|
PIK3CA* [HSA_VAR:5290v1] [HSA:5290] [KO:K00922]
|
D11011 Alpelisib (JAN/USAN/INN) <US>
|
PIK3CD [HSA:5293] [KO:K00922]
|
D10560 Idelalisib (JAN/USAN/INN) <US>
D10867 Copanlisib (USAN/INN)
D10797 Copanlisib hydrochloride (USAN)
D10798 Copanlisib hydrochloride hydrate (JAN)
D10555 Duvelisib (USAN/INN)
D11658 Duvelisib hydrate (JAN) <US>
D11437 Parsaclisib (USAN/INN)
D11506 Parsaclisib hydrochloride (JAN/USAN)
D11322 Umbralisib (USAN/INN)
D11323 Umbralisib tosylate (USAN)
D11159 Leniolisib phosphate (JAN/USAN) <US>
D10924 Dezapelisib (USAN/INN)
D11267 Nemiralisib (USAN/INN)
D11354 Nemiralisib succinate (USAN)
D12009 Zandelisib (JAN/USAN/INN)
D12514 Amdizalisib (USAN/INN)
|
PIK3CG [HSA:5294] [KO:K21289]
|
D10555 Duvelisib (USAN/INN)
D11658 Duvelisib hydrate (JAN) <US>
D11896 Eganelisib (USAN)
|
PIK3C [HSA:5290 5291 5293] [KO:K00922]
|
D11158 Leniolisib (USAN/INN)
D10189 Pictilisib (USAN/INN)
D10543 Apitolisib (USAN/INN)
D10552 Dactolisib (USAN/INN)
D10584 Buparlisib (USAN/INN)
D10609 Buparlisib hydrochloride (JAN/USAN)
D10616 Dactolisib tosylate (USAN)
D10635 Gedatolisib (USAN/INN)
D10718 Omipalisib (USAN/INN)
D11440 Bimiralisib (USAN/INN)
D11501 Samotolisib (USAN)
D11727 Voxtalisib (USAN/INN)
D11774 Taselisib (USAN/INN)
|
DNA polymerase [EC:2.7.7.7]
|
POLA [HSA:5422 23649] [KO:K02320 K02321]
|
D03546 Clofarabine (JAN/USAN/INN) <JP/US>
|
Reverse transcriptase [EC:2.7.7.49]
|
TERT [HSA:7015] [KO:K11126]
|
D09629 Imetelstat (USAN/INN)
D09630 Imetelstat sodium (USAN) <US>
D13071 Ateganosine (USAN/INN)
|
Hydrolases (EC3)
|
Carboxylic-ester hydrolases [EC:3.1.1.-]
|
LIPF [HSA:8513] [KO:K14452]
|
D04028 Orlistat (JAN/USP/INN) <US>
|
LIPC [HSA:3990] [KO:K22283]
|
D02047 Dextran sulfate sodium (JAN)
D03343 Dextran sulfate sodium sulfur 5 (JP18)
|
PNLIP [HSA:5406] [KO:K14073]
|
D09208 Cetilistat (JAN/USAN/INN)
|
PNLIP [HSA:5406 5407 5408] [KO:K14073 K14074 K14075]
|
D04028 Orlistat (JAN/USP/INN) <US>
|
PLA2G [HSA:26279 30814 391013 50487 5319 5320 5322 64600 81579 8399 84647] [KO:K01047]
|
D06283 Varespladib sodium (USAN)
|
PLA2G4A [HSA:5321] [KO:K16342]
|
D03938 Ecopladib (USAN/INN)
D06600 Giripladib (USAN)
D06674 Efipladib (USAN)
|
PLA2G7 (LP-PLA2) [HSA:7941] [KO:K01062]
|
D03650 Darapladib (JAN/USAN)
D04368 Goxalapladib (USAN)
D05728 Rilapladib (USAN)
D06283 Varespladib sodium (USAN)
D08107 Varespladib (USAN/INN)
D08221 Varespladib methyl (USAN)
|
ACHE [HSA:43] [KO:K01049]
|
D08094 Itopride (INN)
D02729 Itopride hydrochloride (JAN) <JP>
D08838 Acotiamide hydrochloride (USAN) <JP>
D02292 Gallamine triethiodide (USP)
D02565 Dimetacrine (INN)
D08555 Tacrine (INN)
D02068 Tacrine hydrochloride (USP)
D07869 Donepezil (JAN/INN) <JP>
D00670 Donepezil hydrochloride (JP18/USP) <JP/US>
D03822 Rivastigmine (JAN/USP/INN) <JP/US>
D02558 Rivastigmine tartrate <US>
D04292 Galantamine (USAN/INN)
D02173 Galantamine hydrobromide (JAN/USP) <JP/US>
D09750 Ipidacrine hydrochloride hydrate (JAN)
D12930 Benzgalantamine (USAN/INN)
D12931 Benzgalantamine gluconate (USAN) <US>
D08261 Neostigmine (BAN)
D00995 Neostigmine bromide (JAN/USP/INN) <JP>
D00998 Neostigmine methylsulfate (JP18/USP) <JP/US>
D00487 Pyridostigmine bromide (JP18/USP/INN) <JP/US>
D01228 Distigmine bromide (JP18/INN) <JP>
D01001 Ambenonium chloride (JP18/INN) <JP>
D02193 Echothiophate iodide (USP) <US>
D00667 Demecarium bromide (USP/INN)
D00196 Physostigmine (USP)
D02418 Physostigmine salicylate (JAN/USP)
D03826 Physostigmine sulfate (USP)
D00043 Isoflurophate
D10529 Paraoxon
D00469 Pralidoxime chloride (USP) <US>
D01572 Pralidoxime iodide (JAN/USAN) <JP>
D05590 Pralidoxime mesylate (USAN)
D05215 Obidoxime chloride (USAN)
D00994 Edrophonium chloride (JP18/USP/INN) <JP>
D03239 Ladostigil tartrate (USAN)
D03751 Icopezil maleate (USAN)
D03823 Quilostigmine (USAN/INN)
D05981 Suronacrine maleate (USAN)
D06288 Velnacrine maleate (USAN)
D06365 Zifrosilone (USAN)
D09835 Zanapezil fumarate (JAN)
D09917 Latrepirdine (USAN/INN)
D09918 Latrepirdine dihydrochloride (USAN)
D12318 Buntanetap (USAN)
D12319 Buntanetap tartrate (USAN)
|
BCHE [HSA:590] [KO:K01050]
|
D04435 Hexafluorenium bromide (USAN)
D03822 Rivastigmine (JAN/USP/INN) <JP/US>
D02558 Rivastigmine tartrate <US>
D02193 Echothiophate iodide (USP) <US>
D00043 Isoflurophate
D03239 Ladostigil tartrate (USAN)
|
LIPA* [HSA_VAR:3988v1] [HSA:3988] [KO:K01052]
|
D10377 Sebelipase alfa (USAN) <JP/US>
|
MGLL [HSA:11343] [KO:K01054]
|
D13114 Irafamdastat (USAN)
|
LPL [HSA:4023] [KO:K01059]
|
D02047 Dextran sulfate sodium (JAN)
D03343 Dextran sulfate sodium sulfur 5 (JP18)
D05255 Omega-3-acid ethyl esters (USP) <JP/US>
D03747 Ibrolipim (USAN/INN)
D04268 Elastase ES <JP>
|
LPL* [HSA_VAR:4023v1] [HSA:4023] [KO:K01059]
|
D10843 Alipogene tiparvovec (INN)
|
RPE65 [HSA:6121] [KO:K11158]
|
D11008 Voretigene neparvovec (USAN/INN) <US>
|
RARRES3 (DDX58, RIG1) [HSA:5920] [KO:K23266]
|
D11385 Inarigivir soproxil (USAN)
|
Phosphatases [EC:3.1.3.-]
|
ALPI (IAP) [HSA:248] [KO:K01077]
|
D12277 Ilofotase alfa (USAN/INN)
|
ALPL [HSA:249] [KO:K01077]
|
D12991 Efzimfotase alfa (USAN/INN)
|
ALPL* [HSA_VAR:249v1] [HSA:249] [KO:K01077]
|
D10595 Asfotase alfa (USAN/INN) <JP/US>
|
NT5E (CD73) [HSA:4907] [KO:K19970]
|
D10963 Oleclumab (USAN/INN)
D12373 Quemliclustat (USAN/INN)
D12401 Uliledlimab (USAN/INN)
D13146 Mavrostobart (USAN/INN)
|
PPP2C [HSA:5515 5516] [KO:K04382]
|
D04262 Fostriecin sodium (USAN)
|
PPP3C/PPP3R/CHP [HSA:5530 5532 5533 5534 5535 11261 63928] [KO:K04348 K06268 K17610 K17611]
|
D08556 Tacrolimus (INN)
D00107 Tacrolimus (USP/INN) <JP/US>
D05480 Pimecrolimus (JAN/USAN/INN) <US>
D00184 Cyclosporine (USP) <JP/US>
D09033 Voclosporin (JAN/USAN/INN) <JP/US>
D10983 Ruclosporin (USAN/INN)
|
PPP4C [HSA:5531] [KO:K15423]
|
D04262 Fostriecin sodium (USAN)
|
PTPN1 [HSA:5770] [KO:K05696]
|
D04050 Ertiprotafib (USAN/INN)
D06252 Trodusquemine (USAN/INN)
|
PTPN11 [HSA:5781] [KO:K07293]
|
D12799 Vociprotafib (USAN/INN)
D12892 Migoprotafib (USAN/INN)
|
INPP5D (SHIP1) [HSA:3635] [KO:K03084]
|
D11275 Rosiptor (USAN/INN)
D11276 Rosiptor acetate (USAN)
|
Phosphodiesterases [EC:3.1.4.-]
|
SMPD1* [HSA_VAR:6609v1] [HSA:6609] [KO:K12350]
|
D10820 Olipudase alfa (USAN/INN) <JP/US>
|
PDE [HSA:10846 27115 50940 5136 5137 5138 5139 5140 5141 5142 5143 5144 5150 5151 5153 8622] [KO:K18438 K18436 K13298 K13755 K18283 K19021 K13296 K13293 K18437]
|
D07425 Papaverine (BAN)
D02218 Papaverine hydrochloride (JP18/USP) <JP>
D07439 Papaverine sulfate
D07089 Moxaverine (INN)
D08238 Moxaverine hydrochloride
D07546 Bucladesine (INN)
D01238 Bucladesine sodium (JAN) <JP>
D01220 Trapidil (JP18/INN) <JP>
D07961 Flavoxate (INN)
D00718 Flavoxate hydrochloride (JP18/USP) <JP/US>
D00691 Dyphylline (USP) <JP>
D02017 Oxtriphylline (USP)
D01771 Proxyphylline (JAN/INN)
D00371 Theophylline (JP18) <JP/US>
D01712 Theophylline sodium acetate (JAN)
D06103 Theophylline (USP)
D06104 Theophylline sodium glycinate (USP)
D00227 Aminophylline (USP/INN)
D05429 Aminophylline hydrate (JP18) <JP>
D11630 Aminophylline dihydrate <US>
D03075 Bemoradan (USAN/INN)
D04006 Enprofylline (USAN/INN)
D05278 Oxagrelate (USAN/INN)
D05612 Prinoxodan (USAN/INN)
D06132 Tibenelast sodium (USAN)
D09822 Theosalicin (JAN)
|
PDE [HSA:5153 5138 5139 5140 5141 5142 5143 5144 8654] [KO:K13755 K18283 K19021 K13296 K13293 K13762]
|
D00528 Caffeine (USP) <JP>
D01453 Caffeine hydrate (JP18) <JP>
D07603 Caffeine citrate (USP) <US>
|
PDE1 [HSA:5136 5153 5137] [KO:K13755]
|
D11883 Lenrispodun (USAN)
D11884 Lenrispodun phosphate (USAN)
|
PDE2A [HSA:5138] [KO:K18283]
|
D03898 Doxofylline (USAN/INN)
|
PDE3 [HSA:5139 5140] [KO:K19021 K13296]
|
D01896 Cilostazol (JP18/USP/INN) <JP/US>
D00231 Inamrinone (USP)
D02084 Inamrinone ethylenelactate
D00417 Milrinone (JAN/USP/INN) <JP>
D02085 Milrinone lactate <US>
D04004 Enoximone (USAN/INN)
D04720 Levosimendan (USAN/INN)
D07455 Anagrelide (INN/BAN)
D02933 Anagrelide hydrochloride (USP)
D10255 Anagrelide hydrochloride hydrate (JAN) <JP/US>
D11743 Ensifentrine (USAN/INN) <US>
D01385 Ibudilast (JP18/INN) <JP>
D01133 Pimobendan (JAN/USAN/INN) <JP>
D01198 Toborinone (JAN/USAN/INN)
D01690 Vesnarinone (JAN/USAN/INN)
D02042 Olprinone hydrochloride hydrate (JAN) <JP>
D04508 Imazodan hydrochloride (USAN)
D04529 Indolidan (USAN/INN)
D04628 Isomazole hydrochloride (USAN)
D04751 Lixazinone sulfate (USAN)
D05514 Piroximone (USAN)
D08294 Olprinone (INN)
D09843 Beradilol monoethyl maleate (JAN)
|
PDE4 [HSA:5141 5142 5143 5144] [KO:K13293]
|
D07088 Drotaverine (INN)
D07879 Drotaverine hydrochloride
D05744 Roflumilast (JAN/USAN/INN) <US>
D10873 Crisaborole (USAN/INN) <US>
D08860 Apremilast (JAN/USAN) <JP/US>
D01630 Propentofylline (JAN/INN)
D11743 Ensifentrine (USAN/INN) <US>
D01385 Ibudilast (JP18/INN) <JP>
D01704 Cilomilast (JAN/USAN/INN)
D01783 Rolipram (JAN/USAN/INN)
D02655 Etazolate hydrochloride (USAN)
D02985 Arofylline (USAN/INN)
D03516 Cipamfylline (USAN/INN)
D04185 Filaminast (USAN/INN)
D05474 Piclamilast (USAN/INN)
D09020 Tofimilast (INN/USAN)
D11305 Lotamilast (USAN/INN)
D11314 Difamilast (JAN/USAN) <JP>
D12397 Tranimilast (USAN/INN)
D12822 Idrebormilast (USAN)
|
PDE4A [HSA:5141] [KO:K13293]
|
D00302 Dipyridamole (JP18/USP/INN) <JP/US>
|
PDE4B [HSA:5142] [KO:K13293]
|
D12975 Nerandomilast (JAN/USAN/INN)
|
PDE4D [HSA:5144] [KO:K13293]
|
D12173 Zatolmilast (USAN)
|
PDE5 [HSA:8654] [KO:K13762]
|
D00302 Dipyridamole (JP18/USP/INN) <JP/US>
D08514 Sildenafil (INN)
D02229 Sildenafil citrate (JAN/USP) <JP/US>
D02008 Tadalafil (JAN/USP/INN) <JP/US>
D08668 Vardenafil (USAN/INN)
D02731 Vardenafil dihydrochoride (USAN)
D03260 Vardenafil hydrochloride hydrate (JAN) <JP/US>
D09989 Vardenafil hydrochloride (USP)
D03217 Avanafil (USAN/INN) <US>
D10027 Udenafil (USAN/INN)
D03657 Dasantafil (USAN/INN)
D09621 Gisadenafil (USAN/INN)
D09622 Gisadenafil besylate (USAN)
|
PDE9 [HSA:5152] [KO:K13761]
|
D12203 Tovinontrine (USAN/INN)
D13001 Edelinontrine (USAN/INN)
|
PDE10A [HSA:10846] [KO:K18438]
|
D11171 Mardepodect (USAN/INN)
D11245 Balipodect (USAN/INN)
D13073 Gemlapodect (USAN/INN)
|
ENPP2 (ATX) [HSA:5168] [KO:K01122]
|
D11844 Ziritaxestat (USAN/INN)
|
Sulfatases [EC:3.1.6.-]
|
STS [HSA:412] [KO:K01131]
|
D09915 Irosustat (USAN/INN)
|
GALNS* [HSA_VAR:2588v1] [HSA:2588] [KO:K01132]
|
D10333 Elosulfase alfa (USAN) <JP/US>
|
ARSA [HSA:410] [KO:K01134]
|
D12877 Atidarsagene autotemcel (USAN/INN) <US>
D12462 Cebsulfase alfa (USAN/INN)
|
ARSB* [HSA_VAR:411v1] [HSA:411] [KO:K01135]
|
D06565 Galsulfase (USAN/INN) <JP/US>
|
IDS* [HSA_VAR:3423v1] [HSA:3423] [KO:K01136]
|
D04499 Idursulfase (USAN/INN) <JP/US>
D11025 Idursulfase beta (INN) <JP>
D11812 Pabinafusp alfa (genetical recombination) (JAN) <JP>
D13242 Verenafusp alfa (INN)
D12806 Tividenofusp alfa (USAN/INN)
|
Glycosidases [EC:3.2.1.-]
|
AMY [HSA:279 280] [KO:K01176]
|
D00216 Acarbose (JAN/USAN/INN) <JP/US>
|
GAA [HSA:2548] [KO:K12316]
|
D00216 Acarbose (JAN/USAN/INN) <JP/US>
D00625 Miglitol (JP18/USAN/INN) <JP/US>
D01665 Voglibose (JP18/USAN/INN) <JP>
D09605 Duvoglustat (USAN/INN)
D09606 Duvoglustat hydrochloride (USAN)
D09779 Emiglitate (JAN/INN)
D11828 Clervonafusp alfa (USAN/INN)
|
GAA* [HSA_VAR:2548v1] [HSA:2548] [KO:K12316]
|
D03207 Alglucosidase alfa (USAN/INN) <JP/US>
D11744 Avalglucosidase alfa (USAN/INN) <JP/US>
D11798 Cipaglucosidase alfa (USAN) <JP/US>
|
GANC [HSA:2595] [KO:K12317]
|
D00216 Acarbose (JAN/USAN/INN) <JP/US>
D00625 Miglitol (JP18/USAN/INN) <JP/US>
D01665 Voglibose (JP18/USAN/INN) <JP>
D09779 Emiglitate (JAN/INN)
|
MGAM [HSA:8972] [KO:K12047]
|
D00216 Acarbose (JAN/USAN/INN) <JP/US>
D00625 Miglitol (JP18/USAN/INN) <JP/US>
D01665 Voglibose (JP18/USAN/INN) <JP>
D09779 Emiglitate (JAN/INN)
|
MAN2B1* [HSA_VAR:4125v1] [HSA:4125] [KO:K12311]
|
D11024 Velmanase alfa (USAN/INN) <US>
|
GUSB [HSA:2990] [KO:K01195]
|
D01805 Aceglatone (JAN/INN)
|
GUSB* [HSA_VAR:2990v1] [HSA:2990] [KO:K01195]
|
D11004 Vestronidase alfa (USAN/INN) <JP/US>
|
GLA* [HSA_VAR:2717v1] [HSA:2717] [KO:K01189]
|
D02784 Agalsidase alfa (USAN/INN) <JP>
D03228 Agalsidase beta (INN) <JP/US>
D11685 Pegunigalsidase alfa (USAN/INN) <US>
|
GLA* [HSA_VAR:2717v2] [HSA:2717] [KO:K01189]
|
D05031 Migalastat hydrochloride (JAN/USAN) <JP/US>
|
GBA* [HSA_VAR:2629v1] [HSA:2629] [KO:K01201]
|
D02810 Alglucerase (JAN/USAN/INN)
D03020 Imiglucerase (USAN/INN) <JP/US>
D09029 Velaglucerase alfa (USAN) <JP/US>
D09675 Taliglucerase alfa (USAN/INN) <US>
|
SI [HSA:6476] [KO:K01203]
|
D03342 Camiglibose (USAN)
|
SI* [HSA_VAR:6476v1] [HSA:6476] [KO:K01203]
|
D05782 Sacrosidase (USAN) <US>
|
NAGLU* [HSA_VAR:4669v1] [HSA:4669] [KO:K01205]
|
D11199 Lesinidase alfa (USAN/INN)
|
IDUA* [HSA_VAR:3425v1] [HSA:3425] [KO:K01217]
|
D04670 Laronidase (USAN) <JP/US>
|
HPSE [HSA:10855] [KO:K07964]
|
D11764 Necuparanib (USAN/INN)
D11765 Necuparanib sodium (USAN)
|
OGA [HSA:10724] [KO:K15719]
|
D12955 Ceperognastat (USAN)
|
ADP-ribosyl cyclase [EC:3.2.2.6]
|
CD38 [HSA:952] [KO:K01242]
|
D10777 Daratumumab (USAN) <JP/US>
D11050 Isatuximab (USAN/INN) <JP/US>
D12315 Ciltacabtagene autoleucel (USAN/INN) <US>
D11945 Mezagitamab (USAN/INN)
D12862 Noraramtide (USAN)
|
Glutaminase [EC:3.5.1.2]
|
GLS [HSA:2744] [KO:K01425]
|
D11738 Telaglenastat (USAN/INN)
D11739 Telaglenastat hydrochloride (USAN)
|
Histone deacetylase [EC:3.5.1.98]
|
HDAC [HSA:3065 3066 8841 9759 10014 10013 51564 55869 9734 83933 79885] [KO:K06067 K11404 K11406 K11407 K11408 K11405 K11409 K18671 K11418]
|
D06320 Vorinostat (JAN/USAN) <JP/US>
D06637 Romidepsin (JAN/USAN/INN) <JP/US>
D10319 Panobinostat (USAN/INN)
D10019 Panobinostat lactate (JAN)
D08870 Belinostat (USAN/INN) <US>
D09338 Entinostat (JAN/USAN/INN)
D13021 Resminostat (INN)
D12742 Givinostat (USAN/INN)
D12743 Givinostat hydrochloride (USAN) <US>
D10060 Abexinostat (USAN)
D10084 Abexinostat hydrochloride (USAN)
D10321 Quisinostat (USAN/INN)
D10322 Quisinostat hydrochloride (USAN)
D10977 Remetinostat (USAN/INN)
D12551 Bocodepsin (USAN)
D12552 Bocodepsin besylate (USAN)
|
HDAC1 [HSA:3065] [KO:K06067]
|
D10993 Tucidinostat (JAN/USAN/INN) <JP>
D05988 Tacedinaline (USAN/INN)
D09357 Mocetinostat dihydrobromide (USAN)
D09641 Mocetinostat (USAN/INN)
D11182 Tinostamustine (USAN/INN)
D11319 Fimepinostat (USAN/INN)
D11442 Nanatinostat (USAN)
|
HDAC2 [HSA:3066] [KO:K06067]
|
D10993 Tucidinostat (JAN/USAN/INN) <JP>
D09357 Mocetinostat dihydrobromide (USAN)
D09641 Mocetinostat (USAN/INN)
D11182 Tinostamustine (USAN/INN)
D11319 Fimepinostat (USAN/INN)
D11442 Nanatinostat (USAN)
|
HDAC3 [HSA:8841] [KO:K11404]
|
D10993 Tucidinostat (JAN/USAN/INN) <JP>
D09357 Mocetinostat dihydrobromide (USAN)
D09641 Mocetinostat (USAN/INN)
D11182 Tinostamustine (USAN/INN)
D11319 Fimepinostat (USAN/INN)
D11442 Nanatinostat (USAN)
|
HDAC4 [HSA:9759] [KO:K11406]
|
D11319 Fimepinostat (USAN/INN)
|
HDAC5 [HSA:10014] [KO:K11406]
|
D11319 Fimepinostat (USAN/INN)
|
HDAC6 [HSA:10013] [KO:K11407]
|
D10661 Ricolinostat (USAN/INN)
D10918 Citarinostat (USAN/INN)
D11182 Tinostamustine (USAN/INN)
D11319 Fimepinostat (USAN/INN)
|
HDAC7 [HSA:51564] [KO:K11408]
|
D11319 Fimepinostat (USAN/INN)
|
HDAC8 [HSA:55869] [KO:K11405]
|
D09357 Mocetinostat dihydrobromide (USAN)
D09641 Mocetinostat (USAN/INN)
D11319 Fimepinostat (USAN/INN)
D11442 Nanatinostat (USAN)
|
HDAC9 [HSA:9734] [KO:K11409]
|
D11319 Fimepinostat (USAN/INN)
|
HDAC10 [HSA:83933] [KO:K18671]
|
D10993 Tucidinostat (JAN/USAN/INN) <JP>
D11319 Fimepinostat (USAN/INN)
|
HDAC11 [HSA:79885] [KO:K11418]
|
D09357 Mocetinostat dihydrobromide (USAN)
D09641 Mocetinostat (USAN/INN)
|
Fatty acid amide hydrolase [EC:3.5.1.99]
|
FAAH [HSA:2166] [KO:K15528]
|
D13114 Irafamdastat (USAN)
|
Arginase [EC:3.5.3.1]
|
ARG1 [HSA:383] [KO:K01476]
|
D11792 Numidargistat (USAN/INN)
|
ARG1* [HSA_VAR:383v1] [HSA:383] [KO:K01476]
|
D11695 Pegzilarginase (USAN/INN)
|
Adenosine deaminase [EC:3.5.4.4]
|
ADA [HSA:100] [KO:K01488]
|
D00155 Pentostatin (JAN/USAN/INN) <US>
|
ADA* [HSA_VAR:100v1] [HSA:100] [KO:K01488]
|
D11017 Elapegademase (USAN/INN) <JP/US>
|
Cytidine deaminase [EC:3.5.4.5]
|
CDA [HSA:978] [KO:K01489]
|
D11679 Cedazuridine (USAN/INN)
|
ATPase [EC:3.6.3.-]
|
ATP1A [HSA:476 477 478 480] [KO:K01539]
|
D06881 Acetyldigitoxin (INN)
D07555 Acetyldigoxin
D00297 Digitoxin (JAN/USP/INN)
D00298 Digoxin (JP18/USP) <JP/US>
D01972 Lanatoside C (JAN/INN)
D01240 Deslanoside (JP18/USP/INN) <JP>
D09847 Metildigoxin (INN)
D02587 Metildigoxin (JP18) <JP>
D07147 Gitoformate (INN)
D01379 Proscillaridin (JAN/USAN/INN)
D00112 G-Strophanthin (JAN)
D00645 Bretylium tosylate (USP)
D07520 Bepridil (INN)
D00631 Bepridil hydrochloride (USAN) <JP>
D07556 beta-Acetyldigoxin
|
ATP2A [HSA:487 488 489] [KO:K05853]
|
D10715 Mipsagargin (USAN/INN)
|
ATP4 [HSA:495 496] [KO:K01542 K01543]
|
D00455 Omeprazole (JP18/USP/INN) <JP/US>
D01207 Omeprazole sodium (USAN)
D05261 Omeprazole sodium injection (JAN) <JP>
D05259 Omeprazole magnesium (USP) <US>
D05353 Pantoprazole (USAN/INN)
D02593 Pantoprazole sodium (USP) <US>
D00355 Lansoprazole (JP18/USP/INN) <JP/US>
D08463 Rabeprazole (INN)
D00724 Rabeprazole sodium (JP18/USP) <JP/US>
D07917 Esomeprazole (INN)
D01984 Esomeprazole magnesium (USP) <JP/US>
D04056 Esomeprazole sodium (USAN) <US>
D09339 Esomeprazole potassium (USAN)
D10120 Esomeprazole strontium (USAN) <US>
D11114 Esomeprazole magnesium dihydrate <US>
D08903 Dexlansoprazole (INN/USAN) <US>
D12816 Dexlansoprazole sesquihydrate <US>
D11784 Vonoprazan (USAN/INN)
D10466 Vonoprazan fumarate (JAN/USAN) <JP/US>
D12246 Tegoprazan (INN)
D13012 Fexuprazan (INN)
D13013 Ilaprazole (INN)
D13240 Zastaprazan (INN)
D01920 Tenatoprazole (JAN/INN)
D05722 Revaprazan hydrochloride (USAN)
D05900 Timoprazole (INN)
D05901 Picoprazole (INN)
D05906 Leminoprazole (INN)
D09837 Penaprazole sodium hydrate (JAN)
D13197 Linaprazan glurate (USAN/INN)
D13198 Linaprazan glurate hydrochloride (USAN)
|
Lyases (EC4)
|
Carboxy-lyases [EC:4.1.1.-]
|
GAD [HSA:2571 2572] [KO:K01580]
|
D00399 Valproic acid (USP) <US>
D00304 Divalproex sodium (USP) <US>
D00710 Valproate sodium (USAN) <JP/US>
D08667 Calcium valproate
|
ODC1 [HSA:4953] [KO:K01581]
|
D07883 Eflornithine (INN)
D00829 Eflornithine hydrochloride (USAN) <US>
|
HDC [HSA:3067] [KO:K01590]
|
D07405 Tritoqualine (INN)
D03158 Brocresine (USAN/INN)
|
DDC [HSA:1644] [KO:K01593]
|
D00558 Carbidopa (USP) <US>
D01653 Benserazide hydrochloride (JP18)
D03082 Benserazide (USAN/INN)
D04997 Methyldopate hydrochloride (USP)
|
DDC* [HSA_VAR:1644v1] [HSA:1644] [KO:K01593]
|
D12407 Eladocagene exuparvovec (USAN/INN) <US>
|
AMD1 [HSA:262] [KO:K01611]
|
D07258 Mitoguazone (INN)
|
GGCX [HSA:2677] [KO:K10106]
|
D07457 Anisindione (INN)
|
Aldehyde-lyases [EC:4.1.2.-]
|
CA [HSA:759 760 761 762 763 11238 765 766 767 768 771 377677 23632] [KO:K01672 K18245 K18246]
|
D01822 Clofenamide (JAN/INN)
D00218 Acetazolamide (JP18/USP/INN) <JP/US>
D01196 Acetazolamide sodium (JAN) <JP/US>
D00518 Dichlorphenamide (USP) <US>
D07871 Dorzolamide (INN)
D00653 Dorzolamide hydrochloride (JP18/USP) <JP/US>
D00655 Methazolamide (JAN/USP/INN) <US>
D02441 Ethoxzolamide
D03845 Sezolamide hydrochloride (USAN)
|
CA2 [HSA:760] [KO:K18245]
|
D00537 Topiramate (JAN/USP/INN) <JP/US>
D00652 Brinzolamide (JAN/USP/INN) <JP/US>
|
CA4 [HSA:762] [KO:K18246]
|
D00537 Topiramate (JAN/USP/INN) <JP/US>
|
CA9 [HSA:768] [KO:K01672]
|
D09593 Girentuximab (USAN/INN)
D09632 Iodine I 124 girentuximab (USAN/INN)
|
Hydro-lyases [EC:4.2.1.-]
|
CBS [HSA:875] [KO:K01697]
|
D12197 Pegtibatinase (USAN)
|
Phosphorus-oxygen lyases [EC:4.6.1.-]
|
ADCY [HSA:107 108 109 196883 111 112 113 114 115 55811] [KO:K08041 K08042 K08043 K08044 K08045 K08046 K08047 K08048 K08049 K11265]
|
D01697 Colforsin daropate hydrochloride (JAN) <JP>
D03584 Colforsin (USAN/INN)
|
GUCY1A [HSA:2977 2982] [KO:K12318]
|
D01810 Nicorandil (JP18/USAN/INN) <JP>
D11051 Vericiguat (JAN/USAN/INN) <JP/US>
D09572 Riociguat (JAN/USAN/INN) <JP/US>
D00517 Amyl nitrite (JP18/USP) <JP>
D07577 Cinaciguat (JAN/INN)
D11274 Praliciguat (USAN/INN)
D11475 Olinciguat (USAN/INN)
D12516 Zagociguat (USAN/INN)
D13034 Avenciguat (USAN/INN)
|
GUCY1B [HSA:2983] [KO:K12319]
|
D01810 Nicorandil (JP18/USAN/INN) <JP>
D11051 Vericiguat (JAN/USAN/INN) <JP/US>
D09572 Riociguat (JAN/USAN/INN) <JP/US>
D00517 Amyl nitrite (JP18/USP) <JP>
D07577 Cinaciguat (JAN/INN)
D11274 Praliciguat (USAN/INN)
D11475 Olinciguat (USAN/INN)
D12516 Zagociguat (USAN/INN)
D13034 Avenciguat (USAN/INN)
|
GUCY2C [HSA:2984] [KO:K12320]
|
D09355 Linaclotide (JAN/USAN) <JP/US>
D06612 Linaclotide acetate (USAN)
D09948 Plecanatide (USAN/INN) <US>
D10976 Recanaclotide (USAN/INN)
D11233 Dolcanatide (USAN/INN)
|
Moco biosynthesis enzyme [EC:4.1.99.2 4.6.1.17]
|
MOCS1* [HSA_VAR:4337v1] [HSA:4337] [KO:K20967]
|
D11779 Fosdenopterin (USAN)
D11780 Fosdenopterin hydrobromide (USAN) <US>
|
Isomerases (EC5)
|
Peptidylprolyl isomerase [EC:5.2.1.8]
|
PPIA [HSA:5478] [KO:K03767]
|
D10087 Alisporivir (USAN)
|
Prostaglandin-E synthase [EC:5.3.99.3]
|
PTGES [HSA:9536] [KO:K15729]
|
D01545 Aceclofenac (JAN/INN)
|
Thromboxane-A synthase [EC:5.3.99.5]
|
TBXAS1 (CYP5A1) [HSA:6916] [KO:K01832]
|
D07140 Picotamide (BAN)
D01220 Trapidil (JP18/INN) <JP>
D01683 Ozagrel hydrochloride hydrate (JAN) <JP>
D01684 Ozagrel sodium (JP18) <JP>
D03661 Dazmegrel (USAN/INN)
D03663 Dazoxiben hydrochloride (USAN)
D04276 Furegrelate sodium (USAN)
D05502 Pirmagrel (USAN/INN)
D05727 Ridogrel (USAN/INN)
D06077 Terbogrel (USAN/INN)
D08327 Ozagrel (INN)
|
DNA topoisomerase [EC:5.99.1.-]
|
TOP1 [HSA:7150] [KO:K03163]
|
D08618 Topotecan (BAN)
D02168 Topotecan hydrochloride (USAN) <JP/US>
D08086 Irinotecan (INN)
D01061 Irinotecan hydrochloride (USP) <JP/US>
D10642 Irinotecan sucrosofate (USAN)
D10367 Etirinotecan pegol (USAN/INN)
D10422 Etirinotecan pegol tetrahydrochloride (USAN)
D10427 Etirinotecan pegol tetratriflutate (USAN)
D03225 Belotecan hydrochloride (USAN)
D02756 Aclarubicin (USAN/INN)
D01911 Aclarubicin hydrochloride (JP18) <JP>
D11529 Trastuzumab deruxtecan (USAN/INN) <JP/US>
D10985 Sacituzumab govitecan (USAN/INN) <JP/US>
D12359 Datopotamab deruxtecan (USAN/INN) <JP/US>
D12184 Patritumab deruxtecan (USAN/INN)
D12753 Ifinatamab deruxtecan (USAN/INN)
D01432 Exatecan mesylate (USAN)
D03954 Edotecarin (USAN/INN)
D03977 Elsamitrucin (USAN/INN)
D04031 Rubitecan (USAN/INN)
D04822 Lurtotecan dihydrochloride (USAN)
D05385 Pegamotecan (USAN)
D09327 Cositecan (USAN)
D09679 Tenifatecan (USAN/INN)
D10464 Firtecan pegol (USAN/INN)
D12919 Samrotecan (USAN/INN)
D12927 Puxitatug samrotecan (USAN/INN)
D12977 Pamirtecan (USAN)
D12978 Trastuzumab pamirtecan (USAN)
D13047 Brengitecan (USAN)
D13053 Izalontamab brengitecan (USAN/INN)
D13067 Tilatamig samrotecan (USAN/INN)
D13069 Raludotatug deruxtecan (USAN/INN)
D13150 Tocentecan (USAN/INN)
D13202 Precemtabart tocentecan (USAN/INN)
|
TOP2 [HSA:7153 7155] [KO:K03164]
|
D00125 Etoposide (JP18/USP/INN) <JP/US>
D04107 Etoposide phosphate (USAN) <US>
D02698 Teniposide (USP/INN)
D03899 Doxorubicin (USAN/INN)
D01275 Doxorubicin hydrochloride (JP18/USP) <JP/US>
D07776 Daunorubicin (INN)
D01264 Daunorubicin hydrochloride (JP18/USP) <JP/US>
D10787 Daunorubicin citrate
D07901 Epirubicin (INN)
D02214 Epirubicin hydrochloride (JP18/USP) <JP/US>
D02756 Aclarubicin (USAN/INN)
D01911 Aclarubicin hydrochloride (JP18) <JP>
D06386 Zorubicin hydrochloride (USAN)
D08062 Idarubicin (INN)
D01747 Idarubicin hydrochloride (JP18/USP) <JP/US>
D08224 Mitoxantrone (INN)
D02166 Mitoxantrone hydrochloride (JAN/USP) <JP/US>
D01885 Pirarubicin (JP18/INN)
D08386 Pirarubicin hydrochloride <JP>
D02697 Valrubicin (USP/INN) <US>
D08854 Amrubicin (USAN/INN)
D07100 Amrubicin hydrochloride (JAN/USAN) <JP>
D05522 Pixantrone (USAN/INN)
D09654 Pixantrone dimaleate (USAN)
D02321 Amsacrine (USAN/INN)
D08024 Vosaroxin (USAN)
D03730 Dexrazoxane (JAN/USAN/INN) <JP/US>
D07807 Dexrazoxane hydrochloride <US>
D01404 Sobuzoxane (JAN) <JP>
D03220 Becatecarin (USAN/INN)
D03602 Crisnatol mesylate (USAN)
D03977 Elsamitrucin (USAN/INN)
D04262 Fostriecin sodium (USAN)
D04498 Idronoxil (USAN/INN)
D04685 Ledoxantrone trihydrochloride (USAN)
D04783 Losoxantrone hydrochloride (USAN)
D04914 Menogaril (USAN/INN)
D05054 Mitindomide (USAN/INN)
D05510 Piroxantrone hydrochloride (USAN)
D06059 Teloxantrone hydrochloride (USAN)
D06167 Tirapazamine (USAN/INN)
D06190 Topixantrone (USAN/INN)
D08871 Berubicin hydrochloride (USAN)
D08981 Quarfloxin (USAN)
D10090 Amonafide (USAN)
D10091 Amonafide l-malate (USAN)
D10383 Aldoxorubicin (USAN/INN)
D10384 Aldoxorubicin Hydrochloride (USAN)
D12844 Naxtarubicin (USAN)
|
Ligases (EC6)
|
Aminoacyl tRNA synthase [EC:6.1.1.-]
|
EPRS1 [HSA:2058] [KO:K14163]
|
D12794 Bersiporocin (USAN/INN)
D12795 Bersiporocin hydrochloride (USAN)
|
HARS [HSA:23438 3035] [KO:K01892]
|
D12612 Efzofitimod (INN)
|
Ubiquitin activating enzyme [EC:6.2.1.45]
|
UBLE1 [HSA:10055 10054] [KO:K10684 K10685]
|
D12268 Subasumstat (USAN/INN)
|
GART [EC:6.3.4.13 2.1.2.2 6.3.3.1]
|
GART [HSA:2618] [KO:K11787]
|
D07472 Pemetrexed (INN) <US>
D03828 Pemetrexed disodium (USAN) <US>
D06503 Pemetrexed sodium hydrate (JAN) <JP/US>
D10596 Pemetrexed sodium hemipentahydrate (JAN) <JP/US>
D11352 Pemetrexed tromethamine (USAN)
D13147 Pemetrexed dipotassium heptahydrate <US>
D04766 Lometrexol sodium (USAN)
D05400 Pelitrexol (USAN/INN)
|
Carbamoyl-phosphate synthase [EC:6.3.4.16]
|
CPS1 [HSA:1373] [KO:K01948]
|
D07130 Carglumic acid (JAN/USAN/INN) <JP/US>
|
Acetyl-CoA carboxylase [EC:6.4.1.2]
|
ACACA [HSA:31] [KO:K11262]
|
D11186 Olumacostat glasaretil (USAN/INN)
D11640 Firsocostat (USAN/INN)
D11902 Clesacostat (USAN)
D11903 Clesacostat tromethamine (USAN)
|
ACACB [HSA:32] [KO:K01946]
|
D11186 Olumacostat glasaretil (USAN/INN)
D11640 Firsocostat (USAN/INN)
D11902 Clesacostat (USAN)
D11903 Clesacostat tromethamine (USAN)
|
|
Nucleic acids
|
RNAs
|
MicroRNAs
|
MIR155 [HSA:406947] [KO:K17009]
|
D11163 Cobomarsen (USAN/INN)
D11164 Cobomarsen sodium (USAN)
|
|
Not elsewhere classified
|
Genetic information processing
|
Transcription factor
|
NFE2L2 [HSA:4780] [KO:K05638]
|
D10964 Omaveloxolone (USAN/INN) <US>
|
AHR [HSA:196] [KO:K09093]
|
D11365 Tapinarof (JAN/USAN) <JP/US>
|
HIF1A [HSA:3091] [KO:K08268]
|
D10464 Firtecan pegol (USAN/INN)
|
HIF2A (EPAS1) [HSA:2034] [KO:K09095]
|
D11954 Belzutifan (JAN/USAN/INN) <JP/US>
D13003 Imdatifan (USAN/INN)
|
MYC [HSA:4609] [KO:K04377]
|
D08956 Omacetaxine mepesuccinate (USAN)
|
SP1 [HSA:6667] [KO:K04684]
|
D09014 Terameprocol (INN/USAN)
|
EGR1 [HSA:1958] [KO:K09203]
|
D11286 Brivoligide sodium (USAN)
D11341 Brivoligide (USAN)
|
WT1 (WT33) [HSA:7490] [KO:K09234]
|
D11057 Adegrapepimut-S (USAN)
D11058 Adegramotide acetate (JAN)
D11059 Elatipepimut-S (USAN)
D11060 Nelatimotide trifluoroacetate (JAN)
|
NANOG [HSA:79923] [KO:K10164]
|
D10903 Amcasertib (USAN/INN)
|
NFKB1 [HSA:4790] [KO:K02580]
|
D01146 Iguratimod (JAN/INN) <JP>
D12932 Bezisterim (USAN/INN)
|
STAT3 [HSA:6774] [KO:K04692]
|
D10717 Napabucasin (JAN/USAN/INN)
|
TP53 (p53) [HSA:7157] [KO:K04451]
|
D08887 Cenersen sodium (USAN)
|
TP53* (p53) [HSA_VAR:7157v1] [HSA:7157] [KO:K04451]
|
D12982 Rezatapopt (USAN/INN)
|
RELA (NKFB3, p65) [HSA:5970] [KO:K04735]
|
D12181 Edasalonexent (USAN/INN)
|
IKZF1/3 [HSA:10320 22806] [KO:K09220]
|
D12858 Zelebrudomide (USAN)
|
Translation factor
|
EIF2B [HSA:1967 8892 8891 8890 8893] [KO:K03239 K03754 K03241 K03680 K03240]
|
D13118 Fosigotifator (USAN/INN)
D13119 Fosigotifator sodium tromethamine (USAN)
|
EIF2S2 [HSA:8894] [KO:K03238]
|
D13104 Comtifator (USAN)
|
EIF4A3 [HSA:9775] [KO:K13025]
|
D11837 Zotatifin (USAN/INN)
|
EIF4E [HSA:1977] [KO:K03259]
|
D10614 Briciclib (USAN/INN)
D10694 Briciclib sodium (USAN)
|
Chaperone and folding catalyst
|
HSP90 [HSA:3320 3326 7184] [KO:K04079 K09487]
|
D06554 Alvespimycin hydrochloride (USAN)
D06650 Tanespimycin (USAN)
D09375 Retaspimycin (USAN/INN)
D09376 Retaspimycin hydrochloride (USAN)
D10126 Ganetespib (USAN)
D10646 Luminespib (USAN/INN)
D10647 Luminespib mesylate (USAN)
D10719 Onalespib (USAN/INN)
D11766 Onalespib lactate (USAN)
D11920 Pimitespib (JAN) <JP>
|
HSP90B1 (GP96) [HSA:7184] [KO:K09487]
|
D06667 Vitespen (USAN)
|
CLU [HSA:1191] [KO:K17252]
|
D09403 Custirsen sodium (USAN)
|
APCS (SAP) [HSA:325] [KO:K23267]
|
D11464 Miridesap (USAN/INN)
D11471 Dezamizumab (USAN/INN)
D12402 Zinpentraxin alfa (USAN/INN)
|
Spliceosome
|
NCBP [HSA:4686 22916 392517] [KO:K12882 K12883]
|
D12345 Obefazimod (USAN)
|
SMN1 [HSA:6606] [KO:K13129]
|
D11559 Onasemnogene abeparvovec (USAN/INN) <US>
|
SMN2 [HSA:6607] [KO:K13129]
|
D10881 Nusinersen (USAN/INN)
D10791 Nusinersen sodium (JAN) <JP/US>
D11406 Risdiplam (JAN/USAN/INN) <JP/US>
D12272 Branaplam (USAN/INN)
D12273 Branaplam hydrochloride (USAN)
|
Environmental information processing
|
G protein
|
RAC1 [HSA:5879] [KO:K04392]
|
D11032 Plitidepsin (INN)
|
KRAS [HSA:3845] [KO:K07827]
|
D12639 Divarasib (USAN/INN)
D12640 Divarasib adipate (USAN)
D12853 Olomorasib (USAN)
|
KRAS* [HSA_VAR:3845v1] [HSA:3845] [KO:K07827]
|
D12055 Sotorasib (JAN/USAN) <JP/US>
D12301 Adagrasib (USAN/INN) <US>
D13038 Opnurasib (USAN/INN)
|
Signaling adaptor
|
ARRB [HSA:408 409] [KO:K04439]
|
D11214 Oliceridine (USAN/INN) <US>
|
GRB2 [HSA:2885] [KO:K04364]
|
D11165 Prexigebersen (USAN/INN)
|
mTOR signaling
|
CASTOR [HSA:652968 729438] [KO:K23080 K23081]
|
D11183 Sapanisertib (USAN/INN)
|
Wnt signaling
|
SOST [HSA:50964] [KO:K16834]
|
D10156 Romosozumab (USAN) <JP/US>
D10094 Blosozumab (USAN)
D13105 Setrusumab (USAN/INN)
|
RSPO3 [HSA:84870] [KO:K23098]
|
D11369 Rosmantuzumab (USAN)
|
CTNNB1 [HSA:1499] [KO:K02105]
|
D12445 Foscenvivint (JAN/INN)
|
SFRP4 [HSA:6424] [KO:K02185]
|
D13162 Remigromig (USAN)
|
Notch signaling
|
NOTCH1 [HSA:4851] [KO:K02599]
|
D11151 Crenigacestat (USAN/INN)
D11229 Brontictuzumab (USAN/INN)
|
NOTCH2 [HSA:4853] [KO:K20994]
|
D11775 Tarextumab (USAN/INN)
|
NOTCH3 [HSA:4854] [KO:K20995]
|
D11775 Tarextumab (USAN/INN)
|
DLL3 [HSA:10683] [KO:K06051]
|
D12234 Tarlatamab (USAN) <JP/US>
D10981 Rovalpituzumab tesirine (USAN/INN)
D11117 Rovalpituzumab (USAN)
D13161 Peluntamig (USAN/INN)
|
DLL4 [HSA:54567] [KO:K06051]
|
D10353 Demcizumab (USAN/INN)
D10460 Enoticumab (USAN/INN)
D11126 Navicixizumab (USAN/INN)
D11642 Dilpacimab (USAN/INN)
|
TGF-beta signaling
|
SMAD7 [HSA:4092] [KO:K19631]
|
D10955 Mongersen sodium (USAN)
D10956 Mongersen (INN)
|
LRRC32 [HSA:2615] [KO:K26316]
|
D12793 Livmoniplimab (USAN/INN)
|
Calcium signaling
|
CALM [HSA:801 805 808 810 91860 51806 163688] [KO:K02183]
|
D04789 Lubeluzole (USAN/INN)
|
Cellular process
|
Cell cycle
|
CCND1 [HSA:595] [KO:K04503]
|
D08956 Omacetaxine mepesuccinate (USAN)
|
Apoptosis
|
BCL2 [HSA:596] [KO:K02161]
|
D08290 Oblimersen (INN)
D05216 Oblimersen sodium (USAN)
D08954 Obatoclax mesylate (USAN)
D12883 Sonrotoclax (USAN/INN)
D13082 Surzetoclax (USAN/INN)
|
BCL2* [HSA_VAR:596v1] [HSA:596] [KO:K02161]
|
D10679 Venetoclax (JAN/USAN/INN) <JP/US>
|
BCL2L [HSA:598 599 4170 597] [KO:K04570 K02163 K02539 K02162]
|
D09935 Navitoclax (JAN/USAN/INN)
D09936 Navitoclax dihydrochloride (USAN)
|
MCL1 [HSA:4170] [KO:K02539]
|
D08956 Omacetaxine mepesuccinate (USAN)
D11962 Murizatoclax (USAN/INN)
D11963 Tapotoclax (USAN/INN)
D13131 Zamzetoclax (USAN/INN)
|
Membrane trafficking
|
GPNMB [HSA:10457] [KO:K20732]
|
D09623 Glembatumumab (USAN/INN)
D09912 Glembatumumab vedotin (USAN)
|
MSLN [HSA:10232] [KO:K20733]
|
D09767 Amatuximab (USAN)
|
RTN4 [HSA:57142] [KO:K20720]
|
D10331 Ozanezumab (USAN/INN)
|
SNCA [HSA:6622] [KO:K04528]
|
D11420 Prasinezumab (USAN/INN)
D11467 Cinpanemab (USAN)
D12796 Minzasolmin (USAN/INN)
D12965 Indenebart (USAN/INN)
D13126 Amlenetug (USAN/INN)
|
LINGO1 [HSA:84894] [KO:K23533]
|
D11767 Opicinumab (USAN/INN)
|
SORT1 [HSA:6272] [KO:K12388]
|
D12427 Latozinemab (USAN/INN)
D12580 Sudotaxel zendusortide (USAN/INN)
D12581 Zendusortide (USAN/INN)
D13210 Nivisnebart (USAN/INN)
|
PMEL (gp100) [HSA:6490] [KO:K17304]
|
D12296 Tebentafusp (USAN/INN) <US>
|
Cytoskeleton
|
MYL2 [HSA:4633] [KO:K10351]
|
D12253 Aficamten (USAN/INN)
D12949 Delocamten (USAN)
|
MYL3 [HSA:4634] [KO:K12749]
|
D12253 Aficamten (USAN/INN)
D12949 Delocamten (USAN)
|
MYL4 [HSA:4635] [KO:K12750]
|
D12253 Aficamten (USAN/INN)
D12949 Delocamten (USAN)
|
MYH [HSA:4619 4620 4621 4622 57644 4626 8735 22989] [KO:K24220]
|
D12902 Sevasemten (USAN/INN)
|
MYH6_7 [HSA:4624 4625] [KO:K17751]
|
D04510 Imciromab pentetate (USAN)
D12253 Aficamten (USAN/INN)
D12949 Delocamten (USAN)
|
MYH7 [HSA:4625] [KO:K17751]
|
D12265 Mavacamten (JAN/USAN/INN) <JP/US>
|
TNNC1 [HSA:7134] [KO:K05865]
|
D12804 Nelutroctiv (USAN/INN)
|
TNNC2 [HSA:7125] [KO:K12042]
|
D11363 Reldesemtiv (USAN)
|
TNNI2 [HSA:7136] [KO:K12043]
|
D11363 Reldesemtiv (USAN)
|
TNNI3 [HSA:7137] [KO:K12044]
|
D12804 Nelutroctiv (USAN/INN)
|
TNNT2 [HSA:7139] [KO:K12045]
|
D12804 Nelutroctiv (USAN/INN)
|
TNNT3 [HSA:7140] [KO:K12046]
|
D11363 Reldesemtiv (USAN)
|
DMD [HSA:1756] [KO:K10366]
|
D10114 Drisapersen (USAN)
D10115 Drisapersen sodium (JAN/USAN)
D11918 Renadirsen sodium (JAN)
D12966 Brogidirsen (JAN/USAN/INN)
|
DMD* [HSA_VAR:1756v1] [HSA:1756] [KO:K10366]
|
D09900 Eteplirsen (USAN/INN) <US>
D11707 Golodirsen (USAN/INN) <US>
D11528 Viltolarsen (JAN/USAN) <JP/US>
D11988 Casimersen (USAN/INN) <US>
D12633 Delandistrogene moxeparvovec (USAN/INN) <US>
|
TUBB [HSA:10381 10382 10383 203068 347688 347733 7280 81027 84617] [KO:K07375]
|
D11691 Tirbanibulin (JAN/USAN/INN) <US>
D11692 Tirbanibulin mesylate (USAN)
D08675 Vinblastine (INN)
D01068 Vinblastine sulfate (JP18/USP) <JP/US>
D08679 Vincristine (INN)
D02197 Vincristine sulfate (JP18/USP) <JP/US>
D06304 Vindesine (USAN/INN)
D01769 Vindesine sulfate (JAN/USAN) <JP>
D08680 Vinorelbine (INN)
D01935 Vinorelbine tartrate (USP) <JP/US>
D09032 Vinflunine ditartrate (USAN)
D00491 Paclitaxel (JAN/USP/INN) <JP/US>
D07866 Docetaxel (JAN/INN) <JP/US>
D02165 Docetaxel (USP) <JP/US>
D05333 Paclitaxel poliglumex (USAN/INN)
D09755 Cabazitaxel (USAN/INN)
D10452 Cabazitaxel acetonate (JAN) <JP/US>
D04645 Ixabepilone (JAN/USAN/INN) <US>
D09980 Trastuzumab emtansine (USAN/INN) <JP/US>
D09587 Brentuximab vedotin (USAN/INN) <JP/US>
D11525 Enfortumab vedotin (USAN) <JP/US>
D11595 Belantamab mafodotin (USAN) <JP>
D11814 Tisotumab vedotin (USAN/INN) <JP/US>
D10954 Mirvetuximab soravtansine (USAN/INN) <US>
D04066 Estramustine (USAN/INN)
D02398 Estramustine phosphate sodium (USAN)
D06397 Estramustine phosphate sodium hydrate (JAN) <JP>
D08914 Eribulin mesylate (USAN) <JP/US>
D00570 Colchicine (JP18/USP) <JP/US>
D01919 Soblidotin (JAN/INN)
D03059 Batabulin sodium (USAN)
D03364 Cantuzumab mertansine (USAN)
D04864 Maytansine (USAN)
D05062 Mivobulin isethionate (USAN)
D06001 Taltobulin (USAN/INN)
D06009 Tasidotin hydrochloride (USAN)
D06305 Vinepidine sulfate (USAN)
D06306 Vinglycinate sulfate (USAN)
D06307 Vinleurosine sulfate (USAN)
D06308 Vinrosidine sulfate (USAN)
D06309 Vinzolidine sulfate (USAN)
D06560 Batabulin (USAN/INN)
D06576 Cevipabulin fumarate (USAN)
D08889 Cevipabulin succinate (USAN)
D09691 Vedotin (USAN)
D09912 Glembatumumab vedotin (USAN)
D09927 Lorvotuzumab mertansine (USAN/INN)
D10013 Indibulin (USAN/INN)
D10029 Verubulin (USAN/INN)
D10030 Verubulin hydrochloride (USAN)
D10073 Lexibulin (USAN)
D10454 Cantuzumab ravtansine (USAN/INN)
D11228 Soravtansine (USAN)
D11232 Denintuzumab mafodotin (USAN/INN)
D11238 Lifastuzumab vedotin (USAN/INN)
D11494 Lisavanbulin (USAN/INN)
D11681 Avanbulin (USAN/INN)
D12183 Farletuzumab ecteribulin (USAN)
D12210 Ozuriftmab vedotin (USAN)
D12220 Mecbotamab vedotin
D12310 Tusamitamab ravtansine (USAN/INN)
D12519 Sabizabulin (USAN/INN)
D12520 Sabizabulin hydrochloride (USAN)
D12582 Opadotin (USAN)
D12583 Anvatabart opadotin (USAN/INN)
D12916 Oberotatug ravtansine (USAN/INN)
D12989 Disitamab vedotin (USAN/INN)
D13007 Sigvotatug vedotin (USAN/INN)
D13164 Sonesitatug vedotin (USAN/INN)
|
KIF11 [HSA:3832] [KO:K10398]
|
D04640 Ispinesib mesylate (USAN)
D09636 Litronesib (USAN/INN)
|
MAPT (TAU) [HSA:4137] [KO:K04380]
|
D11427 Hydromethylthionine (USAN/INN)
D11384 Hydromethylthionine mesylate (USAN)
D11210 Flortaucipir F 18 (USAN) <JP/US>
D11293 Gosuranemab (USAN)
D11533 Zagotenemab (USAN)
D11687 Semorinemab (USAN/INN)
D11840 Tilavonemab (USAN/INN)
D12228 Bepranemab (USAN/INN)
D12636 Posdinemab (USAN/INN)
D12848 Etalanetug (USAN)
|
FLNA [HSA:2316] [KO:K04437]
|
D12003 Simufilam (USAN)
D12004 Simufilam hydrochloride (USAN)
|
Ubiquitin system
|
NAE1 [HSA:8883] [KO:K04532]
|
D10413 Pevonedistat (USAN/INN)
D10654 Pevonedistat hydrochloride (JAN/USAN)
|
KEAP1 [HSA:9817] [KO:K10456]
|
D03846 Dimethyl fumarate (JAN/USAN) <JP/US>
|
DIABLO (SMAC) [HSA:56616] [KO:K10522]
|
D12565 Xevinapant (JAN/USAN/INN)
|
CRBN [HSA:51185] [KO:K11793]
|
D12000 Mezigdomide (JAN/USAN)
D12324 Golcadomide (USAN/INN)
D12832 Golcadomide hydrochloride (JAN/USAN)
D12933 Cemisidomide (USAN/INN)
|
RAD51 [HSA:5888] [KO:K04482]
|
D12558 Emzadirib (USAN)
|
Chromatin
|
BMI1 [HSA:648] [KO:K11459]
|
D11889 Unesblin (USAN)
|
MEN1 [HSA:4221] [KO:K14970]
|
D12728 Revumenib (USAN/INN)
D12729 Revumenib citrate (USAN) <US>
D12419 Ziftomenib (USAN/INN) <US>
D12727 Icovamenib (USAN)
D13193 Enzomenib (USAN/INN)
D13194 Enzomenib tartrate (USAN)
|
EED [HSA:8726] [KO:K11462]
|
D12782 Pociredir (USAN/INN)
|
Cilia formation
|
CEP290 [HSA:80184] [KO:K16533]
|
D12488 Sepofarsen (USAN/INN)
|
Organismal systems
|
Complement and coagulation
|
F8 [HSA:2157] [KO:K03899]
|
D00291 Desmopressin (INN)
D02235 Desmopressin acetate (USP) <JP/US>
|
F8* [HSA_VAR:2157v1] [HSA:2157] [KO:K03899]
|
D08798 Freeze-dried human blood-coagulation factor VIII <JP>
D05401 Octocog alfa (INN)
D05409 Rurioctocog alfa (genetical recombination) (JAN) <JP>
D08232 Moroctocog alfa (INN)
D10227 Turoctocog alfa (INN) <JP>
D10539 Efraloctocog alfa (genetical recombination) (JAN) <JP>
D10758 Turoctocog alfa pegol (genetical recombination) (JAN) <JP>
D10759 Damoctocog alfa pegol (INN) <JP>
D10760 Rurioctocog alfa pegol (genetical recombination) (JAN) <JP>
D10771 Octocog beta (genetical recombination) (JAN) <JP>
D10818 Lonoctocog alfa (INN) <JP>
D10830 Efmoroctocog alfa (INN)
D10831 Susoctocog alfa (INN) <JP>
D10842 Simoctocog alfa (INN) <JP>
D12441 Efanesoctocog alfa (INN) <JP>
D12434 Valoctocogene roxaparvovec (USAN/INN) <US>
|
VWF [HSA:7450] [KO:K03900]
|
D11160 Caplacizumab (USAN/INN) <JP/US>
D09892 Egaptivon pegol (USAN)
D12863 Rondaptivon pegol
|
VWF* [HSA_VAR:7450v1] [HSA:7450] [KO:K03900]
|
D08798 Freeze-dried human blood-coagulation factor VIII <JP>
|
GP6 [HSA:51206] [KO:K06264]
|
D12413 Glenzocimab (USAN/INN)
|
CFP [HSA:5199] [KO:K15412]
|
D12823 Tarperprumig (USAN/INN)
|
Acute phase protein
|
SAA [HSA:6288 6289] [KO:K17310]
|
D12482 Anselamimab (USAN/INN)
|
Immune system
|
FCGRT [HSA:2217] [KO:K24019]
|
D11876 Efgartigimod alfa (USAN/INN) <JP/US>
D12182 Rozanolixizumab (USAN/INN) <JP/US>
D11666 Nipocalimab (USAN) <JP/US>
D11983 Batoclimab (USAN/INN)
D12144 Orilanolimab (USAN/INN)
|
FCGR2B (CD32) [HSA:2213] [KO:K12560]
|
D11339 Valziflocept (USAN)
|
FCER1A [HSA:2205] [KO:K08089]
|
D05251 Omalizumab (USAN/INN) <JP/US>
D03095 Benzylpenicilloyl polylysine (USP)
|
FCER1G [HSA:2207] [KO:K07983]
|
D03095 Benzylpenicilloyl polylysine (USP)
|
FCRL5 [HSA:83416] [KO:K06727]
|
D11984 Cevostamab (USAN/INN)
|
ALOX5AP [HSA:241] [KO:K20735]
|
D05671 Quiflapon sodium (USAN)
D06664 Veliflapon (USAN/INN)
D10069 Fiboflapon (USAN)
D10122 Fiboflapon sodium (USAN)
|
LGALS3 [HSA:3958] [KO:K06831]
|
D11495 Belapectin (USAN)
D12221 Olitigaltin (USAN)
D12763 Selvigaltin (USAN/INN)
|
MAGEA4 [HSA:4103] [KO:K24127]
|
D12951 Afamitresgene autoleucel (USAN/INN) <US>
|
Circulatory system
|
HBA [HSA:3039 3040] [KO:K13822]
|
D03436 Cellulose, oxidized (JAN/USP)
D06456 Cellulose, oxidized regenerated (USP)
|
HBB [HSA:3043] [KO:K13823]
|
D03436 Cellulose, oxidized (JAN/USP)
D06456 Cellulose, oxidized regenerated (USP)
|
ALB [HSA:213] [KO:K16141]
|
D12823 Tarperprumig (USAN/INN)
D13054 Lunsekimig (USAN/INN)
D13155 Donzakimig (USAN/INN)
D13160 Galvokimig (USAN/INN)
D13227 Sonelokimab (USAN/INN)
|
Digestive system
|
MTTP [HSA:4547] [KO:K14463]
|
D09637 Lomitapide (USAN/INN)
D09638 Lomitapide mesylate (USAN) <JP/US>
D05060 Mitratapide (USAN/INN)
|
APOB [HSA:338] [KO:K14462]
|
D08946 Mipomersen sodium (USAN)
|
APOC3 [HSA:345] [KO:K08759]
|
D11648 Volanesorsen (USAN/INN)
D11650 Volanesorsen sodium (USAN)
D13023 Olezarsen sodium (USAN) <US>
D13206 Plozasiran sodium (USAN) <US>
|
COL7A1 [HSA:1294] [KO:K16628]
|
D12632 Beremagene geperpavec (USAN/INN) <US>
D13121 Prademagene zamikeracel (INN) <US>
|
APOL1 [HSA:8542] [KO:K23585]
|
D12964 Inaxaplin (USAN/INN)
|
Nervous system
|
SNAP25 [HSA:6616] [KO:K18211]
|
D00783 Botulinum toxin type A (JAN) <JP/US>
D02735 RimabotulinumtoxinB (USAN) <US>
D10012 Incobotulinumtoxin A (JAN/USAN) <JP/US>
D10921 DaxibotulinumtoxinA (USAN)
D10949 LetibotulinumtoxinA (USAN) <US>
D11405 PrabotulinumtoxinA (USAN) <US>
|
RGMA [HSA:56963] [KO:K23096]
|
D11355 Elezanumab (USAN/INN)
D12649 Unasnemab (USAN/INN)
|
HTT [HSA:3064] [KO:K04533]
|
D12970 Votoplam (USAN/INN)
|
HTT* [HSA_VAR:3064v1] [HSA:3064] [KO:K04533]
|
D12012 Tominersen sodium (JAN)
D12013 Tominersen (USAN/INN)
|
APP [HSA:351] [KO:K04520]
|
D12873 Sabirnetug (USAN/INN)
D13075 Usilnetug (USAN/INN)
|
Amyloid beta [CPD:C16514 C16515] [HSA:351] [KO:K04520]
|
D11678 Lecanemab (USAN) <JP/US>
|
TMEM97 (S2R) [HSA:27346] [KO:K26171]
|
D13086 Zervimesine (USAN)
|
TREM2 [HSA:54209] [KO:K14378]
|
D12996 Iluzanebart (USAN/INN)
|
Sensory system
|
RBP4 [HSA:5950] [KO:K18271]
|
D12351 Tinlarebant (USAN)
|
Unclassified
|
Newly added
|
DLG4 (PSD95) [HSA:1742] [KO:K11828]
HMGB1 [HSA:3146] [KO:K10802]
KLRD1 (CD94) [HSA:3824] [KO:K06516]
LRP5 [HSA:4041] [KO:K03068]
PMEL [HSA:6490] [KO:K17304]
SFTPB [HSA:6439] [KO:K26067]
SFTPC [HSA:6440] [KO:K26068]
|
No longer used
|
MAP2K1 (MEK1) [HSA:5604] [KO:K04368]
MAP2K2 (MEK2) [HSA:5605] [KO:K04369]
|